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Search results for: ANTI-INFLAMMATORY ACTIVITY
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Membrane Filtration-Assisted Enzymatic Hydrolysis Affects the Biological Activity of Potato Juice
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Photochemical properties and promising activity against staphylococci of sulfanyl porphyrazines with dendrimeric moieties
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Thymus serpyllum Essential Oil and Its Biological Activity as a Modern Food Preserver
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Synthesis of 5-arylidene-2-amino-4-azolones and evaluation of their anticancer activity
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Synthesis, biological activity and molecular modelling studies of tricyclic alkylimidazo-, pyrimido- and diazepinopurinediones
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The lipophilicity estimation of 5-arylidene derivatives of (2-thio)hydantoin with antimycobacterial activity
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Gender-Selective Interaction Between Aging, Blood Pressure, and Sympathetic Nerve Activity
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Detection of low- and high-frequency rhythms in the variability of skin sympathetic nerve activity
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Central Vagotonic Effects of Atropine Modulate Spectral Oscillations of Sympathetic Nerve Activity
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Relationship Between Muscle Sympathetic Nerve Activity and Diurnal Blood Pressure Profile
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Baroreflex Control of Sympathetic Nerve Activity and Heart Rate in Obstructive Sleep Apnea
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Interactive Effect of Heart Rate and Muscle Sympathetic Nerve Activity on Blood Pressure
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Residual Effects of Different Cropping Systems on Physicochemical Properties and the Activity of Phosphatases of Soil
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The time spent sitting does not always mean a low level of physical activity
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Interleukin 12 and indomethacin exert a synergistic, angiogenesis-dependent antitumor activity in mice
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Effect of UV radiation and chitosan coating on the adsorption-photocatalytic activity of TiO2 particles
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Effect of extraction method on the antioxidative activity of ground elder (Aegopodium podagraria L.)
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Lysozyme increases bactericidal activity of ceragenin CSA-13 against Bacillus subtilis
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Enhanced Suppressive Activity of Regulatory T Cells in the Microenvironment of Malignant Pleural Effusions
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Use of magnetic nanoparticles as a drug delivery system to improve chlorhexidine antimicrobial activity
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Lipidation of Temporin-1CEb Derivatives as a Tool for Activity Improvement, Pros and Cons of the Approach
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Comparison of antifungal activity of extracts from different Juglans regia cultivars and juglone
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Effect of biochar activation by different methods on toxicity of soil contaminated by industrial activity
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Hypsometric changes in urban areas resulting from multiple years of mining activity
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Institutional Settings and their Impact on the IPO Activity: An Exploratory Study Based on Qualitative Modelling
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Spectroscopic and Spectroelectrochemical Studies on Redox Properties of Zinc Sulfide and Their Consequences on Photocatalytic Activity
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Physical Activity vs. Redox Balance in the Brain: Brain Health, Aging and Diseases
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Vimentin immunoexpression and its prognostic activity in colon cancer among Caucasian patients
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<p>Analysis of toxicity and anticancer activity of micelles of sodium alginate-curcumin</p>
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Impact of paint matrix composition and thickness of paint layer on the activity of photocatalytic paints
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Cinnamon powder: an in vitro and in vivo evaluation of antifungal and plant growth promoting activity
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Photocatalytic activity of anatase powders for oxidation of methylene blue in water and diluted NO gas
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Effect of self-assembly on antimicrobial activity of double-chain short cationic lipopeptides
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Synthesis of Usnic Acid Derivatives and Evaluation of Their Antiproliferative Activity against Cancer Cells
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Process control strategy deployment with part measuring activity in a flexible machining cell
PublicationRozwinięto zintegrowany model planowania i sterowania przebiegu procesu w rzeczywistym, zrobotyzowanym elastycznym gnieździe obróbki (EGO) ze współrzędnościową maszyną pomiarową, realizującą funkcje pomiarowo-kontrolne wytwarzanych przedmiotów. Analizowano współzależności wybranych heurystycznych planów kontroli przedmiotów oraz strategii szeregowania operacji procesów technologicznych, z zastosowaniem programowalnych modeli symulacyjnych...
