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Wyniki wyszukiwania dla: RATIONAL DRUG DESIGN
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Accelerated design optimization of miniaturized microwave passives by design reusing and Kriging interpolation surrogates
PublikacjaElectromagnetic (EM) analysis has become ubiquitous in the design of microwave components and systems. One of the reasons is the increasing topological complexity of the circuits. Their reliable evaluation—at least at the design closure stage—can no longer be carried out using analytical or equivalent network representations. This is especially pertinent to miniaturized structures, where considerable EM cross-coupling effects occurring...
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Design process as complex system
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Using anticipatory and drug-evoked appetitive ultrasonic vocalization for monitoring the rewarding effect of amphetamine in a rat model of drug self-administration
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The Significance of MicroRNAs Expression in Regulation of Extracellular Matrix and Other Drug Resistant Genes in Drug Resistant Ovarian Cancer Cell Lines
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Design. Metodology outline and practice
PublikacjaNa tle - uznawanego za typowy - schematu prac składających się na proces projektowania, pokazano przykładowe tworzenie inicjatywy sprawczej oraz rozwój koncepcji dotyczących sformułowania konkretnego zadania projektowego w dziedzinie budowy maszyn.Temat dotyczył obszaru projektowania turbin wodnych.The origin of project initiative, as well as concept development related to formulating a specific design goal, are presented in the...
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Interaction Design in Agile IT Projects
PublikacjaIn recent years, interactive systems, such as various types of software, online services or mobile applications, have become an integral part of everyday life. Interactive systems and digital services should be easy to use and provide a positive User Experience (UX). For this reason, interaction design has recently emerged as a distinct professional area of information technology (IT). Easy interaction and user experience (UX)...
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Systems Software Design 1
Kursy OnlineSystems Software Design
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Computational Approach towards Repetitive Design Tasks: The Case Study of Parking Lot Automated Design
PublikacjaThe study aims to develop and assess an algorithm for efficiently generating parking spot layouts within predefined area outlines. The algorithm is an attempt to streamline the decisionmaking process by producing different design variants and optimizing the utilization of available space. The algorithm’s primary objective is to streamline decision-making by generating diverse design variants while optimizing the use of available...
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Effectiveness of the robust PSS design
PublikacjaThe paper discusses optimal PSS of synchronous generator synthesis. The optimal controller is an Hinf controller, what means that minimises Hinf norm of transfer function between the exogenous signals such as reference inputs and disturbances, and the error signals which are to be minimised to meet the control objective. The dynamic properties of the plant are shaped by choosing appropriate weighting function applied to the plant...
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Machines Design 2 (PG_00042059) 21-22
Kursy OnlineA course in machine design
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Machines Design 2 (PG_00042059) 2023/24
Kursy OnlineA course in machine design
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Molecular modeling and evaluation of novel dibenzopyrrole derivatives as telomerase inhibitors and potential drug for cancer therapy
PublikacjaDuring previous years, many studies on synthesis, as well as on anti-tumor, anti-inflammatory and anti-bacterial activities of the pyrazole derivatives have been described. Certain pyrazole derivatives exhibit important pharmacological activities and have proved to be useful template in drug research. Considering importance of pyrazole template, in current work the series of novel inhibitors were designed by replacing central...
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Design Space Reduction for Expedited Multi-Objective Design Optimization of Antennas in Highly-Dimensional Spaces
PublikacjaA surrogate-based technique for efficient multi-objective antenna optimization is discussed. Our approach exploits response surface approximation (RSA) model constructed from low-fidelity antenna model data (here, obtained through coarse-discretization electromagnetic simulations). The RSA model enables fast determination of the best available trade-offs between conflicting design goals. The cost of RSA model construction for multi-parameter...
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Design Issues
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Design Studies
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Architectural Design
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Design and Culture
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Design Science
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Ergonomics in Design
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Journal of Design
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VLSI DESIGN
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New Design
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Design of dimensionally stable composites using efficient global optimization method
PublikacjaDimensionally stable material design is an important issue for space structures such as space laser communication systems, telescopes, and satellites. Suitably designed composite materials for this purpose can meet the functional and structural requirements. In this paper, it is aimed to design the dimensionally stable laminated composites by using efficient global optimization method. For this purpose, the composite plate optimization...
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Rapid multi-objective design of integrated on-chip inductors by means of Pareto front exploration and design extrapolation
PublikacjaIdentification of the best trade-offs between conflicting design objectives allows for making educated design decisions as well as assessing suitability of a given component or circuit for a specific application. In case of inductors, the typical objectives include maximization of the quality factor and minimization of the layout area, as well as maintaining a required inductance at a given operating frequency. This work demonstrates...
