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Synthesis, Antimicrobial and Mutagenic Activity of a New Class of d-Xylopyranosides
PublikacjaEight N-[2-(2′,3′,4′-tri-O-acetyl-α/β-d-xylopyranosyloxy)ethyl]ammonium bromides, a new class of d-xylopyranosides containing a quaternary ammonium aglycone, were obtained. Their complete structure was confirmed using NMR spectroscopy (1H, 13C, COSY and HSQC) and high-resolution mass spectrometry (HRMS). An antimicrobial activity against fungi (Candida albicans, Candida glabrata) and bacteria (Staphylococcus aureus, Escherichia...
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Optymalizacja systemu zarządzania uszkodzeniami węzłów komutacyjnych.
PublikacjaW referacie przedstawiono wyniki analizy funkcjonalnej ystemu węzłów komutacyjnych systemu 5ESS. Na podstawie tej analizy dokonano oceny funkcjonowania systemu zarządzania i wskazano obszary jegooptymalizacji. Zaproponowano ssposób wykorzystania narzędzia Action Request System do tworzenia bazy danych raportów alarmowych. Zaproponowano strukturę bazy danych raportów alarmowych i formularza zgłaszania problemu do tworzenia w tej...
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Experimental study on earthquake-induced pounding between structural elements made of different building materials
PublikacjaCelem artykułu jest pokazanie wyników dwóch eksperymentów dotyczących zderzeń pomiędzy elementami wykonanymi z różnych materiałów budowlanych, takich jak: stal, beton, drewno i ceramika. Pierwszy z nich polegał na zrzucaniu kul na płaską powierzchnię, drugi dotyczył zderzeń modeli konstrukcji poddanych wymuszeniom sejsmicznym na stole wstrząsowym. Wyniki testów pokazują, iż wpływ materiału elementów kolidujących ze sobą na zachowanie...
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Projekt belki hybrydowej 1a dla firmy H+H Polska sp. z o.o. wariant 2
PublikacjaNiniejsze opracowanie stanowi projekt belki nadprożowej o długości 3,0 m o przekroju poprzecznym belki hybrydowej (beton konstrukcyjny łączony z betonem komórkowym) nawiązującej do wymiaru bloczka z betonu komórkowego firmy H+H Polska sp. z o.o. o wymiarach (szerokość × wysokość × długość): 24 × 24 × 60 cm, odmiany D600 o średniej wytrzymałości na ściskanie 3,0 MPa. Całkowita wysokość belki hybrydowej wynosi 27 cm (wraz z 3 cm...
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Projekt belki hybrydowej 1a dla firmy H+H Polska sp. z o.o.
PublikacjaNiniejsze opracowanie stanowi projekt belki nadprożowej o długości 3,0 m o przekroju poprzecznym belki hybrydowej (beton konstrukcyjny łączony z betonem komórkowym) nawiązującej do wymiaru bloczka z betonu komórkowego firmy H+H Polska sp. z o.o. o wymiarach (szerokość × wysokość × długość): 24 × 24 × 60 cm, odmiany D600 o średniej wytrzymałości na ściskanie 3,0 MPa. Całkowita wysokość belki hybrydowej wynosi 27 cm (wraz z 3 cm...
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Analiza doświadczalna wpływu długości zakotwienia pręta na zachowanie przyczepności w teście pull-out
PublikacjaArtykuł prezentuje badania przyczepności przeprowadzone przy użyciu testu pull-out. Eksperymenty miały na celu ocenę wpływu długości zakotwienia na przyczepność w tym teście. Z przeprowadzonej analizy wynika, że długość styku pręt-beton znacząco wpływa na zachowanie przyczepności. Określa ona typ zniszczenia połączenia, wpływa na rozkład i wartość naprężeń w pręcie oraz rzutuje na przebieg krzywej przyczepność-poślizg, która jest...
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Obliczenia MES zginanych belek betonowych na poziomie skali mezo
PublikacjaW artykule przedstawiono wyniki numeryczne MES modelowanie belek betonowych z nacięciem w czasie zginania 3-punktowego na poziomie skali mezo. Obliczenia wykonano przy wykorzystaniu modelu degradacji sztywności z nielokalnym osłabieniem. Beton został opisany na poziomie skali mezo jako stochastyczny materiał 3-składnikowy złożony z kruszywa, zaczynu cementowego oraz stref kontaktu. Zbadano wpływ rozkładu stochastycznego ziaren...
