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Wyniki wyszukiwania dla: BISPHENOL A ANALOGUES
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The Multiplatform Environment for Simulation and Features Estimation of Mixed-Signal Devices
PublikacjaThe use of simulation laboratories is gaining popularity in thedomains of engineering programs. However, the experience in teaching showsthat the simulation itself is not very effective in didactic processes. Teachingprocesses in thefield of specialist subjects, designed for students of technicaluniversities, should be based on direct operations performed by the student onreal devices. At the same time, at the later stages of didactic...
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Exploring the cocrystallization potential of urea and benzamide
PublikacjaThe cocrystallization landscape of benzamide and urea interacting with aliphatic and aromatic carboxylic acids was studied both experimentally and theoretically. Ten new cocrystals of benzamide were synthesized using an oriented samples approach via a fast dropped evaporation technique. Information about types of known bi-component cocrystals augmented with knowledge of simple binary eutectic mixtures was used for the analysis...
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Anticancer Properties of Amino Acid and Peptide Derivatives of Mycophenolic Acid
PublikacjaBackground: Although Mycophenolic Acid (MPA) is applied as prodrugs in clinic as an immunosuppressant, it also possesses anticancer activity. MPA acts as Inosine-5’-Monophosphate Dehydrogenase (IMPDH) inhibitor, where the carboxylic group at the end of the side chain interacts with Ser 276 of the enzyme via hydrogen bonds. Therefore, MPA derivatives with other polar groups indicated high inhibition too. On the other hand, potent...
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Characterization of recombinant homocitrate synthase from Candida albicans
PublikacjaLYS21 and LYS22 genes from Candida albicans encoding isoforms of homocitrate synthase (HCS), an enzyme catalyzing the first committed step in the L-lysine biosynthetic pathway, were cloned and expressed as NoligoHistagged fusion proteins in Escherichia coli. The purified gene products revealed HCS activity, i.e. catalyzed the condensation of α-ketoglutarate with acetyl-coenzyme A to yield homocitrate. The recombinant enzymes were purified...
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Molecular basis for the DNA damage induction and anticancer activity of asymmetrically substituted anthrapyridazone PDZ-7
Publikacjanthrapyridazones, imino analogues of anthraquinone, constitute a family of compounds with remarkable anti-cancer activity. To date, over 20 derivatives were studied, of which most displayed nanomolar cytotoxicity towards broad spectrum of cancer cells, including breast, prostate and leukemic ones. BS-154, the most potent derivative, had IC50 values close to 1 nM, however, it was toxic in animal studies. Here, we characterize another...
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Comparison of the coordination geometries of Zn(II) and Cd(II) ions in complexes with water, methanol and bulky aryloxysilanethiolate ligands
PublikacjaZinc and cadmium complexes containing silanethiolate anions and methanol or water were synthesized and characterized by X-ray diffraction, FT-IR and NMR spectroscopy, and DFT calculations. Contrary to zinc, the cadmium ion utilizes very weak donors to complete its coordination sphere; it forms contacts to phenyl rings of the silanethiolate ligand. Two zinc analogs of the general formula [Zn{SSi(OAr)3}2(L)2] where L = CH3OH (2)...
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Plastic Debris in the Stomach of the Invasive Signal Crayfish Pacifastacus leniusculus from a Baltic Coastal River
PublikacjaPollution by plastic debris, widely recognized as a growing global problem [1-3] is caused by the production of synthetic polymers. Over recent years, the production of plastics has increased, while in Europe, fossil-based plastics production has decreased, and recycled plastics production has increased [4]. There are different types of plastics. Some types of plastic ingredients, applied in a wide variety of cosmetics and personal...
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Współczesne zmiany klimatyczne i ich wpływ na funkcjonowanie systemów miejskich (na przykładzie miast strefy nadmorskiej Polski)
PublikacjaThe purpose of this article is to present contemporary climatic changes in their actual scale, and to assess their impact on functioning of urban areas situated on the Polish coast. The results of the analysis of variability of hydro-climatic conditions that occurred in the last 65 years (1951-2015) in the area of the Polish coast suggest that important changes were concerning: (1) temperature of the air, and thickness and length...
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Neural networks and deep learning
PublikacjaIn this chapter we will provide the general and fundamental background related to Neural Networks and Deep Learning techniques. Specifically, we divide the fundamentals of deep learning in three parts, the first one introduces Deep Feed Forward Networks and the main training algorithms in the context of optimization. The second part covers Convolutional Neural Networks (CNN) and discusses their main advantages and shortcomings...
