Convenient and Efficient Synthesis of Functionalized 2-Sulfenylindoles

Justyna Doroszuk; Mateusz Musiejuk; Bartosz Jędrzejewski; Juliusz Maksymilian Walczak; Dariusz Witt

doi:10.3390/ma13204492

Convenient and Efficient Synthesis of Functionalized 2-Sulfenylindoles

Abstract

A simple, efficient, and practical sulfenylation at the C2 position of N-tosylindoles under mild conditions was developed. The designed transformation is based on the reaction of N-tosylindoles with BuLi and S-alkyl, and S-aryl phosphorodithioates or thiotosylates to produce 2-sulfenylindoles in moderate to high yields. The presence of additional hydroxy, carboxy, or amino functionalities did not disturb the formation of products

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Articles

Type:

artykuły w czasopismach

Published in:

Materials no. 13,
ISSN: 1996-1944

Language:

English

Publication year:

2020

Bibliographic description:

Doroszuk J., Musiejuk M., Jędrzejewski B., Walczak J., Witt D.: Convenient and Efficient Synthesis of Functionalized 2-Sulfenylindoles// Materials -Vol. 13,iss. 20 (2020), s.4492-

DOI: