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Search results for: BPA ANALOGUES
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Natural Quercetin Analogues Modulate Oxidative Stress Tolerance and Increase Lifespan Extension of S. cerevisiae ( proceeding)
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Spliced analogues of trypsin inhibitor SFTI‐1 and their application for tracing proteolysis and delivery of cargos inside the cells
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Investigation of Serine‐Proteinase‐Catalyzed Peptide Splicing in Analogues of Sunflower Trypsin Inhibitor 1 (SFTI‐1)
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A comparison of geometric analogues of holographic reduced representations, original holographic reduced representations and binary spatter codes
PublicationGeometric Analogues of Holographic Reduced Representations (GA HRR) employ role-filler binding based on geometric products. Atomic objects are real-valued vectors in n-dimensional Euclidean space and complex statements belong to a hierarchy of multivectors. The paper reports a battery of tests aimed at comparison of GA HRR with Holographic Reduced Representation (HRR) and Binary Spatter Codes (BSC). Firstly, we perform a test of...
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The application of isotopically labeled analogues for the determination of small organic compounds by GC/MS with selected ion monitoring
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QSAR, QSPR and QSRR in Terms of 3-D-MoRSE Descriptors for In Silico Screening of Clofibric Acid Analogues
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Docking simulations, Molecular properties and ADMET studies of novel Chromane6,7diol analogues as potential inhibitors of Mushroom tyrosinase
PublicationResearch on inhibition of tyrosinase enzyme has attained significant value, because tyrosinase inhibitors have potential applications in medicine, cosmetics (as whitening agents) and in agriculture (as bioinsecticides). Determination and elucidation of new tyrosinase inhibitors are not only beneficial for medical purposes, but their promising applications in improving food quality and nutritional...
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Peptide conjugates of lactoferricin analogues and antimicrobials—Design, chemical synthesis, evaluation of antimicrobial activity and mammalian cytotoxicity
PublicationEight new peptide conjugates composed of modified bovine lactoferricin truncated analogues (LFcinB) and oneof the three antimicrobials — ciprofloxacin (CIP), levofloxacin (LVX), and fluconazole (FLC) — were synthesized. Four different linkers were applied to connect a peptide and an antimicrobial agent. The FLC-containing peptidic conjugates were synthesized using the “click chemistry” method. This novel approach is reported here...
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Synthesis and biological activity of tuftsin, its analogues and conjugates containing muramyl dipeptides of nor-muramyl dipeptides
PublicationOpisano syntezę koniugatów MDP oraz nor-MDP modyfikowanych w części peptydowej tuftsyną oraz pochodną tuftsyny zawierającą grupę nitrową. Zsyntetyzowane związki zostały przebadane in vitro na ludzkich monocytach i limfocytach w Akademii Medycznej w Gdańsku. Niektóre z nich wykazały szybsze i skuteczniejsze działanie w porównaniu z tuftsyną.
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Semantic memory knowledge acquisition through active dialogues
PublicationSzereg zagadnień językowych nie może zostać rozwiązany bez pamięci semantycznej zawierającej opisy cech obiektów, Automatyczne tworzenie tego rodzaju pamięci jest wielkim wyzwaniem nawet dla prostych obszarów dziedzinowych. Implementacja pamięci semantycznej opartej na reprezentacji wiedzy poprzez powiązania obiektu z jego cechami pokazuje ciekawe zastosowania które nie zostały dotychczas zademonstrowane poprzez bardziej wyszukane...
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Physicochemical and rheological properties of lentil milk/inulin blend—A feta cheese analogue
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On fault diagnosis of analogue electronic circuits based on transformations in multi-dimensional spaces.
PublicationPrzedstawiono ideę nowej klasy metod diagnostycznych opartej na przekształceniu transformującym zmiany parametru układu na krzywe identyfikacyjne w przestrzeniach wielowymiarowych. Rozszerzono również klasę tych metod na diagnostykę uszkodzeń wielokrotnych. Dla takich metod omówiono algorytm lokalizacji i identyfikacji pojedynczych i wielokrotnych uszkodzeń parametrycznych w liniowych układach elektronicznych. Przedstawiono rezultaty...
