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Optimization of Chemical Functionalities of Indole-2-carboxamides To Improve Allosteric Parameters for the Cannabinoid Receptor 1 (CB1)
Publikacja5-Chloro-3-ethyl-N-(4-(piperidin-1-yl)phenethyl)-1H-indole-2-carboxamide (1; ORG27569) is a prototypical allosteric modulator for the cannabinoid type 1 receptor (CB1). Here, we reveal key structural requirements of indole-2-carboxamides for allosteric modulation of CB1: a critical chain length at the C3-position, an electron withdrawing group at the C5-position, the length of the linker between the amide bond and the phenyl ring...
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The searchlight problem for road networks
PublikacjaWe consider the problem of searching for a mobile intruder hiding in a road network given as the union of two or more lines, or two or more line segments, in the plane. Some of the intersections of the road network are occupied by stationary guards equipped with a number of searchlights, each of which can emit a single ray of light in any direction along the lines (or line segments) it is on. The goal is to detect the intruder,...
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The influence of compensate coils on own ship magnetic field
PublikacjaA ferromagnetic object placed in the earth magnetic field causes a local disturbance in this field distribution. The field distribution disturbance is a function of many arguments like the dimensoins and shape of the object, its ferromagnetic properties ande its positon in relation to the earth magnetic field. in order to minimize the influence of this disturbance one places compensate coils on the ship. Some chosen results of...
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Nowy wewnątrzbudynkowy algorytm wyznaczania położenia obiektów
PublikacjaW referacie zaprezentowano nowy wewnątrzbudynkowy algorytm wyznaczania położenia obiektów WAP. W algorytmie tym uwzględnia się właściwości środowiska propagacyjnego, dzięki czemu dokładność estymat położenia obiektów wyznaczonych algorytmem WAP jest większa niż wyznaczonych znanymi algorytmami Chana oraz Foy’a. W referacie przedstawiono wyniki analizy porównawczej tych trzech algorytmów z użyciem rzeczywistych pomiarów odległości...
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Aproksymacja przebiegu trasy kolejowej na przykładzie krzywoliniowego odcinka połączenia Somonino-Gdańsk Osowa
PublikacjaW artykule zaprezentowano wyniki wyznaczenia współrzędnych przebiegu trasy kolejowej metodami aproksymacji wielomianowej i interpolacji krzywą kubiczną w oparciu o pomiary czasu rzeczywistego GPS zrealizowane z wykorzystanie polskiej aktywnej sieci geodezyjnej ASG-EUPOS. Rozważania teoretyczne poparte zostały praktycznym przykładem aplikacyjnym opartym o zrealizowane pomiary inwentaryzacyjne zmodernizowanego odcinka toru kolejowego...
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Asynchronous time difference of arrival (ATDOA) method
PublikacjaA new method for a location service in the asynchronous wireless sensor networks is outlined. This method, which is called asynchronous time difference of arrival (ATDOA), enables calculation of the position of a mobile node without knowledge of relative time differences (RTDs) between measuring sensors. The ATDOA method is based on the measurement of time difference of arrival between the node and the same sensor at the discrete...
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Mowa nienawiści (hate speech) a odpowiedzialność dostawców usług internetowych w orzecznictwie sądów europejskich
PublikacjaThe article analyses the phenomenon of hate speech in the Internet contrasted with the problem of responsability of Internet Service Providers for cases of such abuses of freedom of expression. The text provides an analysis of jurisprudence of two European Courts. On the one hand it presents the position of the European Court of Human Rights on the problem of hate speech: its definition and the liability for it as an exception...
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The use of a genetic algorithm in the process of optimizing the shape of a three-dimensional periodic beam
PublikacjaMechanical periodic structures exhibit unusual dynamic behavior thanks to the periodicity of their structures, which can be attributed to their cellular arrangement. The source of this periodicity may result from periodic variations of material properties within their cells and/or variations in the cell geometry. The authors present the results of their studies on the optimization of physical parameters of a three-dimensional axisymetrical...
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Automatic detection of abandoned luggage employing a dual camera system
PublikacjaA system for automatic detection of events using a system of fixed and PTZ (pan-tilt-zoom) cameras is described. Images from the fixed camera are analyzed by means of object detection and tracking. Event detection system uses a set of rules to analyze data on the tracked moving objects and to detect defined events. A PTZ camera is used to obtain a detailed view of a selected object. A procedure for conversion between the pixel...