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Experimental and numerical investigations of concrete behaviour at meso-level during quasi-static splitting tension.
PublikacjaArtykuł omawia wyniki numeryczne dotyczące pękania betonu uzyskane stosując metodę elementów dyskretnych. Dwuwymiarowe obliczenia wykonano dla próbek betonowych podczas rozłupywania. Beton został opisany jako model 4-fazowy. Mikrostruktura betonu odpowiadała zdjęciom tomograficznym. Zbadano wpływ warunków brzegowych na proces pękania. W obliczeniach zwrócono uwagę na porzebieg zjawisk mikrostrukturalnych przebieg pękania. Wyniki...
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Membrane Sterols Modulate the Binding Mode of Amphotericin B without Affecting Its Affinity for a Lipid Bilayer
PublikacjaMembrane-active antibiotics are known to selectively target certain pathogens based on cell membrane properties, such as fluidity, lipid ordering, and phase behavior. These are in turn modulated by the composition of a lipid bilayer and in particular by the presence and type of membrane sterols. Amphotericin B (AmB), the golden standard of antifungal treatment, exhibits higher activity toward ergosterol-rich fungal membranes, which...
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Enhancing chain-elongating microbiomes: Sequential fungi-bacteria cooperation for efficient food waste upgrading using endogenous electron donors
PublikacjaThe upgrading of organic waste such as food waste (FW) into medium-chain carboxylates (MCC) is within a bio-based circular economy concept. An efficient chain elongation (CE) microbiome is difficult to obtain, which normally requires long-term acclimatization and an exogenous supplement of electron donor (ED, especially ethanol). In this study, the CE microbiome was rapidly shaped within 18 days and an efficient endogenous ethanol-based...
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Selektywne chłodzenie mózgu noworodka po Niedotlenieniu okołoporodowym. Część 1. Medyczne fakty oraz przegląd dostępnych rozwiązań systemów selektywnego chłodzenia mózgu
PublikacjaMózg ludzki jest organem delikatnym, dlatego tak ważne jest zadbanie o to, aby już w momencie przyjścia na świat noworodek miał zapewnioną, w razie konieczności możliwość minimalizacji uszkodzeń neurologicznych, spowodowanych niedotlenieniem okołoporodowym. Niedotlenienie to w dramatyczny sposób zaburza homeostazę mózgu, który jako organ najbardziej energochłonny potrzebuje najwięcej tlenu. Zapoczątkowane brakiem tlenu procesy...
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Prognozowanie krzywej osiadania pala wierconego z iniekcją ciśnieniową pod podstawą
PublikacjaArtykuł jest kontynuacją tematyki autora dotyczącą mechanizmu działania iniekcji ciśnieniowej pod podstawą pala wierconego. W poprzednich publikacjach, autor wykazał, że iniekcja ta w głównej mierze uaktywnia zwiększone opory gruntu wzdłuż pobocznicy pala. Na tej podstawie w niniejszym artykule zaprezentowano procedurę obliczeniową prognozowania krzywą osiadania pala wierconego z iniekcją ciśnieniową pod podstawą. Przedstawiono...
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Workflow patterns applicable to virtual knowledge-based organizations
PublikacjaWorkflow is a term specifying how to automate a business process, in whole or part during which documents, information or tasks are passed from one participant to another for action, according to a set of procedural rules. Workflow is therefore directly applicable in virtual knowledge-based organizations, where information is exchanged via electronic documents. In the literature, is presented a complete list of workflow control-flow...
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MutL protein as a constituent of vsp, ner and mmr repair systems
PublikacjaMutS and MutL proteins are renowned mostly for their functions in well-characterized, post-DNA replication mis- match repair system (MMR). However, there is growing evidence that MMR system is not the only field of action for these pro- teins. Moreover, the participation in MMR does not even have to be their primary function. There are some reports indicat- ing involvement of MutL in BER, NER and VSP (very short patch repair)....
