Filters
total: 2192
displaying 1000 best results Help
Search results for: INVERSE AGONIST
-
Conformation-activity relationships of cyclo-constrained μ/5 opioid agonists derived from the N-terminal tetrapeptide segment of dermorphin/deltorphin
Publication -
Metrological analysis of an computerized system of protection against electric shock in circuits with variable speed drives
PublicationDrive systems, that can be operated at variable speed, are equipped with power electronics converters. This causes distortion of the earth current, and consequently the need to take into account the use of proper protective devices in relation to earth current harmonics. This paper presents a system for protection against electric shock in circuits with power electronics converters and metrological analysis indicating the requirements...
-
Protective Effect of Black Tea Against Ethanol-Induced Oxidative Modifications of Liver Proteins and Lipids
Publication -
Synergistic action of extracts from carnivorous plants and synthetic peptides against plant pathoghenic bacteria
Publicationw pracy przedstawiono rezultaty badań nad sprawdzeniem aktywności przeciwbakteryjnej ekstraktów z roślin Drosera capensis i Dionaea muscipula w połączeniu z dwoma syntetycznymi peptydami: CAMEL oraz pexiganan. Najwyższą aktywnością przeciwbakteryjną odznaczał się chloroformowy ekstrakt z D. muscipula z peptydem CAMEL.
-
Workforce mobility against the background of labour market duality theory – the example of selected OECD countries
PublicationThe paper aims to present an empirical study of labour market segmentation (LMS) hypothesis. According to the dual labour market theory jobs can be divided into two groups: primary and secondary jobs, with enter barriers into the first one. The primary jobs are usually described with relative high wages, whereas secondary jobs provide lower level of wages. In this paper we first examine the main sectors (according to the ISIC rev....
-
The Level of FGF 21 as a New Risk Factor for the Occurrence of Cardiometabolic Disorders amongst the Psoriatic Patients
Publication -
Renoprotective and Cardioprotective Potential of Moricandia sinaica (Boiss.) against Carbon Tetrachloride-Induced Toxicity in Rats
Publication -
The effect of PWM frequency on the effectiveness of protection against electric shock using residual current devices
PublicationW artykule przedstawiono analizę widmową odkształconego prądu ziemnozwarciowego z obwodu silnika o regulowanej prędkości obrotowej za pomocą przemiennika częstotliwości. Oceniono skuteczność ochrony przeciwporażeniowej wykorzystującej wyłączniki różnicowoprądowe przy różnych wartościach częstotliwości PWM przemiennika. Przedstawiono charakterystykę działania proponowanego wyłącznika różnicowoprądowego.
-
The effect of PWM frequency on the effectiveness of protection against electric shock using residual current devices
PublicationW referacie przedstawiono analizę widmową odkształconego prądu ziemnozwarciowego z obwodu silnika o regulowanej prędkości obrotowej za pomocą przemiennika częstotliwości. Oszacowano wpływ tego odkształcenia na próg fibrylacji serca. Analizowano skuteczność ochrony przeciwporażeniowej wykorzystującej wyłączniki różnicowoprądowe przy różnych wartościach częstotliwości PWM przemiennika. Przedstawiono charakterystykę działania zaproponowanego...
-
The Activity of Isoquinoline Alkaloids and Extracts from Chelidonium majus against Pathogenic Bacteria and Candida sp.
Publication -
Response to Claudio Schuftan on “Three decades of fighting against hunger in Africa: Progress, challenges and opportunities”
Publication -
Phytochemical Profiling and Larval Control of Erythrina variegata Methanol Fraction against Malarial and Filarial Vector
Publication -
Evaluation of antimicrobial activities of powdered cuttlebone against Klebsiella oxytoca, Staphylococcus aureus, and Aspergillus flavus
PublicationBackground: The presence of medicines in the environment is considered as a serious threat to the human health. The entrance of these substances into the water sources causes soil pollution, which eventually leads to the environmental pollution and it creates some problems for the public health. Also, increasing antibiotic resistant bacteria has attracted the attention of researchers to the use of natural resources such as marine...