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The use of Response Surface Methodology for reliability estimation of aluminum silo subjected to wind load
PublikacjaAn axisymmetric aluminum silo model with a single, standardized geometric imperfection of its lateral surface is considered. The silo is wind – loaded only. The paper is focused on the critical, or limit value of wind pressure, both producing a loss of stability of the silo. This value is affected by vertical coordinate (position) of the imperfection and the angular relation between the imperfection and the wind direction. Reliability...
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Hydrogen sulphide electrocatalytic gas sensor
PublikacjaIn this article measurement results of the electrocatalytic gas sensor in different concentrations of hydrogen sulphide are presented. Working principle of such sensor is based on electric current acquisition, while voltage ramp is applied to the sensor. During voltage sweep oxidation and reduction reactions occurs on the sensor electrodes. Obtained current-voltage plot has unique shape connected...
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Accuracy of Trajectory Tracking Based on Nonlinear Guidance Logic for Hydrographic Unmanned Surface Vessels
PublikacjaA new trend in recent years for hydrographic measurement in water bodies is the use of unmanned surface vehicles (USVs). In the process of navigation by USVs, it is particularly important to control position precisely on the measuring profile. Precise navigation with respect to the measuring profile avoids registration of redundant data and thus saves time and survey costs. This article addresses the issue of precise navigation...
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Leader election for anonymous asynchronous agents in arbitrary networks
PublikacjaWe consider the problem of leader election among mobile agents operating in an arbitrary network modeled as an undirected graph. Nodes of the network are unlabeled and all agents are identical. Hence the only way to elect a leader among agents is by exploiting asymmetries in their initial positions in the graph. Agents do not know the graph or their positions in it, hence they must gain this knowledge by navigating in the graph...
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Validation of atmospheric aerosols sampling in equivalent fractions
PublikacjaPhysical properties and chemical composition of atmospheric aerosols are of extreme importance, in many fields of interest, namely the Environment even with legal implications. Atmospheric sampling poses inherent problems with consequent demands on sampling optimisation, with sampling strategies requiring validation. In this work a study was conducted aiming at validating the collection of atmospheric aerosols in equivalent fractions....
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Trophic Transfer of Mercury in a Temperate Marine Food Web, Southern Baltic Sea
PublikacjaMercury (Hg) is considered to be one of the most dangerous global environmental pollutants. The toxicity and bioavailabilityof Hg depend on its chemical form, and the greatest hazard is posed by the organomercurial compounds. Hg is introduced into the human body primarily through the consumption of fish and seafood. Despite numerous studies on Hg in marine organisms, there is still a gap in the knowledge on Hg uptake and...
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The evaluation of eGlasses eye tracking module as an extension for Scratch
PublikacjaIn this paper we present the possibility of using eGlasses eye tracking module as an extension for Scratch programming tool which is a visual programming language supporting computer skills learning. The main concept behind this project is to setup the interface for rapid interaction design. Eye tracking is a powerful tool for hands free communication but for that requires a dedicated software. This software is rarely tailored...
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The geodetic monitoring of the engineering structure – a practical solution of the problem in 3D space
PublikacjaThe study raises the issues concerning the automatic system designed for the monitoring of movement of controlled points, located on the roof covering of the Forest Opera in Sopot. It presents the calculation algorithm proposed by authors. It takes into account the specific design and location of the test object. High forest stand makes it difficult to use distant reference points. Hence the reference points used to study the stability...
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Experimental studies on the impact of changing the pipe material on the propagation of the pressure wave during water hammer
PublikacjaAim of the paper is to present the results studying the water hammer phenomenon in pipes made of different materials, and to show the impact of changing the type of material of the pipe on the velocity of the pressure wave during the transient flow in the pipes. In terms of research material and methods, pipes made of galvanized steel and high-density polyethylene were tested. Measurements were made using strain gauges with a high...
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Pupil detection supported by Haar feature based cascade classifier for two-photon vision examinations
PublikacjaThe aim of this paper is to present a novel method, called Adaptive Edge Detection (AED), of extraction of precise pupil edge coordinates from eye image characterized by reflections of external illuminators and laser beams. The method is used for monitoring of pupil size and position during psychophysical tests of two-photon vision performed by dedicated optical set-up. Two-photon vision is a new phenomenon of perception of short-pulsed...
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Person Tracking in Ultra-Wide Band Hybrid Localization System Using Reduced Number of Reference Nodes
PublikacjaIn this article a novel method of positional data integration in an indoor hybrid localization system combining inertial navigation with radio distance measurements is presented. A point of interest is the situation when the positional data and the radio distance measurements are obtained from less than thee reference nodes and it is impossible to unambiguously localize the moving person due to undetermined set of positional equations....
