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General, Mild, and Metal-Free Functionalization of Indole and Its Derivatives Through Direct C3-Selenylation
PublicationA very mild method for the introduction of functionalized alkylselenyl group at C-3 position of the indole ring was developed. The proposed procedure consists of an electrophilic substitution of indole and its derivatives with bis(O,O-diisopropoxyphosphorothioyl) diselenide and subsequent cleavage of the P–Se bond with tetrabutylammonium fluoride in the presence of various electrophilic reagents. This method can be successfully...
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Opioid Growth Factor and its Derivatives as Potential Non-toxic Multifunctional Anticancer and Analgesic Compounds
PublicationIn this paper, we review the structure-activity relationship of OGF and its analogues. We highlight also OGF derivatives with analgesic, immunomodulatory activity and the ability to penetrate the blood-brain barrier and may be used as safe agents enhancing chemotherapy efficacy and improving quality of life in cancer patients. The reviewed papers indicate that Met-enkephalin and its analogues are interesting candidates for the...
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Computational Complexity and Its Influence on Predictive Capabilities of Machine Learning Models for Concrete Mix Design
PublicationThe design of concrete mixtures is crucial in concrete technology, aiming to produce concrete that meets specific quality and performance criteria. Modern standards require not only strength but also eco-friendliness and production efficiency. Based on the Three Equation Method, conventional mix design methods involve analytical and laboratory procedures but are insufficient for contemporary concrete technology, leading to overengineering...
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INTRODUCING GREENERY INTO A BUILDING BASED ON ITS IMPACT ON HUMAN WELLBEING - REVIEW OF THEORIES AND METHODS IN ARCHITECTURE
PublicationGreenery around and within buildings is an integral part of architectural space. Although science is providing more and more knowledge about the impact of greenery on human well-being, there is still a lack of guidelines on how to apply this knowledge in architectural design. The purpose of this review article is to prepare the ground for further research on how to support architectural design in integrating greenery as a co-creative...
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Lead In drinking water: Adsorption method and role of zeolitic imidazolate frameworks for its remediation: A review
PublicationDue to various characteristics properties lead(II) metal is utilized in many applications like lead ion batteries, water pipes, ammunition and paints. For this reason, concentration of lead(II) ions in water is increasing days by days which is alarming for water pollution. Water pollution is a major problem worldwide which affects biosphere badly, and causes continuous reduction of accessible sources of fresh water and ground water, available...
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Validated GC–MS method for determination of bisphenol a and its five analogues in dietary and nutritional supplements
PublicationBisphenol A (BPA) and its analogues showing structural and functional similarity to BPA are commonly applied in various industrial applications and thus are becoming ubiquitous in the environment. At the same time there is increasing scientific evidence that exposure to these chemicals may lead to adverse health effects in human and wildlife. In recent years dietary and nutritional supplements dedicated for athletes have become...
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The biological role of prolyl oligopeptidase and the procognitive potential of its peptidic inhibitors from food proteins
PublicationProlyl oligopeptidase (POP) is a conserved serine protease belonging to proline-specific peptidases. It has both enzymatic and non-enzymatic activity and is involved in numerous biological processes in the human body, playing a role in e.g., cellular growth and differentiation, inflammation, as well as the development of some neurodegenerative and neuropsychiatric disorders. This article describes the physiological and pathological...
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Cavitation erosion behavior of 18/8 stainless steel after its laser alloying of manganese
PublicationW pracy przedstawiono wyniki badań własności kawitacyjnych stali nierdzewnej gatunku 18/8 po jej laserowym stopowaniu różną zawartością manganu. Stwierdzono, że przy zawartości Mn w ilości 7,13% występuje największy wzrost twardości po stopowaniu a głębokość umacniania na skutek działania obciążeń kawitacyjnych jest najmniejsza.
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Review and Indication of Key Activities for Energy Management Improvement in DC Microgrids
PublicationDC MicroGrids (MG) must have Energy Management Systems (EMS) to guarantee efficient, dependable, and environmentally friendly electricity. The application of Model Predictive Control (MPC), proved to be helpful due to its adaptability and capacity to use non-linear models. This paper, based on an extensive literature review, identifies and discusses the three key activities to improve the characteristics of DC microgrids, i.e.:...
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Structural change in New Member States (1995-2005): shift-share analysis of productivity growth and its determinants
PublicationThe chapter focuses on the latest developments in ten New MemberStates (presented vis-à-vis EU-15countries), seen from the perspective of structural change and quality upgrading of their economic structures. In particular, recently released disaggregated labor statistics are used,allowing to analyse the process of labor reallocation and productivitychanges associated with inter-and intra-industrystructural change. Since the mid-1990s...