-
THE PROTECTIVE MEASURES AGAINST SARS-COV-2 INFECTION IN THE SEAFOOD COMPANY FROM THE PERSPECTIVE OF THE EMPLOYEES
PublicationPurpose: To identify and discuss the protective measures implemented to prevent SARS-CoV-2 infection among employees. Design/methodology/approach: The four-stage course of research. Case study and structured interviews with all employees, directly and indirectly, involved in food processing. Research questions: (R1) What measures have been taken to prevent the risk of infection among employees? (R2) What activities and responsibilities...
-
Testing the positioning accuracy of GNSS solutions during the tramway track mobile satellite measurements in diverse urban signal reception conditions
Publication -
Evaluation of reverse osmosis for improving quality of water utilized in hemodialysis devices (case study: Kerman University of Medical Sciences' hospitals)
Publication -
Evaluation of reverse osmosis for improving quality of water utilized in hemodialysis devices (case study: Kerman University of Medical Sciences' hospitals).
Publication -
Separation of Monovinyl and Divinyl Protochlorophyllides Using C30 Reverse Phase High Performance Liquid Chromatography Column: Analytical and Preparative Applications
Publication -
Diverse behavioral, monoaminergic and Fos protein responses to opioids in Warsaw high-alcohol preferring and Warsaw low-alcohol preferring rats
Publication -
Testing the Positioning Accuracy of GNSS Solutions during the Tramway Track Mobile Satellite Measurements in Diverse Urban Signal Reception Conditions
PublicationMobile Global Navigation Satellite System (GNSS) measurements carried out on the railway consist of using satellite navigation systems to determine the track geometry of a moving railway vehicle on a given route. Their purposes include diagnostics, stocktaking, and design work in railways. The greatest advantage of this method is the ability to perform measurements in a unified and coherent spatial reference system, which...
-
Cytotoxicity of chitosan hydrogels aginst L929 cells
Open Research DataThis study presents absorbance values of formazan product (converted from MTT) which corresponds to the cytotoxicity of chitosan compounds (dissolved in carbonic acid, dissolved in carbonic acid endotoxin free, and dissolved in hydroxyacetic acid) aginst adult mouse fibroblast L929 cells. The experiments were carried out according to the ISO 10993-5:2009(E)...
-
Corrigendum to “Impact of intense rains and flooding on mercury riverine input to the coastal zone” [Mar. Pollut. Bull. 127 (2018) 593–602]
Publication -
Diverse Expression of Selected SMN Complex Proteins in Humans with Sporadic Amyotrophic Lateral Sclerosis and in a Transgenic Rat Model of Familial Form of the Disease
Publication -
Anticancer potential of acetone extracts from selected Potentilla species against human colorectal cancer cells
Publication -
In Vitro Anticancer Potential of Jasione montana and Its Main Components against Human Amelanotic Melanoma Cells
Publication -
Phytochemical analysis of Brasolia, Elleanthus, and Sobralia. Three genera of orchids with antibacterial potential against Staphylococcus aureus
Publication -
Bio-fabrication of Zinc Oxide nanoparticles to rescue Mung Bean against Cercospora leaf spot disease
Publication -
Bactericidal effect of photodynamic inactivation against methicillin-resistant and methicillin-susceptible Staphylococcus aureus is strain-dependent
Publication -
Targeted Nano-Drug Delivery of Colchicine against Colon Cancer Cells by Means of Mesoporous Silica Nanoparticles
Publication -
Chocolate desserts with ricotta hydrolysates: In vitro study of inhibitory activity against angiotensin‐converting enzyme and cholinesterase
Publication -
The Antimicrobial Activity of Omiganan Alone and In Combination against Candida Isolated from Vulvovaginal Candidiasis and Bloodstream Infections
Publication -
In Vitro Evaluation of Polihexanide, Octenidine and NaClO/HClO-Based Antiseptics against Biofilm Formed by Wound Pathogens
Publication -
The ability of selected plant essential oils to enhance the action of recommended antibiotics against pathogenic wound bacteria
Publication -
Panax quinquefolium hairy root extracts and their effect in connections with antibiotics against pathogenic bacteria – preliminary study
Publication -
Comparison of usefulness of three emergent macrophytes for surface waterprotection against pollution and eutrophication:case study, Bielikowo,Poland.
