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Wyniki wyszukiwania dla: AGENCI MOBILNI
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Cytochromes P450 and Skin Cancer: Role of Local Endocrine Pathways
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Synthesis of Combretastatin A-4 Analogs and their Biological Activities
PublikacjaCombretastatin A-4 (CA-4) is a natural product, which consists of two phenyl rings, linked by an ethylene bridge. CA-4, inhibitor of polymerization of tubulin to microtubules, possesses a strong antitumor and anti-vascular properties both in vitro and in vivo. Previous studies showed that disodium phosphate salt of CA-4, a water-soluble prodrug is well tolerated at therapeutically useful doses. However, it should be noted that...
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The gaseous messenger carbon monoxide is released from the eye into the ophthalmic venous blood depending on the intensity of sunlight
PublikacjaCircadian and seasonal rhythms in daylight affect many physiological processes. In the eye, energy of intense visible light not only initiates a well-studied neural reaction in the retina that modulates the secretory function of the hypothalamus and pineal gland, but also activates the heme oxygenase (HO) to produce carbon monoxide (CO). This study was designed to determine whether the concentration of carbon monoxide (CO) in the...
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Anticancer Properties of Amino Acid and Peptide Derivatives of Mycophenolic Acid
PublikacjaBackground: Although Mycophenolic Acid (MPA) is applied as prodrugs in clinic as an immunosuppressant, it also possesses anticancer activity. MPA acts as Inosine-5’-Monophosphate Dehydrogenase (IMPDH) inhibitor, where the carboxylic group at the end of the side chain interacts with Ser 276 of the enzyme via hydrogen bonds. Therefore, MPA derivatives with other polar groups indicated high inhibition too. On the other hand, potent...
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Optical method supported by machine learning for dynamics of C‐reactive protein concentrations changes detection in biological matrix samples
PublikacjaIn this article we present the novel spectroscopy method supported with machine learning for real-time detection of infectious agents in wastewater. In the case of infectious diseases, wastewater monitoring can be used to detect the presence of inflammation biomarkers, such as the proposed C-reactive protein, for monitoring inflammatory conditions and mass screening during epidemics for early detection in communities of concern,...
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A Biofeedback System that Uses the Game to Study Electrical Muscle Activity
PublikacjaThe aim of this project was to design a system that will allow performing repetitive muscle exercises using a biofeedback device. It is supposed to enhance the motivation and attractiveness of the performed tasks thanks to an interactive game developed for mobile devices with the Android operating system. The built-in calibration mechanisms enable the users to play a game that is independent of their abilities which evens out the...
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Are deep eutectic solvents useful in chromatography? A short review
PublikacjaA literature update has been done concerning Deep Eutectic Solvents (DES) use in chromatography applications. The literature survey was based on the period from 2010 till 2020 and manuscripts reported in the data bases Web of Science and Scopus. The use of DES as mobile phase and mobile phase additives, stationary phases and solid phase modifiers and the use of DES as reaction solvents for chromatography use, were evaluated. Emphasis...
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Properties of a lithium solid electrolyte gas sensor based on reaction kinetics
PublikacjaW artykule przedstawiono zasadę działania, budowę i właściwości czujnika gazu na bazie elektrolitu stałego z mobilnymi jonami litu. Czujnik został przygotowany w technologii grubowarstwowej. Przedstawiono wyniki badań czujnika w mieszaninach gazów toksycznych.
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Hydrauliczne układy napędowe w drogowych maszynach roboczych
PublikacjaW maszynach roboczych, określanych jako mobilne, w tym także w maszynach drogowych ważną rolę pełnią hydrauliczne układy napędowe i sterownicze. Ciekawymi rozwiązaniami konstrukcyjnymi, wartymi ich opublikowania są napędy walca wibracyjnego frezarki do nawierzchni drogowych, miniładowarki oraz kombinowanych walców drogowych. W oparciu o przedstawione konstrukcje budowy układów hydraulicznych, omówione zostaną zasady działania niektórych...
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Investigation on structural, optical and anti-bacterial properties of organic additives iron oxide prepared by chemical route method
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Zbigniew Łubniewski dr hab. inż.