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Solution conformational study of Scyliorhinin I analogues with conformational constraints by two-dimensional NMR and theoretical conformational analysis
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Use of NMR and Fluorescence Spectroscopy as well as Theoretical Conformational Analysis in Conformation-activity Studies of Cyclic Enkephalin Analogues
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Interactions of vasopressin and oxytocin receptors with vasopressin analogues substituted in position 2 with 3,3′-diphenylalanine - a molecular docking study
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Micelle-bound conformations of neurohypophyseal hormone analogues modified with a Cα-disubstituted residue: NMR and molecular modelling studies
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Highly Potent Antidiuretic Antagonists: Conformational Studies of Vasopressin Analogues Modified with 1-Naphthylalanine Enantiomers at Position 2
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Electrodes consisting of PEDOT modified by Prussian Blue analogues deposited onto titania nanotubes – Their highly improved capacitance
PublicationIn this work we present the outstanding energy storage of prepared inorganic-organic heterojunction where hydrogenated ordered titania nanotubes (H-TiO2NT) were modified by the hybrid made of poly(3,4-ethylenedioxythiophene) (pEDOT) and iron hexacyanoferrate centres (Fehcf, Prussian Blue). The material TiO2NT/pEDOT:Fechf was obtained electrochemically by means of: anodization, hydrogenation and finally, electropolymerization of...
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Application of cross-priming amplification (CPA) for detection of fowl adenovirus (FAdV) strains
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Modernizm gdyński - modernizm europejski. Inspiracje i analogie
PublicationModernizm gdyński znajduje swe wyraźne korzenie w nurtach architektury europejskiej okresu międzywojennego.Głównymi ośrodkami kształtowanie się tych nurtów były artystyczne stolice europejskie, takie jak Paryż, Berlin, Wiedeń, Amsterdam, Rotterdam,Bruksela, Stuttgard i Hamburg. Artykuł wskazuje na analogie między wybitnymi realizacjami europejskimi a architekturą gdyńskiego moderizmu.
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Synthesis of Combretastatin A-4 Analogs and their Biological Activities
PublicationCombretastatin A-4 (CA-4) is a natural product, which consists of two phenyl rings, linked by an ethylene bridge. CA-4, inhibitor of polymerization of tubulin to microtubules, possesses a strong antitumor and anti-vascular properties both in vitro and in vivo. Previous studies showed that disodium phosphate salt of CA-4, a water-soluble prodrug is well tolerated at therapeutically useful doses. However, it should be noted that...
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Phase Centre Corrections of GNSS Antennas and Their Consistency with ATX Catalogues
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Structural studies on radiopharmaceutical DOTA-minigastrin analogue (CP04) complexes and their interaction with CCK2 receptor
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Evaluation of Chemotherapeutic Activity of the Selected Bases’ Analogues of Nucleic Acids Supported by ab initio Various Quantum Chemical Calculations
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The quantification of bisphenols and their analogues in wastewaters and surface water by an improved solid-phase extraction gas chromatography/mass spectrometry method
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Raman and surface-enhanced Raman spectroscopy investigation of vasopressin analogues containing 1-aminocyclohexane-1-carboxylic acid residue
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Influence of bulky 3,3′-diphenylalanine enantiomers replacing position 2 of AVP analogues on their conformations: NMR and molecular modeling studies
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A study on the protection of methionine and the reduction of methionine sulfoxide in methionine-containing analogues of the growth-modeling factor Gly-His-Lys
PublicationThe protection of methionine and the reduction of methionine sulfoxide in methionine-containing analogues of Gly-His-Lys are described. The peptides were synthesized by a solid-phase method using the standard Fmoc procedure. Simultaneous deprotection of the peptide side chain and liberation from the resin were achieved using an appropriate TFA cocktail. The TFA cocktail was selected to minimize oxidation of the methionine residue....