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Relationship between Chemical Structure and Biological Activity Evaluated In Vitro for Six Anthocyanidins Most Commonly Occurring in Edible Plants
PublikacjaNumerous studies have provided evidence that diets rich in anthocyanins show a broad spectrum of health benefits. Anthocyanins in nature are usually found in the form of glycosides. Their aglycone forms are called anthocyanidins. The chemical structure of anthocyanins is based on the flavylium cation, but they differ in the position and number of substituents. However, the bioactives and foods that contain them are frequently treated...
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Collision‐Aware Routing Using Multi‐Objective Seagull Optimization Algorithm for WSN‐Based IoT
PublikacjaIn recent trends, wireless sensor networks (WSNs) have become popular because of their cost, simple structure, reliability, and developments in the communication field. The Internet of Things (IoT) refers to the interconnection of everyday objects and sharing of information through the Internet. Congestion in networks leads to transmission delays and packet loss and causes wastage of time and energy on recovery. The routing protocols...
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The electronic excited states of dichloromethane in the 5.8-10.8 eV energy range investigated by experimental and theoretical methods
PublikacjaWe present a comprehensive experimental high-resolution vacuum ultraviolet (VUV) photoabsorption spectrum of dichloromethane, CH 2 Cl 2 , with absolute cross sections determined for the full 5.8–10.8 eV energy-range. The calculations on the vertical excitation energies and oscillator strengths were performed using the equation-of-motion coupled cluster method, restricted to the single and double excitations level (EOM-CCSD), and...
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An electric ring thruster as auxiliary manoeuvring propulsion system for watercraft - construction analysis
PublikacjaThe reported project aimed at examining properties and purposefulness of use of modern electromagneticbearings for a screw propeller in a prototype version of a synchronous ring motor with rare earths magnets.Bearings of this type generate electromagnetic forces which keep the rotor in a state of levitation. Therotating machine with magnetic bearings can work in any environment which reveals diamagnetic properties(air, vacuum,...
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FAILURE OF MAGNETIC FLUID SEALS OPERATING IN WATER: PRELIMINARY CONCLUSIONS
PublikacjaThe article analyses properties of magnetic fluid seals installed in rotary sealing no des which operate in the utility water environment. Seals of this type have been examined as a possible solution to the problem with ship manoeuvring propulsion sealing. The present analysis bases on laboratory durability tests of magnetic fluid seals expo sed to long - term utility water loads, at different water pressures and shaft revolutions....
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Two-phase optimizing approach to design assessments of long distance heat transportation for CHP systems
PublikacjaCogeneration or Combined Heat and Power (CHP) for power plants is a method of putting to use waste heat which would be otherwise released to the environment. This allows the increase in thermodynamic efficiency of the plant and can be a source of environmental friendly heat for District Heating (DH). In the paper CHP for Nuclear Power Plant (NPP) is analyzed with the focus on heat transportation. A method for effectivity and feasibility...
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Performance Analysis and Quantification of BeiDou Navigation Satellite System (BDS-3)
PublikacjaPositioning, Navigation, and Timing (PNT) information play a vital role in everyday life of common persons. People greatly rely on Global Navigation Satellite System (GNSS)-enabled applications for navigation to reach their desired destination. However, GNSS navigation performance is highly degraded in urban environments due to the high probability of signal interruption, multipath (MP), and/or non-line-of-sight (NLOS) signal...
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ZASTOSOWANIE FILTRACJI CZĄSTECZKOWEJ DO ESTYMACJI POŁOŻENIA W SYSTEMIE LOKALIZACYJNYM UWB
PublikacjaNiniejszy artykuł dotyczy kwestii poprawy dokładności estymacji położenia w systemie lokalizacji wewnątrzbudynkowej, bazującym na radiowych pomiarach odległości realizowanych przez modemy UWB. Proponuje się zastosowanie metody filtracji cząsteczkowej do zmniejszenia błędu wyznaczania pozycji obiektu przy braku bezpośredniej widoczności ze stacją referencyjną. W artykule opisano algorytm filtru cząsteczkowego, jego przykładową implementację...
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How much is Impact Factor worth?
PublikacjaThe purpose of this work is to present an aspect of counting citations, which is correlated to the Impact Factor, very important for journals in scientific communication, and provides information about the position of a scientific journal in a particular research area. Sometimes citations don’t count in a research output, e.g. if an article is published in a predatory journal. Those journals ...
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Tool Wear Prediction in Single-Sided Lapping Process
PublikacjaSingle-sided lapping is one of the most effective planarization technologies. The process has relatively complex kinematics and it is determined by a number of inputs parameters. It has been noted that prediction of the tool wear during the process is critical for product quality control. To determine the profile wear of the lapping plate, a computer model which simulates abrasive grains trajectories was developed in MATLAB. Moreover,...
