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Design, synthesis and high antitumor potential of new unsymmetrical bisacridine derivatives towards human solid tumors, specifically pancreatic cancers and their unique ability to stabilize DNA G-quadruplexes
PublikacjaNew promising unsymmetrical bisacridine derivatives (UAs), have been developed. Three groupsincluding 36 compounds were synthesized by the condensation of 4-nitro or 4-methylacridinone, imi-dazoacridinone and triazoloacridinone derivatives with 1-nitroacridine compounds linked with anaminoalkyl chain. Cytotoxicity screening revealed the high potency of these compounds against severaltumor cell lines. Particularly, imidazoacridinone-1-nitroacridine...
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In vitro biological evaluation of a novel folic acid-targeted receptor quantum dot−β−cyclodextrin carrier for C-2028 unsymmetrical bisacridine in the treatment of human lung and prostate cancers
PublikacjaTraditional small-molecule chemotherapeutics usually do not distinguish tumors from healthy tissues. However, nanotechnology creates nanocarriers that selectively deliver drugs to their site of action. This work is the next step in the development of the quantum dot−β−cyclodextrin−folic acid (QD−β−CD−FA) platform for targeted and selected delivery of C−2028 unsymmetrical bisacridine in cancer therapy.Herein, we report an initial...
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Career and Technical Education Research (Formerly: Journal of Vocational Education Research)
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Cahiers de l'institut de linguistique de Louvain
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CANADIAN JOURNAL OF SOCIOLOGY-CAHIERS CANADIENS DE SOCIOLOGIE
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Cahiers de Recherches Médiévales (A Journal of medieval studies)
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Cahiers de Psychologie Cognitive / Current Psychology of Cognition
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Cahiers des amis de Pierre Benoit (Les)
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Cahiers de l’association internationale des études françaises
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Cahiers d'Histoire et de Philosophie des Sciences
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Cahiers d Etudes du Religieux-Recherches Interdisciplinaires
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REVUE DE METALLURGIE-CAHIERS D INFORMATIONS TECHNIQUES
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Inter Applied Chemistry Programme 1 Morrison Forensic
Kursy OnlineInter Applied Chemistry Programme 1 Lecture 1 background reading Read the following : Chapter 1 Introduction to Forensic Science ( From Jackson, Jackson, Mountain and Brealey, Forensic Science, Pearson 4th Ed (2016)) Very general professional guidance/Introduction United Nations can be found within these guides, (these are mainly for reference purposes) https://www.unodc.org/documents/scientific/Crime_scene_awareness__Ebook.pdf https://www.unodc.org/documents/justice-and-prison-reform/cjat_eng/Forensic_services_and_infrastructure.pdf Task...
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Factors influencing the selection of the ideal employer
Dane BadawczeThis dataset contains the results of research that were carried out by the Wrocław University of Science and Technology in March and April 2016, using an anonymous "on-line" questionnaire. 1,320 people took part in the study entitled "My ideal employer" - students and doctoral students of all faculties of the university (including those fields of study...
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Piotr Rajchowski dr inż.
OsobyPiotr Rajchowski (Member, IEEE) was born in Poland, in 1989. He received the E.Eng., M.Sc., and Ph.D. degrees in radio communication from the Gdańsk University of Technology (Gdańsk Tech), Poland, in 2012, 2013, and 2017, respectively. Since 2013, he has been working at the Department of Radiocommunication Systems and Networks, Faculty of Electronics, Telecommunications and Informatics, Gdańsk University of Technology, as a IT...
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Artur Gańcza dr inż.
OsobyI received the M.Sc. degree from the Gdańsk University of Technology (GUT), Gdańsk, Poland, in 2019. I am currently a Ph.D. student at GUT, with the Department of Automatic Control, Faculty of Electronics, Telecommunications and Informatics. My professional interests include speech recognition, system identification, adaptive signal processing and linear algebra.
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Personal Branding—A New Competency in the Era of the Network Economy. Corporate Brand Performance Implications
PublikacjaPrimary assets of the network economy are information, network, re-lationships, knowledge, and a virtual environment. The competency of personal branding exercised by knowledge workers, also thought of as knowledge producers, is becoming a natural consequence of the business environment where the significance of hierarchies is constantly decreasing. Knowledge workers are powerful as never be-fore and can exist as separate actors...
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Professional Practice, ET, sem.6, summer 24/25 (PG_000549757)
Kursy OnlineProfessional internships for students include design, workshop and operational work in the field of energy.
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Investigation of tracking systems properties in CAVE-type virtual reality systems
PublikacjaIn recent years, many scientific and industrial centers in the world developed a virtual reality systems or laboratories. One of the most advanced solutions are Immersive 3D Visualization Lab (I3DVL), a CAVE-type (Cave Automatic Virtual Environment) laboratory. It contains two CAVE-type installations: six-screen installation arranged in a form of a cube, and four-screen installation, a simplified version of the previous one. The...
