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Search results for: conformational studies
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Calcium electroporation for treatment of sarcoma in preclinical studies
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Application of bioassays in studies on the impact of pharmaceuticals on the environment
PublicationDrug interactions are often desirable particularly in medicine, when treatment of a patient requires using a mixture of drugs in specific doses to produce the adequate therapeutic effect. Unfortunately, interactions between drugs in the environment are not as desirable, despite the fact that drugs are present in the environment at low concentration levels [1]. Pharmaceuticals are present in the environment in a mixture of compounds,...
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Applying case studies to teaching architectural investment
PublicationCase studies enable students to encounter practical issues during their education. Experiments conducted in class employing this method often feature simplified models of real-world situations. However, they still enable students to encounter actual problems, to which theoretical knowledge is applied. In architectural education, students carrying out semester projects usually rely on data provided by the teacher, without wondering...
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The long-term studies of osmotic membrane distillation
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Surface studies of twinned of YBa2Cu3O7−δ crystals
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The structure of liquid lead: EXAFS and MD studies
PublicationPraca poświecona jest analizie widm XAFS zmierzonych na krawędzi L3dla ciekłego ołowiu. W analizie strukturalnej EXAFS zastosowano podejście GNXAS. Przetestowano kilka modeli strukturalnych, zarówno numerycznych (MD-DLE, MD-TB), jak i tych otrzymanych doświadczalnie (ND, XRD) i ostatecznie zrekonstruowano pierwszy pik w parowej funkcji rozkładu, g(r). Zweryfikowano wcześniejsze doniesienia o obserwownym za pomocą metody XAFS gwałtownym...
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Isolation and Self-Association Studies of Beta-Lactoglobulin
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In vitro toxicity studies of biodegradable, polyelectrolyte nanocapsules
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Adsorption and calorimetric studies of hydrothermally modified carbosils
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CRI board for CBM experiment: preliminary studies
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Design of Experiments in metabolomics-related studies: An overview
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Application of LC-MS technique in environmental studies
PublicationW ciągu ostatnich 10-15 lat obserwuje się ciągły wzrost zainteresowania możliwościami, jakie stwarza technika LC-MS, w związku z czym dokonano przeglądu prac badawczych zrealizowanych na Wydziale Chemicznym PG związanych z użyciem tej techniki. Szczególną uwagę zyskały: kwasy fenoksyoctowe i chlorofenole, które są stosowane w rolnictwie i które mogą zanieczyszczać wody gruntowe; cjanotoksyny, które są emitowane podczas zakwitów...
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The issues of participation in didactics of design. Case studies
PublicationThis article seeks to present and assess the usefulness of didactic methods aimed at preparing future architects for their role in the process of social participation. The article focuses on [a] a general overview of selected participation methods and tools, along with the examples of their application in the context of spatial management in Poland; [b] an overview of teaching methods used with a view to enhancing participation...
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Molecular dynamics studies of polyurethane nanocomposite hydrogels
PublicationPolyurethane PEO-based hydrogels have a broad range of biomedical applicability. They are attractive for drug-controlled delivery systems, surgical implants and wound healing dressings. In this study, a PEO based polyurethane hydrogels containing Cloisite R 30B, an organically modified clay mineral, was synthesized. Structure of nanocomposite hydrogels was determined using XRD technique. Its molecular dynamics was studied by means...
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The carbohydrate glycosylphosphatidylinositol anchor chain under mechanical stress
PublicationCarbohydrates have quite complicated micro heterogenic structure which may undergo different structural transitions. Due to their extreme flexibility it is very difficult to investigate such structural changes experimentally. In these studies we want to predict what structural and conformational changes are possible in the carbohydrate
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Structural and Dynamic Properties of Water within the Solvation Layer around Various Conformations of the Glycine-based Polypeptide
PublicationSeveral conformations of the solvated glycine-based polypeptides were investigated using molecular dynamics simulations. Some properties of water in the neighboring space around these molecules were investigated. It was found that water forms a well-defined layer—the first solvation shell—around the peptide molecule, and thickness of this layer is independent of the peptide structure and is equal to approximately 0.28 nm. Within...
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Structural and dynamic properties of water within the solvation layer around various conformations of the glycine-based polypeptide
PublicationSeveral conformations of the solvated glycine-based polypeptides were investigated using molecular dynamics simulations. Some properties of water in the neighbouring space around these molecules were investigated. It was found, that water forms a well-defined layer - the first solvation shell - around the peptide molecule, and thickness of this layer is independent of the peptide structure, and it equals to approximately 0.28 nm....
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Physics-Based Potentials for the Coupling between Backbone- and Side-Chain-Local Conformational States in the United Residue (UNRES) Force Field for Protein Simulations
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Conformational latitude – activity relationship of KPPR tetrapeptide analogues toward their ability to inhibit binding of vascular endothelial growth factor 165 to neuropilin‐1
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Studi Emigrazione / Migration Studies
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Conformation analysis and semiclassical dynamics study of charge exchange process induced by collision of C2+ ions with tetrahydrofuran
PublicationWe present the results of recent investigations of charge transfer processes in the collisions of C²⁺ ions with heterocyclic molecules of tetrahydrofuran.
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Insightful studies of AuCu nanostructures deposited on Ti platform: Effect of rapid thermal annealing on photoelectrochemical activity supported by synchrotron radiation studies
PublicationIn this work, we present the influence of annealing atmospheres during rapid thermal annealing (40◦C/s) on nanostructured Ti platforms modified by 10 nm layer of AuCu alloy obtained via magnetron sputtering. The AuCu/Ti platform annealed under hydrogen atmosphere exhibits the best photoelectrochemical activity under visible light, i.e. 27 times higher photocurrent than for pure Ti dimpled platform, and the lowest reflectance with minimum...
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Intelligence Augmentation and Amplification: Approaches, Tools, and Case Studies
PublicationMost experts agree that truly intelligent artificial system is yet to be developed. The main issue that still remains a challenge is imposing trust and explainability into such systems. However, is full replication of human intelligence really desirable key aim in intelligence related technology and research? This is where the concept of augmented intelligence comes into play. It is an alternative conceptualization of artificial...
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Electrochemical and acoustic emission studies of aluminum pitting corrosion
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The preparation method of experimental studies of the wood sawing process
PublicationW artykule przedstawiono sposoby działania, mające na celu przygotowanie badań doświadczalnych procesu przecinania drewna sosnowego na małogabarytowej pilarce ramowej PRW15M. Proces przygotowania badań podzielono na kilka etapów: przygotowanie próbek, pomiar własności fizycznych drewna (wilgotności drewna, gęstość drewna), pomiar własności strukturalnych drewna (średniej szerokości przyrostów rocznych oraz średniego udziału drewna...
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An odor-sensing system - powerful technique for foodstuff studies
PublicationThis work examines gas sensor array technology combined with multivariate data processing methods and demonstrates a promising potential for rapid, non-destructive analysis of food. Main attention is focused on detailed description of sensor used in e-nose instruments, construction, and principle of operation of these systems. Moreover, this paper briefly reviews the progress in the field of artificial olfaction and future trends...
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DFT studies of the refractive index of boron-doped diamond
PublicationThe density functional theory is one of the optimal solutions in calculation of optical properties of materials on the quantum scale. In this paper, we have investigated the refractive index of a boron-doped diamond structure with the usage of Atomistic Toolkit software from Synopsys. During this study, various methods and pseudopotentials were checked to obtain an optimal performanceaccuracy method for calculation of such materials....
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Application of the Optimum Dataset Method in Archeological Studies on Barrows
PublicationLight Detection and Ranging (LiDAR) became one of the technologies used in archaeological research. It allows for relatively easy detection of archaeological sites that have their own field form, e.g.: barrows, fortresses, tracts, ancient fields [1]. As a result of the scanning, the so-called point cloud is obtained, often consisting of millions of points. Such large measurement datasets are very time-consuming and labor-intensive...
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Biochemical, Structural Analysis, and Docking Studies of Spiropyrazoline Derivatives
PublicationIn this study, we evaluated the antiproliferative potential, DNA damage, crystal struc‐ tures, and docking calculation of two spiropyrazoline derivatives. The main focus of the research was to evaluate the antiproliferative potential of synthesized compounds towards eight cancer cell lines. Compound I demonstrated promising antiproliferative properties, especially toward the HL60 cell line, for which IC50 was equal to 9.4 μM/L....
