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Wyniki wyszukiwania dla: in vitro metabolizm
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Electrophoretic deposition and characterization of composite chitosan/Eudragit E 100 or poly(4-vinylpyridine)/mesoporous bioactive glass nanoparticles coatings on pre-treated titanium for implant applications
PublikacjaTitanium implants are surface-modified to achieve bioactivity and often antibacterial properties. Such surface coatings may increase corrosion degradation and be weakly attached to the substrate. In the present research, biodegradable composite coatings, investigated so far as smart environment-sensitive, slowly releasing silver to the implant neighborhood, were produced as a combination of chitosan (CS) with Eudragit E 100 (EE100)...
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Obliczanie nośności i osiadania pali pojedynczych na podstawie badań sondą Statyczną CPT.
PublikacjaOmówiono metodę obliczania nośności i osiadania pali z uwzględnieniem bezpośredniego wykorzystania wyników badań sondą statyczną CPT. Dla oceny krzywej osiadania zastosowano funkcje transformacyjne. Przedstawiono analizę wykorzystując wyniki próbnych obciążeń statycznych dla 94 pali Vibro-Fundex. Zaproponowane korelacje zostały zweryfikowane przy wykorzystaniu procedury weryfikacji hipotez statystycznych.
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State of the art in sample preparation for human breast milk metabolomics—merits and limitations
PublikacjaHuman breast milk (HBM) contains metabolites that are diverse in chemical structure and concentration. These metabolites range from high-abundance to low-abundance compounds and from polar to nonpolar. This complex nature of HBM makes HBM samples difficult to analyze, especially in global metabolomic studies for the determination and characterization of complete sets of metabolites. In this review, the state of the art in sample...
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Structural factors affecting affinity of cytotoxic oxathiole-fused chalcones toward tubulin
PublikacjaSynthesis, in vitro cytotoxic activity, and interaction with tubulin of (E)-1-(6-alkoxybenzo[d][1,3]oxathiol- 5-yl)-3-phenylprop-2-en-1-one derivatives (2) are described. Some of the compounds demonstrated cytotoxic activity at submicromolar concentrations, and the activity could be related to interaction with tubulin at the colchicine binding site. Interaction of selected derivatives with tubulinwas evaluated using molecular modeling,...
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Antimicrobial Activity of Chimera Peptides Composed of Human Neutrophil Peptide 1 (HNP-1) Truncated Analogues and Bovine Lactoferrampin
PublikacjaThree chimera peptides composed of bovine lactoferrampin and the analogue of truncated human neutrophil peptide 1 were synthesized by the solid-phase method. In two compounds peptide chains were connected via isopeptide bond, whereas in the third one disulfide bridge served as a linker. All three chimeras displayed significantly higher antimicrobial activity than the constituent peptides as well as their equimolar mixtures. The...
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Badania bioaktywności z wykorzystaniem komórek kościotwórczych na tytanie pokrytym chitozanem = Bioactivity studies using osteogenic cells on titanium coated with chitosan
PublikacjaChitosan is a natural polymer from the group of polysaccharides, which has found wide application in biomedical applications to induce bioactivity of implant. The studies described were carried out test imposition of chitosan membranes with varying degrees of deacetylation on the surface of titanium, and then check the bioactivity of the material in vitro, using osteogenic cells MC3T3-E1. Titanium surface before imposition of...
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Molecular Umbrella as A Nanocarrier for Antifungals
PublikacjaA molecular umbrella composed of two O‐sulfated cholic acid residues was applied for the construction of conjugates with cispentacin, containing a “trimethyl lock” (TML) or o‐dithiobenzylcarbamoyl moiety as a cleavable linker. Three out of five conjugates demonstrated antifungal in vitro activity against C. albicans and C. glabrata but not against C. krusei, with MIC90 values in the 0.22–0.99 mM range and were not hemolytic. Antifungal...
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Studies of the effects of antifungal cationic derivatives of amphotericin B on human erythrocytes.