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Polityka i porządek prawny w polskiej energetyce na tle polityki Unii Europejskiej
PublicationW artykule przeanalizowano rozwój wspólnotowego rynku energii elektrycznej, polityk ę energetyczną Polski i UE, sytuację i działania Polski na wspólnotowym rynku energii elektrycznej, a następnie przeanalizowano nowe regulacje prawne dla współpracy rozproszonych źródeł energii elektrycznej i sieci inteligentnych z systemem krajowym, dla zwrotu energii odzyskiwanej z systemów elektromechanicznych do zasilającej...
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Speech formant frequency and pitch estimation using instantaneous complex frequency
PublicationW pracy opisany został algorytm estymacji częstotliwości podstawowej oraz częstotliwości środkowych i pasm formantów mowy z wykorzystaniem zespolonej pulsacji chwilowej. W artykule przedstawiono również wyniki działania algorytmu dla polskich samogłosek.
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Porównanie działania metod YIN i MAWT w estymacji tonu krtaniowego mowy zaburzonej
PublicationW pracy przedstawiono i dokonano porównania dwóch metod estymacji tonu krtaniowego, YIN i MAWT, ze szczególnym uwzględnieniem tych cech, które mają znaczenie w przetwarzaniu mowy zaburzonej. Algorytmy zaimplementowane w środowisku MATLAB poddano testom za pomocą odpowiednio dobranych nagrań mowy zaburzonej i niezaburzonej. Niniejsza praca zawiera wyniki tych testów oraz sporządzoną na ich podstawie analizę porównawczą.
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On the use of instantaneous complex frequency for pitch and formant tracking.
PublicationW pracy opisano algorytm śledzenia częstotliwości podstawowej i formantów mowy z wykorzystaniem zespolonej pulsacji chwilowej. Działanie algorytmu przetestowano na nagraniach polskich samogłosek, których wysokość zmieniała się płynnie. Wyniki testów wraz z porównaniem działania opisanej metody i metody predykcji liniowej zawarto w artykule.
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Instantaneous complex frequency for pipeline pitch estimation
PublicationIn the paper a pipeline algorithm for estimating the pitch of speech signal is proposed. The algorithm uses instantaneous complex frequencies estimated for four waveforms obtained by filtering the original speech signal through four bandpass complex Hilbert filters. The imaginary parts of ICFs from each channel give four candidates for pitch estimates. The decision regarding the final estimate is made based on the real parts of...
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On the use of instantaneous complex frequency for analysis and modification of simple sounds
PublicationW pracy przedstawiono możliwości wykorzystania zespolonej pulsacji chwilowej do analizy i modyfikacji prostych dźwięków. Opisywany algorytm składa się z dwóch kroków: bifaktoryzacji sygnału na obwiednię minimalnofazową i fazor dodatnipskrętny, a następnie estymacja i modyfikacja zespolonej pulsacji chwilowej obu czynników faktoryzacji.
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Oxidative Dimerisierung von Phosphanen und Hinweise auf das intermediare Auftreten des Phosphinophosphinidens tBu2P-P in Reaktionen von [(eta^5^-C5H5)2TiCl2] und [(eta^5^-C5H5)(eta^5^-C5Me5)TiCl2] mit tBu2P-P(SiMe3)Li und tBu2P-P(Li)-P-tBu2. Bildung von Titan(III)- Fulvalen-Komplexen.
PublicationReakcja dichlorku tytanocenu z tBu2P-P(Li)-P-tBu2 albo tBu2P-P(SiMe3)Li prowadzi do kompleksów Ti(III). Jednocześnie grupy fosfanowe dimeryzują dając (tBu2P)2P-P(P-tBu2)2 lub (tBu2P-PSiMe3)2. Znaleźliśmy produkty, które sugerują przejściowe występowanie tBu2P-P.
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Civil liability for artificial intelligence products versus the sustainable development of CEECs: which institutions matter?
PublicationThe aim of this paper is to conduct a meta-analysis of the EU and CEECs civil liability institutions in order to find out if they are ready for the Artificial Intelligence (AI) race. Particular focus is placed on ascertaining whether civil liability institutions such as the Product Liability Directive (EU) or civil codes (CEECs) will protect consumers and entrepreneurs, as well as ensure undistorted competition. In line with the...