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Education Towards The Use Of BIM On The Example Of Polish Universities
PublikacjaBIM (Building Information Modeling) has been one of the rapidly developing fields of digital techniques supporting the realization of construction projects in recent years. Further development, and especially the use of these techniques, depends to a large extent on the qualifications of young construction engineers who start their professional careers in this field. The article attempts to synthetically list and compare subjects,...
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Using Moodle as a Solution to Interdisciplinary E-collaboration Issues
PublikacjaRapid technological development in recent years has contributed to numerous changes in many areas of life, including education and communication. Establishing interdisciplinary collaboration brings many benefits, however, it is often associated with numerous problems and inconveniences, as well as the need of constant improvement, lifelong learning, professional development (CPD) and finding an effective way of information transferring....
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Teaching Architecture – contemporary challenges and threats in the complexity of built environment
PublikacjaThe complexity of the modern built environment is a problem n ot only of architectural and urban issues. This issue extends to many othe r disciplines as well as covering a wide range of social engagements. The idea of writing this pa per is generally initiated by the debate which took place in Gdańs k on 22.01.2016, and was prepar ed in order to meet representatives of the four circles of interest...
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Nuclear Magnetic Resonance data for the synthesis of esterase cleavable antifungal conjugates containing fatty acids as molecular carriers
Dane BadawczeNMR data for novel organic compounds - conjugates composed of C2-18 fatty acid (FA) residues as a molecular carrier and 5-fluorocytosine (5-FC) as an active agent, released upon the action of intracellular esterases on the ester bond between FA and “trimethyl lock” intramolecular linker.
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Skłonność do rywalizacji a intencje przedsiębiorcze – o różnicach międzypłciowych
PublikacjaAccording to the person-environment fit model people are more inclined to choose particular careers paths over other depending on their individual characteristics. They are also more likely to be satisfied with a career path that matches their characteristics and less likely to experience negative consequences including strain. In previous research several characteristics of entrepreneurs which differentiate them from non-entrepreneurs...
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Daniel Chuchała dr hab. inż.
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High prevalence of carriers of variant c.1528G>C of HADHA gene causing long-chain 3-hydroxyacyl-CoA dehydrogenase deficiency (LCHADD) in the population of adult Kashubians from North Poland
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Daily oligofructose-enriched inulin intake impacts bone turnover markers but not the cytokine profile in pediatric patients with celiac disease on a gluten-free diet: Results of a randomised, placebo-controlled pilot study
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Theory vs. practice. Searching for a path of practical education
PublikacjaThe introduction of a three-tier model of higher education (the Bologna model) has led to considerable changes in the 1st- and 2nd-tier technical courses at universities. At present, a student with a bachelor’s degree can be employed in his / her profession after completing only 7 semesters of study. A search is under way for methods of combining theoretical knowledge taught at universities with practical knowledge gained afterwards....
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Lifelong Learning Idea in Architectural Education
PublikacjaThe recent advances in IT and technology are forcing changes in the approach to educating society. In the 20th century, life-long learning was understood as educating adults in order to improve their occupational qualifications. Life-long learning allows the needs of the present-day world to be addressed through providing the individual with education at every stage of his/her life various forms. The search for a new model...
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PROJEKTOWANIE STANOWISK LABORATORYJNYCH WSPIERAJĄCYCH PROCES SZKOLENIA PRAKTYCZNEGO KADR MORSKICH DZIAŁU MASZYNOWEGO W ŻEGLUDZE MIĘDZYNARODOWEJ, PRZYBRZEŻNEJ I KRAJOWEJ
PublikacjaWithin the article a design offer of the Department of Ship and Power Plants of the Faculty of Ocean Engineering And Ship Technology at the Gdansk University of Technology has been presented. The offer concerns designing laboratory stations which might stand for the equipment of a didactic base of maritime educational centers i.e. maritime (naval) academies and schools as well as maritime affairs' professional training centers,...
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New Molecular Markers Involved in Regulation of Ovarian Granulosa Cell Morphogenesis, Development and Differentiation during Short-Term Primary In Vitro Culture—Transcriptomic and Histochemical Study Based on Ovaries and Individual Separated Follicles
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Nina Rizun dr
OsobyNina Rizun jest adiunktem na Wydziale Zarządzania i Ekonomii Politechniki Gdańskiej. W październiku 1999 r. uzyskała stopień doktora nauk technicznych za specjalizacją Gospodarka przedsiębiorstwa i organizacja produkcji. W latach 1993–2000 pracowała na Wydziale Informatyki Ekonomicznej w Akademji Metalurgicznej, Dnipro, Ukraina. W latach 2000–2016 – na Wydziale Cybernetyki Ekonomicznej i Metod Matematycznych na Uniwersytecie Alfreda...
