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- Publikacje 1407 wyników po odfiltrowaniu
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Wyniki wyszukiwania dla: ACTIVE PHARMACEUTICAL INGREDIENTS
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Probing the Magnetic Anisotropy of Co(II) Complexes Featuring Redox-Active Ligands
PublikacjaCoordination complexes that possess large magnetic anisotropy (otherwise known as zero-field splitting, ZFS) have possible applications in the field of magnetic materials, including single molecule magnets (SMMs). Previous studies have explored the role of coordination number and geometry in controlling the magnetic anisotropy and SMM behavior of high-spin (S = 3/2) Co(II) complexes. Building upon these efforts, the present work...
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Application of surface active amino acid ionic liquids as phase-transfer catalyst
PublikacjaFive structurally related morpholinium derived ionic liquids containing N-acetyl-glycinate anion were synthesized and their thermal stability, surface properties and activity as phase transfer catalysts investigated. The thermal properties were studied by differential scanning calorimetry, while the adsorption at the air/water interface and micellization behavior was analyzed by surface tension measurements, conductometry and isothermal...
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Voriconazole-Based Salts Are Active against Multidrug-Resistant Human Pathogenic Yeasts
PublikacjaVoriconazole (VOR) hydrochloride is unequivocally converted into VOR lactates and valinates upon reaction with silver salts of organic acids. This study found that the anticandidal in vitro activity of these compounds was comparable or slightly better than that of VOR. The Candida albicans clinical isolate overexpressing CaCDR1/CaCDR2 genes, highly resistant to VOR, was apparently more susceptible to VOR salts. On the other hand,...
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Quantitative active dynamic thermal Ir-Imaging and thermal tomography in medical diagnostics
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Solid electrolyte gas sensors based on cyclic voltammetry with one active electrode
PublikacjaW artykule przedstawiono wyniki badań elektrokatalitycznego czujnika gazów toksycznych z jedną elektrodą aktywną.
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Generation of chirality in 4,4'-azopyridine by co-crystallization with optically active dicarboxylic acids
PublikacjaOtrzymano kokryształy anti-4,4'-azopirydyny z optycznie czynnymi kwasai: 9,10-dihydro-9,10-etanoantraceno-11,12-dikarboksylowym i trans-1,2-cykloheksnodikarboksylowym. Następnie pomierzono dichroizm kołowy otrzymanych kryształów. Dodatni znak efektu Cottona, odpowiadający niskoenergetycznemu wzbudzeniu elektronowemu n-pi*, został skorelowany z M helikalnością skręconego chromoforu Ar-N=N. Absolutna konfiguracja skręconej cząsteczki...
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Smart MV/LV distribution transformer for Smart Grid with active prosumer participation
PublikacjaWraz z rozwojem sieci dystrybucyjnych i ich stopniowym przekształcaniem w inteligentne sieci typu Smart Grid będzie rosłoznaczenie i udział sterowanych układów przekształtnikowych mocy stosowanych jako interfejsy pomiędzy źródłami energii a sieciąoraz pomiędzy siecią a odbiorcami. W artykule rozwinięto koncepcję wymiany konwencjonalnych transformatorów dystrybucyjnych50 Hz na inteligentne transformatory dystrybucyjne. Zaproponowano...
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Improving the accuracy of bearing in active sonar with cylindrical array using spectrum estimation.
PublikacjaThe articles presents a method for improving the accuracy of bearing in multibeam sonar with a cylindrical array. Based on a known spatial spectrum estimation technique, the method has been successfully used in linear array systems. Its accuracy of bearing is satisfactory and ensures a relatively low computational effort. The article discusses certain simplifications and assumptions to adapt the spatial spectrum estimation technique...
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Quantitative Active Dynamic Thermal IR-Imaging and Thermal Tomography in Medical Diagnostics
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Continuous-Time Active-RC Filter Model for Computer-Aided Design and Optimization
PublikacjaW pracy przedstawiono ogólny model filtru aktywnego RC opartego na wzmacniaczach odwracajacych faze. Model analizowany jest przy użyciu równań macierzowych. Podano jawną formułę określającą funkcję przenoszenia filtru w ogólnym przypadku. Przedstawiono rozszerzenia modelu pozwalające uwzgledniać nieidealność wzmacniaczy operacyjnych, w tym skończone wzmocnienie i pasmo przenoszenia oraz niezerową rezystancję wyjściową. Wyprowadzono...
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Highly Active TiO2 Microspheres Formation in the Presence of Ethylammonium Nitrate Ionic Liquid
PublikacjaSpherical microparticles of TiO2 were synthesized by the ionic liquid-assisted solvothermal method at different reaction times (3, 6, 12, and 24 h). The properties of the prepared photocatalysts were investigated by means of UV-VIS diffuse-reflectance spectroscopy (DRS), Brunauer–Emmett–Teller (BET) surface area measurements, scanning electron microscopy (SEM), X-ray diffraction analysis (XRD), and X-ray photoelectron spectroscopy...