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Novel luminescent calixarene-based lanthanide materials: From synthesis and characterization to the selective detection of Fe3+
PublicationCalix[n]arene-based coordination networks are an emerging class of materials with intriguing properties resulted from the presence of the cavity-like structure of the macrocycle and metallic nodes. In this work, four novel luminescent materials based on calix[4]arene-carboxylate and lanthanides (Eu3þ and Tb3þ) were prepared by two synthetic approaches, solvothermal (CDA-Eu-ST) and slow diffusion (CDA-Eu-RT, CDA-Tb-RT, CTA-Tb-complex)...
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Empirical investigation on labour market interactions in an enlarged Europe
PublicationThis paper proposes an empirical assessment of economic interactions between the labour markets ofthe integrating EU over the period of time 1995-2005. Drawing on recently made available industrystatistics, we provide a sector level study (13 tradable sectors, including manufacturing and services),analysing the contemporary evolution of domestic and trade partners' employment levels. Given theintensification of trade relations...
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Ochrona powietrza - europejskie standardy
PublicationCurrent regulations in EU oblige every member country to cover the protection of the air as well as determine, in a bright and clear way, the responsibilities of the governments to monitor the condition and introduce ways of protection of the air from pollution. If the responsibilities imposed by the directive on evaluation and management of the air quality are obeyed by the respective organs of member countries of EU, then the...
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Assessment of the Global and Regional Land Hydrosphere and Its Impact on the Balance of the Geophysical Excitation Function of Polar Motion
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Changes of Power Output and Velocity During Successive Sets of the Bench Press With Different Duration of Eccentric Movement
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Ammonia in Fly Ashes from Flue Gas Denitrification Process and its Impact on the Properties of Cement Composites
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Experimental validation of the use of energy transfer ratio (ETR) for damage diagnosis of steel-concrete composite beams
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Antifungal Activity of Capridine β as a Consequence of Its Biotransformation into Metabolite Affecting Yeast Topoisomerase II Activity
PublicationIn the last few years,increasing importance is attached to problems caused by fungal pathogens. Current methods of preventing fungal infections remain unsatisfactory. There are several antifungal compounds whichare highly effective in some cases, however, they have limitations in usage: Nephrotoxicity and other adverse effects. In addition, the frequent use of available fungistatic drugs promotes drug resistance....
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Minimal Sets of Lefschetz Periods for Morse-Smale Diffeomorphisms of a Connected Sum of g Real Projective Planes
PublicationThe dataset titled Database of the minimal sets of Lefschetz periods for Morse-Smale diffeomorphisms of a connected sum of g real projective planes contains all of the values of the topological invariant called the minimal set of Lefschetz periods, computed for Morse-Smale diffeomorphisms of a non-orientable compact surface without boundary of genus g (i.e. a connected sum of g real projective planes), where g varies from 1 to...
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The extracellular loop of Man-PTS subunit IID is responsible for the sensitivity of Lactococcus garvieae to garvicins A, B and C
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The Non-Lantibiotic Bacteriocin Garvicin Q Targets Man-PTS in a Broad Spectrum of Sensitive Bacterial Genera
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Multivariable optimization of ultrasound-assisted solvent extraction of bee pollen prior to its element analysis by FAAS
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Quantification of methadone and its metabolites: EDDP and EMDP determined in autopsy cases using LC‐MS/MS
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Corrigendum: Contrast Tempo of Movement and Its Effect on Power Output and Bar Velocity During Resistance Exercise
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Antioxidant potential of various solvent extract from Morus alba fruits and its major polyphenols composition
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Immunohistochemical detection of galectin-1 in renal biopsy specimens of children and its possible role in proteinuric glomerulopathies
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Parameter of nonlinearity B/A of three-component systems with separate volumes of liquid, its vapor and a neutral gas
PublicationOtrzymane zostało wyrażenie dla zaburzenia entropii substancji o trzech komponentach jako funkcja zaburzeń jej ciśnienia i gęstości. Na podstawie wzoru prędkość i parametru nieliniowosci fali akustycznej zostały wyliczone jako funkcje i ciśnienia i koncentracji pary i powietrza. Rezultaty są przedstawione w postaci wykresów.
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Synthesis and biological activity of tuftsin, its analogues and conjugates containing muramyl dipeptides of nor-muramyl dipeptides
PublicationOpisano syntezę koniugatów MDP oraz nor-MDP modyfikowanych w części peptydowej tuftsyną oraz pochodną tuftsyny zawierającą grupę nitrową. Zsyntetyzowane związki zostały przebadane in vitro na ludzkich monocytach i limfocytach w Akademii Medycznej w Gdańsku. Niektóre z nich wykazały szybsze i skuteczniejsze działanie w porównaniu z tuftsyną.
