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Search results for: combretastatyna a-4
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Fluorescent analogs of trypsin inhibitor SFTI-1 isolated from sunflower seeds-synthesis and applications
PublicationThis article describes the synthesis and enzymatic study of newly synthesized analogs of trypsin inhibitors SFTI-1 that were fluorescent labeled on their N-terminal amino groups. Two fluorescent derivatives of benzoxazole (3-[2-(4-diphenylaminophenyl) benzoxazol-5-yl]-L-alanine[(4NPh(2)) Ph] Box-Ala and 3-[2-(2', 4', 5'-trimethoxyphenyl) benzoxazol-5-yl]-l-alanine-[2,4,5-(OMe)3Ph] Box-Ala) were used as efficient fluorescent labels....
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The complexity of minimum-length path decompositions
PublicationWe consider a bi-criteria generalization of the pathwidth problem, where, for given integers k, l and a graph G, we ask whether there exists a path decomposition P of G such that the width of P is at most k and the number of bags in P, i.e., the length of P, is at most l. We provide a complete complexity classification of the problem in terms of k and l for general graphs. Contrary to the original pathwidth problem, which is fixed-parameter...
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The influence of the type of halogen substituent and its position on the molecular conformation, intermolecular interactions and crystal packing for a series of 1-benzoyl-3-(halogenophenyl)thioureas
PublicationBy the reaction of benzoyl chloride, potassium isothiocyanate and the appropriate halogenoaniline, i.e. 2/3/4-(bromo/iodo)aniline, we have obtained five new 1-benzoyl-3-(halogenophenyl)thioureas, namely, 1-benzoyl-3-(2-bromophenyl)- thiourea and 1-benzoyl-3-(3-bromophenyl)thiourea, C14H11BrN2OS, and 1-benzoyl-3-(2-iodophenyl)thiourea, 1-benzoyl-3-(3-iodophenyl)thiourea and 1-benzoyl-3-(4-iodophenyl)thiourea, C14H11IN2OS. Structural...
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Submicron inorganic particles as an additional filler in hybrid epoxy matrix composites reinforced with glass fibres
PublicationIn this study, the effect of selected submicron metal oxide (zinc oxide, titanium oxide) or non-metal oxide (silicon dioxide) particles on mechanical and thermo-mechanical properties of epoxy/glass composites was investigated. The applied epoxy resin was a diglycidyl ether of bisphenol-A cured with triethylenetetramine. As a reinforcement twill weave E-glass fabric was used. Hybrid composites (contained particulate and fibrous...
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Distinct hippocampal-prefrontal neural assemblies coordinate memory encoding, maintenance, and recall
PublicationShort-term memory enables incorporation of recent experience into subsequent decision-making. This processing recruits both the prefrontal cortex and hippocampus, where neurons encode task cues, rules, and outcomes. However, precisely which information is carried when, and by which neurons, remains unclear. Using population decoding of activity in rat medial prefrontal cortex (mPFC) and dorsal hippocampal CA1, we confirm that mPFC...
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No-Wait & No-Idle Open Shop Minimum Makespan Scheduling with Bioperational Jobs
PublicationIn the open shop scheduling with bioperational jobs each job consists of two unit operations with a delay between the end of the first operation and the beginning of the second one. No-wait requirement enforces that the delay between operations is equal to 0. No-idle means that there is no idle time on any machine. We model this problem by the interval incidentor (1, 1)-coloring (IIR(1, 1)-coloring) of a graph with the minimum...
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Acid-catalysed synthesis of oxathiolone fused chalkones. Comparison of their activity toward various microrganisms and human cancer lines
PublicationOtrzymano podstawione pochodne oksationolowych sprzężonych chalkonów w wyniku kondensacji 4-acetylo-5-metoksy-2-0ksobenz[1,3]oksatiolu z aldehydem benzoesowym w środowisku kwaśnym. Badano właściwości biologiczne otrzymanych związków. Trzy z otrzymanych pochodnych wykazały umiarkowaną aktywność wobec komórek HeLa, dwa były aktywne wobec Micrococcus luteus i Staphylococcus aureus, a jeden wobec Mycobacterium tuberculosis.