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Antitumor 1-nitroacridine derivative C-1748 induces significant apoptosis in pancreatic cancer cells.
PublikacjaPancreatic cancer is the fifth leading cause of cancer death and has the lowest survival rate of any solid cancer in the industrial countries. The poor prognosis of pancreatic cancer results from its tendency for late presentation, aggressive invasion, early metastasis, and resistance to chemotherapy. Gemcitabine still remains the best chemotherapeutic agent available for the treatment of advanced pancreatic cancer. However, gemcitabine...
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Wyszukiwarka internetowa z bazą wiedzy
PublikacjaW artykule scharakteryzowano program wspomagający klienta w wyborze najbardziej go satysfakcjonującej wycieczki ze zbioru ofert biura turystycznego. Zakładamy, że agencja podróży oferuje szeroki i bardzo różnorodny zakres usług a klienci nie mają jasno sprecyzowanej wizji wycieczek.
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International Symposium on Modelling and Optimization in Mobile, Ad Hoc, and Wireless Networks
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Deflection measurement of field section with pavement with base course made of Cement Bitumen Treated Material Mixture C3E4 (28, 180, 270, 365 days after compaction)
Dane BadawczeDataset presents data of deflections determined for pavement with base course made of cold recycled mixture – cement bitumen treated material mixture with following binding agents: 3% cement, 4% emulsion (C3E4). Mixture was designed according to Polish requirements for the base course of pavement. Mixture was mixed in stationary plant and compacted...
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Fatigue data of Cement Bitumen Treated Material Mixture C3E5.5 (Direct tension, over 28 days of curing at 20C)
Dane BadawczeFatigue data of Cement Bitumen Treated Material Mixture C3E5.5 (Direct tension, over 28 days of curing at 20C)
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Model of management of knowledge bases in the information technology evaluation environment
PublikacjaThe paper presents the model of management of knowledge bases in multi-agent system for evaluation of information technologies (IT_MAS). Such system is being developed in Gdansk Uni-versity of Technology by Information Technology Management Team. Multi-agent system is supposed to support manager level specialists during decision processes when there is identified need to buy or change any information technology. The main goal of...
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Marta Łabuda dr hab. inż.
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The AFM topographic measurements of the surface heterogeneity of iron hexacyanoferrate on a steel surface
Dane BadawczeMeasurements in semi-contact mode. NTEGRA Prima (NT-MDT) device. NSG 01 probe.
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Płyta czołowa mobilnej stacji pomiarowej
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Metabolic transformation of antitumor acridinone C-1305 but not C-1311 via selective cellular expression of UGT1A10 increases cytotoxic response: implications for clinical use.
PublikacjaThe acridinone derivates C-1305 and C-1311 are promising antitumor agents with high activity against several experimental cellular and tumor models and which are under evaluation in pre-clinical and early phase clinical trials. Recent evidence from our laboratories has indicated that both compounds were conjugated by several UGT isoforms with the most active being extrahepatic UGT1A10. The present studies were designed to test...
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Governmental supported space internship programmes in new ESA member states - Polish perspective
PublikacjaOver last 10 years ve new countries - Czech Republic, Romania, Poland, Hungary and Estonia - have joined the European Space Agency. These countries are currently experiencing a considerable increase of space activities aiming to take part in the European and Global space market. New companies, start-ups and consortiums have been created alongside oces of foreign entities have opened their premises in these countries. All of them...
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Projekt stanowiska badawczego do wyznaczania charakterystyki ogólnej silnika spalinowego ZS przy wykorzystaniu hydraulicznego układu odbioru mocy
PublikacjaPrzedstawiono projekt stanowiska badawczego służącego do wyznaczania charakterystyki ogólnej silnika pojazdu ciężarowego, wykorzystując przystawkę odbioru mocy do napędu układu hydraulicznego generującego obciążenie silnika w różnych punktach jego pracy. Przedstawiono założenia projektowe oraz ograniczenia konstrukcyjne. Omówiono zasadę działania stanowiska i metodę wyznaczania charakterystyki. Opisano układ hydrauliczny oraz układ...
