Filtry
wszystkich: 2110
wybranych: 1647
-
Katalog
- Publikacje 1647 wyników po odfiltrowaniu
- Czasopisma 6 wyników po odfiltrowaniu
- Osoby 173 wyników po odfiltrowaniu
- Wynalazki 3 wyników po odfiltrowaniu
- Projekty 17 wyników po odfiltrowaniu
- Zespoły Badawcze 1 wyników po odfiltrowaniu
- Kursy Online 45 wyników po odfiltrowaniu
- Wydarzenia 2 wyników po odfiltrowaniu
- Dane Badawcze 216 wyników po odfiltrowaniu
Filtry wybranego katalogu
wyświetlamy 1000 najlepszych wyników Pomoc
Wyniki wyszukiwania dla: N,O‐ ANDN,N‐DONORS
-
2,4,6-Trimethylbenzamide.
PublikacjaAnaliza rentgenograficzna monokryształu 2,4,6-trimetylobenzamidu wykazała, że cząsteczki imidu oddziałują ze sobą poprzez wiązania wodorowe typu N-H...O=C tworząc motyw C(4). Takie uporządkowanie cząsteczek w sieci krystalicznej jest dodatkowo stabilizowane poprzez słabe oddziaływanie typu N-H...pi pomiędzy atomem syn-H grupy amidowej a pierścieniem aromatycznym. Wzajemne ułożenie grupy amidowej i pierścienia aromatycznego jest...
-
W-like bound entangled states and secure key distillation
PublikacjaWe construct multipartite entangled states with underlying W-type structuresatisfying positive partial transpose (PPT) condition under any (N −1)|1 partition. Then we showhow to distill a N-partite secure key from the states using two different methods: direct applicationof local filtering and novel random key distillation scheme in which we adopt the idea from recentresults on entanglement distillation. Open problems and possible...
-
Ex situ XANES, XPS and Raman studies of poly(3,4-ethylenedioxythiophene)modified by iron hexacyanoferrate
PublikacjaPraca dotyczy badań XANES, XPS i Ramana polimeru przewodzącego poli(3,4-etylenodioksytiofenu) modyfikowanego heksacyjanożelazianem żelaza. Badania XANES potwierdziły oktaedryczne otoczenie atomu żelaza, którego najbliższymi sąsiadami są atomy węgla oraz atomy azotu. Badania XPS wykazały istnienie wiązań Fe-C, Fe-N oraz chemicznego oddziaływania między atomem siarki polimeru a atomem żelaza błękitu pruskiego. Obecność oddziaływań...
-
The selective salinity and hydrazine parameters for the start-up of non-anammox-specific biomass SBR
PublikacjaThe presence of ammonium (NH 4+ ) in wastewater above the permissible limits leads to undesirable ecological impact and public health concerns. In this study, the anaerobic ammonium oxidizing (anammox) bacteria-mediated nitrogen removal was investigated using a sequential batch reactor (SBR). Effects of different salinity levels were evaluated on the bacterial activity at: mild (below 0.2 g NaCl/L), elevated (18.2 g NaCl/L) and...
-
Interactions between polyphenolic antioxidants quercetin and naringenin dictate the distinctive redox-related chemical and biological behaviour of their mixtures
PublikacjaFood synergy concept is suggested to explain observations that isolated antioxidants are less bioactive than real foods containing them. However, mechanisms behind this discrepancy were hardly studied. Here, we demonstrate the profound impact of interactions between two common food flavonoids (individual: aglycones quercetin—Q and naringenin—N− or their glycosides rutin—R and naringin—N+ vs. mixed: QN− and RN+) on their electrochemical...
-
Application of the Electronic Nose Technique to Differentiation between Model Mixtures with COPD Markers
PublikacjaABSTRACT The paper presents the potential of an electronic nose technique in the field of fast diagnostics of patients suspected of Chronic Obstructive Pulmonary Disease (COPD). The investigations were performed using a simple electronic nose prototype equipped with a set of six semiconductor sensors manufactured by FIGARO Co. They were aimed at verification of a possibility of differentiation between model reference mixtures with...
-
The influence of chemical composition of amide block on the thermal properties and structure of terpoly(ester-b-ether-b-amide) elastomers
PublikacjaMultiblock terpolymers-(PBT-b-PTMO-b-PA12,10)(n)- constituting the polymer systems, in which one of the three blocks (PBT) does not dissolve in PA12,10 block (hard phase) and, depending on its molecular weight is slightly soluble in PTMO block (soft phase), have been obtained. The DSC method was applied to investigate the thermal properties of these polymers and it was found that PBT block acts as an element that produces stiffness...