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Hybrid analogues of SFTI-1 modified in P1 position by β- and γ-amino acids and N-substituted β-alanines
PublicationA series of compounds containing either non-proteinogenic beta-/gamma-amino acids or N-substituted beta-alanine residues (beta-peptoid units) in P-1 specificity position were synthesized based on the structure of sunflower trypsin inhibitor 1 (SFTI-1). The compounds were synthesized on a solid support; the N-substituted beta-alanines (beta Nhlys and beta Nhphe) were introduced into a peptidomimetic chain via a two-step approach...
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Introduction of Pro and Its Analogues in the Conserved P1 Position of Trypsin Inhibitor SFTI-1 Retains Its Inhibitory Activity
PublicationA number of monocyclic SFTI-1 analogues modified in the conserved inhibitor P1 position by Pro, its L-hydroxyproline (Hyp) derivative as well as mimetics with different ring size were synthesized by the solid-phase method. Replacement of Ser6 by Pro, Hyp, and a four-member ring, L-azetidine-2-carboxylic acid (Aze), retained trypsin or chymotrypsin inhibitory activity. The determined association equilibrium constants of these analogues...
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Inhibitory activity of double‐sequence analogues of trypsin inhibitor SFTI‐1 from sunflower seeds: an example of peptide splicing
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Antimicrobial Activity of Chimera Peptides Composed of Human Neutrophil Peptide 1 (HNP-1) Truncated Analogues and Bovine Lactoferrampin
PublicationThree chimera peptides composed of bovine lactoferrampin and the analogue of truncated human neutrophil peptide 1 were synthesized by the solid-phase method. In two compounds peptide chains were connected via isopeptide bond, whereas in the third one disulfide bridge served as a linker. All three chimeras displayed significantly higher antimicrobial activity than the constituent peptides as well as their equimolar mixtures. The...
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Analysis of Video Transmission Capabilities in a Simulated OFDM-Based Supplementary BPL-PLC System
PublicationThe design and maintenance of a reliable communication system, especially in harsh working conditions for the oil and mining industry, brings many challenges. With the use of a video transmission system, one can monitor the crew and their working environment. Broadband over power line–power line communication (BPL-PLC) seems an ideal medium for such a service, since it enables the use of the existing wired infrastructure for supplementary...
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Two bacterial small heat shock proteins, IbpA and IbpB, form a functional heterodimer
PublicationSmall heat shock proteins (sHsps) are a conserved class of ATP-independent chaperones which in stress conditions bind to unfolded protein substrates and prevent their irreversible aggregation. Substrates trapped in sHsps-containing aggregates are efficiently refolded into native structures by ATP-dependent Hsp70 and Hsp100 chaperones. Most γ-proteobacteria possess a single sHsp (IbpA), while in a subset of Enterobacterales, as...
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Investigation on air quality of specific indoor environments—spa salons located in Gdynia, Poland
PublicationDue to excessive application of essential oils and scented products in spa salons during aromatherapy and massage sessions, the elevated concentration of total volatile organic compounds (TVOCs), particularly terpenes, which are known as secondary organic aerosol (SOA) precursors, is expected there. This study was aimed at determination of VOCs with a particular regard to terpenes in air samples collected in selected spa salons...
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Subjective Quality Evaluation of Speech Signals Transmitted via BPL-PLC Wired System
PublicationThe broadband over power line – power line communication (BPL-PLC) cable is resistant to electricity stoppage and partial damage of phase conductors. It maintains continuity of transmission in case of an emergency. These features make it an ideal solution for delivering data, e.g. in an underground mine environment, especially clear and easily understandable voice messages. This paper describes a subjective quality evaluation of...
