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Search results for: CHIRAL PHARMACEUTICALS
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New approach based on solid-phase extraction for the assessment of organic compound pollutions in so-called pharmaceutically pure water
PublicationOpisano mozliwość zastosowania nowej procedury analitycznej opartej na wykorzystaniu techniki ekstrakcji do fazy stałej (na etapie izolacji i wzbogacania analitów) do oznaczania śladowych ilości zanieczyszczeń organicznych w wodzie specjalnej czystości używanej do celów farmaceutycznych.Próbka badanej wody jest przepuszczana przez złoże sorbenta, które jest osuszane za pomocą strumienia oczyszczonego powietrza, przed etapem termicznej...
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Chiralne katalizatory tiomocznikowe w reakcji stereoselektywnego alkilowania związków heteroaromatycznych
PublicationNiniejsza praca doktorska podzielona jest na trzy zasadnicze części: wstęp teoretyczny, badania własne oraz część eksperymentalną. Studium literaturowe obejmuje przegląd doniesień z ostatnich lat z dziedziny organokatalizy niekowalenycjnej. Zaprezentowano zakres zastosowań organokatalizatorów tiomocznikowych jednofunkcyjnych i dwufunkcyjnych z uwzględnieniem ograniczeń w strukturze reagentów, roli dodatków katalitycznych i mechanizmu...
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Exploration of the Solubility Hyperspace of Selected Active Pharmaceutical Ingredients in Choline- and Betaine-Based Deep Eutectic Solvents: Machine Learning Modeling and Experimental Validation
PublicationDeep eutectic solvents (DESs) are popular green media used for various industrial, pharmaceutical, and biomedical applications. However, the possible compositions of eutectic systems are so numerous that it is impossible to study all of them experimentally. To remedy this limitation, the solubility landscape of selected active pharmaceutical ingredients (APIs) in choline chloride- and betaine-based deep eutectic solvents was...
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A Novel Electrochemical Sensor Based on Graphene Oxide Nanosheets and Ionic Liquid Binder for Differential Pulse Voltammetric Determination of Droxidopa in Pharmaceutical and Urine Samples
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Artemisia abrotanum L. (Southern Wormwood)—History, Current Knowledge on the Chemistry, Biological Activity, Traditional Use and Possible New Pharmaceutical and Cosmetological Applications
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Elemental characteristics of mushroom species cultivated in China and Poland
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Determination of electrode impedance by means of exponential chirp signal
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Economic significance of initial public offerings in China and India
PublicationRapid economic growth in China and India has attracted attention of many researchers, focusing on various social and economic factors underlying the success of these countries. One of the key components of country’s economy is financial system which consists of segments such as banking sector and equity market. The topic of initial public offerings (IPOs), one of the corporate financing sources, involving raising funds through...
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Determination of electrode impedance by means of exponential chirp signal.
PublicationPrzedstawiona została nowa metoda pomiaru impedancji elektrodowej. Jako pobudzenie zastosowany został niestacjonarny sygnał napięciowy, którego częstotliwość jest ekspotencjalną funkcją czasu. Zastosowanie zmodyfikowanej któtko-czasowej transformaty Fouriera (STFT) w analizie napięciowego pobudzenia i odpowiedzi prądowej pozwala na otrzymanie widma impedancyjnego.
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Efficacy of intralesional bleomycin in treatment resistant viral warts
PublicationIntroduction Optimal management of treatment-refractory viral warts caused by human papillomavirus is unknown. One of the treatment methods is intralesional bleomycin solution. Objective To determine risk factors for resistant viral warts (not responding to conventional treatments for ≥ 6 months), to determine the effectiveness and safety of intralesional bleomycin in a group of patients with viral warts resistant to conventional...
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Monosaccharides as internal probes for the determination of the absolute configuration of 2-butanol
PublicationD-dlukoza, D-mannoza i L-ramnoza zostały poddane reakcji z mieszaniną racemiczną 2-butanolu. Otrzymane w ten sposób glikozydy były analizowane za pomocą spektroskopii NMR, z wykorzystaniem eksperymentów COSY i NOESY. Analiza konformacyjna wiązania glikozydowego (dokonana w oparciu o modelowanie molekularne i heteronuklearne stałe sprzężenia) wraz z analizą sprzężeń dipolowych obserwowanych w widmie NOESY umożliwiła określenie konfiguracji...
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Development of factors and measurement of personnel risk in the marketing services of four Polish pharmaceutical companies
Open Research DataThis text contains the presentation and analysis of research results in relation to four companies (A, B, C, D), according to the adopted case study method.Further considerations should be preceded by the assumption that personal risk factors often affect the level of this risk in various directions, so their final impact is the result of the shaping...