-
3,3'-Dibenzoyl-1,1'-dibenzyl-1,1'-(ethane-1,2-diyl)dithiourea
PublikacjaIn the title compound, C32H30N4O2S2, the carbonyl and thiocarbonyl groups are found in a rare synclinal conformation, with an S-C···C-O pseudo-torsion angle of 62.6(2)°. The molecule has Ci = S2 point-group symmetry with a crystallographic center of inversion located in the middle of the ethylene bridge. One of the symmetry-independent phenyl...
-
On a Recurrence Arising in Graph Compression
PublikacjaIn a recently proposed graphical compression algorithm by Choi and Szpankowski (2012), the following tree arose in the course of the analysis. The root contains n balls that are consequently distributed between two subtrees according to a simple rule: In each step, all balls independently move down to the left subtree (say with probability p) or the right subtree (with probability 1p). A new node is created as long as...
-
Systemic modulation of stress and immune parameters in patients treated for prostate adenocarcinoma by intensity-modulated radiation therapy or stereotactic ablative body radiotherapy
Publikacja -
Dissociation and fragmentation of furan by electron impact
PublikacjaDissociation and fragmentation processes that produce electronically excited atomic and molecular fragments, following electron impact excitation, have been studied in furan. The optical excitation technique has been employed over the electron incident energy range 15-95 eV. Formation of excited hydrogen atoms H(n) in the n = 4-10 states has been detected by observation of the Balmer series. The diatomic CH fragments are formed...
-
Radzenie sobie ze stresem w warunkach różnego stopnia zagrożenia zdrowia.
PublikacjaCelem pracy była ocena zróżnicowania podejmowanych strategii zaradczych oraz siły poczucia koherencji u kobiet w różnym stanie zdrowia. W badaniu uczestniczyły kobiety zdrowe (n=79), zagrożone chorobą nowotworową (n=41) oraz chore na nowotwór narządów rodnych (n=118). Stwierdzono, że w stanach deficytu zdrowia preferowane są strategie emocjonalne, a w zdrowiu - instrumentalne. Dominującą strategią w radzeniu sobie z chorobą nowotworową...
-
Interactions in Ternary Aqueous Solutions of NMA and Osmolytes—PARAFAC Decomposition of FTIR Spectra Series
PublikacjaIntermolecular interactions in aqueous solutions are crucial for virtually all processes in living cells. ATR-FTIR spectroscopy is a technique that allows changes caused by many types of such interactions to be registered; however, binary solutions are sometimes difficult to solve in these terms, while ternary solutions are even more difficult. Here, we present a method of data pretreatment that facilitates the use of the Parallel...
-
Interactions of amphotericin B derivative of low toxicity with biological membrane components - the Langmuir monolayer approach
PublikacjaMetodą monowarstw Langmuira zbadano naturę oddziaływań nowej pochodnej antybiotyku przeciwgrzybowego amfoterycyny B o niskiej toksyczności, tj. estru metylowego N-metylo-N-D-fruktopiranozyloamfoterycyny B (MF-AME)z komponentami błon biologicznych: ergosterolem, występującym w komórkach grzybowych i cholesterolem występującym w komórkach zwierzęcych oraz z modelowym fosfolipidem DPPC i na tej podstawie stwierdzono, że zróżnicowanie...
-
Cytotoxic and Antioxidant Activities of Benzohydroxamic Acid Analogues
Publikacja20 benzohydroxamic acid analogues were synthesized and evaluated for their in vitro cytotoxicities against mouse mammary tumor cells as well as antioxidant activities against DPPH radical and superoxide anion. It was found that benzothiohydroxamic acids exhibit greater cytotoxicities than benzohydroxamic acids and N-isopropyl derivatives are more active than N-methyl ones. On the other hand, benzothiohydroxamic acids show more...
-
Polyhedral Ramsey Numbers
PublikacjaGiven two polygons or polyhedrons P1 and P2, we can transform these figures to graphs G1 and G2, respectively. The polyhedral Ramsey number Rp(G1,G2) is the smallest integer n such that every graph, which represents polyhedron on n vertices either contains a copy of G1 or its complement contains a copy of G2. Using a computer search together with some theoretical results we have established some polyhedral Ramsey numbers, for example...