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New vitamin D analogs as potential therapeutics in melanoma
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Phosphate and Thiophosphate Biphenyl Analogs as Steroid Sulfatase Inhibitors
PublicationIn the present work, we report convenient methods for the synthesis and biological evaluation of phosphate and thiophosphate biphenyl derivatives exhibiting steroid sulfatase (STS) activity. The described synthesis is based on straightforward preparation of biphenyl-4-ol and 40-hydroxybiphenyl- 4-carboxylic acid ethyl ester modified with various phosphate or thiophosphate moieties. The inhibitory effects of these compounds were...
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Phase Transitions and Structural Changes in DPPC Liposomes Induced by a 1-Carba-Alpha-Tocopherol Analogue
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An initial assessment of correlations between host- and virus-related factors affecting analogues antiviral therapy in HBV chronically infected patients
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Arginine-, d-arginine-vasopressin, and their inverso analogues in micellar and liposomic models of cell membrane: CD, NMR, and molecular dynamics studies
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Synergistic catalysis of Fe3O4/CuO bimetallic catalyst derived from Prussian blue analogues for the efficient decomposition of various organic pollutants
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Helicity discrimination in N,N'-dibenzoyl-1,2,3,4,7,8,9,10-octahydro-1,10-phenanthrolines and their thiono- and selenocarbonyl analogues by inclusion complexation with chiral diols
PublicationX-ray crystallographic analysis of the title compounds revealed that they assume a folded helical con- formation of an approximate C2 symmetry in the solid state. Dithioamide, diselenoamide and monoselenoamide were resolved to enantiomers by inclusion crystallization with optically active diols (TADDOLs). The absolute configuration of the guest molecules in the complexes was assigned as P. The optical activity of the resolved compounds...
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Internet w służbie historii. Zbiory muzealne Sekcji Historycznej BPG w przestrzeni internetowej
PublicationChoć liczne są funkcje, jakie mogą pełnić strony internetowe –zadania informacyjne, marketingowe, kontaktowe (komunikacyjne),społecznościowe, płatnicze czy rezerwujące – każda witryna WWWzostała przede wszystkim stworzona do przekazywania informacji. Zatakie możemy również uznać informacje na temat posiadanych przezmuzea zbiorów, a dynamiczny rozwój Internetu jako globalnego mediumwymusza...
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Ce-modified zeolite BEA catalysts for the trichloroethylene oxidation. The role of the different and necessary active sites
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Anomalous pressure dependence of acoustic phonons of AgGaSe2 investigated by inelastic neutron scattering to 4.3 GPa
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Quality Evaluation of Voice Transmission Using BPL Communication System in MV Mine Cable Network
PublicationThis article presents results of a quality evaluation study, considering voice transmission in a 6 kV medium voltage cable network using the BPL (Broadband over Power Line) communication system. The tests are carried out under real mining conditions for the selected power cable without voltage, earthed at both sides. Such a method of monitoring work conditions is of great importance, especially during a disaster. Power cables are...
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Attempt to a Video-Transmission Capability in MV Mine Cable Network Using BPL-PLC Technology
PublicationThis article presents and discusses the attempt to transmit video content using the BPL-PLC (Broadband over Power Line - Power Line Communication) technology. It includes simulation results of a specially developed digital transmitter and receiver, dedicated to a given predefined 6 kV mining power cable. The effect of two different transmission modes (2-7 MHz and 3-7.5 MHz) and two types of coupling (capacitive-inductive and induction-inductive),...
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Równoległa realizacja dostępu ISDN-BRA i transmisji danych xDSL w sieci dostępowej
PublicationPrzedstawiono możliwości zrealizowania dostępu ISDN-BRA z wykorzystaniem wydzielonej części przepływności w standardowych systemach xDSL. Jednoczesny dostęp do usług ISDN i do usług szerokopasmowych przy użyciu techniki xDSL we wspólnej sieci dostępowej o przewodach miedzianych można uzyskać korzystając z rozdziału zakresu częstotliwości, wykorzystując wyodrębnienie niezależnych kanałów cyfrowych (STM) w strukturze ramki xDSL lub...
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Effect of resveratrol analogue, DMU-212, on antioxidant status and apoptosis-related genes in rat model of hepatocarcinogenesis
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