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Wyniki wyszukiwania dla: PO MARKER PEPTIDES
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Peptide conjugates of lactoferricin analogues and antimicrobials—Design, chemical synthesis, evaluation of antimicrobial activity and mammalian cytotoxicity
PublikacjaEight new peptide conjugates composed of modified bovine lactoferricin truncated analogues (LFcinB) and oneof the three antimicrobials — ciprofloxacin (CIP), levofloxacin (LVX), and fluconazole (FLC) — were synthesized. Four different linkers were applied to connect a peptide and an antimicrobial agent. The FLC-containing peptidic conjugates were synthesized using the “click chemistry” method. This novel approach is reported here...
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Synthesis and structure-activity studies of peptide-acridine/acridone conjugates
PublikacjaW artykule opisano strukturę, syntezę i biologiczną aktywność peptydowych koniugatów akrydyny i akrydonu jako potencjalnych leków o aktywności przeciwnowotworowej i przeciwwirusowej.
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Nutritional value, protein and peptide composition of edible cricket powders
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Elusive π-helical peptide foldamers spotted by chiroptical studies
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Gemcitabine Peptide-Based Conjugates and Their Application in Targeted Tumor Therapy
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Bladder cancer detection using a peptide substrate of the 20S proteasome
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Structural Analysis of a Peptide Fragment of Transmembrane Transporter Protein Bilitranslocase
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Membrane structure and interactions of peptide hormones with model lipid bilayers
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The influence of substrate peptide length on human β‐tryptase specificity
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Coulomb-Assisted Dissociative Electron Attachment: Application to a Model Peptide
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Simulating Electron Transfer Attachment to a Positively Charged Model Peptide
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Dynamics of Antimicrobial Peptide Encapsulation in Carbon Nanotubes: The Role of Hydroxylation
PublikacjaIntroduction: Carbon nanotubes (CNTs) have been widely employed as biomolecule carriers, but there is a need for further functionalization to broaden their therapeutic application in aqueous environments. A few reports have unraveled biomolecule–CNT interactions as a measure of response of the nanocarrier to drug-encapsulation dynamics. Methods: Herein, the dynamics of encapsulation of the antimicrobial peptide HA-FD-13 (accession...
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DMSO and TMAO—Differences in Interactions in Aqueous Solutions of the K-Peptide
PublikacjaInteractions between a solvent and their co-solute molecules in solutions of peptides are crucial for their stability and structure. The K-peptide is a synthetic fragment of a larger hen egg white lysozyme protein that is believed to be able to aggregate into amyloid structures. In this study, a complex experimental and theoretical approach is applied to study systems comprising the peptide, water, and two co-solutes: trimethylamide...
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New Peptide Based Fluconazole Conjugates with Expanded Molecular Targets
PublikacjaInfections of Candida spp. etiology are frequently treated with azole drugs. Among azoles, the most widely used in the clinical scenario remains fluconazole (FLC). Promising results in treatment of dangerous, systemic Candida infections demonstrate the advantages of combined therapies carried out with combinations of at least two different antifungal agents. Here, we report five conjugates composed of covalently linked FLC and...
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Anticancer Properties of Amino Acid and Peptide Derivatives of Mycophenolic Acid
PublikacjaBackground: Although Mycophenolic Acid (MPA) is applied as prodrugs in clinic as an immunosuppressant, it also possesses anticancer activity. MPA acts as Inosine-5’-Monophosphate Dehydrogenase (IMPDH) inhibitor, where the carboxylic group at the end of the side chain interacts with Ser 276 of the enzyme via hydrogen bonds. Therefore, MPA derivatives with other polar groups indicated high inhibition too. On the other hand, potent...
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Immunosuppressive properties of amino acid and peptide derivatives of mycophenolic acid
PublikacjaMycophenolic acid (MPA) was coupled with amino acids and biologically active peptides including derivatives of tuftsin to modify its immunosuppressive properties. Both amino acid unit in the case of simple MPA amides and modifications within peptide moiety of MPA - tuftsin conjugates influenced the observed activity. Antiproliferative potential of the obtained conjugates was investigated in vitro and MPA amides with threonine methyl...
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Optimised expression cassettes of hpt marker gene for biolistic transformation of Miscanthus sacchariflorus
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314 Osteopontin as a Potential Serum Marker in Early Breast Cancer-Preliminary Results
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Prediction of Bioactive Peptides From Chicken Feather and Pig Hair Keratins Using In Silico Analysis Based on Fragmentomic Approach
PublikacjaBackground: Keratin is among the most abundant structural proteins of animal origin, however it remains broadly underutilized. Objective: Bioinformatic investigation was performed to evaluate selected keratins originating from mass-produced waste products, i.e., chicken feathers and pig hair, as potential sources of bioactive peptides. Methods: Pepsin, trypsin, chymotrypsin, papain, and subtilisin were used for in silico keratinolysis...
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The concept of rule model of the internet mortgage market
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A decentralised model of the regulating ancillary services market
PublikacjaThe article presents a model of regulating ancillary services provision in a dencetralised manner. A concept of the operation of local markets for ancillary services is presented.
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Differentiation of the european insurance market (Polish example)
PublikacjaRynek usług ubezpieczeniowych jako część systemu finansowego każdej gospodarki odgrywa istotną rolę w stymulowaniu wzrostu gospodarczego. Jego sprawne funkcjonowanie w krajach Unii umożliwi realizację idei Jednolitego Rynku Ubezpieczeniowego. Dotychczasowy stan rzeczy wskazuje jednak na istotne zróżnicowanie poziomu rozwoju rynku ubezpieczeniowego w różnych krajach członkowskich Unii.