-
Electron impact fragmentation of pyrrole molecules studied by fluorescence emission spectroscopy
PublikacjaThe fluorescence emission spectroscopy using electron impact excitation technique was employed to study fragmentation processes of the gas phase pyrrole molecules. The following excited fragmentation species were observed by detection of their fluorescence decay: the atomic hydrogen H(n), n = 4-7 and the diatomic CH(A2Δ), CN(B2Σ+), NH(A3Π) and C2(d3Πg) fragments. These atomic and molecular products differ from those previously...
-
Asynchronous time difference of arrival (ATDOA) method
PublikacjaA new method for a location service in the asynchronous wireless sensor networks is outlined. This method, which is called asynchronous time difference of arrival (ATDOA), enables calculation of the position of a mobile node without knowledge of relative time differences (RTDs) between measuring sensors. The ATDOA method is based on the measurement of time difference of arrival between the node and the same sensor at the discrete...
-
Fluctuation of nitrogen fraction during wastewater treatment in a multistage treatment wetland
PublikacjaFactors influencing COD and removal and transformation of N fractions have been investigatedin the conditions of horizontal (SSHF) and vertical (SSVF) flow reed beds. Multistage treatment wetlandin Wiklino ensured a stable and very effective removal of all the analysed pollutants. Based onthe resultsof investigation, it could be assumed that the working conditions of SSHF beds play an importantrole in the transformation of particulate...
-
Amides as models to study the hydration of proteins and peptides — spectroscopic and theoretical approach on hydration in various temperatures
PublikacjaInteractions with water are one of the key factors which determine protein stability and activity in aqueous solutions. However, the protein hydration is still insufficiently understood. N-methylacetamide (NMA) is regarded as a minimal part of the peptide backbone and the relative simplicity of its structure makes it a good model for studies on protein–water interactions. In this paper, the influence of NMA and N,N-dimethylacetamide...
-
Novel nitrogen precursors for electrochemically driven doping of titania nanotubes exhibiting enhanced photoactivity
PublikacjaNitrogen doped titania nanotubes were successfully sensitized by electrochemical method, i.e. as-anodized titania was immersed in different amine (diethyleneamine-DETA, triethyleneamine-TEA, ethylenediamine-EDA) and urea (U) solution and a constant potential was applied. The highly ordered morphology of fabricated N-TiO2 was investigated by using scanning electron microscopy. Spectroscopic techniques, i.e. UV-Vis spectroscopy,...
-
(R,R)-1-Acetyl-1'-(2,4,6-trinitrophenyl)-2,2'-bipyrrolidine
Publikacja(R,R)-1-Acetyl-1'-(2,4,6-trinitrophenyl)-2,2'-bipyrrolidine has been synthesized and its rentgenostructure has been determined. The structure of the title molecule, C16H19N5O7, is mainly determined by the steric effect of a bulky 2,4,6-trinitrophenyl group attached to the N atom of a pyrrolidine ring. Both pyrrolidine rings adopt an envelope conformation, with one of the methylene C atoms as the flap in each case, and the N-C-C-N...
-
Collision-Free Network Exploration
PublikacjaA set of mobile agents is placed at different nodes of a n-node network. The agents synchronously move along the network edges in a collision-free way, i.e., in no round may two agents occupy the same node. In each round, an agent may choose to stay at its currently occupied node or to move to one of its neighbors. An agent has no knowledge of the number and initial positions of other agents. We are looking for the shortest possible...
-
Concentrations of alfa- and gamma- tocopherols in human breast milk during the first months of lactation and in infant formulas
PublikacjaThe aim of this study was to determine the concentrations of alpha- and gamma-tocopherols in human breast milk samples from different periods of lactation and to compare them with tocopherol content in commercially available formulas for infants at corresponding ages. The study included 93 breast milk samples obtained on the 2nd (colostrum, n=17), 14th (n=30), 30th (n=27) and 90th day of lactation (n=19), along with 90 samples...
-
Population-based case-control study of alpha 1-antitrypsin and SLC11A1 in Crohn's disease and ulcerative colitis.
PublikacjaBackground: Crohn’s disease (CD) and ulcerative colitis (UC) are chronic inflammatory diseases of the digestive tract. Genetic factors and an abnormal immune response to infections are suspected to be involved in inflammatory bowel diseases. Methods: In the present study 300 blood samples from CD patients (n 100), UC patients (n 100), and healthy controls (n 100) were taken from a population-based case-control study. PCR assays...