PublikacjaBadano nową grupę kationowych pochodnych amfoterycyny B pod kątem zależności pomiędzy ich zdolnością do asocjacji i selektywną toksycznością. We wszystkich przypadkach stosowano amfoterycynę B jako związek odniesienia. Jako miarę efektu toksycznego in vitro badanych związków stosowano wypływ wewnątrzkomórkowego potasu oraz hemolizę. Miarą aktywności przeciwgrzybowej był MIC i utrata potasu wewnatrzkomórkowego. Do oceny stopnia...
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Smart acoustic band structures
PublikacjaSmart acoustic band structures exhibit very interesting and non-standard physical properties due to the periodic nature of their certain characteristic on different scale levels. They manifest mostly in their frequency spectra as socalled frequency band-gaps or stop-bands, what has a great impact on the behaviour of these structures in relation to the propagation of vibro-acoustic signals that can be transmitted through the structures...
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The occurence and diagnosis of biomarkers of ethyl alcohol consumption
PublikacjaEthyl alcohol is a legal and a widely available psychoactive drug. However, its excessive consumption causes addiction. This leads to aggressive behaviors, family battery, difficulties in interpersonal relations, legal offences, suicides, car accidents and deterioration in labor productivity, what causes financial problems. Despite many social actions against alcohol consumption, this problem is still unresolved. Therefore, fast...
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Białka prokariotycznego systemu MMR: rola oraz interakcje
PublikacjaUszkodzenia komórkowego DNA w postaci błędnie sparowanych lub niesparowanych zasad azotowych są wynikiem niewłaściwie zachodzących procesów metabolizmu DNA, takich jak replikacja, rekombinacja oraz naprawa DNA. Utrwalenie tego rodzaju zmian prowadzi do powstania mutacji. System MMR (ang. DNA mismatch repair) usuwa te uszkodzenia przyczyniając się do zwiększenia wierności replikacji DNA oraz utrzymania stabilności genomu komórki....
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Fast-SEC coupled to ICP-MS for selected metal determination and its stability over time in polish wine
PublikacjaMetal ions contribute to the wine browning (as reaction catalysts), turbidity (in complexes), and astringency (due to inter- action with tannins). Being aware that bioavailability and metabolism of metal ions in the human body are strictly related with their concentration and the form they occur it is important to monitor not only the total content of metals but also their speciation. Thus, we can obtain more information about...
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Determination of the bearing capacity of pile foundations based on CPT test results
PublikacjaAnalityczne określanie pełnej krzywej obciążenie - osiadanie na podstawie parametrów geotechnicznych wciąż stanowi bardzo trudne zadanie naukowe i inżynierskie. W pracy przedstawiono metodę bezpośredniego wykorzystania oporów na stożku sondy statycznej do określania pełnej krzywej osiadania dla pali Vibro-Fundex. W sumie jako materiał weryfikacyjny wykorzystano 94 próbne obciążenia statyczne pali.
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Bioactive Ingredients with Health-Promoting Properties of Strawberry Fruit (Fragaria x ananassa Duchesne)
PublikacjaStrawberries (Fragaria x ananassa Duchesne) belong to the berry group and are characterized primarily by delightful sensory properties. Due to their chemical composition, these fruits are a rich source of bioactive compounds that can modify the metabolic and physiological functions of the body. The aim of this work is to present the current state of research on bioactive ingredients found in these fruits in the context of their...
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Prime-Boost Vaccination with Toxoplasma Lysate Antigen, but Not with a Mixture of Recombinant Protein Antigens, Leads to Reduction of Brain Cyst Formation in BALB/c Mice
PublikacjaIntroduction Infection with the ubiquitous parasite Toxoplasma gondii is a threat for immunocompro- mised patients and pregnant women and effective immune-prophylaxis is still lacking. Methods Here we tested a mixture of recombinant T . gondii antigens expressed in different develop- mental stages, i.e., SAG1, MAG1 and GRA7 (SMG), and a lysate derived from T . gondii tachyzoites (TLA) for prophylactic vaccination against cyst formation....
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Process of convergence in EU
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Process Engineering in Circular Economy
Kursy OnlineKurs jest przeznaczony dla doktorantów szkoły doktorskiej w dyscyplnach: inżynieria lądowa i transport (SzD), III stopnia, stacjonarne inżynieria środowiska, górnictwo i energetyka (SzD), III stopnia, stacjonarne The course is addressed to PhD students of the doctoral school in disciplines: civil engineering and transport environmental engineering, mining and power engineering Course type: lecture Total hours of...