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Uniwersalny Kontroler Radiowy w systemie STRADAR
PublikacjaOpisano praktyczne rozwiązanie uniwersalnego kontrolera radiowego UKR – jednego z podstawowych elementów funkcjonalnych systemu STRADAR – który obsługuje sensory wykorzystywane na granicy morskiej państwa. Jest on także odpowiedzialny za komunikację personelu Straży Granicznej. UKR ma dwie wersje, jedną mobilną – na jednostki pływające, pojazdy lądowe i jednostki latające, drugą stacjonarną – na stałe punkty obserwacyjne rozmieszczone...
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Identification and antimicrobial susceptibility of fecal coliforms isolated from surface water
Publikacjaof 274 fecal coliforms isolated from two watercourses influencing the costal water quality of the gdańsk and the puck bay, 265 were identified as escherichia coli. the remained strains belonged to: acinetobacter spp. (n=1), enterobacter spp. (n=3), klebsiella spp. (n=4) and shigella spp. (n=1). the susceptibility of 222 e. coli was tested against 19 antimicrobial agents: aminoglycosides, carbapenems, cephalosporines, folate antagonists,...
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9,10-Dioxoanthracenyldithiocarbamates effectively inhibit the proliferation of non-small cell lung cancer by targeting multiple protein tyrosine kinases
PublikacjaAnthraquinones have attracted considerable interest in the realm of cancer treatment owing to their potent anticancer properties. This study evaluates the potential of a series of new anthraquinone derivatives as anticancer agents for non-small-cell lung cancer (NSCLC). The compounds were subjected to a range of tests to assess their cytotoxic and apoptotic properties, ability to inhibit colony formation, pro-DNA damage functions,...
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Polymer biodegradable coatings as active substance release systems for urological applications
PublikacjaCatheter-associated urinary tract infections are the result of catheterization of the bladder. The risk of infection is directly proportional to the length of the bladder catheterization. Bacteria cells have the ability to adhere and create the biofilm on the surface of catheter materials. Bacteria’s biofilm is an extremely beneficial environment of existence for microorganisms. Microorganisms that are an integral part of the biofilm...
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Data-Centric Dempster-Shafer Theory-Based Selfishness Thwarting via Trust Evaluation in MANETs and WSNs
PublikacjaPrzedstawiono ramy wymiany informacji reputacyjnej pomiędzy terminalami sieci mobilnej ad hoc lub sensorowej, prowadzące do efektywnej lokalizacji terminali egoistycznych i jednocześnie zapobiegające skutkom fałszywych rekomendacji. Integrację miar zaufania i rekomendacji reputacyjnych oparto na teorii Dempstera-Shafera.
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Ryszard Katulski prof. dr hab. inż.
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Disturbances of Earth magnetic field caused by eddy currents of airplane
PublikacjaThe uniform magnetic field of the Earth in the surrounding of a mobile, metallic object undergoes deformation by eddy currents. The influence of the moving, conducting object on the Earth's total magnetic field depends on the object's shape, position and speed of the changes relative to the magnetic field vector of the Earth, as well as the electric conductivity and the relative magnetic permeability of the material. Disturbances...
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pH -Tunable equilibria in azocrown ethers with histidine moieties, Bioelectrochemistry
PublikacjaThe crown ethers with electro- and photoactive azo moieties containing substituents with mobile protons such as in the –COOH groups of histidine, show unique effect of pH switched on/off presence of the azo form. The differences observed for the electrochemical behavior of azocrown ethers with N-acetylhistidine and imidazole moieties reveal the interference of a chemical reduction pathway in strongly acidified solutions. This...
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Detection of dialogue in movie soundtrack for speech intelligibility enhancement
PublikacjaA method for detecting dialogue in 5.1 movie soundtrack based on interchannel spectral disparity is presented. The front channel signals (left, right, center) are analyzed in the frequency domain. The selected partials in the center channel signal, which yield high disparity with left and right channels, are detected as dialogue. Subsequently, the dialogue frequency components are boosted to achieve increased dialogue intelligibility....
