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Novel approaches in the synthesis of batracylin and its analogs: rebirth of an old player?
PublikacjaW pracy opisano batracylinę (BAT), jej syntezę i aktywność biologiczną oraz otrzymane analogi. BAT została wyselekcjonowana przez NCI (Bethesda, USA) w programie poszukiwań nowych potencjalnych leków przeciwnowotworowych. Związek ten w badaniach in vivo na myszach okazał się bardzo aktywny przeciw nowotworowi okrężnicy 38 (Colon 38), trudnemu do wyleczenia przez dotychczas znane leki przeciwnowotworowe. Jest ona skuteczna również...
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THE ART OF VIRTUAL INFORMATION EXCHANGE AND ITS INFLUENCE ON REAL CITY SPACE
PublikacjaThe paper investigates the impact of the new genres of contemporary public art based on the virtual information exchange in real spaces of the cities. On the basis of theoretical approaches, trans-disciplinary surveys and case studies, the paper focuses on the art that not only relies on the technological support but also refers to the new public sphere, where people are co-creators of the art object giving their personal input...
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THE PANTOGRAPH AND ITS GEOMETRIC TRANSFORMATIONS - A FORMER POPULAR TOOL FOR COPYING AND SCALING
PublikacjaDevelopment of digital technology has resulted in significant transformations of designer workshops. Computer applications replaced the previously existing tools and methods for drawing up of projects. Professional, sophisticated drawing instruments and tools for manual plotting, as well as basic drawing aids, have gradually fallen into oblivion and become relicts of a bygone era - the objects of collectors' interest. Gdansk University...
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Structural Health Monitoring of Composite Shell Footbridge for Its Design Validation
PublikacjaThe paper presents the structural health monitoring system of the composite bridge for pedestrians and cyclists. The footbridge was designed and manufactured within the FOBRIDGE project. It is the first bridge in the world, which is classified as a consistent single element structural girder, made of sandwich shells, entirely produced in a single cycle. The developed structural health monitoring system, supported design process,...
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Multi-level Virtualization and Its Impact on System Performance in Cloud Computing
PublikacjaThe results of benchmarking tests of multi-level virtualized environments are presented. There is analysed the performance impact of hardware virtualization, container-type isolation and programming level abstraction. The comparison is made on the basis of a proposed score metric that allows you to compare different aspects of performance. There is general performance (CPU and memory), networking, disk operations and application-like...
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The Effect of Circular Saw Blade Clamping Diameter on its Resonant Frequencies
PublikacjaIn this paper results of comparison of characteristic resonant frequencies of circular saw blades as a function of the saw clamping diameter from the impact test are presented. Obtained results revealed that proportionally with the increase of the saw clamping diameter also the dynamical stiffness of the saw blade increased. As a consequence of that the resonant frequencies of the saw blade move to higher values. Moreover, with...
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The effect of circular saw blade clamping diameter on its resonant frequencies
PublikacjaIn this paper results of comparison of characteristic resonant frequencies of circular saw blades as a function of saw clamping diameter from the impact test are presented. Obtained results revealed that proportionally with the increase of the saw clamping diameter also the dynamical stiffness of the saw blade increased. As a consequence of that the resonant frequencies of the saw blade move to higher values. Moreover, with the...
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Thermal ablation modeling via the bioheat equation and its numerical treatment
PublikacjaThe phenomenon of thermal ablation is described by Pennes’ bioheat equation. This model is based on Newton’s law of cooling. Many approximate methods have been considered because of the importance of this issue. We propose an implicit numerical scheme which has better stability properties than other approaches.
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“Project-factor-decision”. Decisive factors in IT projects and their impact on its success
PublikacjaThe aim of this article is to indicate the need for a deepening, systematizing and codifying of the theoretical and practical knowledge on IT project management, in the area of management decision-making processes. The scope of decisions made by managers is constantly on the increase. Project managers make decisions not only within the classic triangle of constraints, which consists of a schedule, a budget and the project scope,...
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Sources of Market Information, Its Quality and New Product Financial Performance
PublikacjaWhile we observe a growing interest in the role of market information in new product development (NPD), existing research has still largely ignored the quality of market information that is a crucial issue in the era of the information society. What does affect the quality of market information in new product development projects, and how does this quality influence the financial performance of new products? In this paper, we address...
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Pantographic metamaterials: an example of mathematically driven design and of its technological challenges
PublikacjaIn this paper, we account for the research efforts that have been started, for some among us, already since 2003, and aimed to the design of a class of exotic architectured, optimized (meta) materials. At the first stage of these efforts, as it often happens, the research was based on the results of mathematical investigations. The problem to be solved was stated as follows: determine the material (micro)structure governed by those...