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Change Detection in Signals 2023
Kursy OnlineChange Detection in Signals - files for students.
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Spectroscopy Methods in Nanotechnology 2023
Kursy OnlineCourse for 2nd degree Students of Nanotechnology, specialization Nanostructures and computer simulations in materials science, sem. 2. The aim of the course is to discuss the basic theoretical and practical issues of spectroscopy and presentation of the various types of spectroscopic methods and ways to interpret spectra, with particular attention paid to the possibility of their use in the study of nanostructured systems.
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[ZiJ] Empirical research in Management
Kursy OnlineDyscyplina: nauki o zarządzaniu i jakości Zajęcia obowiązkowe dla doktorantów I i II roku Prowadzący: dr inż. Wioleta Kucharska Liczba godzin: 30 Forma zajęć: laboratoria Discipline: management and quality Obligatory course for 1st and 2nd-year PhD students Academic teacher: dr inż. Wioleta Kucharska Total hours of training: 30 teaching hours Course type: laboratories
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Passive Methods in Heat Transport
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Law and Ethics in Science
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ICT in Management, Spring 2022
Kursy Online„ ICT w zarządzaniu licencjami” dla studentów studiów z zarządzania, edycja 2022 „ ICT w sklepie ” dla studentów BiM edycja 2022
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IT project management in business
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Corrosion in Theory and Practice
Kursy Onlinestopień: II, semestr: II
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Spectroscopy Methods in Nanotechnology 2022
Kursy OnlineCourse for 2nd degree Students of Nanotechnology, specialization Nanostructures and computer simulations in materials science, sem. 2. The aim of the course is to discuss the basic theoretical and practical issues of spectroscopy and presentation of the various types of spectroscopic methods and ways to interpret spectra, with particular attention paid to the possibility of their use in the study of nanostructured systems.
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Forecasting and optimalization in logistics
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Management in space industry WiMiO
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Surrogate methods in system engineering
Kursy Online{mlang pl} Dyscyplina: Automatyka, Elektronika i Elektrotechnika Zajęcia fakultatywne dla doktorantów II roku Prowadzący: dr hab. inż. Adrian Bekasiewicz Liczba godzin: 15 h Forma zajęć: wykład {mlang} {mlang en} Discipline: control, electronic and electrical engineering Facultative course for 2nd year PhD students Academic teacher: dr hab. inż. Adrian Bekasiewicz Total hours of training: 15 teaching hours Course...
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[EiF] Empirical research in Economics
Kursy Online{mlang pl} Dyscyplina: EiF Zajęcia obowiązkowe dla doktorantów I roku Prowadzący: A. Parteka / J. Wolszczak - Derlacz, F. Venturini Liczba godzin: 30 Forma zajęć: laboratoria {mlang} {mlang en} Discipline: EiF Obligatory course for 1st-year PhD students Academic teacher: A. Parteka / J. Wolszczak - Derlacz, F. Venturini Total hours of training: 30 teaching hours Course type: Laboratories {mlang}
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Ecological solutions in contemporary architecture
Kursy OnlineThis lecture aims to equip you with a comprehensive understanding of ecological architecture and inspire you to integrate these principles into your future projects.
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HR management - Bachelor in management
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Process engineering in circular economy
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Advances in Functional Materials 2024
Kursy OnlineOur summer school on Advances in Functional Materials 2024 aims to bring together young scientists (Ph.D. and MSc students) with specialists in materials engineering. You will be able to follow our lectures, and laboratory classes so you can practice what you have learned. This course consists of 40 hours of direct contact classes - 30 hours of lectures and 10 hours of laboratory classes delivered by our specialists from the Advanced...
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ICT in Management - Spring 2024
Kursy OnlineICT in Management course for Bachelor in Management students (Spring 2024 edition)
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2024 Microscopy in Environmental Monitoring
Kursy OnlineThe online repository will be used to teach students by presenting them lectures about variable aspects of microscopy techniques used in environmental monitoring.
