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wszystkich: 521
Wyniki wyszukiwania dla: ASI
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Synthesis and biological evaluation of thiophosphate tricyclic coumarin derivatives as steroid sulfatase inhibitors
PublikacjaSteroid sulfatase (STS) enzyme inhibition is an important approach to the management of hormone-dependent breast cancer. In this paper, we report convenient methods for the synthesis and biological evaluation of thiophosphate tricyclic coumarin analogs exhibiting STS activity. The described methods are based on the straightforward preparation of 7-hydroxy-2,3-dihydro-1H-cyclopenta[c]chromen-2-one, 3-hydroxy- 7,8,9,10-tetrahydro-6H-benzo[c]chromen-6-one,...
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New potent STS inhibitors based on fluorinated 4-(1-phenyl-1H-[1,2,3]triazol-4-yl)-phenyl sulfamates
PublikacjaA series of fluorinated analogs based on the frameworks of 4-(1- phenyl-1H-[1,2,3]triazol-4-yl)-phenyl sulfamates have been synthesized as steroid sulfatase (STS) inhibitors. The design of chemical structures of new potential STS inhibitors was supported by molecular docking techniques to identify potential interactions between inhibitors and amino acid residues located in the STS active site. The STS inhibitory potency was evaluated...
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Association for Computer-Aided Architectural Design Research in Asia (CAADRIA) annual conference
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Asia Conference on Information, Computer and Communications Security (ACM Symposium on Information, Computer and Communications Security)
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Asia Pacific Symposium on Intelligent and Evolutionary Systems (Australia-Japan Joint Workshop on Intelligent and Evolutionary Systems)
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Zespół Systemów Mikroelektronicznych
Zespoły Badawcze* projektowania I optymalizacji układów i systemów mikroelektronicznych * zaawansowane metody projektowania i optymalizacji analogowych filtrów aktywnych * programowanie układów scalonych (FPGA, CPLD, SPLD, FPAA) * układy specjalizowane ASIC * synteza systemów o małym poborze mocy * projektowanie topografii układów i zagadnień kompatybilności elektromagnetycznej * modelowania przyrządów półprzewodnikowych * modelowania właściwości...
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Influence of a Lighting Column in the Working Width of a W-Beam Barrier on TB51 Crash Test
PublikacjaRoad equipment, such as, e.g., road safety barriers and lighting columns, are subject to certification according to the EN1317 standard to be allowed for use on European roads. In engineering practice, due to the terrain conditions, there are cases where other road equipment is installed within the working width of road safety barriers. Such situations are not considered during the certification process. Hence, the aim of this...
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The LS-index: A Survey
PublikacjaNiniejszy przegląd jest oparty na wykładach autora wygłoszonych na NATO-ASI-SMS w 2004 roku na University of Montreal w Kanadzie.Niech H będzie przestrzenią Hilberta. Rozważmy pole wektorowe f zdefiniowane na H postaci f(x)=L(x)+K(x), gdzie L jest silnie nieokreślonym, ograniczonym operatorem liniowym, a K jego pełnociągłym zaburzeniem. W tej pracy prezentujemy rozszerzenie klasycznego indeksu Conley'a na potoki generowane przez...
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Alan Turower dr inż.
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18th European Symposium on Radiopharmacy and Radiopharmaceuticals
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Safety of Bariatric Surgery in ≥ 65-Year-Old Patients During the COVID-19 Pandemic
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30-Day Morbidity and Mortality of Bariatric Surgery During the COVID-19 Pandemic: a Multinational Cohort Study of 7704 Patients from 42 Countries
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Effect of BMI on safety of bariatric surgery during the COVID-19 pandemic, procedure choice, and safety protocols – An analysis from the GENEVA Study
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30-day morbidity and mortality of sleeve gastrectomy, Roux-en-Y gastric bypass and one anastomosis gastric bypass: a propensity score-matched analysis of the GENEVA data
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Handling of the Covid-19 Pandemic and Its Effects on Bariatric Surgical Practice: Analysis of GENEVA Study Database
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Surgical site infection after gastrointestinal surgery in high-income, middle-income, and low-income countries: a prospective, international, multicentre cohort study
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Effects of hospital facilities on patient outcomes after cancer surgery: an international, prospective, observational study
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Global variation in postoperative mortality and complications after cancer surgery: a multicentre, prospective cohort study in 82 countries
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Elective surgery system strengthening: development, measurement, and validation of the surgical preparedness index across 1632 hospitals in 119 countries
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Global variation in anastomosis and end colostomy formation following left‐sided colorectal resection
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Pooled analysis of WHO Surgical Safety Checklist use and mortality after emergency laparotomy
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