Filters
total: 1512
-
Catalog
displaying 1000 best results Help
Search results for: controlled drug delivery
-
Antimicrobials Are a Photodynamic Inactivation Adjuvant for the Eradication of Extensively Drug-Resistant Acinetobacter baumannii
Publication -
Interactions of dissolved dsDNA with intercalating drug by anodic voltammetry and spectroscopy. Influence of pH
PublicationOddziaływanie związku przeciwnowotworowego C-1305 z DNA było badane przy pomocy impulsowej voltametrii różnicowej oraz spektroskopii UV/Vis. Triazoloakrydon C-1305 oddziałuje z DNA na dwóch drogach: przez interkalacje pomiedzy pary zasad oraz przez wiązanie sie w małym rowku helisy. W fizjologicznym pH (7,4) stałe wiązania wynoszą: K1=3,36E+5 i K2=0,18E+5 [1/M] a wielkość miejsca wiązania: n1=2,5 i n2=4,0, odpowiednio dla pierwszego...
-
Regenerative Drug Discovery Using Ear Pinna Punch Wound Model in Mice
PublicationThe ear pinna is a complex tissue consisting of the dermis, cartilage, muscles, vessels, and nerves. Ear pinna healing is a model of regeneration in mammals. In some mammals, including rabbits, punch wounds in the ear pinna close spontaneously; in common-use laboratory mice, they remain for life. Agents inducing ear pinna healing are potential regenerative drugs. We tested the effects of selected bioactive agents on 2 mm ear pinna...
-
Molecular mechanism of the enzymatic oxidation investigated for imidazoacridinone antitumor drug C-1311.
PublicationPraca miala na celu określenie molekularnego mechanizmu enzymatycznej utleniającej aktywacji wymienionego związku przeciwnowotworowego w takim układzie modelowym, w którym wcześniej wykazano jego kowalencyjne wiązanie się do DNA. Badania struktur chemicznych produktów enzymatycznej aktywacji wykazały, że dwa z nich powstają w wyniku dealkilacji łańcucha bocznego cząsteczki, natomiast dwa inne w wyniku aktywacji pierścienia imidazoakrydonu....
-
Optimizing Last-Mile Delivery: A Multi-Criteria Approach with Automated Smart Lockers, Capillary Distribution and Crowdshipping
Publication -
Spliced analogues of trypsin inhibitor SFTI‐1 and their application for tracing proteolysis and delivery of cargos inside the cells
Publication -
Trans-endocardial delivery of progenitor cells to compromised myocardium using the “needle technique”and risk of myocardial injury
Publication -
A Method for the Evaluation of Urban Freight Transport Models as a Tool for Improving the Delivery of Sustainable Urban Transport Policy
PublicationThe article presents a method which helps local authorities to evaluate urban freight transport models. Given the complex requirements for input data and the inability to supply them for most cities, a proper quantitative evaluation of model functionality may be quite difficult for local authorities. Freight transport models designed to support sustainable urban freight transport objectives are a particular example. To overcome...
-
A Decade of Wishes-Changes in Maternal Preference of the Mode of Delivery among Polish Women over the Last Decade
Publication -
Preoperative nutritional support in cancer patients with no clinical signs of malnutrition—prospective randomized controlled trial
Publication -
The impact of an electronic monitoring and reminder device on patient compliance with antihypertensive therapy: a randomized controlled trial
Publication -
The effects of statins on blood pressure in normotensive or hypertensive subjects — A meta-analysis of randomized controlled trials
Publication -
Safety and efficacy of lenabasum in a phase 2 randomized, placebo-controlled trial in adults with cystic fibrosis
Publication -
Melatonin and clonidine premedication has similar impact on the pharmacokinetics and pharmacodynamics of propofol target controlled-infusions
Publication -
Mechatronics in the design of three wheeled mobile platform controlled by surveillance system at energy performance index
PublicationPraca jest poświęcona projektowaniu mechatronicznemu trójkołowej platformy mobilnej, sterowanej systemem nadzorowania bazującym na energetycznym wskaźniku jakości. Zdefiniowany zakres badań i silna nieliniowość obiektu wymagały niezawodnego systemu sterowania. Warunki deterministyczne i zastosowany algorytm wpłynęły na wybór metody opracowania systemu. Przedstawione techniki projektowania mechatronicznego i przeprowadzone warianty...
-
Efficacy of the Whole-Body Cryotherapy as Add-on Therapy to Pharmacological Treatment of Depression—A Randomized Controlled Trial
Publication -
Intercalation complex of imidazoacridinone C-1311, a potential anticancer drug, with DNA helix d(CGATCG)2: stereostructural studies by 2D NMR spectroscopy.
PublicationImidazoacridinone C-1311 (Symadex®) is a powerful antitumor agent, which successfully made its way through the Phase I clinical trials and has been recommended for Phase II few a years ago. It has been shown experimentally that during the initial stage of its action C-1311 forms a relatively stable intercalation complex with DNA, yet it has shown no base-sequence specificity while binding to DNA. In this paper, the d(CGATCG)2:C-1311...