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Grip strength is associated with markers of central hemodynamics
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Usefulness of selected laboratory markers in ulcerative colitis
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Forecasts of the managed futures market – an empirical analysis
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Innovations in the payment card market: The case of Poland
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Segmentation of Passenger Electric Cars Market in Poland
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Regional Labour Market and Tourist Enterprises in Malopolska
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Identification of inertia and activity in the market behaviour of enterprises
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Markers of Anemia in Children with Type 1 Diabetes
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The point forecast of the situation of the examined company on the market
PublikacjaOkreślono sytuację badanego przedsiębiorstwa na rynku za pomocą analizy portfolio, w aspektach wzrostu rynku oraz względnego udziału badanego przedsiębiorstwa w rynku. Analiza objęła zarówno okres retrospektywny jak i prognozowany.
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GENDER INEQUALITY IN THE LABOUR MARKET IN KAZAKHSTAN AND UZBEKISTAN
PublikacjaThe aim of the following article is to present gender inequality in the labour market in Kazakhstan and Uzbekistan. Gender inequality was researched by analyzing documents providing rights for women and men in Kazakhstan and Uzbekistan. The author presented the unequal treatment of women in the labour market by examining the causes of the level of employment of women and men - contract workers, higher unemployment among women,...
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The investment risk forecasting in a local energy market
PublikacjaThe paper considers the general problems faced when evaluating the risk of investing in a local energy market by computer tools. The proposal formulated for the emerging local energy markets suggests broadening the method of evaluating investment risk so as to include elements of cluster analysis. The paper also discusses the significance of estimating investment risk in market terms and the importance and range of the local energy...
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Quality of graphical markers for the needs of eyewear devices
Publikacjain this paper we propose to cast the problem of identification of people, objects or places into an application for smart glasses that decodes information from graphical markers. We focus on analyzing different factors that can have influence on the processes of the automatic recognition of information from a code. The research we present aims at reviewing recognition performances in function of: size of a marker, distance from/to...
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Modelling processes for Polish civil aviation market
PublikacjaThe present , paper is the first step in research of Polish civil aviation market, focusing on the area of civil, legacy airlines. First, the market is described with its players, current conditions and its main problems. Next, the tools which are currently used for the prognosis processes are presented. Finally, the idea of a new model (fuzzy model) for the process of prognosis is presented.
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The situation of young mothers in the Polish labour market
PublikacjaThe purpose of the article is to present the situation of young women combining professional and paternal responsibilities in the Polish labour market. The papaer presents the results of interviews conducted with six young mothers.
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The (lack of) momentum effect in the UAE stock market
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A note on value investing in the UAE stock market
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Is there a low-risk anomaly in the UAE stock market?
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CONTAINER SHIPPING MARKET IN THE BALTIC SEA REGION
PublikacjaThe following article presents the situation on the maritime container transport market in the Baltic Sea Region. In the first part the author focuses on describing the specifics of the economic and geopolitical area of the Baltic Sea. The following parts include the market container shipping description along with its individual participants, such as carriers or seaports. Finally, the dynamic development of Polish container ports...
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Market Regeneration in Line with Sustainable Urban Development
PublikacjaThis article presents the study of the optimal design solutions for regeneration of marketplaces. It examines the design variants for the revitalisation of the marketplace, in particular, investment in their modernisation in order to find the most optimal model for transforming these public spaces to have a significant impact on the city’s development. The research is a comparative analysis of the implementation of regeneration...
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Different sources of market information and product innovativeness
PublikacjaThe purpose of this study is to identify whether the gathering of market information from different sources – i.e. from customers, competitors and other entities – is related to product innovativeness. The relationships proposed so far have not been empirically investigated but they can have important theoretical and practical implications for product innovation. To achieve the purpose of the paper data concerning 287 new products...
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CURRENT SITUATION ON THE POLAND REAL ESTATE MARKET
PublikacjaIn recent years the polish real estate market has been characterised by a significant increase in supply and demand. This was facilitated by a number of macroeconomic factors. In recent years, housing has been commissioned as 30 years ago. Therefore, the depth analysis issue of the causes and consequences for the Polish economy of these trends is now relevant. Among the reasons are significant economic growth, low interest rates...
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Synergistic action of extracts from carnivorous plants and synthetic peptides against plant pathoghenic bacteria
Publikacjaw pracy przedstawiono rezultaty badań nad sprawdzeniem aktywności przeciwbakteryjnej ekstraktów z roślin Drosera capensis i Dionaea muscipula w połączeniu z dwoma syntetycznymi peptydami: CAMEL oraz pexiganan. Najwyższą aktywnością przeciwbakteryjną odznaczał się chloroformowy ekstrakt z D. muscipula z peptydem CAMEL.
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Retro analog concept: comparative study on physico-chemical and biological properties of selected antimicrobial peptides
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Effect of Marination Time on the Antioxidant Properties of Peptides Extracted from Organic Dry-Fermented Beef
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Possible mechanisms for protecting NCα bonds in helical peptides from electron-capture (or transfer) dissociation
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Amides as models to study the hydration of proteins and peptides — spectroscopic and theoretical approach on hydration in various temperatures
PublikacjaInteractions with water are one of the key factors which determine protein stability and activity in aqueous solutions. However, the protein hydration is still insufficiently understood. N-methylacetamide (NMA) is regarded as a minimal part of the peptide backbone and the relative simplicity of its structure makes it a good model for studies on protein–water interactions. In this paper, the influence of NMA and N,N-dimethylacetamide...
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World Research Journal of Peptide and Protein
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Current Topics in Peptide and Protein Research
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