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Wyniki wyszukiwania dla: PROTEASE ACTIVITY
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The LD loop as an important structural element required for transmission of the allosteric signal in the HtrA (DegP) protease from Escherichia coli
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Regulation of the First Committed Step in Lipopolysaccharide Biosynthesis Catalyzed by LpxC Requires the Essential Protein LapC (YejM) and HslVU Protease
PublikacjaWe previously showed that lipopolysaccharide (LPS) assembly requires the essential LapB protein to regulate FtsH-mediated proteolysis of LpxC protein that catalyzes the first committed step in the LPS synthesis. To further understand the essential function of LapB and its role in LpxC turnover, multicopy suppressors of ΔlapB revealed that overproduction of HslV protease subunit prevents its lethality by proteolytic degradation...
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Structure-activity relationship studies on the antimicrobial activity of novel edeine a and d analogues
PublikacjaOpisano syntezę 4 nowych analogów peptydowego antybiotyku, edeiny a i d z wykorzystaniem klasycznej syntezy w roztworze. Stosowano metodę estrów aktywnych oraz metodę azydową do tworzenia wiązań peptydowych. Zbadano także aktywność przeciwgrzybową i przeciwbakteryjną opisanych połączeń.
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Bladder cancer detection using a peptide substrate of the 20S proteasome
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An update on medium- and low-abundant blood plasma proteome of horse
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Effects of Primary Processing and Pre-Salting of Baltic Herring on Contribution of Digestive Proteases in Marinating Process
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Screening of potential inhibitors for COVID-19 main protease from phytoconstituents of Tectona grandis Linn: application of molecular modeling studies
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Substrate profiling of Finegoldia magna SufA protease, inhibitor screening and application to prevent human fibrinogen degradation and bacteria growth in vitro
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Development of potent and effective SARS-CoV-2 main protease inhibitors based on maleimide analogs for the potential treatment of COVID-19
PublikacjaIn the present work, we report a new series of potent SARS-CoV-2 Main Protease (Mpro) inhibitors based on maleimide derivatives. The inhibitory activities were tested in an enzymatic assay using recombinant Mpro (3CL Protease from coronavirus SARS-CoV-2). Within the set of new Mpro inhibitors, 6e demonstrated the highest activity in the enzymatic assay with an IC50 value of 8.52 ± 0.44 mM. The IC50 value for Nirmatrelvir (PF-07321332,...
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Innovative activity of SMEs In Poland
PublikacjaInnovative activity of enterprises is determined by many factors. On one hand, these are external factors creating a sort of innovative climate in the economy, on the other hand - there are many internal factors stimulating or reducing the intensity of innovative activities. What influences the innovativeness of enterprises is the effectiveness of the system supporting innovations, which was stated by for example Pyciński and Żołnierski...
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Photocatalytic Activity ofTiO2-WO3Composites
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Antimicrobial activity of Potentilla species
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Effect of chronic mild stress and imipramine on the proteome of the rat dentate gyrus
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Human proteinase 3 resistance to inhibition extends to alpha‐2 macroglobulin
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Design of selective substrates of proteinase 3 using combinatorial chemistry methods
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Proteome changes upon in ovo stimulation with Lactobacillus synbiotic in chicken liver
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On practical problems in estimation of antioxidant activity of compounds by DPPH method (Problems in estimation of antioxidant activity)
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The Physical Activity Environment Policy Index for monitoring government policies and actions to improve physical activity
PublikacjaBackground A multifaceted response, including government action, is essential to improve population levels of physical activity (PA). This article describes the development process of the ‘Physical Activity Environment Policy Index’ (PA-EPI) monitoring framework, a tool to assess government policies and actions for creating a healthy PA environment. Methods An iterative process was undertaken. This involved a review of policy...
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Structure–activity relationships study on biological activity of peptides as dipeptidyl peptidase IV inhibitors by chemometric modeling
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Antifungal Activity of Capridine β as a Consequence of Its Biotransformation into Metabolite Affecting Yeast Topoisomerase II Activity
PublikacjaIn the last few years,increasing importance is attached to problems caused by fungal pathogens. Current methods of preventing fungal infections remain unsatisfactory. There are several antifungal compounds whichare highly effective in some cases, however, they have limitations in usage: Nephrotoxicity and other adverse effects. In addition, the frequent use of available fungistatic drugs promotes drug resistance....
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A. Computational analysis by molecular docking of thirty alkaloid compounds from medicinal plants as potent inhibitors of SARS-CoV-2 main protease(2020).
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The effect of previous storage condition on the diffusion and contribution of digestive proteases in the ripening of marinated Baltic herring (Clupea harengus)
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Lupine embryo axes under salinity stress. II. Mitochondrial proteome response
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A Peptidomimetic Fluorescent Probe to Detect the Trypsin β2 Subunit of the Human 20S Proteasome
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Novel internally quenched substrate of the trypsin-like subunit of 20S eukaryotic proteasome
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Inhibition of Human and Yeast 20S Proteasome by Analogues of Trypsin Inhibitor SFTI-1
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The new fluorogenic substrates of neutrophil proteinase 3 optimized in prime site region
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A new proteinase 3 substrate with improved selectivity over human neutrophil elastase
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Urinary Proteome of Newborn Calves—New Potential in Non-Invasive Neonatal Diagnostic
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Different Patterns of mRNA Nuclear Retention during Meiotic Prophase in Larch Microsporocytes
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Declared and actual students’ physical activity
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Novel dendrimeric lipopeptides with antifungal activity
PublikacjaZaprojektowano, zsyntezowano i scharakteryzowano serię nowych kationowych lipopeptydów zawierających rozgałęziony, amfifilowy polarny rdzeń strukturalny pochodzący od dendronu (Lys)(Lys)(Lys) oraz łańcuchy C8 i C12 na C-końcu. Otrzymane zwiazki wykazywały aktywność przeciwdrobnoustrojową, w tym szczególnie przeciwgrzybową wobec drożdżaków z rodzaju Candida. Najwyższą aktywność, selektywną wobec drobnoustrojów grzybowych, wykazywały...
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Hydroacustic activity of the ship propeller operation
PublikacjaPraca przedstawia działanie śrub okretowych jako źródła sygnałów hydroakustycznych, związanych przede wszystkim z różnymi formami kawitacji występującymi podczas pracy śrub.
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Antifungal Activity of Homoaconitate and Homoisocitrate Analogs
PublikacjaThirteen structural analogs of two initial intermediates of the L-alpha-aminoadipate pathway of L-lysine biosynthesis in fungi have been designed and synthesized, including fluoro- and epoxy-derivatives of homoaconitate and homoisocitrate. Some of the obtainedcompounds exhibited at milimolar range moderate enzyme inhibitory properties against homoaconitase and/or homoisocitrate dehydrogenase of Candida albicans. The structural...
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The market and the fair as a traditional activity of the city
PublikacjaThe modern commercial center with its impersonal form still on the squares and streets appear traditional markets and its annual versions – fairs, which similarly to the historical commerce - gather different activities of the inhabitants.
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Extracellular proteolytic activity of Deinococcus geothermalis
PublikacjaProduction of extracellular protease by extremophilic bacteria Deinococcus geothermalis cultivated in liquid media containing 0.1% (w/v) of peptone K, 0.1% yeast extract and 0.2% marine salt reached a maximum in 14 h of the cell growth at 45°C and pH 8.0. The enzyme was purified by a two-step procedure using fractionation by a graded ammonium sulphate precipitation technique and gel filtration on Sephadex G-100 column. Protease...
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Muramyl peptides - synthesis and biological activity
PublikacjaArtykuł przeglądowy opisujący syntezę i aktywność biologiczną muramylopeptydów.
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Anthracenedione analogues - synthesis and biological activity
PublikacjaW artykule opisano syntezę i aktywność biologiczną analogów antracenedionowych.
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Green Physical Activity Indicator: Health, Physical Activity and Spending Time Outdoors Related to Residents Preference for Greenery
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THE EFFECT OF WATER ACTIVITY AND TEMPERATURE ON THE GROWTH AND LIPOLYTIC ACTIVITY OF PENICILLIUM CHRYSOGENUM (THOM) AND EUROTIUM HERBARIORUM (WIGG.) STRAINS
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Molecular modeling study of tectoquinone and acteoside from Tectona grandis linn: a new SARS-CoV-2 main protease inhibitor against COVID-19
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The effects of p53 gene inactivation on mutant proteome expression in a human melanoma cell model
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Identification of serum proteome signatures of locally advanced and metastatic gastric cancer: a pilot study
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An Insight into the Proteome of Uveal Melanoma-Derived Ectosomes Reveals the Presence of Potentially Useful Biomarkers
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Changes in the Cell Wall Proteome of Leaves in Response to High Temperature Stress in Brachypodium distachyon
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Modification of ileal proteome in growing pigs by dietary supplementation with inulin or dried chicory root
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Dietary Inclusion of Dried Chicory Root Affects Cecal Mucosa Proteome of Nursery Pigs
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Lactose-rich milk replacer modifies the proteome of bloodplasma in 2-week-old calves
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Nuclear retention of pre-mRNA involving Cajal bodies during meiotic prophase in plants
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EFFECT OF WATER ACTIVITY AND TEMPERATURE ON GROWTH AND LIPOLYTIC ACTIVITY OF PENICILLIUM CHRYSOGENUM STRAINS IN LIQUID CULTURE MEDIA WITH PLANT OILS
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