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Heterogeneity of quaternary structure of glucosamine-6-phosphate deaminase from Giardia lamblia
PublicationThe oligoHis-tagged versions of glucosamine-6- phosphate deaminase from Giardia lamblia (GlmNagB-HisN, GlmNagB-HisC) were constructed and purified to hear homogeneity, and their kinetic and structural properties were compared to those of the wild-type enzyme (GlmNagB). Introduction of the oligoHis tag at the GlmNagB C-terminus resulted in almost complete loss of the catalytic activity, while the catalytic properties of GlmNagB-HisN...
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Engineering Candida albicans glucosamine-6-phosphate synthase for efficient enzyme purification
PublicationRationally designed muteins of Candida albicans glucosamine-6-phosphate synthase, an enzyme known as a promising target for antifungal chemotherapy, were constructed, overexpressed in Escherichia coli and purified to near homogeneity. To facilitate and to optimize the purification of the enzyme, three recombinant versionscontaining internal oligoHis fragments were constructed: (i) by substituting residues 343 - 348...
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Inhibitors of glucosamine-6-phosphate synthase as potential antimicrobials or antidiabetics – synthesis and properties
PublicationGlucosamine-6-phosphate synthase (GlcN-6-P synthase) is known as a promising target for antimicrobial agents and antidiabetics. Several compounds of natural or synthetic origin have been identified as inhibitors of this enzyme. This set comprises highly selective L-glutamine, amino sugar phosphate or transition state intermediate cis-enolamine analogues. Relatively low antimicrobial activity of these inhibitors, poorly penetrating...
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Influence of Operation Conditions on Temperature Hazard of Lithium-Iron-Phosphate (LiFePO4) Cells
PublicationThe article presents and discusses the results of research on hazard, especially temperature, for selected lithium-ion-phosphate cells operated in accordance with the manufacturer’s recommendations but used under onerous mining conditions. This applies to the performance of cells in battery sets without the application of any management system (BMS). On the basis of the obtained test results, first of all, the influence of the...
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Polarimetric studies of L-arginine-doped potassium dihydrogen phosphate single crystals
PublicationConoscopic interference patterns, channelled spectra and polarimetric techniques have been used for the characterization of pure and doped (with L-arginine amino acid) potassium dihydrogen phosphate (KDP) single crystals. Experimental polarimetric data have been obtained for the frequently used wavelength of 633 nm and for two close wavelengths of 532 and 543 nm in a high-accuracy dual-wavelength polarimeter. The measurement of...
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Multi-objective electric distribution network reconfiguration solution using runner-root algorithm
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Damage Detection in Composite Materials Using Hyperspectral Imaging
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Condition monitoring and fault detection in wind turbines based on cointegration analysis of SCADA data
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Towards homoscedastic nonlinear cointegration for structural health monitoring
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An Experimental Study on the Effect of Temperature on Acoustic Emission Characteristics in Metallic Structures
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Nonlinear Cointegration Approach for Condition Monitoring of Wind Turbines
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Regulatory B Cells Involvement in Autoimmune Phenomena Occurring in Pediatric Graves’ Disease Patients
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Surface phenomena in discotic liquid crystals investigated using polarized FTIR transmission spectroscopy
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Parallel simulations of electrophysiological phenomena in myocardium on large 32 and 64-bit Linux clusters.
PublicationW pracy podjęto badania i przeprowadzono symulacje zjawisk elektrofizjologicznych w mięśniu sercowym z wykorzystaniem wytworzonego w tym celu oprogramowania równoległego opartego na MPI. Zaimplementowano i zbadano ulepszenia kodu prowadzące do uzyskania dobrej skalowalności oraz przeprowadzono testy wydajności na najnowszych 32 i 64-bitowych klastrach linuksowych. Praca stanowi próbę równoległej implementacji znanego podejścia...
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The influence of azide and imidazole on the properties of Mn- and Cd-based networks: conductivity and nonlinear phenomena
PublicationWe report a study on a family of four new Mn- and Cd-azide-imidazolate-based compounds with various crystal architectures. Notably, three of these compounds display noncentrosymmetric crystal arrangements at room temperature, a rare phenomenon in hybrid organic–inorganic materials. Both nonlinear optical (NLO) and electrical phenomena in these compounds are observed. The NLO processes include second and third harmonic generation,...
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Case studies of resonance phenomena in high voltage overhead power lines with shunt reactors
PublicationMisguided design of the towers of power transmission lines can lead to serious problems such as voltage asymmetry, overvoltages, electric arc extinction difficulties or resonance – in case of double circuit line with shunt reactors. The paper points out those threats on example of 400 kV double circuit overhead transmission line with shunt reactors.