-
Przemiany azotu organicznego w komunalnych oczyszczalniach ścieków
PublikacjaW pracy przedstawiono przemiany koloidalnego i rozpuszczonego azotu organicznego w komorach osadu czynnego czterech komunalnych oczyszczalni ścieków zlokalizowanych w Polsce północnej. Średnie stężenia DON i CON w ściekach oczyszczonych mechanicznie zmieniały się w zakresie 1,8-2,9 g N/m3 oraz 7,6-13,6 g N/m3, co stanowiło odpowiednio 4,9-8,3% oraz 16,6-41,1% azotu organicznego. W ściekach oczyszczonych biologicznie zaobserwowano...
-
Computational analysis of substituent effects on proton affinity and gas-phase basicity of TEMPO derivatives and their hydrogen bonding interactions with water molecules
PublikacjaThe study investigates the molecular structure of 2,2,6,6-tetramethylpiperidine-1-oxyl (TEMPO) and its derivatives in the gas phase using B3LYP and M06-2X functional methods. Intermolecular interactions are analyzed using natural bond orbital (NBO) and atoms in molecules (AIM) techniques. NO2-substituted TEMPO displays high reactivity, less stability, and softer properties. The study reveals that the stability of TEMPO derivatives...
-
Combined effect of nitrogen-doped functional groups and porosity of porous carbons on electrochemical performance of supercapacitors
PublikacjaIn this work, nitrogen-doped porous carbons obtained from chitosan, gelatine, and green algae were investigated in their role as supercapacitor electrodes. The effects of three factors on electrochemical performance have been studied— of the specific surface area, functional groups, and a porous structure. Varying nitrogen contents (from 5.46 to 10.08 wt.%) and specific surface areas (from 532 to 1095 m2g−1) were obtained by modifying...
-
European Multicenter Evaluation of High-Density DNA Probe Arrays for Detection of Hepatitis B Virus Resistance Mutations and Identification of Genotypes
Publikacja -
Dielectric Spectroscopy Studies and Modelling of Piezoelectric Properties of Multiferroic Ceramics
PublikacjaCompounds and solid solutions of bismuth ferrite (BiFeO3)—barium titanate (BaTiO3) system are of great scientific and engineering interest as multiferroic and potential high-temperature lead-free piezoelectric materials. In the present paper, the results of research on the synthesis and characterisation of 0.67Bi1.02FeO3–0.33BaTiO3 (67BFBT) ceramics in terms of crystal structure and dielectric and piezoelectric properties are reported....
-
Global defensive sets in graphs
PublikacjaIn the paper we study a new problem of finding a minimum global defensive set in a graph which is a generalization of the global alliance problem. For a given graph G and a subset S of a vertex set of G, we define for every subset X of S the predicate SEC ( X ) = true if and only if | N [ X ] ∩ S | ≥ | N [ X ] \ S | holds, where N [ X ] is a closed neighbourhood of X in graph G. A set S is a defensive alliance if and only if for...
-
Effect of lag screw on stability of first metatarsophalangeal joint arthrodesis with medial plate
PublikacjaBackground: First metatarsophalangeal joint (MTP-1) arthrodesis is a commonly performed procedure in the treatment of disorders of the great toe. Since the incidence of revision after MTP-1 joint arthrodesis is not insignificant, a medial approach with a medially positioned locking plate has been proposed as a new technique. The aim of the study was to investigate the effect of the application of a lag screw on the stability and...
-
Incorporation of the sulfur cycle in sustainable nitrogen removal systems - A review
PublikacjaIn wastewater treatment systems, sulfur (S) removal processes are generally based on heterotrophic sulfate (SO42−) reduction by sulfate reducing bacteria and S-dependent autotrophic denitrification by sulfur oxidizing bacteria. A combination of either two cycles (N and S) or three cycles (N, S and C) appears to be a viable approach to sustainable wastewater treatment, resulting in energy savings and reduction of sludge production....
-
Automatic Regularization by Quantization in Reducible Representations of CCR: Point-Form Quantum Optics with Classical Sources
PublikacjaElectromagnetic fields are quantized in a manifestly covariant way by means ofa class of reducible "center-of-mass N-representations" of the algebra of canonical commutationrelations (CCR). The four-potential Aa(x) transforms in these representations as aHermitian four-vector field in Minkowski four-position space (without change of gauge), butin momentum space it splits into spin-1 massless photons and two massless scalars. Whatwe...
