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Diminished toxicity of C-1748, 4-methyl-9-hydroxyethylamino-1-nitroacridine, compared with its demethyl analog, C-857, corresponds to its resistance to metabolism in HepG2 cells
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Diminshed toxicity of C-1748, 4-methyl-9-hydroxyethylamino-1-nitroacridine, compared with its demethyl analog, C-857, corresponds to its resistance to metabolism in HepG2 cells
PublicationThe narrow "therapeutic window" of anti-tumour therapy may be the result of drug metabolism leading to the activation or detoxification of antitumour agents. The aim of this work is to examine (i) whether the diminished toxicity of a potent antitumour drug, C-1748, 9-(2'-hydroxyethylamino)-4-methyl-1-nitroacridine, compared with its 4-demethyl analogue, C-857, results from the differences between the metabolic pathways for the...
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Modelling long-term technological transition of Polish power system using MARKAL: Emission trade impact
PublicationThe need for technological transition of electricity production becomes a global problem. However, in coal-dominated Polish power system this need is even more crucial than anywhere, since technical lifetime of the most domestic power plants is ending. In this paper, the impact of the EU Emission Trading Scheme (EU ETS) for CO2 combined with sulfur dioxide (SO2) and nitrogen oxides (NOx) emission trading mechanism on power technology...
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On the application of magnetoelastic properties measureme nts for plastic level determination in martensitic steels
PublicationThe change in the dislocation density, induced by plastic deformation, influences strongly the magnetic domain structure inside the material. Being so, classic parameters, like the coercivity or magnetic permeability, can be a good measure of the deformation level, yet their reliable determination in a non-destructive way in industrial environment is problematic. The magnetoacoustic emission (MAE) which results from the non-180...
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Regulated Assembly of LPS, Its Structural Alterations and Cellular Response to LPS Defects
PublicationDistinguishing feature of the outer membrane (OM) of Gram-negative bacteria is its asymmetry due to the presence of lipopolysaccharide (LPS) in the outer leaflet of the OM and phospholipids in the inner leaflet. Recent studies have revealed the existence of regulatory controls that ensure a balanced biosynthesis of LPS and phospholipids, both of which are essential for bacterial viability. LPS provides the essential permeability...
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A PRELIMINARY STUDY ON THE OPTIMAL CHOICE OF AN IMPLANT AND ITS ORIENTATION IN VENTRAL HERNIA REPAIR
PublicationThis paper addresses the problem of ventral hernia repair. The main goals are to find an optimal surgical mesh for hernia repair and to define its optimal orientation in the abdominal wall to minimise the maximum force at the tissue-implant juncture. The optimal mesh is chosen from a set of orthotropic meshes with different stiffness ratios for typical hernia placement in the abdominal area. The implant is subjected to an anisotropic...
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The compositional space of exhaled breath condensate and its link to the human breath volatilome
PublicationBreath analysis is commonly understood to target gaseous or volatile organic compounds (VOCs) for the characterization of different pathologies. Targeted analysis is most effective if a working hypothesis can be based on a plethora of data. The recently published volatilome builds an optimal basis for organizing powerful target sets. However, the origin and pathways of biosynthesis of many VOCs are not known, which complicates...
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Modern remote sensing and the challenges facing education systems in terms of its teaching
PublicationCurrently the fastest growing area of geodesy is undoubtedly remote sensing. The importance that it has recently conducted on the effectiveness of worldwide research determines its huge success. Examination of the specific characteristics of objects without direct contact with them is a key feature has opened the way to the new very interesting areas of contemporary research. In this light, it seems reasonable to say that there...
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Equitable and semi-equitable coloring of cubic graphs and its application in batch scheduling
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Mercury fractionation in marine macrofauna using thermodesorption technique: Method and its application
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The Design Development of the Sliding Table Saw Towards Improving Its Dynamic Properties
PublicationCutting wood with circular saws is a popular machining operation in the woodworking and furniture industries. In the latter sliding table saws (panel saws) are commonly used for cutting of medium density fiberboards (MDF), high density fiberboards (HDF), laminate veneer lumber (LVL), plywood and chipboards of different structures. The most demanded requirements for machine tools are accuracy and precision, which mainly depend on...
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The effect of dehydration/rehydration of bacterial nanocellulose on its tensile strength and physicochemical properties
PublicationBacterial nanocellulose (BNC) is a natural biomaterial with a wide range of biomedical applications. BNC contains 99 % of water which makes it too thick to be used as a bioimplant material. The aim of the work was to determine the effect of the BNC dehydration followed by rehydration on its mechanical and physicochemical properties, in the context of the use of BNC as bio-prostheses in the cardiovascular system. Dehydration involved the...