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MUTL PROTEIN AS A COMMON CONSTITUENT OF VSP, BER, NER AND MMR REPAIR SYSTEMS
PublikacjaMutS and MutL proteins are renowned mostly for their functions in well-characterized, post-DNA replication mismatch repair system (MMR). However, there is growing evidence that MMR system is not the only field of action of these proteins. Moreover, involvement in MMR does not even have to be their primary function. There are some reports indicating involvement of MutL in BER, NER and VSP (very short patch repair). MutL protein...
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Mathematical modelling of implant in an operated hernia for estimation of the repair persistence
PublikacjaThis paper presents mathematical modelling of an implanted surgical mesh used in the repair process of the abdominal hernia. The synthetic implant is simulated by a membrane structure. The author provides a material modelling of the implant based on the dense net model appropriate for technical fabrics. The accuracy of the proposed solution is evaluated by comparing the simulations of the dynamic behaviour of the system with the...
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Comparative molecular modelling of biologically active sterols
PublikacjaMembrane sterols are targets for a clinically important antifungal agent – amphotericin B. The relatively specific antifungal action of the drug is based on a stronger interaction of amphotericin B with fungal ergosterol than with mammalian cholesterol. Conformational space occupied by six sterols has been defined using the molecular dynamics method to establish if the conformational features correspond to the preferential interaction...
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Low temperature processed MnCo2O4 and MnCo1.8Fe0.2O4 as effective protective coatings for solid oxide fuel cell interconnects at 750 °C
PublikacjaIn this study two materials, MnCo2O4 and MnCo1.8Fe0.2O4 are studied as potential protective coatings for Solid Oxide Fuel Cell interconnects working at 750 °C. First powder fabrication by a modified Pechini method is described followed by a description of the coating procedure. The protective action of the coating applied on Crofer 22 APU is evaluated by following the area specific resistance (ASR) of the scale/coating for 5500...
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Effect of culinary treatment on chnages in the contents of selected nutrients and non-nutrients in curly kale (Brassica oleracea var. acephala)
PublikacjaKale has a great nutritive value, very high antioxidant activity and pro-healthypotential. The level of phytochemicals and related bioactive compounds arestrongly dependent on pre and postharvest stages of production chain (domestic orindustrial). The study investigated changes in the levels of vitamin C, b-carotene,total polyphenols, antioxidant activity, degradation products of glucosinolates aswell as nitrates and nitrites in...
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Aminy w środowisku - niebezpieczeństwo czy jego naturalny element?
PublikacjaA lot of amines and their compounds are used in the industry. First of all they are used for the preparation of medicines, plant protection agents, fertilizers and plastics. Amines are also released into the environment as a result of natural biological processes such as the release of certain species of flowers to lure insects, and also biochemical breakdown of amino acids in the protein during decomposition of organic matter. Unfortunately,...
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Hydrogen effects in duplex stainless steel welded joints - electrochemical studies
PublikacjaIn this work results on the influence of hydrogen on passivity and corrosion resistance of 2205 duplex stainless steel (DSS) welded joints are described. The results were discussed by taking into account three different areas on the welded joint: weld metal (WM), heat-affected zone (HAZ) and parent metal. The corrosion resistance was qualified with the polarization curves registered in a synthetic sea water. The conclusion is that,...
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Cell-penetrating peptides – mechanism of transduction and synthesis – short review
PublikacjaPotential antimicrobial agents may be effective if they are delivered efficiently to their site of action. In many cases, lack of permeability through the cell membrane is the main problem. One of the possible solutions could be a novel intracellular delivery system involving cell-penetrating peptides (CPPs), which may improve the efficiency of many new biophar-maceuticals. Among other things, CPPs are capable of trans-porting...
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Small Urban Hacks - Big Impact! Tackling major urban challenges through acupunctural smallness
PublikacjaSmall urban hacks, acupunctural action and process-oriented planning approaches might appear to address quite a socio-romantic attitude towards our urban environments. In this chapter, our aim is to remedy such a biased view, demonstrating the impact and potential of smallness in the context of major urban challenges. Small urban hacks and their multi-faceted and creativity-driven approaches of small is beautiful are selected from...