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Structure of solvation water around the active and inactive regions of a type III antifreeze protein and its mutants of lowered activity
PublikacjaWater molecules from the solvation shell of the ice-binding surface are considered important for the antifreeze proteins to perform their function properly. Herein, we discuss the problem whether the extent of changes of the mean properties of solvation water can be connected with the antifreeze activity of the protein. To this aim, the structure of solvation water of a type III antifreeze protein from Macrozoarces americanus (eel...
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A Novel Electrochemical Sensor Based on Graphene Oxide Nanosheets and Ionic Liquid Binder for Differential Pulse Voltammetric Determination of Droxidopa in Pharmaceutical and Urine Samples
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Artemisia abrotanum L. (Southern Wormwood)—History, Current Knowledge on the Chemistry, Biological Activity, Traditional Use and Possible New Pharmaceutical and Cosmetological Applications
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A novel cold-active β-D-galactosidase with transglycosylation activity from the Antarctic Arthrobacter sp. 32cB - gene cloning, purification and characterization
PublikacjaA gene encoding a novel β-D-galactosidase from the psychrotolerant Antarctic bacterium Arthrobacter sp. 32cB was isolated, cloned and expressed in Escherichia coli. The active form of recombinant β-D-galactosidase consists of two subunits with a combined molecular weight of approximately 257 kDa. The enzyme's maximum activity towards o-nitrophenyl-β-D-galactopyranoside was determined as occurring at 28 °C and pH 8.0. However, it...
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Fabrication of Gold and Silver Nanoparticles Supported on Zinc Imidazolate Metal–Organic Frameworks as Active Catalysts for Hydrogen Release from Ammonia Borane
PublikacjaWell-dispersed Au and Ag nanoparticles (NPs) have been immobilized on a zinc imidazolate metal−organic framework, Zn(mim), using the “one-pot” method and tested as catalysts in ammonia borane hydrolysis. The AuNPs@Zn(mim) and AgNPs@Zn(mim) materials were characterized by FTIR, XRD, ICP-OES, TGA, BET, SEM, and TEM. The AgNPs@Zn(mim) catalyst showed a high yield (98.5%) and high hydrogen generation rate (3352.71 mL min−1 gAg−1) in...
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Comparative analysis of three‐phase dual active bridge converter with different transformer topology and modern universal control for DC microgrids
PublikacjaThe presented work discusses issues related to the use of modern multiphase topologies of Dual Active Bridge (DAB)-type converters. Converters of this type are widely used in most DC microgrid applications. The introduction emphasizes a comparative analysis between single-phase and multi-phase DAB topologies within high-power DC microgrids, delving into their respective advantages, drawbacks, design procedures, and considerations...
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Determination of pharmaceutical residues in drinking water in Poland using a new SPE-GC-MS(SIM) method based on Speedisk extraction disks and DIMETRIS derivatization
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Determination of mefenamic acid in urine and pharmaceutical samples by HPLC after pipette-tip solid phase microextraction using zinc sulfide modified carbon nanotubes
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Ecotoxicological equilibria of triclosan inMicrotox, XenoScreen YES/YAS, Caco2, HEPG2 and liposomal systems are affected by the occurrence of other pharmaceutical and personal care emerging contaminants
PublikacjaContaminants of emerging concernmay be considered as any chemicals or factorswhose unintended continuous release and persistence in the environmentmay lead to any observable undesirable response of living beings. Still not much is known on reciprocal toxicological impact of given chemicals when present in binary or more complex mixtures. In thiswork, an attemptwas thus undertaken to study the impact of butylparaben,methylparaben and...
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Burn depths evaluation based on active dynamic IR thermal imaging - A preliminary study
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Higuchi fractal dimension analysis of surface EMG signals and determination of active electrode positions
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Effect of Active Mining Impact On Properties with Engineering Structures – Forecast and Final Result Discrepancies
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High power, zero ripples active filtering system with power modules operating in parallel
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A hybrid, coupled reactors based 18-pulse diode rectifier with active power filter
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From Democratic (Citizenship) Education to Participative Democracy? Youth’s Difficult Way to Active Citizenship
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ALD thin ZnO layer as an active medium in a fiber-optic Fabry–Perot interferometer
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Selective monoprotection of 1,4,7,10-tetraazacyclododecane via direct reactions with 4-nitrophenyl active esters
Publikacja1,4,7,10-tetraazacyklododekan jest cykliczną tetraaminą. Z chemicznego punktu widzenia wszystkie atomy azotu posiadają takie same właściwości fizykochemiczne. Jedyną różnicę stanowią ich właściwości kwasowo-zasadowe. Cyklen posiada dwa atomy azotu o obniżonej zasadowości. Właściwość ta z powodzeniem wykorzystywana jest w reakcjach jednoczesnej selektywnej substytucji dwóch atomów w pozycji 1 i 7. W przypadku bezpośredniej reakcji...
