Wyszukiwarka
dr hab. Piotr F.J. Lipiński
Zatrudnienie
- 2013 - present Assistant Professor w Neuropeptides Department
Obszary badawcze
- Brak danych
Publikacje
Filtry
wszystkich: 48
Katalog Publikacji
Rok 2024
Rok 2023
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Docking is not enough: 17-trifluoromethylphenyl trinor PGF2α is only a very weak ligand of neurokinin-1 receptor
Publikacja -
Gαi-derived peptide binds the µ-opioid receptor
Publikacja -
Moving out of CF3‐Land: Synthesis, Receptor Affinity, and in silico Studies of NK1 Receptor Ligands Containing a Pentafluorosulfanyl (SF5) Group
Publikacja -
NK1 receptor binding of a few low molecular weight 3,5-bistrifluoromethylbenzene derivatives
Publikacja -
Quantitative chirality in the binding of androgens to their receptor
Publikacja -
Synthesis of Fentanyl Triazole Derivatives and their Affinity for Mu-Opioid and Sigma-1 Receptors
Publikacja -
The influence of a synthetic growth hormone‐releasing hormone analogue G11 and opioid peptide biphalin on selected fibroblasts parameters relevant to wound healing
Publikacja
Rok 2022
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Bifunctional Opioid/Melanocortin Peptidomimetics for Use in Neuropathic Pain: Variation in the Type and Length of the Linker Connecting the Two Pharmacophores
Publikacja -
Correcting a widespread error: Neuroprotectant N-acetyl-L-tryptophan does not bind to the neurokinin-1 receptor
Publikacja -
Fentanyl Structure as a Scaffold for Opioid/Non-Opioid Multitarget Analgesics
Publikacja -
In Vitro Biological Evaluation of Aprepitant Based 177Lu-Radioconjugates
Publikacja -
Novel NK1R-Targeted 68Ga-/177Lu-Radioconjugates with Potential Application against Glioblastoma Multiforme: Preliminary Exploration of Structure–Activity Relationships
Publikacja
Rok 2021
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On Raman optical activity sign-switching between the ground and excited states leading to an unusual resonance ROA induced chirality
Publikacja -
PSMA-D4 Radioligand for Targeted Therapy of Prostate Cancer: Synthesis, Characteristics and Preliminary Assessment of Biological Properties
Publikacja -
Synthesis, Pharmacological Evaluation, and Computational Studies of Cyclic Opioid Peptidomimetics Containing β3-Lysine
Publikacja -
Virtual screening for small molecular non-covalent binders of the SARS-CoV-2 main protease
Publikacja
Rok 2020
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Antinociceptive and Cytotoxic Activity of Opioid Peptides with Hydrazone and Hydrazide Moieties at the C-Terminus
Publikacja -
Enantioselective sensing of (S)-Thalidomide in blood plasma with a chiral naphthalene diimide derivative
Publikacja -
Evaluation of Receptor Affinity, Analgesic Activity and Cytotoxicity of a Hybrid Peptide, AWL3020
Publikacja -
In Vivo, In Vitro and In Silico Studies of the Hybrid Compound AA3266, an Opioid Agonist/NK1R Antagonist with Selective Cytotoxicity
Publikacja -
Pharmacological Profile and Molecular Modeling of Cyclic Opioid Analogues Incorporating Various Phenylalanine Derivatives
Publikacja -
Radiochemical Synthesis and Evaluation of Novel Radioconjugates of Neurokinin 1 Receptor Antagonist Aprepitant Dedicated for NK1R-Positive Tumors
Publikacja -
The analgesic hybrid of dermorphin/substance P and analog of enkephalin improve wound healing in streptozotocin‐induced diabetic rats
Publikacja -
β2-Homo-Amino Acid Scan of µ-Selective Opioid Tetrapeptide TAPP
Publikacja
Rok 2019
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Affinity of fentanyl and its derivatives for the σ1-receptor
Publikacja -
Fentanyl Family at the Mu-Opioid Receptor: Uniform Assessment of Binding and Computational Analysis
Publikacja -
Molecular dynamics of fentanyl bound to μ-opioid receptor
Publikacja -
Triazolopeptides Inhibiting the Interaction between Neuropilin-1 and Vascular Endothelial Growth Factor-165
Publikacja
Rok 2018
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Branched pentapeptides as potent inhibitors of the vascular endothelial growth factor 165 binding to Neuropilin-1: Design, synthesis and biological activity
Publikacja -
Structural Insights into σ1 Receptor Interactions with Opioid Ligands by Molecular Dynamics Simulations
Publikacja -
Structural studies on radiopharmaceutical DOTA-minigastrin analogue (CP04) complexes and their interaction with CCK2 receptor
Publikacja -
Substituent Effect in the First Excited Singlet State of Monosubstituted Benzenes
Publikacja -
The influence of the position of a chiral substituent on undecathiophene chain. A DFT study
Publikacja
Rok 2017
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Conformational latitude – activity relationship of KPPR tetrapeptide analogues toward their ability to inhibit binding of vascular endothelial growth factor 165 to neuropilin‐1
Publikacja -
Hydrazone Linker as a Useful Tool for Preparing Chimeric Peptide/Nonpeptide Bifunctional Compounds
Publikacja -
SCRAMBLE’N’GAMBLE: a tool for fast and facile generation of random data for statistical evaluation of QSAR models
Publikacja -
Structure-activity relationship study of a small cyclic peptide H-c[Lys-Pro-Glu]-Arg-OH: a potent inhibitor of Vascular Endothelial Growth Factor interaction with Neuropilin-1
Publikacja -
Structure-activity relationship study of tetrapeptide inhibitors of the Vascular Endothelial Growth Factor A binding to Neuropilin-1
Publikacja -
The FMO analysis of the molecular interaction of fentanyl derivatives with the μ-opioid receptor
Publikacja
Rok 2016
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Conformation of six fentanyls revisited
Publikacja -
Design, synthesis and in vitro biological evaluation of a small cyclic peptide as inhibitor of vascular endothelial growth factor binding to neuropilin-1
Publikacja -
On splitting of the NICS(1) magnetic aromaticity index
Publikacja -
Substituent effect in theoretical ROA spectra
Publikacja
Rok 2014
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Local chirality measures in QSPR : IR and VCD spectroscopy
Publikacja -
Substituent effect in theoretical VCD spectra
Publikacja -
α-Amino Acids In Water: A Review Of VCD And ROA Spectra
Publikacja
Rok 2012
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Chirality Measures of α-Amino Acids
Publikacja
wyświetlono 511 razy