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Consumerism and the Quality of Life
PublikacjaHigh level of consumption, driven by marketing activities, the pleasure and joy of possession and the accumulation of material goods are often associated with prosperity, sense of happiness and fulfilment in life. On a broader scale, economic indicators related to production and consumption are used to define the well-being and quality of life in societies. Unfortunately, the phenomenon of consumerism entails negative social and...
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LNG TANK IN ŚWINOUJŚCIE: NONLINEAR ANALYSIS OF THE TANK DOME ELEMENTS BEHAVIOUR
PublikacjaIn this paper, the dome of a tank in the Świnoujście LNG terminal is analysed. Some of the rafter ribs at the connection with hangers were not mounted during construction of the tank dome. Therefore, it has become necessary to estimate its response, which has been done with the aid of some computational models of the dome, that have been created in the finite element method environment. Different local models are studied, aiming...
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Generic invariant measures for iterated systems of interval homeomorphisms
PublikacjaIt is well known that iterated function systems generated by orientation preserving homeomorphisms of the unit interval with positive Lyapunov exponents at its ends admit a unique invariant measure on (0, 1) provided their action is minimal. With the additional requirement of continuous differentiability of maps on a fixed neighbourhood of {0,1} { 0 , 1 } , we present a metric in the space of such systems which renders it complete....
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Phytoremediation—From Environment Cleaning to Energy Generation—Current Status and Future Perspectives
Publikacja:Phytoremediationis a technology based on the use of green plants to remove, relocate, deactivate, or destroy harmful environmental pollutants such as heavy metals, radionuclides, hydrocarbons, and pharmaceuticals. Under the general term of phytoremediation, several processes with distinctively different mechanisms of action are hidden. In this paper, the most popular modes of phytoremediation are described and discussed. A broad...
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Dynamics of the small-span railway bridge under moving loads
PublikacjaThe paper presents the results of dynamic analysis of the small-span railway bridge, subjected to an action of moving trains. Numerical simulations were performed using three different load models: series of moving forces, series of moving single-mass and double-mass oscillators. The parameters of the vehicle were taken from the existing EN57 train. The parameters of the bridge were taken from the existing steel span of 10,24 m...
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VARIANT DESIGNING IN the PRELIMINARY SMALL SHIP DESIGN PROCESS
PublikacjaShip designing is a complex process, as the ship itself is a complex, technical multi-level object which operates in the air/water boundary environment and is exposed to the action of many different external and internal factors resulting from the adopted technical solutions, type of operation, and environmental conditions. A traditional ship design process consists of a series of subsequent multistage iterations, which gradually...
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A convergence result for mountain pass periodic solutions of perturbed Hamiltonian systems
PublikacjaIn this work, we study second-order Hamiltonian systems under small perturbations. We assume that the main term of the system has a mountain pass structure, but do not suppose any condition on the perturbation. We prove the existence of a periodic solution. Moreover, we show that periodic solutions of perturbed systems converge to periodic solutions of the unperturbed systems if the perturbation tends to zero. The assumption on...
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Consistency of Quantum Computation and the Equivalence Principle.
PublikacjaThe equivalence principle, being one of the building blocks of general relativity, seems to be crucial for analysis of quantum effects in gravity. In this paper we consider the relation between the equivalence principle and the consistency of quantum information processing in gravitational field. We propose an analysis with a looped evolution consisting of steps both in the gravitational field and in the accelerated reference frame....
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Meso-mechanical modelling of damage in concrete using discrete element method with porous ITZs of defined width around aggregates.
PublikacjaArtykuł omawia wyniki obliczeń numerycznych pękania dla betonu stosując metodę elementów dyskretnych. Beton był opisany jako materiał 4-fazowy i był poddany zginaniu. W obliczeniach uwzględniono strefy ITZ o skończonej szerokości dookoła wszystkich ziaren kruszywa. Nacisk położono na przebieg mikropęknięć przy kruszywie. Wyniki porównano bezpośrednio z doświadczeniami. Obliczenia wykonano także dla szorstkich ziaren kruszywa....