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Caravelle. Cahiers du monde hispanique et luso-brésilien
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Cahiers d’études des cultures ibériques et latino-américaines
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Magdalena Barańska dr
OsobyNauczyciel akademicki, doradca zawodowy, pedagog, adiunkt w Zakładzie Kształcenia Ustawicznego i Doradztwa Zawodowego WSE UAM. Doktor nauk społecznych w zakresie pedagogiki. Od poczatku swojej kariery związana jestem z Wydziałem Studiów Edukacyjnych. Moje zainteresowania naukowe oraz badawcze koncentrują się wokół problematyki kształcenia ustawicznego, edukacji akademickiej i uniwersytetów, planowania kariery edukacyjno–zawodowej,...
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Employing economical methods for pavement defects estimation
PublikacjaIt is a common practise that measurements of road surface conditions are made using professional and expensive apparatus. Typically a van or a truck equipped with a set of professional sensors i.e. laser scanners of surface is used, therefore the measurement update period is often quite long. Two alternative low-cost methods for estimating road pavement defects and failures were proposed and investigated by the authors. The first...
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Risking It All or Here Comes the Flood
PublikacjaThe professional reality is interdisciplinary! When city transformation and evolution starts, what are the tools for successful strategies for urban interventions? How does digital planning for digital fabrication processes look like? How dedicated are the new professionals? And how does this all influence the future of bridge design? More than 60 students representing various disciplines of built environment and working together...
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“The Guardians of the Truth”: Journalists’ Resistance to the Algorithmization of Journalism
PublikacjaRegardless of the term used, be it “robot journalism,” “automated journalism,” “algorithmic journalism” or “machine-written journalism,” the process of automatic content creation and distribution is progressing in the newsrooms. Meanwhile, exercising control over the creation and distribution of news is considered a fundamental element of journalists’ professional identity. The article presents the results of research on the perception...
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Aleksandra Szewczyk mgr
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Monika Downar mgr
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Study on Speech Transmission under Varying QoS Parameters in a OFDM Communication System
PublikacjaAlthough there has been an outbreak of multiple multimedia platforms worldwide, speech communication is still the most essential and important type of service. With the spoken word we can exchange ideas, provide descriptive information, as well as aid to another person. As the amount of available bandwidth continues to shrink, researchers focus on novel types of transmission, based most often on multi-valued modulations, multiple...
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Autodesk Robot Structural Analysis = Wymiarowanie Konstrukcji Stalowych i Żelbetowych : Przyklady Obliczeń
PublikacjaW pracy przedstawiono przykłady wymiarowania konstrukcji stalowych i żelbetowych z wykorzystaniem programu Autodesk Robot Structural Analysis Professional.
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How to enhance perception of reassembled but incomplete works of ancient art? Eye-tracking study of virtual anastylosis.
Publikacjan 1964 the Venice Charter described anastylosis as the only acceptable method of reassembly of architectural remains. Although the scientific community has agreed with the Charter’s decision, many questions pertaining to the technical and aesthetic aspects of anastylosis remain unanswered. Virtual anastylosis seems one of the most promising digital solutions to finding at least some answers, as it permits testing various solutions...
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The Urban Mentoring as a New Method of Participatory Urban Planning in Poland
PublikacjaTwenty-five years after the return of democracy and the beginning of basing the country's economy on neoliberal developmental paradigm, Poland adopted the regulations regarding management of urban policy, which had been wait for over a decade (accession to the EU). The National Urban Policy as well as the Act on revitalization have defined, in a modern manner, the field of cooperation between the local government, the administration...
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Emotional experiences of family caregivers of children with Dravet syndrome
PublikacjaBackground: Since the psychosocial implications of Dravet syndrome (DS) are much more serious and far-reaching than in other types of epilepsy, caring for a DS child seriously affects the entire family. This study describes the emotional experiences of family caregivers of DS children and evaluates the way caregiving affects their perceived quality of life. Methods: An anonymous, self-administered...
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Job Demands, Engagement, and Turnover Intentions in Polish Nurses: The Role of Work-Family Interface
PublikacjaBackground: Poland has lower ratios of employed registered nurses per 1,000 inhabitants than the EU average. Polish nurses work under miserable conditions without assisting personnel, and they reconcile their professional demands with responsibilities for their families; 96% of them are women. Rationale/Aims: This study uses Hobfoll’s conservation of resources (CORs) theory to explain the role of various resources in the improvement...
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PROFESSIONAL PRACTICE [2020/21]
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The situation of young mothers in the Polish labour market
PublikacjaThe purpose of the article is to present the situation of young women combining professional and paternal responsibilities in the Polish labour market. The papaer presents the results of interviews conducted with six young mothers.
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InSitu-Revista Cientifica do Programa de Mestrado Profissional em Projeto Producao e Gestao do Espaco Urbano
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Cahiers Franz Schubert. Revue de musique classique et romantique
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