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Bridge Ergonomic Design: A Review
PublikacjaHuman error remains the most common cause of marine incidents and it is worth emphasizing that navigator’s performance is directly affected by ergonomic factors on the bridge. Studies regarding influence of bridge design and work environment on the operator are rare, thus the main purpose of this paper is to fill in this gap. Documents issued by recognized organizations, research publications and additional sources were reviewed...
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Big Data in Regenerative Urban Design
PublikacjaWhy the use of Big Data in regenerative planning matters? The aim of this chapter is to study under what conditions Big Data can be integrated into regenerative design and sustainable planning? Authors seek to answer how – when related to the ecosystem and to human activities – Big Data can be used to: • both shape policies that support the development of regenerative human settlements, • support restorative design for practitioners...
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Determination of amikacin and ciprofloxacin by liquid chromatography with pre-column derivatization to evaluate sustained delivery of antibiotics from Drug-Eluting Biopsy Needle
PublikacjaDetermination of chosen antibacterial antibiotics: amikacin and ciprofloxacin was carried out by HPLC-UV after derivatization with 9-fluorenylmethyl chloroformate and in their native form by HPLC-MS/MS. Developed methods have been applied to control the kinetics of antibiotic release from polymer-based controlled drug delivery system.
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Theory of Achitectural Design I. 2020/2021
Kursy OnlineLectures on architectural composition and architectural design
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Safety-based approach in multifunctional building design
PublikacjaABSTRACT: The modern trend in design of the public buildings is to create multifunctional environments in one building, hosting a variety of functions. Multifunctional buildings entertain large number of visitors. The complexity and vulnerability of this type of public space are the main reasons to use within their design process the performance based approach including the recognition of hazards. Safety and reliability approach...
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Feasibility study of a Raman spectroscopic route to drug detection
PublikacjaWe present an surface-enhanced Raman spectroscopy (SERS) approach for detection of drugs of abuse in whole human blood. We utilize a near infrared laser with 830 nm excitation wavelength in order to reduce the influence of fluorescence on the spectra of blood. However, regular plasmon resonance peak of plasmonic nanoparticles, such as silver or gold fall in a much lower wavelength regime about 400 nm. Therefore, we have shifted...
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Computer modeling and design of materials 2022/2023
Kursy OnlineComputer modeling and design of materials, kierunek: Nanotechnologia, specjalność: Mathematics for new materials design, II stopień, semestr 3
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Rational Pharmacotherapy in Cardiology [ Рациональная фармакотерапия в кардиологии ]
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Modelling in machine design (PG_00057377)_2024
Kursy OnlineMachine Design - selected problems is a subject in which we will deepen understanding of selected topics from FMD course
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Light4Health eLearning Course: health research for interior lighting design. Re-thinking design approaches based on science
PublikacjaThis paper presents the results of 'Light4Health' (L4H), a three-year EU Erasmus+ Strategic Partnership grant project (2019-2021), which investigated, systematized and taught health-related research on the impact of natural and artificial light on human health and well-being relevant to indoor lighting design. The objective was to re-think evidence-based lighting design approaches for residential, working/educational, and healthcare...
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Computationally-efficient design optimisation of antennas by accelerated gradient search with sensitivity and design change monitoring
PublikacjaElectromagnetic (EM) simulation tools are of primary importance in the design of contemporary antennas. The necessity of accurate performance evaluation of complex structures is a reason why the final tuning of antenna dimensions, aimed at improvement of electrical and field characteristics, needs to be based on EM analysis. Design automation is highly desirable and can be achieved by coupling EM solvers with numerical optimisation...
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Natalia Sokół dr inż.
OsobyBACKGROUND Master of Science in Light and Lighting (2008-2009/11) The UCL Bartlett School of Graduate Studies, Faculty of the Built Environment, London, UK, www.bartlett.ucl.ac.uk MA Degree in Interior Architecture (1999-2004), The Academy of Fine Arts, Poznan, Poland, www.uap.edu.pl MA Degree in Art Education (1997-2002), Academy of Fine Arts, Poznan, Poland, www.uap.edu.pl MAIN RESEARCH AREAS · ...
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Unraveling Luminescent Energy Transfer Pathways: Futuristic Approach of Miniature Shortwave Infrared Light-Emitting Diode Design
Dane BadawczePhosphor-converted shortwave infrared phosphor light-emitting diodes (pc-SWIR LEDs, 900–1700 nm) are promising next-generation portable light sources for spectroscopy, security, optical communication, and medical applications. A typical design strategy involves energy transfer from Cr3+ to Ni2+, and thus, energy transfer from Cr3+–Cr3+ pairs to Ni2+...
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Prediction of Overall In Vitro Microsomal Stability of Drug Candidates Based on Molecular Modeling and Support Vector Machines. Case Study of Novel Arylpiperazines Derivatives
PublikacjaOther than efficacy of interaction with the molecular target, metabolic stability is the primary factor responsible for the failure or success of a compound in the drug development pipeline. The ideal drug candidate should be stable enough to reach its therapeutic site of action. Despite many recent excellent achievements in the field of computational methods supporting drug metabolism studies, a well-recognized procedure to model...
