Filters
total: 2515
-
Catalog
- Publications 2050 available results
- Journals 164 available results
- People 52 available results
- Inventions 5 available results
- Projects 4 available results
- Laboratories 1 available results
- Research Teams 2 available results
- e-Learning Courses 99 available results
- Events 29 available results
- Open Research Data 109 available results
displaying 1000 best results Help
Search results for: drugi gradient
-
Controlled Drug Release by the Pore Structure in Polydimethylsiloxane Transdermal Patches
Publication -
Pharmaceutical and forensic drug applications of chiral supercritical fluid chromatography
PublicationTHE SUPERCRITICAL FLUID IS AN EXCELLENT CHOICE AS THE CHROMATOGRAPHIC MOBILE PHASE BECAUSE IT ALLOWS RAPID SEPARATION WITH HIGH EFFICIENCY AND APPLICATIONS INVOLVING ENANTIORESOLUTION ARE COMMON. SUPERCRITICAL FLUID CHROMATOGRAPHY (SFC) IS INCREASINGLY USED FOR ANALYTICAL, SEMI-PREPARATIVE AND PREPARATIVE PURIFICATION OF CHIRAL COMPOUNDS, INCLUDING PRODUCTION OF ENANTIOMERS THAT ARE MAINLY ENCOUNTERED DURING DRUG DEVELOPMENT. SFC...
-
Mesoporous silica nanoflakes – Biocompatibility, cellular uptake and drug transport
Publication -
The Role of miRNA-7 in the Biology of Cancer and Modulation of Drug Resistance
Publication -
Diatomaceous earth as a drug-loaded carrier in a glass-ionomer cement
PublicationThe effect of a natural filler (diatomaceous earth [DE], a promising drug-delivery agent) and its content was investigated on the performance of a model glass-ionomer cement (GIC). Three sample series, differing in DE content (0, 2.5 and 5 wt%), were prepared using a commercial GIC as a matrix (3M Ketac Molar Easymix). The resultant surface microhardness and roughness, wear performance, and compressive strength of the samples were...
-
Phosphorus pools and internal loading in a eutrophic lake with gradients in sediment geochemistry created by land use in the watershed
Publication -
An Assessment of RASSCF and TDDFT Energies and Gradients on an Organic Donor−Acceptor Dye Assisted by Resonance Raman Spectroscopy
PublicationThe excitation energies and gradients in the ground and the first excited state of a novel donor−(π- bridge)−acceptor 4-methoxy-1,3-thiazole-based chromophore were investigated by means of MS-RASPT2/RASSCF and TDDFT in solution. Within both methods, the excitation energies strongly depend on the employed equilibrium structures, whose differences can be rationalized in terms of bond length alternation indexes. It is shown that functionals with...
-
STUDENTS' PERCEPTION OF E-GRADING: INFORMATICS COURSE CASE STUDY
PublicationUsing computers for grading can simplify work for teachers. However it is a sensitive part of their work and must be performed carefully. More information is required on students' reception and opinions about e-grading. This paper is a case study of e-grading used in Informatics course and discusses results obtained from surveying the students after being graded by a teacher and a computer.
-
ANALYSIS OF CLIMATIC ZONES IN POLAND WITH REGARD TO ASPHALT PERFORMANCE GRADING
PublicationTowards the end of the last century a new system of bitumen grading was developed and implemented as part of the American Strategic Highway Research Program (SHRP). Its aim was to better adjust the testing methods and requirements for road bitumens to the actual conditions in which those bitumens serve in road pavements. Currently in Poland, similarly as in the other EU countries, road bitumens are tested and classified with regard...
-
Torsional stability capacity of a nano-composite shell based on a nonlocal strain gradient shell model under a three-dimensional magnetic field
PublicationThis paper considers a single-walled composite nano-shell (SWCNS) exposed in a torsional critical stability situation. As the magnetic field affects remarkably nanostructures in the small size, a three-dimensional magnetic field is assessed which contains magnetic effects along the circumferential, radial and axial coordinates system. Based on the results of the nonlocal model of strain gradient small-scale approach and the first-order...