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CROWDSOURCING A KOMUNIKACJA Z KONSUMENTAMI
PublikacjaRozdział prezentuje wybrane modele komunikacji w Internecie oraz crowdsourcing jako nową metodę pozyskiwania pomysłów i informacji od konsumentów. W ciągu ostatnich 5 lat rozwój technologii komunikacyjnych znacząco zmienił sposób komunikowania się ludzi, a w konsekwencji również organizacji z konsumentami. Nie tylko firmy z branży IT mogą wzmocnić swoją markę, reputację oraz zwiększyć przychody dzięki opracowaniu atrakcyjnej, społecznie...
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New Unsymmetrical Bisacridine Derivatives Noncovalently Attached to Quaternary Quantum Dots Improve Cancer Therapy by Enhancing Cytotoxicity toward Cancer Cells and Protecting Normal Cells
PublikacjaThe use of nanoparticles for the controlled drug delivery to cells has emerged as a good alternative to traditional systemic delivery. Quantum dots (QDs) offer potentially invaluable societal benefits such as drug targeting and in vivo biomedical imaging. In contrast, QDs may also pose risks to human health and the environment under certain conditions. Here, we demonstrated that unique combination of nanocrystals core components...
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A three-dimensional meso-scale approach to concrete fracture based on combined DEM with x-ray micro-CT images
PublikacjaArtykuł omawia wyniki numeryczne uzyskane stosując 3-wymiarowy mezoskopowy model do opisu pękania w betonie na poziomie kruszywa w belce z nacięciem podczas zginania. Do obliczeń użyto metodę elementów dyskretnych. Beton został opisany jako materiał 4-fazowy złożony z kruszywa, zaprawy, makro-porów i stref przejściowych miedzy kruszywem a zaprawą. Kształt i położenia kruszywa przyjęto na podstawie skanów z mikro-tomografu. Uzyskano...
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Influence of a lipid bilayer on the conformational behavior of amphotericin B derivatives - A molecular dynamics study.
PublikacjaAmphotericin B (AmB) is an effective but very toxic antifungal antibiotic. In our laboratory a series of AmB derivatives of improved selectivity of action was synthesized and tested. To understand molecular basis of this improvement, comparative conformational studies of amphotericin B and its two more selectivederivatives were carried out in an aqueous solution and in a lipid membrane. These molecular simulation studies revealed...
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Sources and Fate of PAHs and PCBs in the Marine Environment
PublikacjaThe assessment of a hazard resulting from the pollution of the environment by chemical compounds is in principle limited to the determination of their concentrations in its various compartments. But for solving many problems in this context, knowledge of the emission sources, transport pathways, and sites of deposition is of great benefit. By far the largest amounts of pollutants, regardless of where they were discharged, end up...
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Compensation of pressure peaks in pwk-type hydraulic pumps
Publikacjahydraulic axial pumps equipped with cam-driven commutation unit (pwk pumps) proved their high efficiency up to 55 mpa and ability to work self-sucking, even at high speed. displacement of pwk pump may easily be changed by moving its control cam. full discharge from hydrostatic forces makes such control possible by direct action of a low-energy actuator like proportional electromagnet or stepping motor. that eliminates heavy and...
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Optical recognition elements: macrocyclic imidazole chromoionophores entrapped in silica xerogel
PublikacjaMaterials containing new chromoionophores consisting of crown residue and azole moiety as partsof macrocycles were encapsulated by the sol-gel procedure in silica xerogel matrices and proposed aschemical recognition elements especially for such metal ions as Li+, Cs+ and Cu2+. Action of these recognition elements is in principle based on changes of reflectance. The recognition elements containing 21-membered chromogenic...
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Occurrence and Determination of Volatile Fatty Acids in Landfill Leachate and Gas
PublikacjaIn landfills containing biological matter volatile fatty acids (VFAs) are generated at high rate at the early stage of waste disposal and their content in leachate is high as compared to the leachate from old parts of landfill since they are converted to methane gas. Monitoring of the leachate for the content of VFAs can help determine the processes occurring in waste and possible effect of the leachate on the environment in the...
