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dr hab. Piotr F.J. Lipiński
Employment
- 2013 - present Assistant Professor at Neuropeptides Department
Research fields
- No data
Publications
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total: 48
Catalog Publications
Year 2024
Year 2023
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Docking is not enough: 17-trifluoromethylphenyl trinor PGF2α is only a very weak ligand of neurokinin-1 receptor
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Gαi-derived peptide binds the µ-opioid receptor
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Moving out of CF3‐Land: Synthesis, Receptor Affinity, and in silico Studies of NK1 Receptor Ligands Containing a Pentafluorosulfanyl (SF5) Group
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NK1 receptor binding of a few low molecular weight 3,5-bistrifluoromethylbenzene derivatives
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Quantitative chirality in the binding of androgens to their receptor
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Synthesis of Fentanyl Triazole Derivatives and their Affinity for Mu-Opioid and Sigma-1 Receptors
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The influence of a synthetic growth hormone‐releasing hormone analogue G11 and opioid peptide biphalin on selected fibroblasts parameters relevant to wound healing
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Year 2022
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Bifunctional Opioid/Melanocortin Peptidomimetics for Use in Neuropathic Pain: Variation in the Type and Length of the Linker Connecting the Two Pharmacophores
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Correcting a widespread error: Neuroprotectant N-acetyl-L-tryptophan does not bind to the neurokinin-1 receptor
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Fentanyl Structure as a Scaffold for Opioid/Non-Opioid Multitarget Analgesics
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In Vitro Biological Evaluation of Aprepitant Based 177Lu-Radioconjugates
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Novel NK1R-Targeted 68Ga-/177Lu-Radioconjugates with Potential Application against Glioblastoma Multiforme: Preliminary Exploration of Structure–Activity Relationships
Publication
Year 2021
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On Raman optical activity sign-switching between the ground and excited states leading to an unusual resonance ROA induced chirality
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PSMA-D4 Radioligand for Targeted Therapy of Prostate Cancer: Synthesis, Characteristics and Preliminary Assessment of Biological Properties
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Synthesis, Pharmacological Evaluation, and Computational Studies of Cyclic Opioid Peptidomimetics Containing β3-Lysine
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Virtual screening for small molecular non-covalent binders of the SARS-CoV-2 main protease
Publication
Year 2020
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Antinociceptive and Cytotoxic Activity of Opioid Peptides with Hydrazone and Hydrazide Moieties at the C-Terminus
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Enantioselective sensing of (S)-Thalidomide in blood plasma with a chiral naphthalene diimide derivative
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Evaluation of Receptor Affinity, Analgesic Activity and Cytotoxicity of a Hybrid Peptide, AWL3020
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In Vivo, In Vitro and In Silico Studies of the Hybrid Compound AA3266, an Opioid Agonist/NK1R Antagonist with Selective Cytotoxicity
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Pharmacological Profile and Molecular Modeling of Cyclic Opioid Analogues Incorporating Various Phenylalanine Derivatives
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Radiochemical Synthesis and Evaluation of Novel Radioconjugates of Neurokinin 1 Receptor Antagonist Aprepitant Dedicated for NK1R-Positive Tumors
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The analgesic hybrid of dermorphin/substance P and analog of enkephalin improve wound healing in streptozotocin‐induced diabetic rats
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β2-Homo-Amino Acid Scan of µ-Selective Opioid Tetrapeptide TAPP
Publication
Year 2019
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Affinity of fentanyl and its derivatives for the σ1-receptor
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Fentanyl Family at the Mu-Opioid Receptor: Uniform Assessment of Binding and Computational Analysis
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Molecular dynamics of fentanyl bound to μ-opioid receptor
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Triazolopeptides Inhibiting the Interaction between Neuropilin-1 and Vascular Endothelial Growth Factor-165
Publication
Year 2018
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Branched pentapeptides as potent inhibitors of the vascular endothelial growth factor 165 binding to Neuropilin-1: Design, synthesis and biological activity
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Structural Insights into σ1 Receptor Interactions with Opioid Ligands by Molecular Dynamics Simulations
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Structural studies on radiopharmaceutical DOTA-minigastrin analogue (CP04) complexes and their interaction with CCK2 receptor
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Substituent Effect in the First Excited Singlet State of Monosubstituted Benzenes
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The influence of the position of a chiral substituent on undecathiophene chain. A DFT study
Publication
Year 2017
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Conformational latitude – activity relationship of KPPR tetrapeptide analogues toward their ability to inhibit binding of vascular endothelial growth factor 165 to neuropilin‐1
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Hydrazone Linker as a Useful Tool for Preparing Chimeric Peptide/Nonpeptide Bifunctional Compounds
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SCRAMBLE’N’GAMBLE: a tool for fast and facile generation of random data for statistical evaluation of QSAR models
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Structure-activity relationship study of a small cyclic peptide H-c[Lys-Pro-Glu]-Arg-OH: a potent inhibitor of Vascular Endothelial Growth Factor interaction with Neuropilin-1
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Structure-activity relationship study of tetrapeptide inhibitors of the Vascular Endothelial Growth Factor A binding to Neuropilin-1
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The FMO analysis of the molecular interaction of fentanyl derivatives with the μ-opioid receptor
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Year 2016
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Conformation of six fentanyls revisited
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Design, synthesis and in vitro biological evaluation of a small cyclic peptide as inhibitor of vascular endothelial growth factor binding to neuropilin-1
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On splitting of the NICS(1) magnetic aromaticity index
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Substituent effect in theoretical ROA spectra
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Year 2014
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Local chirality measures in QSPR : IR and VCD spectroscopy
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Substituent effect in theoretical VCD spectra
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α-Amino Acids In Water: A Review Of VCD And ROA Spectra
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Year 2012
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Chirality Measures of α-Amino Acids
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