Publication.
-
Expert opinion on the effectiveness of protection against electric shock in case of fault in an installation for electric vehicles charging
PublicationThe opinion concerns the use of residual current devices for protection against electric shock by automatic disconnection of supply in a Norwegian installation intended for charging of electric vehicles.
-
Collective action against same-sex marriages_online research in Poland
Open Research DataThe study was conducted in the context of people opposing the equality of sexual minorities. At the beginning of the survey, each respondent was asked to mark their support for the equality of rights of heterosexual and homosexual persons, on a scale from -3 (definitely not) to 3 (definitely yes). The subsequent questions of the survey were formulated...
-
Inhibiting activity of HIV-1: protease, reverse transcriptase and integrase all together by novel compounds using computational approaches (flexible and rigid docking)
PublicationAcquired immunodeficiency syndrome (AIDS), caused by human immunodeficiency virus type 1 (HIV-1) infection, is one of the most challenging diseases in recent decades. Nevertheless the shortcomings of chemical drugs such as toxicity, lack of curative effects, the search for more potent anti-HIV agents have been focused in our study. In current study, novel scaffold was designed having a benzyl and imidazole in it which are very...
-
Simultaneous determination of hydrophobicity and dissociation constant for a large set of compounds by gradient reverse phase high performance liquid chromatography–mass spectrometry technique
Publication -
The Leaderless Bacteriocin Enterocin K1 Is Highly Potent against Enterococcus faecium: A Study on Structure, Target Spectrum and Receptor
Publication -
Systems of General Grants for Local Governments in Selected EU Countries Against the Background of the General Theory of Fiscal Policy
PublicationFiscal policy, including its expenditure aspect, is often discussed and analysed from a variety of angles in the literature on public finances, undoubtedly due to the major importance of this topic. However, not all areas of the expenditure part of fiscal policy have been subjected to in-depth analysis. One of the less discussed tools of fiscal policy consists of general purpose transfers, which are a certain type of expenditure...
-
Effectiveness of E-Beam Radiation against Saccharomyces cerevisiae, Brettanomyces bruxellensis, and Wild Yeast and Their Influence on Wine Quality
Publication -
Robust effectiveness behavior of synthesized cobalt doped Prussian blue graphene oxide ferrite against EMI shielding
Publication -
Chemical Composition and Antimicrobial Activity of Selected Essential Oils against Staphylococcus spp. Isolated from Human Semen
Publication -
S-seco-porphyrazine as a new member of the seco-porphyrazine family – Synthesis, characterization and photocytotoxicity against cancer cells
Publication -
Optical properties of a series of pyrrolyl-substituted porphyrazines and their photoinactivation potential against Enterococcus faecalis after incorporation into liposomes
Publication -
Novel 2019 coronavirus structure, mechanism of action, antiviral drug promises and rule out against its treatment
Publication -
Pd-catalysed general access to 7-membered N/O-heterocyclic compounds as potential agents against inflammation
Publication -
Social and economic aspects of the transformation of pomorskie region against the background of changes in the polish economy in the years 1990-2010
PublicationPrzemiany społeczno-gospodarcze, które nastąpiły w Polsce w latach 1990-2010 i ich tempo należy oceniać w świetle totalnego, permanentnego kryzysu, który nasilił się w latach osiemdziesiątych XX w. W tym aspekcie 20 lat realizacji reform w Polsce przyniosło zasadniczy postęp zarówno w odniesieniu do wzrostu społeczno-gospodarczego, jak i umiędzynarodowieniu polskiej gospodarki. Do niekorzystnych zjawisk tego okresu zaliczyć należy...
-
Chemical composition and antifungal activity of Chelidonium majus extracts – antagonistic action of chelerythrine and sanguinarine against Botrytis cinerea
Publication