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Post-Activation Performance Enhancement: Save Time With Active Intra-Complex Recovery Intervals
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A rapid, selective, and ultrasensitive voltammetric and gravimetric protocol for MMP-1 active form detection
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Treatment of high-quality groundwater by means of one-stage filtration on active filtration beds
PublikacjaPrzeprowadzone badania pilotowe uzdatniania wody podziemnej wysokiej jakości, wykazały, że wody o niewielkich stężeniach żelaza (< 0,6 mgl) i manganu (<0,1 mg/l) można uzdatniać stosując napowietrznie i jednostopniową filtrację, w układzie zamkniętym, przez aktywne złoża filtracyjne. Wszystkie przebadane złoża (jednowarstwowe z piasku kwarcowego; dwuwarstwowe z piasku kwarcowego i piroluzytu oraz trzywarstwowe z antracytu, piasku...
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Edu Inspiracje WZiE: Active Learning, czyli o mocy aktywnego przetwarzania informacji
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The use of a static electrical energy meter as a transducer of active power to a pulse frequency signal
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Differentiating between Inactive and Active States of Rhodopsin by Atomic Force Microscopy in Native Membranes
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New Insights into Dietary Supplements Used in Sport: Active Substances, Pharmacological and Side Effects
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Methods of decreasing the lasing thresholds of optical resonators with periodically structured active nano wires
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A new approach to active noise and vibration control - [Part I: the known frequency case]
PublikacjaThis paper presents a new approach to rejection of complex-valued sinusoidal disturbances acting at the output of a discrete-time stable linear plant with unknown dynamics. It is assumed that the frequency of the sinusoidal disturbance is known, and that the output signal is contaminated with wideband measurement noise. The disturbance rejection control rule is first derived and analyzed for a nominal plant model, different from...
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A new approach to active noise and vibration control - [Part II: unknown frequency case]
PublikacjaThis paper presents a new approach to rejection of complex-valued sinusoidal disturbances acting at the output of a discrete-time stable linear plant with unknown and possibly timevarying dynamics. It is assumed that both the instantaneous frequency of the sinusoidal disturbance and its amplitude may be slowly varying with time and that the output signal is contaminated with wideband measurement noise. It is not assumed that a...
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ALD thin ZnO layer as an active medium in a fiber-optic Fabry-Perot interferometer
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Influence of Protonation State on the Excited State Dynamics of a Photobiologically Active Ru(II) Dyad
PublikacjaThe influence of ligand protonation on the photophysics of a ruthenium (Ru) dyad bearing the 2-(1-pyrenyl)-1H-imidazo[4,5-f][1,10]-phenanthroline (ippy) ligand was investigated by time-resolved transient absorption spectroscopy. It was found that changes in the protonation state of the imidazole group led to changes in the electronic configuration of the lowest lying excited state. Formation of the fully deprotonated imidazole...
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Active Linear Tunable Resistance Element and Application to Feedforward Linearization of CMOS Transconductance Amplifier
PublikacjaW pracy przedstawiono koncepcję układową przestrajalnego rezystora liniowego MOS wykorzystującego tranzystory pracujące w zakresie triodowym. Opracowana struktura, jak wykazały symulacje komputerowe, charakteryzuje się dobrymi właściwościami zarówno jeżeli chodzi o zakres przestrajania jak i liniowość charakterystyk przejściowych. Pozwoliło to efektywnie wykorzystać prezentowany element do linearyzacji operacyjnego wzmacniacza...
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The effect of UV-C irradiation on lipids and selected biologically active compounds in human milk
PublikacjaThe effect of UV-C irradiation of human milk on lipid oxidation, content of antioxidants (vitamin C and catalase, CAT) and bactericidal compounds (lysozyme), as well as the total antioxidant capacity (TAC), of the breast milk was investigated. In parallel, the extent of inactivation of some bacteria was also determined. UV-C at doses from 85 to 740 J L−1 caused total inactivation of Escherichia coli and Staphylococcus aureus, but...
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Comparative analysis of seismic response reduction in multi-storey buildings equipped with base isolation and passive/active friction-tuned mass dampers
PublikacjaThis study presents an innovative approach to mitigating seismic responses in multi-storey buildings equipped with a base-isolation (BI) system and passive friction-tuned mass dampers (PFTMDs). The key innovation lies in the combined use of a BI system and a PFTMD system, as well as the activation of this mechanical system by controllers. Additionally, the research design optimizes the parameters of these devices specifically for...
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Jundishapur Journal of Natural Pharmaceutical Products
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International Journal of Pharmaceutical Sciences and Research
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World Journal of Pharmacy and Pharmaceutical Sciences
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Journal of Advanced Pharmaceutical Technology & Research
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International Journal of Pharmaceutical and Phytopharmacological Research
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International Journal of Pharmaceutical and Healthcare Marketing
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International Journal of Innovations in Pharmaceutical Sciences
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