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PARAMETERS OF THE ELECTROPHORETIC DEPOSITION PROCESS AND ITS INFLUENCE ON THE MORPHOLOGY OF HYDROXYAPATITE COATINGS. REVIEW
PublicationMetallic materials intended for bone implants should exhibit not only appropriate mechanical properties, but also high biocompatibility. The surface treatment modifications, for example acidic treatment, laser treatment, ion implantation and deposition of highly biocompatible coatings, are practiced. One of the most popular methods of surface modification is to deposit hydroxyapatite (HAp) coatings. HAp naturally occurs in human...
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Possible directions for development of C-ITS services in cities on the example of the TRISTAR System
PublicationDuring the previous EU financial perspective (2007 - 2013), we observed an intensification of the evelopment of transport management systems using ITS services in Polish cities. One of the biggest territorially and functionally system is Tri-city TRISTAR system, the implementation of which was completed in 2015. The concept of the TRISTAR system and its architecture was developed in the years 2002-2007. Currently, we can observe...
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Effect of aeration of antibiotic-loaded bone cement on its properties and bactericidal effectiveness
PublicationBACKGROUND: Antibiotic-loaded bone cements are now widely used in medicine. They are able to locally deliver antibiotic particles and they allow treat or protect against infection. It is assumed that the bactericidal effectiveness of bioactive bone cements depend on the parameters of its production. Hence, the aim of this study was to check the effect of aeration of bone cement before mixing the components on its properties as...
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A Novel Approach of Using Selected Unconventional Geodesic Methods of Estimation on VTS Areas
PublicationThe Vessel Traffic Service (VTS) systems belong to the fundamental tools used in ensuring a high level of safety across sea basins with heavy traffic, where the presence of navigational hazards poses a great risk of collision or a ship running aground. In order to determine the mutual location of ships, VTS systems obtain information from different facilities, such as coastal radar stations, AIS, and vision systems. Fixing a ship’s...
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Water uptake in protective organic coatings and its reflection in measured coating impedance
PublicationWater uptake in commercially available epoxy coating on mild steel using impedance spectroscopy and gravimetry was studied. The water content in the coating was determined using the Brasher-Kingsbury equation and various methods of coating capacitance calculation used in the literature. The obtained results were compared with reference gravimetric data. An overestimation of values obtained from impedance data in relation to gravimetric...
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Standard deviation as the optimization criterion in the OptD method and its influence on the generated DTM
PublicationReduction of the measurement dataset is one of the current issues related to constantly developing technologies that provide large datasets, eg. laser scanning. It could seems that presence and evolution of processors computer, increase of hard drive capacity etc. is the solution for development of such large datasets. And in fact it is, however, the “lighter” datasets are easier to work with. Additionally, reduced datasets can...
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Geometry optimization of steroid sulfatase inhibitors - the influence on the free binding energy with STS
PublicationIn the paper we review the application of two techniques (molecular mechanics and quantum mechanics) to study the influence of geometry optimization of the steroid sulfatase inhibitors on the values of descriptors coded their chemical structure and their free binding energy with the STS protein. We selected 22 STS-inhibitors and compared their structures optimized with MM+, PM7 and DFT B3LYP/6–31++G* approaches considering separately...
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Relationship between microstructure of laser alloyed C45 steel and its cavitation resistance.
PublicationW pracy przedstawiono badania wpływu laserowo kształtowanej mikrostruktury na stali C45 po stopowniu różnymi kompozycjami proszków metali na własności kawitacyjne warstwy wierzchniej. Badania prowadzono w początkowym stadium erozji kawitacyjnej. Stwierdzono, że lepszą odporność kawitacyjną osiąga się gdy mikrostruktura jest podatna do umacniania odkształceniowego np. w obecności pewnej ilości austenitu w strukturze.
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On the possibility of estimating fish length distribution from its target strength statistics.
PublicationArtykuł przedstawia koncepcję odtwarzania rozkładu długości ryb na podstawie danych z przeszukiwań akustycznych. Wykorzystując metody odwrotne w statystycznym przetwarzaniu rozkładu siły celu ryb pokazano, że przy pewnych założeniach co do rozkładu położenia ryb w wiązce, możliwa jest estymacja szukanego rozkładu długości ryb.
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Relationship between microstructure of laser alloyed of C45 steel and its cavitation resistance.
PublicationPrzedstawiono badania odporności kawitacyjnej stali C45 po laserowym stopowaniu jej powierzchni proszkami Mn., Ni, Cr, Nb, Mo, Co. Stwierdzono, że warstwa wierzchnia posiada wyższą odporność kawitacyjną jeśli w jej mikrostrukturze występuje pewna ilość austenitu zwiększająca podatność do wzmacniania odkształceniowego.