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THE POSSIBILITIES OF ESTIMATING THE RELIABILITY OF SHIP PIPELINES’ ELEMENTS INCLUDING DESTRUCTIVE PHENOMENA ACTING ON THEM
PublicationIn the article an approach to the problem of estimating reliability data based on physical models is proposed. The possibility of reliability assessment for selected elements of ship pipelines, based on the recognition of the destructive physical phenomena taking place in them, is discussed. To do this, an overview of these phenomena has been made. In addition, a preliminary review of existing measures of destruction of materials...
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Characteristics of microstructural phenomena occurring on the surface of protective gloves by the action of mechanical and chemical factors
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Standing Acoustic Waves and Relative Nonlinear Phenomena in a Vibrationally Relaxing Gas-Filled Resonator
PublicationStanding acoustic waves in one-dimensional resonator filled with vibrationally relaxing gas, are studied. Two regimes of excitation of molecular vibrational degrees of freedom are considered, equilibrium and nonequilibrium. The acoustic energy enlarges with time in the non-equilibrium regime and decreases otherwise before formation of discontinuity. After that, it decreases due to nonlinear absorption and tends to zero in equilibrium...
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Predicting Ice Phenomena in a River Using the Artificial Neural Network and Extreme Gradient Boosting
PublicationForecasting ice phenomena in river systems is of great importance because these phenomena are a fundamental part of the hydrological regime. Due to the stochasticity of ice phenomena, their prediction is a difficult process, especially when data sets are sparse or incomplete. In this study, two machine learning models—Multilayer Perceptron Neural Network (MLPNN) and Extreme Gradient Boosting (XGBoost)—were developed to predict...
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Artificial Neural Network in Forecasting the Churn Phenomena Among Costumers of IT and Power Supply Services
PublicationThis paper presents an attempt to use an artificial neural network to investigate the churn phenomenon among the customers of a telecommunications operator. An attempt was made to create a data model based on the customer lifetime value (CLV) rather than on activity alone. A multilayered artificial neural network was used for the experiments. The results yielded a 99% successful identification rate for customers in no danger of...
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Metal dusting phenomena of 501 AISI furnace tubes in refinery fractional distillation unit
PublicationThe purpose of this investigation was to conduct the failure analysis of 501 AISI furnace tubes places before distillation column in fractional distillation unit. The investigated furnace tubes were planned to work for ten years however after just two years of exploitation <30% of the material left. The observed corrosion process had the intense and complex character. The well-adhered shiny black deposits and deep, round pits were...
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Thermal and Hydrodynamic Phenomena in the Stagnation Zone — Impact of the Inlet Turbulence Characteristics on the Numerical Analyses
PublicationOne of the methods of heat transfer enhancement is utilization of the turbulent impinging jets, which were recently applied, for example, in the heat exchangers. Their positive impact on the heat transfer performance was proven, but many questions related to the origin of this impact are still unanswered. In general, the wall-jet interaction and the near-wall turbulence are supposed to be its main reason, but their accurate numerical...
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Publicationes Universitatis Miskolciensis. Sectio philosophica
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Introduction to Higher Physics (PG_00055138), Design and Production Engineering, sem. 01, 2023/24
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CURRENT OPINION IN PHARMACOLOGY
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CLINICAL PHARMACOLOGY & THERAPEUTICS
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Current Vascular Pharmacology
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BRITISH JOURNAL OF PHARMACOLOGY
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Bangladesh Journal of Pharmacology
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CANCER CHEMOTHERAPY AND PHARMACOLOGY
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JOURNAL OF CLINICAL PHARMACOLOGY
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BMC Pharmacology & Toxicology
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FUNDAMENTAL & CLINICAL PHARMACOLOGY
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POLISH JOURNAL OF PHARMACOLOGY
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International Journal of Pharmacology
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Current Molecular Pharmacology
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ENVIRONMENTAL TOXICOLOGY AND PHARMACOLOGY
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Journal of Pharmacology & Pharmacotherapeutics
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Current Clinical Pharmacology
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BMC Pharmacology & Toxicology
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EUROPEAN JOURNAL OF PHARMACOLOGY
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Oral Therapeutics and Pharmacology
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Pharmacology Research & Perspectives
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Translational and Clinical Pharmacology
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Journal of HerbMed Pharmacology
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ALIMENTARY PHARMACOLOGY & THERAPEUTICS
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Current Pharmacology Reports
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Current Topics in Pharmacology
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Journal of Experimental Pharmacology
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