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Structure activity relationship for a series of peptidomimetic antimicrobial prodrugs containing glutamine analogues.
PublicationZbadano specyficzność transporterów Dpp i Opp w stosunku do peptydów zawierających FMDP. Przy pomocy modelowania cząsteczkowego zaproponowano najbardziej prawdopodobne struktury konformerów peptydów i skorelowano je z aktywnością przeciwbakteryjną oraz specyficznością transporterów peptydowych.
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Molecular modelling of membrane activity of amphotericin B, a polyene macrolide antifungal antibiotic
PublicationPraca dotyczy różnego typu modelowań molekularnych cząsteczki przeciwgrzybowego antybiotyku (amfoterycyny B). Praca przeglądowa obejmuje opis badań nad właściwościami molekularnymi samej cząsteczki antybiotyku, jej oddziaływań z powierzchnią błony oraz struktur kanałowych jakie tworzą cząsteczki amfoterycyny wewnątrz błony lipidowej.
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A Redundant Role of Human Thyroid Peroxidase Propeptide for Cellular, Enzymatic, and Immunological Activity
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The propeptide of human thyroid peroxidase is not required for its cellular, enzymatic or immunological activity
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Effect of Cobalt Addition on the Activity of Nanocrystalline Iron Catalysts in the Cracking of Methane Reaction
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Influence of Magnesium Oxide on the Structure and Catalytic Activity of the Wustite Catalyst for Ammonia Synthesis
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Synthesis and Anticancer Activity of Mitotic-Specific 3,4-Dihydropyridine-2(1H)-thiones
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Antinociceptive and Cytotoxic Activity of Opioid Peptides with Hydrazone and Hydrazide Moieties at the C-Terminus
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The Chemometric Evaluation of Antitumor Activity of Novel Benzensulfonamide Derivatives Based on their Physiochemical Properties
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Biological Activity of Compounds Exhibiting Local Anesthetics's Properties Evaluated by QSAR Approach
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Variation in Total Polyphenolics Contents of Aerial Parts of Potentilla Species and Their Anticariogenic Activity
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Activity evaluation of some psychoactive drugs with the application of QSAR/QSPR modeling methods
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N-acylpeptides with glucosamine-6-phosphate synthase inhibitors - synthesisand antifungal activity
PublicationOpracowano syntezę kilku peptydów (di i tripeptydów) zawierających inhibitory syntazy glukozamino-6-fosforanu oraz przeprowadzono je w N-acylopochodne (acetylowe, heksanoilowe, dekanoilowe) oraz zbadano ich aktywność przeciwgrzybową w stosunku do szczepów Candida albicans z opornością wielolekową. Stwierdzono, że N-acylopeptydy wykazują aktywność przeciwgrzybową oraz określono wartości MIC.
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Facilitated diffusion of glucosamine-6-phosphate synthase inhibitors enhances their antifungal activity
PublicationKwas N-3(4-metoksyfumaroilo)-L-2,3-diaminopropanowy (FMDP) i 2-amino-2-deo-ksy-D-glucitolo-6-fosforan (ADGP) są silnymi inhibitorami syntazy glukoza-mino-6-fosforanu, istotnego enzymu grzybowego, jednak ich aktywność przeciwgrzybowa jest słaba, ze względu na powolną penetrację tych związków przez błonę cytoplazmatyczną. W tej pracy badaliśmy możliwość poprawy działania przeciwgrzybowego ADGP i FMDP poprzez zwiększenie ich własności...
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Encapsulation of Cs3Bi2Br9 perovskite photocatalyst with polythiophene for prolonged activity in oxidizing and humid environment
PublicationDespite their growing popularity in modern technology, halide perovskites suffer from susceptibility to oxidation, limiting their applications. Our aim was to enhance Cs3Bi2Br9 perovskite's performance in humid environments through polythiophene encapsulation. This extended its lifespan while preserving photocatalytic abilities, as demonstrated in toluene decomposition experiments. We confirmed the stability of Cs3Bi2Br9 encapsulated...