-
New Life of an Old Drug: Caffeine as a Modulator of Antibacterial Activity of Commonly Used Antibiotics
Publication -
The Current Use of Mass Spectrometry in Combination with Other Separation Techniques in Drug Discovery Arena
Publication -
Activity of Phage–Lactoferrin Mixture against Multi Drug Resistant Staphylococcus aureus Biofilms
Publication -
Cisplatin filled multiwalled carbon nanotubes – a novel molecular hybrid of anticancer drug container
Publication -
The modulatory effect of green tea catechin on drug resistance in human ovarian cancer cells
Publication -
Acinetobacter baumannii isolated from hospital‐acquired infection: biofilm production and drug susceptibility
Publication -
Fulminant hepatic failure in woman with iron and non-steroidal anti-inflammatory drug intoxication
Publication -
Drug transporter expression profiling in chemoresistant variants of the A2780 ovarian cancer cell line
Publication -
Drug-Releasing Antibacterial Coating Made from Nano-Hydroxyapatite Using the Sonocoating Method
Publication -
Homoisocitrate dehydrogenase from Candida albicans: properties, inhibition, and targeting by an antifungal pro-drug
PublicationThe LYS12 gene from Candida albicans, coding for homoisocitrate dehydrogenase was cloned and expressed as a His-tagged protein in Escherichia coli. The purified gene product catalyzes the Mg2+- and K+-dependent oxidative decarboxylation of homoisocitrate to alpha-ketoadipate. The recombinant enzyme demonstrates strict specificity for homoisocitrate. SDS-PAGE of CaHIcDH revealed its molecular mass of 42.6±1 kDa, while in size-exclusion...
-
Glucosamine-6-phosphate synthase,a novel target for antifungalagents.Molecular modelling studies in drug design
PublicationPraca dotyczy modelowania zarówno samych inhibitorów syntazy glukozamino-6-fosforanu jak i ich oddziaływania z obydwiema domenami tego enzymu. Enzym syntaza glukozamino-6-fosforanu został zaproponowany jako nowy cel molekularny w chemoterapii infekcji grzybowych. Zaprojektowano i zsyntezowano szereg inhibitorów tego enzymu - potencjalnych nowych leków przeciwgrzybowych. Dzięki modelowaniu molekularnemu udało się wyjaśnić mechanizm...
-
Correction to “Emerging Anticancer Activity of Candidal Glucosamine-6-Phosphate Synthase Inhibitors upon Nanoparticle-Mediated Delivery”
Publication -
Hydrogel Delivery System Containing Calendulae flos Lyophilized Extract with Chitosan as a Supporting Strategy for Wound Healing Applications
Publication -
Twenty‐four‐hour and conventional blood pressure components and risk of preterm delivery or neonatal complications in gestational hypertension
Publication -
DRUG AND CHEMICAL TOXICOLOGY
Journals -
DRUG METABOLISM AND DISPOSITION
Journals -
DRUG DEVELOPMENT RESEARCH
Journals -
DRUG METABOLISM REVIEWS
Journals -
Jarosław Guziński prof. dr hab. inż.
PeopleJaroslaw Guzinski received M.Sc., Ph.D. and D.Sc. degrees from the Electrical Engineering Department at Technical University of Gdansk, Poland in 1994, 2000 and 2011 respectively. Since 2016 he is Associate Professor at Gdansk University of Technology. Currently he is the head of the Department of Electric Drives and Energy Conversion. From 2006 to 2009 he was involved in European Commission Project PREMAID Marie Curie, ‘Predictive...
-
Pressure Algometry Evaluation of Two Occlusal Splint Designs in Bruxism Management-Randomized, Controlled Clinical Trial
Publication -
Hydroacoustic System in a Biomimetic Underwater Vehicle to Avoid Collision with Vessels with Low-Speed Propellers in a Controlled Environment
Publication -
Synthesizing of Sensitizing Glasses in Very Small Volumes and Strictly Controlled Atmospheres for Fiber and Integrated Optic Sensors
Publication -
Preparation of matrix-free materials of volatile analytes based on the controlled decomposition of surface compounds: a new concept
PublicationW publikacji przedstawiono nową koncepcję wytwarzania bezmatrycowych materiałów odniesienia wykorzystującą związki powierzchniowe, które są chemicznie związane z powierzchnią nośnika (żelu krzemionkowego, szkła porowatego, pałeczek szklanych pokrytych żelem krzemionkowym, oraz włókna szklanego), które w określonych warunkach temperaturowych ulegają termicznemu rozkładowi lub przegrupowaniom chemicznym z uwolnieniem ściśle określonej...
-
Effect of hybrid TiO2 nanoparticles with controlled morphology on rheological properties of poly(styrene-co-acrylonitrile) nanocomposites
Publication -
ASSAY AND DRUG DEVELOPMENT TECHNOLOGIES
Journals -
ARZNEIMITTEL-FORSCHUNG-DRUG RESEARCH
Journals -
Expert Opinion On Drug Safety
Journals -
American Health and Drug Benefits
Journals -
Journal of Drug Metabolism & Toxicology
Journals -
International Journal of Drug Discovery
Journals -
Expert Opinion on Drug Discovery
Journals -
FOOD AND DRUG LAW JOURNAL
Journals -
Drug Healthcare and Patient Safety
Journals