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Systemy Inmarsat dla potrzeb radiokomunikacji morskiej - ewolucja technologii i usług
PublicationW pracy przedstawiono ewolucję organizacyjną i technologiczną systemów Inmarsat w obszarze satelitarnej radiokomunikacji morskiej. Zaprezentowano najnowsze satelity Inmarsat-4 w kontekście już istniejącej konstelacji satelitów Inmarsat oraz systemy i usługi realizowane w sieciach Inmarsat w oparciu o te satelity. Przedstawiono również najnowsze trendy rozwojowe w satelitarnej radiokomunikacji morskiej kreowane przez Inmarsat.
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Systemy Inmarsat dla potrzeb radiokomunikacji morskiej - ewolucja technologii i usług
PublicationW pracy przedstawiono ewolucję organizacyjną i technologiczną systemów Inmarsat w obszarze satelitarnej radiokomunikacji morskiej. Zaprezentowano najnowsze satelity Inmarsat-4 w kontekście już istniejącej konstelacji satelitów Inmarsat oraz systemy i usługi realizowane w sieciach Inmarsat w oparciu o te satelity. Przedstawiono również najnowsze trendy rozwojowe w satelitarnej radiokomunikacji morskiej kreowane przez Inmarsat.
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Application of PCA and time series analysis in studies of precipitation in Tricity (Poland).
PublicationPrzedstawiono wyniki monitoringu zanieczyszczenia atmosfery Trójmiasta. Próbki wody opadowej pobierano w cyklach miesięcznych przez 4 lata (1998-2001)w 10 punktach. Wyniki poddano statystycznej i chemometrycznej analizie (szeregi czasowe, analiza wariancji, analiza głównych składowych). Wykazano wpływ lokalizacji punktów monitoringowych i bliskości Morza Bałtyckiego na zawartość jonów nieorganicznych w analizowanych próbkach.
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Interval incidence coloring of subcubic graphs
PublicationIn this paper we study the problem of interval incidence coloring of subcubic graphs. In [14] the authors proved that the interval incidence 4-coloring problem is polynomially solvable and the interval incidence 5-coloring problem is N P-complete, and they asked if χii(G) ≤ 2∆(G) holds for an arbitrary graph G. In this paper, we prove that an interval incidence 6-coloring always exists for any subcubic graph G with ∆(G) = 3.
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Voltage Source Power Line Conditioner for Applications in Local Supply Systems
PublicationThe paper presents the basic principles of operation of voltage source power line conditioners (VSPLC) as well as their energy and filtration properties. A 4-level cascade based Voltage Source Converter (VSC) is used as a voltage source. The advantages of this topology is relatively simple construction and simple way of balancing DC link voltages. Results of the theoretical and experimental investigations confirm good energetic...
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Quaternion Encryption Method for Image and Video Transmission
PublicationQuaternions are hyper-complex numbers of rank 4. They are often applied to mechanics in 3D space and are considered to be one of the best ways of representing rotations. In this paper a quaternion encryption method, based on algorithm by Nagase et al. (2004) has been proposed. According to a computer-based simulation the results of the performed research yield a high level of security, which is additionally strengthened by the...
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Cross sections for electron scattering from furan molecules; measurements and calculations
PublicationZmierzono i policzono przekroje czynne (TCS) na rozproszenie elektronów na drobinach furanu (C4H4O). Całkowite przekroje czynne zmierzono metodą transmisyjną w zakresie energii 0.6 - 400 eV. Sprężysty i jonizacyjny przekrój czyny obliczono dla energii zderzenia do 4 keV; powyżej 70 eV suma obu przekrojów pozostaje w dobrej zgodności z mierzonymi wartościami TCS.
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Prognozowanie mocy skrawania przy przecinaniu polskiego drewna sosnowego na pilarkach tarczowych
PublicationPrzedstawiono metodę określania mocy skrawania dla pilarek tarczowych wykorzystującą w modelu elementy mechaniki pękania. W obliczeniach uwzględniano wiązkość materiału obrabianego oraz jego wytrzymałość na ścinanie. Wykazano, że wspomniane parametry są silnie uzależnione od pochodzenia drewna. Dla jednej operacji przeprowadzono obliczenia dla drewna sosnowego pochodzącego z 4. różnych Krain geograficznych Polski.
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Prognozowanie mocy skrawania przy przecinaniu polskiego drewna sosnowego na pilarkach tarczowych
PublicationPrzedstawiono metodę określania mocy skrawania dla pilarek tarczowych wykorzystującą w modelu elementy mechaniki pękania. W obliczeniach uwzględniano wiązkość materiału obrabianego oraz jego wytrzymałość na ścinanie. Wykazano, że wspomniane parametry są silnie uzależnione od pochodzenia drewna. Dla jednej operacji przeprowadzono obliczenia dla drewna sosnowego pochodzącego z 4. różnych Krain geograficznych Polski.