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Interactions with recognized objects
PublikacjaImplicit interaction combined with object recognition techniques opens a new possibility for gathering data and analyzing user behavior for activity and context recognition. The electronic eyewear platform, eGlasses, is being developed, as an integrated and autonomous system to provide interactions with smart environment. In this paper we present a method for the interactions with the recognized objects that can be used for electronic...
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Remote Spatial Database Access in the Navigation System for the Blind
PublikacjaThe article presents the problem of a database access in the navigation systems. The authors were among the main creators of the prototype navigation system for the blind - “Voice Maps”. In the implemented prototype only exemplary, limited spatial data were used, therefore they could be stored in the mobile device’s memory without any difficulties. Currently the aforementioned system is being prepared for commercialization - the...
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ZAPEWNIENIE SYNCHORNIZACJI CZASU PRZY CZĘŚCIOWYM WSPARCIU SIECI
PublikacjaCelem badań zaprezentowanych w artykule było sprawdzenie czy możliwe jest zapewnienie dużej dokładności synchronizacji czasu przy częściowym wsparciu sieci w oparciu o model HRM-1 składający się z 12 szeregowo podłączonych urządzeń sieciowych wraz z wygenerowanym ruchem sieciowym. Badania wykazały, że dla obecnie stosowanych technologii mobilnych takich jak LTE TDD możliwe jest zapewnienie odpowiedniej jakości synchronizacji czasu....
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ENISA Study: Challenges in Securing Industrial Control Systems
PublikacjaIn 2011, the European Network and Information Security Agency (ENISA) conducted a study in the domain of Industrial Control Systems (ICS). Its objective was to obtain the current view on the ICS protectionprimarily in Europe but also in the international context. The portrait' included threats, risks, and challenges in the area of ICS protection as well as national, pan European, and international initiatives on ICS security. The...
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Magdalena Brzozowska-Woś dr hab. inż.
OsobyMagdalena Brzozowska-Woś jest absolwentką Wydziału Zarządzania i Ekonomii Politechniki Gdańskiej (specjalność: systemy zarządzania). Jest również absolwentką Podyplomowego Studium Reklamy (Wydział Zarządzania i Ekonomii PG) oraz Podyplomowego Studium Public Relations (SWPS Uniwersytet Humanistycznospołeczny). W latach 2000-2003 współpracowała z Panoramą Internetu sp. z o. o. jako specjalista ds. marketingu. Pełniła również obowiązki...
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Examination of the epoxy coating system's resistance to Corrobill
PublikacjaThe tests of the influence of the surface cleaning agent on the epoxy coating were carried out. Electrochemical and corrosion tests were carried out. The effect of the preparation on the adhesion and hardness of the tested coating was tested.
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Conception of interactive information and decision support system - model and evaluation
PublikacjaThis article presents conception of interactive information and decision support system for urban and industrial air quality management. The emphasis of the project is on real-time analysis and multi-media information, and support of distributed and mobile clients through the Internet.
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Zanieczyszczenia olejowe
PublikacjaPrzybliżono problematykę zanieczyszczeń olejowych z punktu widzenia technologii ich likwidacji, mając też na uwadze czystsze technologie oczyszczania środowiska. Agencja Ochrony Środowiska z USA zabrania wykorzystywać ropę naftową do badań i prób likwidacji likwidacji rozlewów w terenie, wymuszając stosowanie przyjaznych środowisku substytutów.
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Knowledge management in the processes of project requirements analysis
PublikacjaAuthors, based on one of popular software project management methods as RUP fo-cused on one of most important discipline in project management as requirements management. Authors decomposed the role of the business analyst and present methodological and realizational processes of knowledge managament in traditional and applied sources of knowledge tied with this role. An experiment was conducted in four project teams of all sizes,...
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Business applications of geolocation - modern solutions and trends
PublikacjaThe technological development of geolocation systems has resulted in the utilization of physical location of users by a growing number of entrepreneurs. As mobile technology develops, the use of geolocation in business is becoming widespread with a new range of geomarketing techniques. Entrepreneurs therefore more often utilize geolocation in their promotional and operational activities. In this article mobile-based geolocation...