-
Cubane Like Structure of a Silanethiol Primary Amine Assembly a Novel, Unusual Hydrogen Bond Pattern.
PublikacjaMetodą rentgenowskiej analizy strukturalnej wyznaczono struktury krystaliczne i cząsteczkowe trzech soli amoniowych: (t-BuO)3SiS(-)H3N(+)Bu-t, (i-PrO)3SiS(-)H3N(+)Bu-t i (t-BuO)3SiS(-)H3N(+)(CH2)2CH(CH3)2. Wszystkie trzy związki w ciele stałym tworzą tetramery w których atomy S i N wyznaczają w przybliżeniu naroża sześcianu. Trwałość tych agregatów, oprócz sił elektrostatycznego przyciągania, zapewnia sieć wiązań wodorowych N-H
-
Characteristic of Morpholinium Ionic Liquids as Gas Chromatography Stationary Phases with McReynolds Constants and Activity Coefficients at Infinite Dilution
PublikacjaIn this work, four ionic liquids based on N-alkyl-N-methylmorpholinium cation ([Mor1,R] where R= 2, 4, 8, 10) and bis(trifluoromethanesulfonyl)imide anion [TFSI] were synthesized. Using gas-liquid chromatography a number of parameters describing the sorption properties of the investigated ionic liquids were determined. The values of Kovats indices, McReynolds constants, and activity coefficients at infinite dilution were the basis...
-
Strategia wektorowej modulacji szerokości impulsów dla wielofazowych falowników napięcia
PublikacjaW artykule zaproponowano strategię wektorowej modulacji szerokości impulsów dla wielofazowych falowników napięcia. Zaproponowane rozwiązanie pozwala na niezależne formowanie napięć wyjściowych w n-fazowym falowniku dwupoziomowym z wykorzystaniem (n-1) wektorów aktywnych. Przedstawiony algorytm modulacji umożliwia dobór sekwencji wektorów aktywnych i pasywnych wymagającej minimalnej liczby przełączeń...
-
Ammonia amendment promotes high rate lactate production and recovery from semi-continuous food waste fermentation
PublikacjaIn this study, a reliable approach using ammonia nitrogen was proposed to increase lactate production during semi-continuous food waste (FW) fermentation under mesophilic conditions. Both free ammonia nitrogen (FAN) and ammonium ion (NH4+-N) were present in mesophilic reactors, with a wide FAN/NH4+-N ratio variation due to the intermittent pH control. The investigation of responsible mechanisms revealed that the increased production...
-
Place Attachment and Collective Action Tendency
PublikacjaThree studies were carried out to examine how place attachment and collective action tendency are related and what role self-expansion and social interactions play in this relationship. In the first study (N = 156) we found that a more active form of attachment – place discovered – is a significant predictor of tendency to engage in collective action in favor of one’s neighborhood. In the second study (N = 197), we focused on...
-
Partially Isolated Multi-Active Bridge DC-DC Converter with Bidirectional EV Charging Ports
PublikacjaThere is a growing interest in multiport converters due to their ability to interconnect various energy sources and loads using reduced number of components. Regarding electric vehicle (EV) chargers connection, existing multiport solutions either lack scalability, featuring only one isolated charging port or the operation of ports depend on each other, complicating the converter control algorithm. This article proposes a partially...
-
Universal Augmentation Schemes for Network Navigability
PublikacjaRozważano problem uzupełniania grafu (reprezentującego np. sieci społeczne) poprzez dodanie w każdym węźle jednego dodatkowego skierowanego połączenia (długodystansowego). Dokładniej, dla każdego węzła definiuje się listę prawdopodobieństw istnienia połączenia wychodzącego z danego węzła do wszystkich pozostałych węzłów; wartości tych prawdopodobieństw muszą sumować się do jedności. Routing zachłanny w takiej sieci polega na przekazywaniu...
-
The role of SSVF and SSHF beds in concentrated wastewater treatment, design recommendation
PublikacjaThe return flows of reject water from sewage sludge dewatering alter the activated sludge process ina conventional WWTP and increase TN concentration in the final effluent from WWTP. The objectiveof the investigation carried out was to consider the application of multistage treatment wetland(MTW) for the treatment of reject water from sewage sludge dewatering in a centrifuge (RWC). Thispaper aims to present the design and performance...