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wycieczka dydaktyczna "KPŚ. spotkania sztuki z architekturą. vol. 2.22"
PublicationWycieczka dydaktyczna włączyła się w wydarzenie NARRACJE # 13. Wybrane zostały 4 spośród propozycji artystycznych przygotowanych na dwa jesienne wieczory (18-19 XI). Spotkanie rozpoczęło się 18 listopada o godzinie 17:00 przed Punktem Info (Siennicka 10a, Gdańsk-Przeróbka). Doświadczaliśmy i analizowaliśmy miejskie emocje, miejskie gry, miejskie historie i miejską przyrodę.
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ASIC Design Example of Complex SoC with FPGA Prototyping
PublicationThe paper presents an example of the System on a Chip design, where the FPGA prototyping has been used. Two FPGA prototypes have been realized. The first FPGA prototype uses AVNET board containing Xilinx Virtex4 device accompanied by custom board with required devices. The second FPGA prototype has been built using the custom PCB with Xilinx Virtex-4 XC4VLX60 FPGA accompanied by all needed external components. The final system...
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A comparison of exhaust emissions from vehicles fuelled with petrol, LPG and CNG
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Carbon dioxide emissions and fuel consumption from passenger cars tested over the NEDC and WLTC – an overview and experimental results from market-representative vehicles
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The effect of a low ambient temperature on the cold-start emissions and fuel consumption of passenger cars
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Force-induced structural changes in non-sulfated carrageenan based oligosaccharides – a theoretical study
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EGATEC: A new high-resolution engineering model of the global atmospheric electric circuit—Currents in the lower atmosphere
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Quantum chemical modeling (DFT) of active species on the VWO catalyst surface in various redox conditions
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The role of tungsten in formation of active sites for no SCR on the V-W-O catalyst surface — quantum chemical modeling (DFT)
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Biology, systematics, and clinical manifestations of Zygomycota infections
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Self-ignition of hydrogen–nitrogen mixtures during high-pressure release into air
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Fabrication of diet supplements components applied in order to reduce body mass
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Tribological synergy between classical ZDDP and innovative MoS2 and MoO3 nanotube additives at elevated temperatures
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Thermal properties of rare earth elements complexes with 1,3,5-benzenetricarboxylic acid
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Evaluation of Influence of the Addition Nanofillers on the Mechanical and Thermal Properties Terpolymers Ester-Ether-Amide
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Some applications of fractional order calculus
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P4018Reduced fibrin clot permeability is associated with an increased risk of both ischemic stroke and major bleeding in atrial fibrillation patients treated with vitamin K antagonists
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Computer modeling and testing of structural metamaterials
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Application of decision–making parametric structures in the analysis of a compound planetary gear
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Transformations of Tetrahydrocannabinol, tetrahydrocannabinolic acid and cannabinol during their extraction from Cannabis sativa L.
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Optimization of Transport Properties of A-Site Ordered LnBa1-xSrxCo2-yFeyO5+ Perovskite-Type Cathode Materials
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Correlation between chosen polymorphisms in genes coding 5HTT, 5HT2A and COMT with obesity.
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Protein transphosphorylation during the mutual interaction between phytochrome a and a nuclear isoform of nucleoside diphosphate kinase is regulated by red light
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Using CFD software for the evaluation of hygrothermal conditions at wall-window perimeters
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Reasons for changes in the value of unit pressure of compression products supporting external treatment
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In vitro anticariogenic effects of aerial parts of Drymocallis rupestris and its phytochemical profile
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Anticariogenic effects of extracts and fractions of Potentilla recta and their antioxidant activity
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Monitoring of fatigue damage development in as-received and exploited 10CrMo9-10 power engineering steel supported by Digital Image Correlation
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Characterization of carbon deposit with controlled carburization degree
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Systematic study on synthesis and purification of double-walled carbon nanotubes synthesized via CVD
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Interlayer defect evolution in an organic coating system on steel under hydromechanical loading
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Joint time–frequency analysis of electrochemical noise
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Investigations of the passive layer cracking by means of Dynamic Electrochemical Impedance Spectroscopy
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Correlation between destruction of the metal surface caused by pitting corrosion and intensity of the observed electrochemical noise (Invited Paper)
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