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Reliable method of assessing fracture properties of asymmetric bonded joints
PublikacjaTwo methods of assessing fracture properties of adhesive joints were studied. Two wedge tests: with continuous deflection and with force measurements were compared. Asymmetric geometry of the bonded joint was considered, i.e. two different plates of aluminium alloys: Al-Cu and Al-Mg, were bonded with epoxy DGEBA adhesive. The analytical model is shown to estimate the values of fracture properties: crack position and critical fracture...
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Modelling of in-plane wave propagation in a plate using spectral element method and Kane-Mindlin theory with application to damage detection
PublikacjaThis paper presents results of experimental and numerical analyses of in-plane waves propagatingin a 5 mm-thick steel plate in the frequency range of 120-300 kHz. For such a thickness/frequency ratio,extensional waves reveal dispersive character. To model in-plane wave propagation taking into account thethickness-stretch effect, a novel 2D spectral element, based on the Kane-Mindlin theory, was formulated. Anapplication of in-plane...
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Intelligent equalizer solution employing music genre and the room characteristics analysis
PublikacjaThe paper presents an intelligent equalizer solution based on room acoustic conditions and music genre analysis. A series of acoustic characteristic measurements are performed for checking the concept proposed. White noise (reference signal) and audio excerpts belonging to six music genres are utilized as excitation signals in measurements. This results in registration of frequency responses of rooms and reverberation times. Signals...
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Selected properties and parameters of radio channel impulse response estimation in ISM 2.4 GHz band
PublikacjaThe article presents experimental research indicating that the impulse response of the communication channel, determined in practice, are not of an universal character, but only represent its approximate value for the frequency on which this measurement was made. Phases for each of the replicas of the measurement signal were determined during the analysis of the received signals in the baseband. Phase changes of individual replicas...
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Dynamic Positioning System with Vectorial Backstepping Controller
PublikacjaThe problem of synthesis a dynamic positioning system for low frequency model of surface vessel was considered in this paper. The recursive vectorial backstepping control design was used to keep a fixed position and heading in presence of wave disturbances. The passive observer was introduced to smooth the measurements and to estimate the velocities needed for the control algorithm. Some parameters of observer were optimized off-line...
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Functionalized azobenzocrown ethers as sensor materials—The synthesis and ion binding properties
PublikacjaNew 13- and 16-membered azobenzocrown ethers with aromatic amino, amide, ether–ester or ether–amide residue in para position to an azo moiety were obtained. Acid–base properties and ion binding ability of the colored compounds were studied by spectroscopic methods: UV–vis, fluorimetry and 1H NMR spectroscopy. Selected azobenzocrowns were tested as ionophores in ion-selective membrane electrodes (ISEs) – classic and miniature all...
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A comprehensive approach to double inverted pendulum modelling
PublikacjaThe problem of mathematical modelling and indication of properties of a DIP has been investigated in this paper. The aim of this work is to aggregate the knowledge on a DIP modelling using the Euler-Lagrange formalism in the presence of external forces and friction. To indicate the main properties important for simulation, model parameters identification and control system synthesis, analytical and numerical tools have been used....
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Autonomous Vehicle Navigation in Dense Urban Area in Global Positioning Context
PublikacjaAutonoumous vehicle services are likely to be adopted in dense urban area. Some research prove that autonomous transport might be capable of improving the transport needs of few times and as a consequence sustainability, congestion and safety may be improved. The world, hopefully is close to a transport revolution age. These studies are perhaps exaggerated, over-optimistic and far fro fully operational. The paper takes into account...
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Komputerowo wspomagana analiza elastycznych siłowników elektrostatycznych dla potrzeb implementacji w systemach mechatroniki
PublikacjaPrzeprowadzone badania naukowe rozpoczęto od szczegółowej analizy układu mechatronicznego dłoni robotycznych, powstałych na przestrzeni ostatnich 40 lat, w celu dokładnego rozpoznania ich głównych wymogów konstrukcyjnych i ograniczeń systemowych. Z uwagi na brak dostępnych narzędzi do symulacji omawianych siłowników, w rozprawie opracowano uniwersalne narzędzie – program do analizy numerycznej. U jego podstawy założono wykorzystanie...
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Optymalizacja doboru prawa konstytutywnego membrany o strukturze plecionej
PublikacjaCelem niniejszej dysertacji jest opracowanie zagadnienia optymalizacyjnego pozwalającego dobrać model konstytutywny opisujący mechaniczne zachowanie membrany technicznej. Do analizy wybrano membrany plecione, stosowane w medycynie, tzw. siatki chirurgiczne. W celu wykonania identyfikacji praw konstytutywnych, wykonano dwuosiowe rozciąganie próbek materiałów, otrzymując wskazanie na nieliniowe anizotropowe zachowanie materiałów....
