Search results for: CHOLINESTERASE INHIBITORY ACTIVITY

• Synthesis and Cholinesterase Inhibitory Activity of N-Phosphorylated /N-Tiophosphorylated Tacrine

  Publication

  • M. Przybyłowska
  • I. Inkielewicz-Stępniak
  • S. Kowalski
  • K. Dzierzbicka
  • S. Demkowicz
  • M. Daśko

  - Medicinal Chemistry - Year 2020

  Novel phosphorus and thiophosphorus tacrine derivatives were designed, synthesized and their biological activity and molecular modeling was investigated as a new potential anti-Alzheimer's disease (AD) agents. All new synthesized compound exhibited lower toxicity against neuroblastoma cell line (SH-SY5Y) in comparison with tacrine. Two analogues in the series, 7 and 9, demonstrated lack of cytotoxicity against hepatocellular cells...

• Variability of Hordeum vulgare L. Cultivars in Yield, Antioxidant Potential, and Cholinesterase Inhibitory Activity

  Publication

  • J. Kobus-Cisowska
  • P. Szulc
  • O. Szczepaniak
  • M. Dziedziński
  • D. Szymanowska
  • K. Szymandera-Buszka
  • E. Goryńska-Goldmann
  • M. Gazdecki
  • A. Telichowska
  • M. Ligaj

  - Sustainability - Year 2020

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• Cholinesterase inhibitory activity, antioxidative potential and microbial stability of innovative liver pâté fortified with rosemary extract (Rosmarinus officinalis)

  Publication

  • A. Bilska
  • J. Kobus-Cisowska
  • D. Kmiecik
  • B. Danyluk
  • R. Kowalski
  • D. Szymanowska
  • A. Gramza-Michałowska
  • O. Szczepaniak

  - ELECTRONIC JOURNAL OF BIOTECHNOLOGY - Year 2019

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• Chocolate desserts with ricotta hydrolysates: In vitro study of inhibitory activity against angiotensin‐converting enzyme and cholinesterase

  Publication

  • J. Kobus‐Cisowska
  • O. Szczepaniak
  • D. Szymanowska
  • M. Przeor
  • M. Jarzębski
  • M. Ligaj
  • A. Gramza‐Michałowska
  • D. Szwajgier
  • J. Foksowicz‐Flaczyk

  - JOURNAL OF FOOD SCIENCE - Year 2020

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• Effect of intensive lipid-lowering therapies on cholinesterase activity in patients with coronary artery disease

  Publication

  • E. Pytel
  • B. Bukowska
  • M. Koter-Michalak
  • M. Olszewska-Banaszczyk
  • P. Gorzelak-Pabiś
  • M. Broncel

  - Pharmacological Reports - Year 2017

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• Composition and In Vitro Effects of Cultivars of Humulus lupulus L. Hops on Cholinesterase Activity and Microbial Growth

  Publication

  • J. Kobus-Cisowska
  • D. Szymanowska-Powałowska
  • O. Szczepaniak
  • D. Kmiecik
  • M. Przeor
  • A. Gramza-Michałowska
  • J. Cielecka-Piontek
  • M. Smuga-Kogut
  • P. Szulc

  - Nutrients - Year 2019

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• Antiplasmodial Activity of Nitroaromatic Compounds: Correlation with Their Reduction Potential and Inhibitory Action on Plasmodium falciparum Glutathione Reductase

  Publication

  • A. Marozienė
  • M. Lesanavičius
  • E. Davioud-Charvet
  • A. Aliverti
  • P. Grellier
  • J. Šarlauskas
  • N. Čėnas

  - MOLECULES - Year 2019

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• Introduction of Pro and Its Analogues in the Conserved P1 Position of Trypsin Inhibitor SFTI-1 Retains Its Inhibitory Activity

  Publication

  • A. Legowska
  • D. Debowski
  • R. Lukajtis
  • E. Sztabkowska
  • A. Mizeria
  • K. Brzozowski
  • M. Wysocka
  • A. Lesner
  • K. Rolka

  - PROTEIN AND PEPTIDE LETTERS - Year 2011

  A number of monocyclic SFTI-1 analogues modified in the conserved inhibitor P1 position by Pro, its L-hydroxyproline (Hyp) derivative as well as mimetics with different ring size were synthesized by the solid-phase method. Replacement of Ser6 by Pro, Hyp, and a four-member ring, L-azetidine-2-carboxylic acid (Aze), retained trypsin or chymotrypsin inhibitory activity. The determined association equilibrium constants of these analogues...

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• Truncation of Huia versabilis Bowman-Birk inhibitor increases its selectivity, matriptase-1 inhibitory activity and proteolytic stability

  Publication

  • A. Gitlin-Domagalska
  • D. Dębowski
  • K. Gucwa
  • D. Starego
  • N. Ptaszyńska
  • A. Sieradzan
  • A. Karczyńska
  • S. Samsonov
  • M. Mangold
  • M. Gütschow... and 2 others

  - BIOCHIMIE - Year 2020

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• Inhibitory activity of double‐sequence analogues of trypsin inhibitor SFTI‐1 from sunflower seeds: an example of peptide splicing

  Publication

  • A. Łęgowska
  • A. Lesner
  • E. Bulak
  • A. Jaśkiewicz
  • A. Sieradzan
  • M. Cydzik
  • P. Stefanowicz
  • Z. Szewczuk
  • K. Rolka

  - FEBS Journal - Year 2010

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