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Occurrence and Determination of Volatile Fatty Acids in Landfill Leachate and Gas
PublikacjaIn landfills containing biological matter volatile fatty acids (VFAs) are generated at high rate at the early stage of waste disposal and their content in leachate is high as compared to the leachate from old parts of landfill since they are converted to methane gas. Monitoring of the leachate for the content of VFAs can help determine the processes occurring in waste and possible effect of the leachate on the environment in the...
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THE ROLE OF NATURE IN PLACEMAKING WITHIN THE LIMITS OF HISTORIC CITIES
PublikacjaThis paper focuses on the role of nature in placemaking within historic cities. There are two different approaches to placemaking – The first is a more traditional approach, i.e. complete building process which entails significant investments. The second is “Lighter, Quicker, Cheaper” approach proposed by the Project for Public Spaces organization. This article discusses the role, importance and place of nature in both approaches....
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New generation of analytical tests based on the assessment of enzymatic and nuclear receptor activity changes induced by environmental pollutants
PublikacjaAnalytical methods show great potential in biological tests. The analysis of biological response that results from environmental pollutant exposure allows: (i) prediction of the risk of toxic effects and (ii) provision of the background for the development of markers of the toxicants presence. Bioanalytical tests based on changes in enzymatic activity and nuclear receptor action provide extremely high specificity and sensitivity....
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Guided waves for monitoring of plate structures with linear cracks of variable length
PublikacjaDamage occurring at the work of plate structures may grow to a considerable size. The joint action – the detection of a defect at the earliest possible stage, the monitoring of its growth and the determination of its critical size in the context of structural reliability allows optimizing the cost of the maintenance and repair of structural elements. Thus the development of monitoring systems for permanent observation of fault...
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RECODIS: Resilient Communication Services Protecting End-user Applications from Disaster-based Failures
PublikacjaDisaster-based failures can seriously disrupt any communication network, making its services unavailable. Such disruptions may be caused by natural disasters, technology-related failures, or malicious attacks, and they are observably increasing in number, intensity and scale. When network services that are a part of critical infrastructure become unavailable, commercial and/or societal problems are inevitable. The issue of limiting...
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Strongly anisotropic surface elasticity and antiplane surface waves
PublikacjaWithin the new model of surface elasticity, the propagation of anti-plane surface waves is discussed. For the proposed model, the surface strain energy depends on surface stretching and on changing of curvature along a preferred direction. From the continuum mechanics point of view, the model describes finite deformations of an elastic solid with an elastic membrane attached on its boundary reinforced by a family of aligned elastic...
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Participatory co-design approach for Greencoin educational tool shaping urban green behaviors.
PublikacjaOur main goal is to prepare assumptions of the Greencoin (GC) cybernetic system, implying pro-ecological attitudes and behavior of city residents. We used qualitative methods, including a literature review and action research -workshops attended by academics, representatives of private and business sectors, urban movements, municipal institutions’ partners, and residents. Our results defined functionalities of the GC, identified...
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Problems and chellenges to determine pesticide residues in bumblebees
PublikacjaBumblebees play an important role in t he pollination process of many crops and flowers. Therefore, taking action to protect and assess the impact of p esticides on these insects is fully justi fied. Pesticides may cause mortality and also sub-lethal effects that are not always directly visible. Bumblebees, like honeybees, can be used as indicators for environmental monitoring contamination. Two approaches are mainly used for the...
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Chiral Pyrazolo[4,3-e][1,2,4]triazine Sulfonamides—Their Biological Activity, Lipophilicity, Protein Affinity, and Metabolic Transformations
PublikacjaReferring to our previous laboratory results related to the tyrosinase and urease inhibition by pyrazolo[4,3-e][1,2,4]triazine sulfonamides, we examined here in silico the mechanism of action at the molecular level of the investigated pyrazolotriazine sulfonamides by the molecular docking method. The studied compounds being evaluated for their cytotoxic effect against cancer cell lines (MCF-7, K-562) and for recombinant Abl and...
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Polyurethanes
PublikacjaHandbook of Thermoset Plastics, Fourth Edition provides complete coverage of the chemical processes, manufacturing techniques and design properties of each polymer, along with its applications. This new edition has been expanded to include the latest developments in the field, with new chapters on radiation curing, biological adhesives, vitrimers, and 3D printing. This detailed handbook considers the practical implications of using...