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Effects of the Origin and Deacetylation Degree of Chitosan on Properties of Its Coatings on Titanium
PublikacjaThe properties of chitosan coatings on titanium surfaces may be influenced by a variety of factors, including their chemical characteristics and the deposition method. The aim of this research was to determine the influence of a chitosan’s origin (a type of shrimp) and deacetylation degree (DD), when deposited on a very smooth titanium surface, on adhesion and biological behavior. The tests were performed using chitosan of a degree...
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Identification of the Agile Mindset and Its Comparison to the Competencies of Selected Agile Roles
PublikacjaIn this paper we present the results of the identification and evalua-tion of the elements of an agile mindset as well as its comparison to the compe-tence models for the roles of Scrum Master, Product Owner and agile analyst. We have identified 70 unique agile mindset elements from literature and 5 in-terviews with experts. Based on an opinion survey among 52 agile practitioners we evaluated the importance of 26 selected elements...
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Broadband communication solutions for maritime ITSs: Wider and faster deployment of new e-navigation services
Publikacjan its initial part, the paper presents an overview of popular technologies and systems currently developed or employed in maritime communication. These solutions are used to provide both ship-to-ship and ship-to-shore communication for the purpose of supporting specific services, often dedicated to maritime safety and e-navigation. Utility of such communication systems have been thoroughly verified over the years and their strengths...
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Diminished toxicity of C-1748, 4-methyl-9-hydroxyethylamino-1-nitroacridine, compared with its demethyl analog, C-857, corresponds to its resistance to metabolism in HepG2 cells
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Diminshed toxicity of C-1748, 4-methyl-9-hydroxyethylamino-1-nitroacridine, compared with its demethyl analog, C-857, corresponds to its resistance to metabolism in HepG2 cells
PublikacjaThe narrow "therapeutic window" of anti-tumour therapy may be the result of drug metabolism leading to the activation or detoxification of antitumour agents. The aim of this work is to examine (i) whether the diminished toxicity of a potent antitumour drug, C-1748, 9-(2'-hydroxyethylamino)-4-methyl-1-nitroacridine, compared with its 4-demethyl analogue, C-857, results from the differences between the metabolic pathways for the...
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Rapid naming ability and its relationship to reading in Polish-speaking children with dyslexia
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Influence of Laser Modification on the Surface Character of Biomaterials: Titanium and Its Alloys—A Review
PublikacjaLaser surface modification is a widely available and simple technique that can be applied to different types of materials. It has been shown that by using a laser heat source, reproducible surfaces can be obtained, which is particularly important when developing materials for medical applications. The laser modification of titanium and its alloys is advantageous due to the possibility of controlling selected parameters and properties...
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Mechanism of Biofilm Formation on Installation Materials and Its Impact on the Quality of Tap Water
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Effect of Long-Term Potato Starch Retention with Citric Acid on Its Properties
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The Advancement of Biodegradable Polyesters as Delivery Systems for Camptothecin and Its Analogues—A Status Report
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A strongly bound OF3- anion and its unstable parent neutral OF3 species
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Improvement of charge separation in TiO 2 by its modification with different tungsten compounds
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The influence of texturing of the surface of concrete substrate on its adhesion to cement mortar overlay
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Fabrication of a Smartphone-Based Spectrophotometer and Its Application in Monitoring Concentrations of Organic Dyes
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Method for Determination of Methyl tert-Butyl Ether and Its Degradation Products in Water
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Thymus serpyllum Essential Oil and Its Biological Activity as a Modern Food Preserver
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The exponential law for partial, local and proper maps and its application to otopy theory
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The mechanism of overcoming multidrug resistance (MDR) of fungi by amphotericin B and its derivatives
PublikacjaPrzeprowadzono badania porównawcze w celu określenia aktywności i cytotoksyczności amfoterycyny B (AmB) i jej pochodnych wobec standardowego szczepu S. cerevisiae i jego transformantów zawierających geny C. albicans kodujące białka oporności wielolekowej (MDR) typu ABC i MFS. Pochodne AmB: amid 3-dimetyloaminopropylowy amfoterycyny B oraz ester metylowy N-metylo-N-D-fruktopiranozylo-amfoterycyny B wykazały efekt fungistatyczny...
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DFT and NBO theoretical study of protonation of tri-tert-butoxysilanethiol and its anion
PublikacjaWykonano obliczenia kwantowo-chemiczne metodą DFT dla tri-tert-butoksysilanotiolu oraz jego protonowanych i deprotonowanych form, zarówno na atomie tlenu jak i siarki. Przeanalizowano bilans energetyczny dla protonowania anionu w próżni i w fazie wodnej (stosując model IPCM). Zaobserwowano skrócenie wiązania Si-S w wyniku protonowania na atomie tlenu. Zmiany długości wiązań Si-O i Si-S zostały zinterpretowane w oparciu o analizę...
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Application of pH measurements for the following the course of biological treatment of wastewater and its control
PublikacjaZaprezentowano wyniki badań przeprowadzonych w skali laboratoryjnej w reaktorze imitującym działanie reaktora SBR. Oczyszczaniu poddano ścieki syntetyczne z dodatkiem glukozy. W trakcie oczyszczania ścieków monitorowano zmiany pH, redox, przewodności oraz stężenia azotu amonowego, azotanów i fosforanów. Stwierdzono korelację między pH i zmianami stężenia fosoranów oraz brak podobnej zależności dla związków azotowych.
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Loads of ship main diesel engine in the aspect of practical assessment of its operation
PublikacjaW artykule przedstawiono koncepcję metody pozwalającej na ocenę działania silnika pracującego na obciążeniu częściowym. Do określenia istniejącego zapasu parametrów użytkowych silnika oraz związanych z degradacją jego stanu technicznego dodatkowych kosztów ponoszonych przez użytkownika wykorzystane zostało wartościujące (ilościowe) ujęcie działania interpretowanego jako pewna wielkość fizyczna.
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Increasing the rate of sustainable change: a call for a redefinition of the concept and the model for its implementation
PublikacjaW pracy dokonano analizy problemu dużej rozbieżności pomiędzy zaproponowanymi strategiami a efektywnością akcji podjętych w celu wprowadzenia w praktyce zasad zrównoważonego rozwoju. Podkreślono konieczność współpracy różnych organizacji i samorządów lokalnych oraz uwzględniono rolę szkół wyższych w procesie wprowadzania zasad zrównoważonego rozwoju.
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Digital Cartographic Generalization – Study of Its Thresholds and Stages in Example of Cartographic Line
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Outdoor Advertising in Public Space and its Legal System in Poland over the Centuries
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Assessment of the Reliability of Wind Farm Device on the Basis of Modeling Its Operation Process
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Vimentin immunoexpression and its prognostic activity in colon cancer among Caucasian patients
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Ambulatory pulse pressure and its contributors in autosomal dominant polycystic kidney disease
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Characterization of a Unique Bordetella bronchiseptica vB_BbrP_BB8 Bacteriophage and Its Application as an Antibacterial Agent
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A Comprehensive Review on Shilajit: What We Know about Its Chemical Composition
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The history of Lake Rzecin and its surroundings drawn on maps as a background to palaeoecological reconstruction
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The question of whether diabetes and its cardiovascular risks can be prevented: A realistic DREAM?
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The influence of UV-radiation on hyaluronic acid and its blends with addition of collagen and chitosan
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Sun shines also in Poland - PV's global market and its future in Poland
PublikacjaNiekorzystne zmiany klimatyczne stanowią wyzwanie do poszukiwania konkurencyjnych ekotechnologii. Fotowoltaika ma szansę stać się ważnym źródłem energii w 21 wieku na całym świecie. Systemy fotowoltaiczne (PV) dostarczają energii elektrycznej w wyniku konwersji energii promieniowania słonecznego i przewiduje się, że wniosą one znaczący wkład w systemy energetyczne dzięki stałemu postępowi technologicznemu w tej dziedzinie i znaczącej...
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Inteligentne systemy transportu ITS na drogach szybkiego ruchu [Rozdział 12]
PublikacjaPrzedstawiono charakterystykę Inteligentnych Systemów Transportowych, architekturę ITS, funkcje systemów ITS na drogach szybkiego ruchu oraz efektywność wdrożenia rozwiązań z zakresu ITS.
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Characteristics, Chemical Modification Processes as well as the Application of Silica and its Modified Forms
PublikacjaThe variety of chemical modifications of the surface of silica and its modified forms cause thesematerials to find a consistently wider scope of application. In the publication, the characteristicsof silica, silica gel, aerogel and xerogel are presented. The obtainment, application and propertiesof these materials are discussed. Methods of chemical modifications of surface structures withthe use of different chemical compounds...
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Shaking table experimental study on diagnosis of damage and its evaluation in steel structure
PublikacjaCelem artykułu jest pokazanie wyników badań eksperymentalnych przeprowadzonych na stole sejsmicznym dotyczących identyfikacji uszkodzeń modelu dwukondygnacyjnej konstrukcji stalowej. Uszkodzenie zdefiniowano poprzez spadek sztywności i symulowano poprzez zamianę słupów modelu na elementy o mniejszym przekroju poprzecznym. Wyniki badań pokazują charakterystyczny spadek wartości naturalnych częstotliwości konstrukcji wraz ze wzrostem...
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Equitable and semi-equitable coloring of cubic graphs and its application in batch scheduling
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Mercury fractionation in marine macrofauna using thermodesorption technique: Method and its application
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The propeptide of human thyroid peroxidase is not required for its cellular, enzymatic or immunological activity
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