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Bezzałogowy kołowy pojazd elektryczny do automatycznego wychodzenia z poślizgów
PublikacjaPojazdy bezzałogowe znajdują zastosowanie w wielu dziedzinach współczesnego świata. Pojazdy autonomiczne wraz z algorytmami wspomagającymi kierowanie pojazdami skupiają uwagę wielu zespołów inżynierskich. Jednym z ważniejszych aspektów bezpieczeństwa na drogach jest wspomaganie zapobiegania i wychodzenia z poślizgów w dynamicznym środowisku. Artykuł przedstawia projekt oraz wykonanie bezzałogowego pojazdu kołowego zdolnego do automatycznego...
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LTE as a Trunking - Dispatch System
PublikacjaIn the paper solutions of trunking-dispatch systems based on the LTE system are presented. The solution in the form of separate LTE/TDD trunking system is discussed, and the concept of the LTE/FDD trunking system operating in the infrastructure of public, mobile networks is characterised.
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Low-volume label-free SARS-CoV-2 detection with the microcavity-based optical fiber sensor
PublikacjaAccurate and fast detection of viruses is crucial for controlling outbreaks of many diseases; therefore, to date, numerous sensing systems for their detection have been studied. On top of the performance of these sensing systems, the availability of biorecognition elements specific to especially the new etiological agents is an additional fundamental challenge. Therefore, besides high sensitivity and selectivity, such advantages...
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Therapeutic intervention by the simultaneous inhibition of DNA repair and type I or type II DNA topoisomerases: one strategy, many outcomes
PublikacjaMany anticancer drugs reduce the integrity of DNA, forming strand breaks. This can cause mutations and cancer or cell death if the lesions are not repaired. Interestingly, DNA repair-deficient cancer cells (e.g., those with BRCA1/2 mutations) have been shown to exhibit increased sensitivity to chemotherapy. Based on this observation, a new therapeutic approach termed 'synthetic lethality' has been developed, in which radiation...
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Adam Wronkowski dr inż.
OsobyDoktor nauk społecznych w dyscyplinie geografia społeczno-ekonomiczna i gospodarka przestrzenna. Adiunkt na Wydziale Geografii Społeczno-Ekonomicznej i Gospodarki Przestrzennej Uniwersytetu im. Adama Mickiewicza w Poznaniu. Należy do Zakładu Gospodarki Przestrzennej i Projektowania Urbanistycznego. Moje zainteresowania naukowe obejmują geografie dzieci i osób młodych, w tym w szczególności niezależną mobilność, sprawczość i wzajemne...
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Performance Analysis of Machine Learning Methods with Class Imbalance Problem in Android Malware Detection
PublikacjaDue to the exponential rise of mobile technology, a slew of new mobile security concerns has surfaced recently. To address the hazards connected with malware, many approaches have been developed. Signature-based detection is the most widely used approach for detecting Android malware. This approach has the disadvantage of being unable to identify unknown malware. As a result of this issue, machine learning (ML) for detecting malware...
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Antitumor Activity of Triazine Mimic Antibiotics for DNA-binding Implications (Impressive Activity in Vitro Against a Variety of Tumor Types in the NCI-60 Screen): NSC 710607 To Fight HCT-116 Human Colon Carcinoma Cell Lines in Vivo Using the Hollow Fiber Assay and Xenograft Mouse Models
PublikacjaPurpose Successful clinical applications of DNA-directed selective cytotoxic agents disrupt the vital replication/transcription processes and ultimately lead to cancer cell death. This study aimed to examine the growth screen of two lead triazine compounds in a number of cell lines and xenografts and to develop anticancer agents with noncovalent binding affinity bringing fewer side effects. Methods The NCI initial hollow...
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Pharmaceutical applications of surfactants
PublikacjaIn this study we focused on biological activity of various surfactants. According to our research, they con act both as carriers as well as therapeutic agents. Depending on their concentration, they can create different structures in a solution, which influence their properties. Liposomes have a significant role in drug delivery system. Surfactants in from of bilayer are analogous to natural biological cell membrane.