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9-(2,6-dichlorophenoxycarbonyl)10-methylacridinium trifluoromethanesulfonate and its precursor 2,6-dichlorophenyl acridine-9-carboxylate
PublicationMetodą rentgenowskiej analizy strukturalnej oznaczono struktury obu tytułowych związków. W ich trójskośnych kryształach występują odpowiednio: układy oddziaływań elektrostatycznych, C-H...O i π-π lub C-H...Cl, π-π i oddziaływań dyspersyjnych.
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The differential impact of a density of Polish pine wood on cutting forces with its origin region taken into consideration
PublicationIn the article the dependence of cutting forces in a function the density of wood with regard to the wood origin are presented. Samples used in experiment were with Scotch pine (Pinus sylvestris L.) originating from four provenances in Poland (Figure 1). Wood density was measured by two methods: stereometric method (global density) and radiometric method (local density). Stereometric method consists in measurements the volume...
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Classifying the transformation products (TPs) of emerging contaminants (ECs) for prioritizing research into their impact on the environment and human health
PublicationOne of the first books to cover transformation products, rather than primary compounds, Transformation Products of Emerging Contaminants in the Environment gathers, specifies, synthesizes, and advances existing knowledge of the most important transformation product (TPs) of the main groups of emerging contaminants with potential concern to human health and the environment. This two-volume set for researchers and professionals covers...
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Tailoring Defects in B, N-Codoped Carbon Nanowalls for Direct Electrochemical Oxidation of Glyphosate and its Metabolites
PublicationTailoring the defects in graphene and its related carbon allotropes has great potential to exploit their enhanced electrochemical properties for energy applications, environmental remediation, and sensing. Vertical graphene, also known as carbon nanowalls (CNWs), exhibits a large surface area, enhanced charge transfer capability, and high defect density, making it suitable for a wide range of emerging applications. However, precise...
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Problems of modelling toxic compounds emitted by a marine internal combustion engine for the evaluation of its structure parameters
PublicationThe paper presents the possibility of using an analytical study of the engine exhaust ignition to evaluate the technical condition of the selected components. Software tools available for the analysis of experimental data commonly use multiple regression model that allows the study of the effects and iterations between model input quantities and one output variable. The use of multi-equation models gives a lot of freedom in the...
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Membrane Sterols Modulate the Binding Mode of Amphotericin B without Affecting Its Affinity for a Lipid Bilayer
PublicationMembrane-active antibiotics are known to selectively target certain pathogens based on cell membrane properties, such as fluidity, lipid ordering, and phase behavior. These are in turn modulated by the composition of a lipid bilayer and in particular by the presence and type of membrane sterols. Amphotericin B (AmB), the golden standard of antifungal treatment, exhibits higher activity toward ergosterol-rich fungal membranes, which...
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Application of Msplit method for filtering airborne laser scanning data sets to estimate digital terrain models
PublicationALS point cloud filtering involves the separation of observations representing the physical terrain surface from those representing terrain details. A digital terrain model (DTM) is created from a subset of points representing the ground surface. The accuracy of the generated DTM is influenced by several factors, including the survey method used, the accuracy of the source data, the applied DTM generation algorithm, and the survey...
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Revitalized Mill Island in Bydgoszcz - the identity of the place created by the Brda River and its tributary named Młynowka
PublicationMill Island in Bydgoszcz, Poland is an example of downtown public space where a meander of the Młynówka creates the identity of the area.Before 2005, the only outstanding local feature was the fact that its south and west ends resembled the Venetian canals. The way the other parts of Mill Island were managed was inappropriate for a downtown.A comprehensive revitalization programme is returning Mill Island public space to residents,...
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Transformation of the countryside into an open-air museum as a way to rescue its spatial layot and to improve the quality of life
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Cigarette smoking and its impact on weight loss after bariatric surgery: A single center, retrospective study
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Paternal Postpartum Bonding and Its Predictors in the Early Postpartum Period: Cross-Sectional Study in a Polish Cohort
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Chemical composition of Polish propolis and its antiproliferative effect in combination with Bacopa monnieri on glioblastoma cell lines
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In Vitro Anticancer Potential of Jasione montana and Its Main Components against Human Amelanotic Melanoma Cells
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Effects of Low Concentration of Selected Analgesics and Successive Bioaugmentation of the Activated Sludge on Its Activity and Metabolic Diversity
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