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THE ARCHİTECTURE AND FASHİON DESİGN – An Examination of the Relationship between Fashion and Architecture Design in light of Technological Advancements
PublikacjaThe article focuses on the mutual relationship between two seemingly distant fields of art - architecture and fashion design. It describes a common basis for the process of creating art in the approach to both fashion and architecture. The following considerations, which are based on principles of composition, attempt to reach beyond just the form and analyze also context or perception. The article quotes famous creators and depicts...
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Application tool for IP QoS network design
PublikacjaDespite the fact that differentiated-service-aware network implementation has been a widely discussed topic for quite some time, network design still proofs nontrivial. Well developed software could put an end to network designer's problems. This chapter describes work, which has been aimed at creating a comprehensive network design tool, offering a fair range of functionality and high reliability. The presented tool is able to...
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Design and investigations of the ethanol microturbine
PublikacjaThe paper presents the results of the design analysis and experimental investigations of the microturbine set consisting of the microturbine with partial admission and permanent magnet generator. The microturbine was designed for operation with the vapour of ethanol as a working fluid. Microturbine unit was tested for different parameters of the working fluid and varying the electrical load. The examples and the comparison between...
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Microbial Drug Resistance
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Footbridges. Dynamic Design – Selected Problems
PublikacjaModern footbridges create challenge in esthetic and structural design. Breaking the proven canons is a recipe for architectural success. However esthetic form has to be also a functional pedestrian bridge. Therefore a good FEM modeling is a key element in engineering part of design. The paper presents selected problems related to the modeling of the dynamic construction of footbridges. Several basic dynamic problems concerning...
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Design of residential buildings in architecture education
PublikacjaThis article is based on an analysis of residential building designs made by students of the Faculty of Architecture at Gdańsk University of Technology (FA-GUT), Poland, and on the results of a survey conducted among these students. The purpose of the survey was to verify the broad, interdisciplinary knowledge of the students required in preparation for taking up design issues, as well as their ability to use this knowledge in...
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A Generative Approach to Hull Design for a Small Watercraft
PublikacjaIn the field of ocean engineering, the task of spatial hull modelling is one of the most complicated problems in ship design. This study presents a procedure applied as a generative approach to the design problems for the hull geometry of small vessels using elements of concurrent design with multi-criteria optimisation processes. Based upon widely available commercial software, an algorithm for the mathematical formulation of...
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Artificial Intelligence Aided Architectural Design
PublikacjaTools and methods used by architects always had an impact on the way building were designed. With the change in design methods and new approaches towards creation process, they became more than ever before crucial elements of the creation process. The automation of architects work has started with computational functions that were introduced to traditional computer-aided design tools. Nowadays architects tend to use specified tools...
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Development of a Peptide Derived from Platelet-Derived Growth Factor (PDGF-BB) into a Potential Drug Candidate for the Treatment of Wounds
PublikacjaObjective: This study evaluated the use of novel peptides derived from platelet-derived growth factor (PDGF-BB) as potential wound healing stimulants. One of the compounds (named PDGF2) was subjected for further research after cytotoxicity and proliferation assays on human skin cells. Further investigation included evaluation of: migration and chemotaxis of skin cells, immunological and allergic safety, the transcriptional analyses...
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Cancer stem cells in drug resistance and drug screening: can we exploit the cancer stem cell paradigm in search for new antitumor agents?
PublikacjaPraca przedstawia przegląd literatury dotyczącej hipotezy komórek pierwotnych nowotworu, w szczególności w ich oporności na istniejące terapie. Dyskutowane jest także zagadnienie możliwości wykorzystania wiedzy o tych komórkach do konstrukcji nowych testów do badań przesiewowych in vitro w celu poszukiwania nowych leków przeciwnowotworowych.
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Test Design Patterns for Embedded Systems,
PublikacjaTest suites for embedded systems are typically created from scratch using dif- ferent, often inadequate methods. In consequence, industry branches dealing with software-intensive embedded systems have to cope with quality problems, even though test processes are particularly time-consuming and costly. Based on an evolving model-based testing methodology we introduce test design patterns for simplifying and accelerating...
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Design optimisation of air-fed full pressurised suits
PublikacjaOpisano szczegóły złożoności zjawisk cieplno-przepływowych pomiędzy wewnętrzną powierzchnią kombinezonu ochronnego i zewnętrznego ubioru. Komplikacja polega na jednoczesnym rozważaniu wymiany masy i ciepła wraz z realistycznymi, trójwymiarowymi geometriami. Dodatkowo rozważany jest ludzki metabolizm. Zrozumienie tych zjawisk i umiejętnośćich symulacji jest konieczna w celu właściwych prac projektowych nad nowymi typami kombinezonów...