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New thiourea organocatalysts and their application for the synthesis of 5-(1H-indol-3-yl)methyl-2,2-dimethyl-1,3-dioxane-4,6-diones a source of chiral 3-indoylmethyl ketenes
PublicationThe stereoselective properties of modified thiourea organocatalysts were tested in the Friedel–Crafts alkylation of indole with 5-arylidene-2,2-dimethyl-1,3-dioxane-4,6-diones, which produces chiral 5-((1H-indol-3-yl)(aryl)methyl)-2,2-dimethyl-1,3-dioxane-4,6-diones. Based on a tentative reaction mechanism for ((S)-N-benzyl-2-(3-(3,5-bis (trifluoromethyl)phenyl)thioureido)-N,3,3-trimethylbutanamide organocatalysts, modifications...
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The Role of NF-κB in Uterine Spiral Arteries Remodeling, Insight into the Cornerstone of Preeclampsia
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A STUDY OF THE ORIGINAL AND CONTEMPORARY LAYOUT OF NAZAR GARDEN WITHIN THE CITY OF SHIRAZ, IRAN
PublicationShiraz city was famous for its beautiful gardens that shaped its landscape. Nazar Garden,with its buildings was designed by Karim Khan in the 18th c. The aim of the research wasto compare the size and layout of the Garden during the Zand Period with its contemporary shape. The research was based on literature sources, available plans and an on-sitesurvey.
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Minimum vertex ranking spanning tree problem for chordal and proper interval graphs
PublicationW pracy rozważamy problem szukania, dla danego grafu prostego, drzewa spinającego, którego uporządkowana liczba chromatyczna jest minimalna. K.~Miyata i inni dowiedli w [Np-hardness proof and an approximation algorithm for the minimum vertex ranking spanning tree problem,Discrete Appl. Math. 154 (2006) 2402-2410], że odpowiedni problem decyzyjny jest NP-trudny już w przypadku pytania o istnienie uporządkowanego 4-pokolorowania....
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Determination of pharmaceutical residues in drinking water in Poland using a new SPE-GC-MS(SIM) method based on Speedisk extraction disks and DIMETRIS derivatization
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Determination of mefenamic acid in urine and pharmaceutical samples by HPLC after pipette-tip solid phase microextraction using zinc sulfide modified carbon nanotubes
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Ecotoxicological equilibria of triclosan inMicrotox, XenoScreen YES/YAS, Caco2, HEPG2 and liposomal systems are affected by the occurrence of other pharmaceutical and personal care emerging contaminants
PublicationContaminants of emerging concernmay be considered as any chemicals or factorswhose unintended continuous release and persistence in the environmentmay lead to any observable undesirable response of living beings. Still not much is known on reciprocal toxicological impact of given chemicals when present in binary or more complex mixtures. In thiswork, an attemptwas thus undertaken to study the impact of butylparaben,methylparaben and...
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Acta Pharmaceutica Sinica B
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International Journal of Applied Pharmaceutics
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Jundishapur Journal of Natural Pharmaceutical Products
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International Journal of Pharmaceutical Sciences and Research
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World Journal of Pharmacy and Pharmaceutical Sciences
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Journal of Advanced Pharmaceutical Technology & Research
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International Journal of Pharmaceutical and Phytopharmacological Research
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International Journal of Pharmaceutical and Healthcare Marketing
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International Journal of Innovations in Pharmaceutical Sciences
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PDA JOURNAL OF PHARMACEUTICAL SCIENCE AND TECHNOLOGY
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Journal of Pharmaceutical Health Care and Sciences
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Indo American Journal of Pharmaceutical Sciences
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International Journal of Advances in Pharmaceutical Analysis
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Journal of Pharmaceutical Health Services Research
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Asian Journal of Biomedical and Pharmaceutical Sciences
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Indian Journal of Pharmaceutical Education and Research
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International Journal of Pharmaceutical Quality Assurance
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Dhaka University Journal of Pharmaceutical Sciences
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International Journal of Research in Pharmaceutical Sciences
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International Journal of Current Pharmaceutical Research
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Journal of Global Trends in Pharmaceutical Sciences
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Asian Journal of Pharmaceutical and Clinical Research
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Journal of Medical Pharmaceutical and Allied Sciences
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International Journal of Pharmaceutical Sciences and Nanotechnology
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European Journal of Parenteral and Pharmaceutical Sciences
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Optimization of impedance measurements using ‘chirp’ type perturbation signal
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Emerging developments in ASEAN–China relations in regional production linkages
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Looking for the sectoral interdependence: evidence from the Visegrad countries and China
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Pathophysiology of Clinical Symptoms in Acute Viral Respiratory Tract Infections
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Price nonsynchronicity, idiosyncratic risk, and expected stock returns in China
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Optimization of impedance measurements using ''chirp'' type perturbation signal
PublicationW pracy przedstawiono innowacyjny sposób pomiaru impedancji przy użyciu sygnału niestacjonarnego "chirp". W procesie akwizycji pobudzenia i odpowiedzi prądowej zastosowano zmienną częstotliwość próbkowania. Podejście takie pozwala zarówno na wielokrotne zmniejszenie ilości niezbędnych do otrzymania widma impedancyjnego rejestrowanych danych jak również upraszcza i przyspiesza proces obliczeniowy. Stwierdzono iż dokładność wyników...