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Planning and simulation studies of cellular-type manufacturing processes
PublicationZaproponowano metodę i algorytmy projektowania struktur organizacyjnych systemów wytwarzania typu gniazdowego, z wykorzystaniem zdefiniowanych modeli zapisu wiedzy technologicznej i zasad grupowej obróbki przedmiotów. Wyznaczono wskaźniki efektywności procesu grupowego przebiegającego w systemach gniazdowych z rozmieszczeniem komórkowym oraz funkcjonalnym stanowisk wg przyjętych formuł analitycznych. Zawarto wyniki zrealizowanych...
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Classification of submandibular salivary stones based on ultrastructural studies
PublicationIntroduction: Sialolithiasis remains a clinical problem with unclear etiopathogenesis, lack of prevention methods, and only surgical treatment. Materials and methods: An ultrastructure examination of submandibular sialoliths obtained from patients with chronic sialolithiasis was conducted using a scanning electron microscope and X-ray photoelectron...
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Theoretical studies of the pyranose ring under mechanical stress
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Recent Results from Studies of Electric Discharges in the Mesosphere
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Experimental studies of circuit breaker drives and mechanisms diagnostics
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Alanine Scanning Studies of the Antimicrobial Peptide Aurein 1.2
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Photophysical and theoretical studies of diphenylacetylene derivatives with restricted rotation
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Pathways and analytical tools in degradation studies of organic pollutants
PublicationWszystkie substancje chemiczne podlegają różnym procesom w wyniku wielu reakcji chemicznych, biochemicznych czy też fotochemicznych. W zależności od elementu środowiska w jakim znajduje się analit (np.: gleba, sedymenty, wody powierzchniowe i podziemne), może on ulegać powolnym przemianom w wyniku różnych procesów. W pracy przedstawiono niektóre drogi degradacji wybranych substancji w różnych warunkach. Omówiono problem identyfikacji...
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Parametric imaging in dynamic glucose metabolism studies in brain
PublicationArtykuł analizuje badania dynamiczne 18FDG-PET, które służą do estymacji metabolizmu glukozy w mózgu. Zbadano w nim wpływ zakłóceń na wyznaczanie interesującego nas parametru LCMRGlc.
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Automatic recognition of the arterial input function in MRI studies
PublicationArtykuł prezentuje opis automatycznej metody detekcji tętniczej funkcji wejście (AIF). Metoda została porównana z klinicznie pomierzonymi seriami obrazów DSC-MRI.
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Hydration of urea and its derivatives - Volumetric and compressibility studies
PublicationThe densities and sound velocities at T = (288.15, 293.15, 298.15, 303.15 and 308.15) K have been measured for aqueous solutions of urea, N,N-dimethylurea, N,N-diethylurea, N-propylurea, N-butylurea. From these data the apparent molar volumes, V the apparent molar isentropic compressions, KS,, and the Passynski solvation numbers of solutes have been determined. The concentration dependencies of the calculated quantities, their...
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Classification of submandibular salivary stones based on ultrastructural studies
PublicationIntroduction: Sialolithiasis remains a clinical problem with unclear etiopathogenesis, lack of prevention methods, and only surgical treatment. Materials and methods: An ultrastructure examination of submandibular sialoliths obtained from patients with chronic sialolithiasis was conducted using a scanning electron microscope and X‐ray photoelectron spectroscopy. Results: Based on the results, we divided sialoliths into three types:...
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Corrosion resistance studies of carbon-encapsulated iron nanoparticles
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In situ thermo-optical studies of polymer:fullerene blend films
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Dielectric and Optical Studies of FLC Sample with Helix Inversion
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Potential applications of plant in vitro cultures in phytoremediation studies
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Human Geomatics in Urban Design—Two Case Studies
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Studies of Exfoliated Graphite (EG) for Heavy Oil Sorption
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Optical absorption studies of (Ga0.1In0.9)2Se3 thin film
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Optical absorption studies of (Ga0.1In0.9)2Se3 thin film
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TG and DSC studies of bone tissue: Effects of osteoporosis
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