-
Odpady z produkcji alkoholu jako alternatywne źródła węgla dla wspomagania denitryfikacji w komunalnych oczyszczalniach ścieków
PublikacjaZaprezentowane w artykule wyniki badań potwierdziły, że produkty odpadowe z destylarni mogą stanowić alternatywę dla komercyjnych źródeł węgla zewnętrznego (np. etanol) stosowanych do wspomagania procesu denitryfikacji. Dozowanie syropu lub odcieku powodowało natychmiastowy wzrost SDN (ponad 3 g N/(kg s.m.o.•h)), natomiast SDN z olejem fuzlowym i niezaadaptowanym osadem czynnym były stosunkowo niskie (< 2 g N/(kg s.m.o.•h)). Należy...
-
A note on the Morse homology for a class of functionals in Banach spaces involving the 2p-area functional
PublikacjaIn this paper we show how to construct Morse homology for an explicit class of functionals involving the 2p-area functional. The natural domain of definition of such functionals is the Banach space W_0^{1,2p}(\Omega), where p > n/2 and \Omega \subet R^n is a bounded domain with sufficiently smooth boundary. As W_0^{1,2p}(\Omega) is not isomorphic to its dual space,critical points of such functionals cannot be non-degenerate...
-
Effects of different external carbon sources and electron acceptors on interactions between denitrification and phosphorus removal in BNR processes
PublikacjaThe effects of two different external carbon sources (acetate, ethanol) and electron acceptors (dissolved oxygen, nitrate and nitrite) were investigated under aerobic and anoxic conditions with non-acclimated process biomass from a full-scale biological nutrient removal activated sludge system. When acetate was added as an external carbon source, phosphate release was observed even in the presence of electron acceptors. The release...
-
On the time behaviour of Okazaki fragments
PublikacjaW pracy wyprowadzono wzory na prawdopodobieństwo, że podczas procesu replikacji DNA w chwili t pojawi się n fragmentów Okazaki.
-
A note on polynomial algorithm for cost coloring of bipartite graphs with Δ ≤ 4
PublikacjaIn the note we consider vertex coloring of a graph in which each color has an associated cost which is incurred each time the color is assigned to a vertex. The cost of coloring is the sum of costs incurred at each vertex. We show that the minimum cost coloring problem for n-vertex bipartite graph of degree ∆≤4 can be solved in O(n^2) time. This extends Jansen’s result [K.Jansen,The optimum cost chromatic partition problem, in:...
-
Cooperative mobile guards in grids
PublikacjaPraca dotyczy problemu strzeżenia dwuwymiarowych krat ortogonalnych, przy założeniu, że obszar widoczności strażnika obejmuje jedną ulicę oraz wszystkie ulice ją przecinające. Rozważano wariant straży słabo współpracujących, w którym dodatkowo każdy strażnik musi widzieć przynajmniej jednego innego strażnika. Podano dowód NP-trudności problemu optymalizacyjnego w przypadku ogólnym, algorytm dokładny o złożoności O(n log n) dla...
-
Bismuth germanate and bismuth silicate glasses in cryogenic detectors.
PublikacjaStwierdzono, że przewodnictwo elektryczne redukowanych szkieł silnie zależy od temperatury, czasu reakcji i koncentracji Bi. Zależność przewodnictwa elektrycznego od temperatury jest dobrze opisana przez funkcję ĺ~exp[-(T0/T)n,gdzie n=1/4. Współczynnik emisji wtórnej elektronów jest praktycznie niezależny od stopnia redukcji ale znacznie rośnie po domieszkowaniu szkieł alkalicznymi jonami. Badania dowiodły, że modyfikowane...
-
Synthesis and biological activity of ester derivatives of mycophenolic acid and acridines/acridones as potential immunosuppressive agents
PublikacjaImproved derivatives of mycophenolic acid (MPA) are necessary to reduce the frequency of adverse effects, this drug exerts in treated patients. In this study, MPA was coupled with N-(x-hydroxyalkyl)-9-acridone-4-carboxamides or N-(x-hydroxyalkyl)acridine-4-carboxamides to give respective ester conjugates upon Yamaguchi protocol. This esterification required protection of phenol group in MPA. Designed conjugates revealed higher...