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Daylight in Architecture 2022/23
Kursy OnlineTutor: Professor Claudia Naves David Amorim (University of Brasilia) Project: 60 h (lectures + online platform + individual consultations) With a support of e-platform NLITED educational content; http://lms.nlited.eu/, Students will become familiar with the different methods of daylight assessment within the built environment. Innovative daylight design is understood as a better user-centred and energy-efficient design strategy. The...
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Spectroscopy Methods in Nanotechnology 2024
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Process engineering in circular economy
Kursy OnlineDefinition and principles of the circular economy (CE). The transition from a linear model to a circular model. Business models for the CE. Circular design and innovation. CE assessment carbon footprint, life cycle assessment. Case studies of the cities implementing the CE concept. CE policy and legislation (EU and Poland). Wastewater treatment plants as an element of the CE. Energy and nutrient recovery technologies in wastewater...
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Recent advances in transcription regulation
Kursy OnlineRecent advances in transcription regulation
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Modern Techniques in Control Theory
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Modelling in machine design (PG_00057377)
Kursy Onlinegoal of the subject is to show how simple enginnering models reflect the reality and how contemporary FEM calulations can illustrate the operation of machine elements
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L23_24 Artificial Intelligence in Healthcare
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Adipokine and cytokine levels in patients with adrenocortical cancer, subclinical Cushing's syndrome and healthy controls
PublikacjaIntroduction In recent years researchers have focused at hormonal activity in Cushing’s syndrome (CS) in connection with metabolic disorders and the role of adipokines and cytokines secreted by the adipose tissue. The aim of the study was to investigate levels of adipokines and cytokines in patients with: subclinical CS (SCS) – in relation to hormonal parameters of hypercortisolemia, and, adrenocortical cancer (ACC). Materials...
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Generation of biodiesel and glycerol from waste of rice industries in Brazil
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Inhibition of amyloid fibril formation of hen egg white lysozyme by trimethylamine N-oxide at low pH
PublikacjaIn vitro inhibition of the formation of fibrous aggregates of proteins (amyloids) has gained increasing attention due to the number of diseases associated with protein misfolding and fibrillation. An interesting group of compounds for which pronounced activity against this phenomenon can be expected consists of low molecular weight substances (osmolytes) which have the ability to change protein stability. Here we investigate the...
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Inhibitors of amino acids biosynthesis as antifungal agents
PublikacjaFungal microorganisms, including the human pathogenic yeast and filamentous fungi, are able to synthesize all proteinogenic amino acids, including nine that are essential for humans. A number of enzymes catalyzing particular steps of human-essential amino acid biosynthesis are fungi specific. Numerous studies have shown that auxotrophic mutants of human pathogenic fungi impaired in biosynthesis of particular amino acids exhibit...
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Bioactive core material for porous load-bearing implants
PublikacjaSo far state of knowledge on biodegradable materials is reviewed. Among a variety of investigated materials, those composed of polymers and ceramics may be considered as only candidates for a core material in porous titanium alloy. The collagen and chitosan among natural polymers, polyhydroxy acids among synthetic polymers, and hydroxyapatite and tricalcium phosphate among ceramics are proposed for further research. Three essential...
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Influence of different cultivation systems on bioactivity of asparagus
PublikacjaEvaluation of functional and bioactive compounds of Asparagus officinalis L. growing in conventional and organic greenhouse and conventional open –field farming was the aim of this research. Polyphenols in cladodes grown conventionally were higher than organic. Flavonoids and carotenoids were the highest in cladodes in open field. Organic spears were richer in total phenolics (+6.9% and +19.1%) and flavonoids (+4.7% and 16.8%)...
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Investigation of an elutable N-propylphosphonic acid chitosan derivative composition with a chitosan matrix prepared from carbonic acid solution
PublikacjaPorous chitosan composites using CO2 dissolution procedure and including water soluble N-propylphosphonic chitosan derivative (p-CHI) were obtained and characterized. In contrast to the control material, composites containing modified chitosan distinguished by a rapid moisture absorption and good adhesion to the skin. The FTIR analysis confirmed the presence of propylphosphonic group in the structure of the polymer. The porosity...