-
On well-posedness of the first boundary-value problem within linear isotropic Toupin–Mindlin strain gradient elasticity and constraints for elastic moduli
PublicationWithin the linear Toupin–Mindlin strain gradient elasticity we discuss the well-posedness of the first boundary-value problem, that is, a boundary-value problem with Dirichlet-type boundary conditions on the whole boundary. For an isotropic material we formulate the necessary and sufficient conditions which guarantee existence and uniqueness of a weak solution. These conditions include strong ellipticity written in terms of higher-order...
-
Badania systemów powstrzymujących pojazd przed wypadnięciem z drogi - cz. II
PublicationW artykule zaprezentowana została tematyka systemów powstrzymujących pojazd przed wypadnięciem z drogi. Podczas codziennego użytkowania dróg występuje szereg zagrożeń, które wpływają na bezpieczeństwo. Badanie, identyfikacja i klasyfikacja zagrożeń stanowią istotny element utrzymania dróg. Artykuł stanowi drugą część podjętej problematyki. Pierwsza została opublikowana w magazynie Mosty nr 3-4/19 str. 66-68.
-
Studies of human and veterinary drugs' fate in environmental solid samples- analytical problems.
PublicationW różnych ośrodkach naukowych na całym świecie trwają prace nad poznaniem losu środowiskowego zanieczyszczeń z grupy farmaceutyków. Obecność pozostałości farmaceutycznych w poszczególnych elementach środowiska stanowi nowe wyzwanie zarówno z punktu widzenia technologii oczyszczania wód i ścieków jak i analityków, których zadaniem jest opracowanie nowych metodyk analitycznych. W publikacji przedstawiono problemy z jakimi stykają...
-
The Comparison Between the Calculated and HPLC-Predicted Lipophilicity Parameters for Selected Groups of Drugs
Publication -
Activity evaluation of some psychoactive drugs with the application of QSAR/QSPR modeling methods
Publication -
European Society of Hypertension Working Group on Obesity: obesity drugs and cardiovascular outcomes
Publication -
Detrimental effects of chemotherapeutics and other drugs on the endothelium: A call for endothelial toxicity profiling
Publication -
Wyznaczanie drogi tarcia w warunkach ślizgania oscylacyjnego o małej amplitudzie.
PublicationW pracy omówiono sposób wyznaczania drogi tarcia w warunkach ruchu oscylacyjnego o małej amplitudzie, która jak wykazały badania, w takim przypadku dla niemetalowych materiałów łożyskowych różni się znacząco od nominalnej drogi ślizgania. Jest to spowodowane postaciowymi odkształceniami materiału umożliwiającymi ruch względny czopa i panwi bez poślizgu na powierzchni styku. Zaproponowana metoda umożliwia uwzględnienie tego zjawiska....
-
Interaction of selected drugs with food in the group of patients over 60 years of age
Publication -
Stable and degradable microgels linked with cystine for storing and environmentally triggered release of drugs
PublicationEnvironmentally sensitive, degradable microgels based on poly(N-isopropylacrylamide) (pNIPA) crosslinked with the diacryloyl derivative of cystine (BISS) were synthesized by applying surfactant-free emulsion polymerization. pNIPA contributed the sensitivity to temperature to the microgels and the cross-linker made them degradable and sensitive to pH. The morphology of the microgels was investigated by using scanning and transmission...
-
Impact of selected drugs and their binary mixtures on the germination of Sorghum bicolor (sorgo) seeds
PublicationThe aim of this study was to assess the toxicological potential of binary drug mixtures and individual drugs under different pH conditions with different inorganic ion additions on the germination of Sorghum bicolor (sorgo) seeds. To assess whether the given drug mixtures were more phytotoxic than the individual compounds, concentration addition (CA) and independent action (IA) approaches were applied to estimate the predicted...