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How Can We Identify Electrophysiological iEEG Activities Associated with Cognitive Functions?
PublikacjaElectrophysiological activities of the brain are engaged in its various functions and give rise to a wide spectrum of low and high frequency oscillations in the intracranial EEG (iEEG) signals, commonly known as the brain waves. The iEEG spectral activities are distributed across networks of cortical and subcortical areas arranged into hierarchical processing streams. It remains a major challenge to identify these activities in...
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Two-spinors, oscillator algebras, and qubits: aspects of manifestly covariant approach to relativistic quantum information
PublikacjaThe first part of the paper reviews applications of 2-spinor methods to relativistic qubits (analogies between tetrads in Minkowski space and 2-qubit states, qubits defined by means of null directions and their role for elimination of the Peres-Scudo-Terno phenomenon, advantages and disadvantages of relativistic polarization operators defined by the Pauli-Lubanski vector, manifestly covariant approach to unitary representations...
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Determination of butyltin stabilizers in PVC using Liquid-Phase microextraction with electrothermal atomic absorption spectrometry
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Neural network approach to 2D Kalman filtering in image processing
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Fixed final time and free final state optimal control problem for fractional dynamic systems – linear quadratic discrete-time case
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Nonlinear control systems modelling: global vs. local
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Adaptive Feedback Control of Fractional Order Discrete State-Space Systems
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Client’s Expectations vs Contractor’s Pricing. Fair Prices or Bid Rigging
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The quality management in precast concrete production and delivery processes supported by association analysis
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Adaptive resolution simulation of liquid para-hydrogen: testing the robustness of the quantum-classical adaptive coupling
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Classical to Path-Integral Adaptive Resolution in Molecular Simulation: Towards a Smooth Quantum-Classical Coupling
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Impact of the medical clothing on the thermal stress of surgeons
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Application of the MSPD Technique for the HPLC Analysis of Rutin in Sambucus nigra L.: The Linear Correlation of the Matrix Solid-Phase Dispersion Process
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Target tracking in RIS
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Effects of lightning and sprites on the ionospheric potential, and threshold effects on sprite initiation, obtained using an analog model of the global atmospheric electric circuit
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Drastically decreased transcription from CII-activated promoters is responsible for impaired lysogenization of the Escherichia coli rpoA341 mutant by bacteriophage λ
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Modeling changes of the ionospheric potential due to lightning and sprites
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Enforced conformational changes in the structural units of glycosaminoglycan (non-sulfated heparin-based oligosaccharides)
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Theoretical estimation of acid–base properties of Lewis and Brønsted centres at the V-W-O catalyst surface: water molecule as the probe in DFT calculations
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A study on transverse shear correction for laminated sandwich panels
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Study of anticorrosion and microwave absorption properties of NiZn ferrite pigments
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Effect of environmental temperature variations on protective properties of organic coatings
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Analysis of electrochemical noise by means of bispectral technique
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DEIS assessment of AISI 304 stainless steel dissolution process in conditions of intergranular corrosion
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OPTIMAL WAVELET CHOICE IN ELECTROCHEMICAL EXPERIMENTS
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Performance evaluation of the construction products as a research challenge. Small error – big difference in assessment?
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The application of Gabor transformation in the harmonic analysis of corrosion processes
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DEIS evaluation of the relative effective surface area of AISI 304 stainless steel dissolution process in conditions of intergranular corrosion
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APPLICATION OF NON-STATIONARY TECHNIQUES IN THE ANALYSIS OF ELECTROCHEMICAL NOISE
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Use of impedance spectroscopy to evaluate the durability of protective coatings after thermal shock
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Accelerated ageing of organic coating systems by thermal treatment
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Impact of sensitization on dissolution process of AISI 304 stainless steel during intergranular corrosion evaluated using DEIS technique
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A comparison of the target tracking in marine navigational radars by means of GRNN filter and numerical filter
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Variability of sea ice deformation rates in the Arctic and their relationship with basin-scale wind forcing
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Thermal properties of poly(vinyl chloride)/polyurethane blends
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Ground-state correlation properties of charged bosons trapped in strongly anisotropic harmonic potentials
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Two-Boson Correlations in Various One-Dimensional Traps
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Thermal properties of polyamide 6/polyurethane blends
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Large eddy simulations of wall-bounded flows using a simplified immersed boundary method and high-order compact schemes
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Generating amplicon reads for microbial community assessment with next‐generation sequencing
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Technology of laser deposition of narrow bead overlays using solid and flux-cored wires
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