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Virtual Whiteboard: A gesture-controlled pen-free tool emulating school whiteboard
PublikacjaIn the paper the so-called Virtual Whiteboard is presented which may be an alternative solution for modern electronic whiteboards based on electronic pens and sensors. The presented tool enables the user to write, draw and handle whiteboard contents using his/her hands only. An additional equipment such as infrared diodes, infrared cameras or cyber gloves is not needed. The user's interaction with the Virtual Whiteboard computer...
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<i>N,N</i>'-diphenylthiourea acetone monosolvate
PublikacjaIn the title compound, C13H12N2S·C3H6O, the phenyl rings of the thiourea molecule are in syn and anti positions in relation to the C=S bond. Two molecules are connected by N-HS=C hydrogen bonds into a centrosymmetric dimer. An additional N-HO=C hydrogen bond to the acetone solvent molecule and some weak C-H interactions reinforce the crystal structure.
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Effect of Time Varying Measurement Conditions on Antenna Pattern in Near Field Measurement and Its Correction Procedure
PublikacjaAuthors present the procedure of taking into account the changes of electrical parameters of setup due to the time drift of temperature during the procedure of near field measurement. It is proposed to make additional measurements in determined positions of probe are next used the results to introduce corrections terms in measured data. Such approach was verified practically in experimental near field measurement system.
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The influence of the development of private air communication on the architecture and urban planning of the 21st century
PublikacjaIn the first part, the article describes the stages of the development of gyroplanes and the influence of wartime policy on the interest in light aircraft. Also presented are links and the possibilities of using gyroplanes in various sectors of the economy. The authors, based on source texts, present the current position of the aviation industry in the Polish economy and attempt to diagnose its development capabilities. As a result,...
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Using Alpha-beta filtration for robustness improvement of a quadrocopter positioning system
PublikacjaQuadrocopter is an unmanned aerial vehicle (UAV) platform. The position of the robot is determined based on readings from an accelerometer and a gyroscope, but the measurement signals contain broadband noise. This article describes a solution for filtering out the noise based on an Alpha – beta filter. It also presents the methodology of designing and implementing such a filter for noise cancellation in measurement signals from...
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Myths and facts about women aged 50+
PublikacjaThis study attempts to confront the three stereotypes attributed to women aged 50+ in Poland: the one related to women being interested in retiring as early as possible, the other related to the lack of educational activity and reluctance to acquire new knowledge and skills, and the third related to the image of a grandmother focused on looking after her grandchildren. The author’s aim is to present rational arguments in favour...
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The Attitude of Polish Entrepreneurs to the Fact of Staging the Mega Sport Event - the Case of Pomeranian SMEs Towards Euro 2012
PublikacjaIn the course of preparations to the 2012 European Football Championship (Euro 2012) many doubts have arisen as to the actual cost-benefit balance affecting the hosting country. The event is accompanied by intense promotion of the agglomeration and the region, especially abroad. In effect, one can anticipate the competitive position of both the region and the businesses operating there to improve. The investigation whether the...
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GPR simulations for diagnostics of a reinforced concrete beam
PublikacjaThe most popular technique for modelling of an electromagnetic field, the finite difference time domain (FDTD) method, has recently become a popular technique as an interpretation tool for ground penetrating radar (GPR) measurements. The aim of this study is to detect the size and the position of damage in a reinforced concrete beam using GPR maps. Numerical simulations were carried out using the finite differ-ence time domain...
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Disturbances of magnetic field in surrounding of mobile, metalic plate
PublikacjaThe uniform magnetic field of the Earth in the surrounding of a mobile, metalic object undergoes deformation by eddy currents. The influence of the moving conducting object on total magnetic field of the Earth depends on the object's shape, position and speed of the changes relative to the magnetic field's vector of the Earth as well as the electric conductivity and the relative magnetic permeability of the material. The disturbances...
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FEX a Fingers Extending eXoskeleton for Rehabilitation and Regaining Mobility
PublikacjaThis paper presents the design process of an exoskeleton for executing human fingers’ extension movement for the rehabilitation procedures and as an active orthosis purposes. The Fingers Extending eXoskeleton (FEX) is a serial, under-actuated mechanism capable of executing fingers’ extension. The proposed solution is easily adaptable to any finger length or position of the joints. FEX is based on the state-of-art FingerSpine serial...