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Toxicity of sediments and its relations with the mobility of pollutants on the basis of studies of Lake Turawskie
PublicationPraca niniejsza jest raportem z badań nad toksycznością i jej powiązaniem z mobilnością zanieczyszczeń. Moblilność zanieczyszczeń uzależniona jest od pH próbki. Próbki pobierano z Jez. Turawskiego, toksyczność była mierzona przy użyciu testu Microtox (AZUR Environmental, USA).
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Nitrogen monitoring in atmospheric deposition and its removal from municipal and industrial wastewater
PublicationBadano zmiany stężenia azotu w opadach atmosferycznych oraz warunki usuwania azotu ze ścieków komunalnych i przemysłowych. Badano wpływ wybranych sulfonamidów na proces nitryfikacji oraz oznaczano ich stopień biodegradacji. Stwierdzono, że sulfonamidy są substancjami, które hamują procesy biologicznego oczyszczania ścieków, jak również w niskim stopniu ulegają biodegradacji.
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Photovoltaic solar cells and modules as the source of electricity in the world and its future in Poland
PublicationJedną z metod ograniczenia emisji CO2 na świecie i w Polsce jest zastępowanie paliw kopalnych odnawialnymi źródłami energii. Systemy fotowoltaiczne, generujące energie elektryczną, są uważane za technologię wpisująca się w politykę zrównoważonego rozwoju dzięki znacznemu postępowi technologicznemu w zakresie ich wytwarzania i znacznej redukcji kosztów tych systemów.W artykule naświetlono postęp, jaki dokonał się w tej dziedzinie...
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The Advancement of Biodegradable Polyesters as Delivery Systems for Camptothecin and Its Analogues—A Status Report
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A strongly bound OF3- anion and its unstable parent neutral OF3 species
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Improvement of charge separation in TiO 2 by its modification with different tungsten compounds
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Digital Cartographic Generalization – Study of Its Thresholds and Stages in Example of Cartographic Line
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Outdoor Advertising in Public Space and its Legal System in Poland over the Centuries
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Comparison of usefulness of different diagnostic procedures in slipped capital femoral epiphysis in cats
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Assessment of the Reliability of Wind Farm Device on the Basis of Modeling Its Operation Process
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Vimentin immunoexpression and its prognostic activity in colon cancer among Caucasian patients
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Ambulatory pulse pressure and its contributors in autosomal dominant polycystic kidney disease
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Characterization of a Unique Bordetella bronchiseptica vB_BbrP_BB8 Bacteriophage and Its Application as an Antibacterial Agent
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A Comprehensive Review on Shilajit: What We Know about Its Chemical Composition
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The history of Lake Rzecin and its surroundings drawn on maps as a background to palaeoecological reconstruction
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The question of whether diabetes and its cardiovascular risks can be prevented: A realistic DREAM?
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The influence of UV-radiation on hyaluronic acid and its blends with addition of collagen and chitosan
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Phenotypic yield and its structure variability of moderately late and late potato cultivars
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In search of environmental role of cylindrospermopsin: A review on global distribution and ecology of its producers
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Chlorpromazine-induced hyperprolactinemia in a young female and its relation with fibrocystic breast disease
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Free-ranging domestic cats are characterized by increased metal content in reproductive tissues
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The influence of texturing of the surface of concrete substrate on its adhesion to cement mortar overlay
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Precise mapping of the magnetic field in the CMS barrel yoke using cosmic rays
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Performance of the CMS hadron calorimeter with cosmic ray muons and LHC beam data
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Calibration of the CMS drift tube chambers and measurement of the drift velocity with cosmic rays
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<title>JTAG test system for RPC muon trigger in the CMS experiment</title>
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Interaction of amphotericin B and its selected derivatives with membranes: molecular modeling studies
PublicationJest to praca przeglądowa obejmująca krytyczną analizę danych dotyczących oddziaływania amfoterycyny B (AmB) i jej wybranych, mniej toksycznych pochodnych, z błonami lipidowymi. Amfoterycyna B jest antybiotykiem przeciwgrzybowym ale ze względu na jej toksyczność trwają prace nad modyfikacjami chemicznymi tego związku. Celem molekularnym dla tego antybiotyku jest błona lipidowa i dlatego różnicowe powinowactwo AmB i jej pochodnych...
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Increasing the rate of sustainable change: a call for a redefinition of the concept and the model for its implementation
PublicationW pracy dokonano analizy problemu dużej rozbieżności pomiędzy zaproponowanymi strategiami a efektywnością akcji podjętych w celu wprowadzenia w praktyce zasad zrównoważonego rozwoju. Podkreślono konieczność współpracy różnych organizacji i samorządów lokalnych oraz uwzględniono rolę szkół wyższych w procesie wprowadzania zasad zrównoważonego rozwoju.