-
Badania systemów powstrzymujących pojazd przed wypadnięciem z drogi - cz. I
PublicationTransportation systems are designed and used so as to effectively and safely relocate people, goods and services. Despite this there are numerous hazards that disrupt or damage these systems. Risks such as extreme weather conditions, terrorist threats, landsliders or earthquakes are difficult to predict, manage and mitigate. One of the hazards for transportation systems are accidents, and their impact on the transport functioning...
-
HYGRO-MAGNETIC VIBRATION OF THE SINGLE-WALLED CARBON NANOTUBE WITH NONLINEAR TEMPERATURE DISTRIBUTION BASED ON A MODIFIED BEAM THEORY AND NONLOCAL STRAIN GRADIENT MODEL
PublicationIn this study, vibration analysis of single-walled carbon nanotube (SWCNT) has been carried out by using a refined beam theory, namely one variable shear deformation beam theory. This approach has one variable lesser than a contractual shear deformation theory such as first-order shear deformation theory (FSDT) and acts like classical beam approach but with considering shear deformations. The SWCNT has been placed in an axial or...
-
Detection ofHelicobacterspecies in liver and stomach tissues of patients with chronic liver diseases using polymerase chain reaction-denaturing gradient gel electrophoresis and immunohistochemistry
Publication -
Simultaneous determination of hydrophobicity and dissociation constant for a large set of compounds by gradient reverse phase high performance liquid chromatography–mass spectrometry technique
Publication -
Damped forced vibration analysis of single-walled carbon nanotubes resting on viscoelastic foundation in thermal environment using nonlocal strain gradient theory
PublicationIn this paper, the damped forced vibration of single-walled carbon nanotubes (SWCNTs) is analyzed using a new shear deformation beam theory. The SWCNTs are modeled as a flexible beam on the viscoelastic foundation embedded in the thermal environment and subjected to a transverse dynamic load. The equilibrium equations are formulated by the new shear deformation beam theory which is accompanied with higher-order nonlocal strain...
-
Modification of gradient HPLC method for determination of small molecules' affinity to human serum albumin under column safety conditions: Robustness and chemometrics study
PublicationIn the early stages of drug discovery, beyond the biological activity screening, determining the physicochemical properties that affect the distribution of molecules in the human body is an essential step. Plasma protein binding (PPB) is one of the most important investigated endpoints. Nevertheless, the methodology for measuring %PPB is significantly less popular and standardized than other physicochemical properties, like lipophilicity....
-
MM/PBSA analysis of molecular dynamics simulations of bovine beta-lactoglobulin: free energy gradients in conformational transitions?
PublicationPraca dotyczy pH zależnych zmian konformacyjnych EF pętli beta-laktoglobuliny. Zmiany te są śledzone za pomocą metod obliczeniowych chemii (dynamika molekularna oraz metody MM/PBSA).
-
BIOPHARMACEUTICS & DRUG DISPOSITION
Journals -
CLINICAL DRUG INVESTIGATION
Journals -
DRUG NEWS & PERSPECTIVES
Journals -
DRUG INFORMATION JOURNAL
Journals -
Drug Target Insights
Journals -
Drug Discoveries and Therapeutics
Journals -
Drug Testing and Analysis
Journals -
CNS DRUG REVIEWS
Journals -
Journal of Drug Delivery
Journals -
DRUG DISCOVERY TODAY
Journals -
DRUG RESISTANCE UPDATES
Journals -
Current Drug Safety
Journals -
BIOINFO Drug targets
Journals -
Drug Metabolism and Pharmacokinetics
Journals -
Current Drug Therapy
Journals -
JOURNAL OF DRUG ASSESSMENT
Journals -
DRUG AND ALCOHOL REVIEW
Journals -
Drug and Therapeutics Bulletin
Journals -
Drug Discovery World
Journals -
Drug Metabolism Letters
Journals -
Drug Delivery Letters
Journals -
WHO Drug Information
Journals