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Approaches Towards Better Immunosuppressive Agents
PublikacjaSeveral classes of compounds are applied in clinics due to their immunosuppressive properties in transplantology and the treatment of autoimmune diseases. Derivatives of mycophe-nolic acid, corticosteroids and chemotherapeutics bearing heterocyclic moieties like methotrexate, azathioprine, mizoribine, and ruxolitinib are active substances with investigated mechanisms of action. However, improved synthetic approaches of known drugs...
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Equivalent Single Layer Models in Free Vibration Analysis of Laminated Multi-Layered Plates
PublikacjaThe performance of selected equivalent single-layer (ESL) models is evaluated within several classical benchmark tests for small amplitude free vibration analysis of multi-layered plates. The authors elaborated their own Finite Element software based on the first-order shear deformation (FOSD) theory with some modifications incorporated including a correction of the transverse shear stiffness and an application of zigzag type functions....
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Amino Acid Based Antimicrobial Agents – Synthesis and Properties
PublikacjaStructures of several dozen of known antibacterial, antifungal or antiprotozoal agents are based on the amino acid scaffold. In most of them, the amino acid skeleton is of a crucial importance for their antimicrobial activity, since very often they are structural analogs of amino acid intermediates of different microbial biosynthetic pathways. Particularly, some aminophosphonate or aminoboronate analogs of protein amino acids are...
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Contemporary Architectural Design in the Context of Historic Remains: The Case of the Old City of Gdańsk
PublikacjaThis article presents several examples of modern developments designed to preserve and coexist with fragments of historic brick buildings. These building projects each faced a similar task; to save and display the historical urban fabric, but they differed significantly in how they chose to achieve that goal. Not all of the projects presented in this study meet the requirements of the Venice Charter equally well. In this field,...
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NONLINEAR VIBRATION ANALYSIS OF BEAM AND PLATE WITH CLOSED CRACK: A REVIEW
PublikacjaThe effect of nonlinearity is high sensitivity in damage detection, especially for closed cracks and delamination. This review illustrates the results of several researchers dealing with nonlinear effects caused by the closure of cracks in the structure, i.e., beam and plate structures. Early detection of damage is an important aspect for the structure and, therefore, continuous progress is being made in developing new and effective...
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Bunker demolition located in a conservation protection zone in the light of technical, national defense, functional-utility and economic conditions
PublikacjaThe paper presents a description of the technical condition of the Bunker building located at the port quay, which has been out of use for several decades. The direct reason for the cessation of exploitation was the deletion of Bunker from the Civil Defense records. The paper contains a detailed analysis of the Bunker's technical condition, also taking into account the national defense, functional and utility aspects and the issues...
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In silico design of telomerase inhibitors.
PublikacjaTelomerase is a reverse transcriptase enzyme involved in DNA synthesis at the end of linear chromosomes. Unlike in most other cells, telomerase is reactivated most cancerous cells and, therefore, has become a promising new anticancer target. Despite extensive research, direct telomerase inhibitors have yet not been introduced to the clinics because of the complexity of this enzyme. Structures of this protein from simple organisms...
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Dynamic mechanical properties and flexing fatigue resistance of tire sidewall rubber as function of waste tire rubber reclaiming degree
PublikacjaA stepwise downsizing method of gel particles in reclaimed rubber to a micro-nano scale and its excellent dynamic performance in tire sidewall were introduced by this work. The results showed that the size of gel particles decreased from several micrometers to micro-nanometers with the increase of reclaiming degree, accompanied by reduced molecular weight and widened molecular weight distribution of sol fraction. The addition of...
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Traffic Noise Analysis Applied to Automatic Vehicle Counting and Classification
PublikacjaProblems related to determining traffic noise characteristics are discussed in the context of automatic dynamic noise analysis based on noise level measurements and traffic prediction models. The obtained analytical results provide the second goal of the study, namely automatic vehicle counting and classification. Several traffic prediction models are presented and compared to the results of in-situ noise level measurements. Synchronized...
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Sensitivity analysis in design process of sandwich U-shaped composite footbridge
PublikacjaThe structure of the sandwich composite footbridge of a 14 metre span length and U-shaped cross-section was analysed. Sensitivity analysis was performed to support the design process of this innovative object. Linear discrete sensitivity analysis was performed by means of finite element method. The influence of vari-ation of several design variables i.e. thicknesses of inner and outer laminates on the mid-span deflection, as-sumed...
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Selected studies of flow maldistribution in a minichannel plate heat exchanger
PublikacjaAnalysis of the state of-the-art in research of minichannel heat exchangers, especially on the topic of flow maldistribution in multiple channels, has been accomplished. Studies on minichannel plate heat exchanger with 51 parallel minichannels with four hydraulic diameters, i.e., 461 μm, 574 μm, 667 μm, and 750 μm have been presented. Flow at the instance of filling the microchannel with water at low flow rates has been visualized. The...
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Technology adoption review for ageing well: analysis of technical solutions
PublikacjaWhile several technological solutions are available for older adults to improve their wellbeing and quality of life, little is known about the gaps between the needs, provided solutions, and their adoption from a more pragmatic perspective. This paper reports on reviewing existing technological solutions for older adults, which span the work life, life in the community, and wellbeing at home. We analyzed 50 different solutions...
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Emotion monitoring system for drivers
PublikacjaThis article describes a new approach to the issue of building a driver monitoring system. Actual systems focus, for example, on tracking eyelid and eyebrow movements that result from fatigue. We propose a different approach based on monitoring the state of emotions. Such a system assumes that by using the emotion model based on our own concept, referred to as the reverse Plutchik’s paraboloid of emotions, the recognition of emotions...
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Systems of Public Higher Education in Poland and Germany. Evidence from Institution Level Data
PublikacjaThe chapter presents a comparative analysis of public higher education systems (HES) in Germany and Poland. Instead of limiting our study to macro indicators such as gross expenditure on higher education or R&D as per cent of GDP, we draw on the evidence based on micro data especially collected for this study and concerning individual higher education institutions (HEIs). Comparative analysis is based on a sample of 71 public...
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Multi-objective optimization of expensive electromagnetic simulation models
PublikacjaVast majority of practical engineering design problems require simultaneous handling of several criteria. For the sake of simplicity and through a priori preference articulation one can turn many design tasks into single-objective problems that can be handled using conventional numerical optimization routines. However, in some situations, acquiring comprehensive knowledge about the system at hand, in particular, about possible...
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Enriching the Context: Methods of Improving the Non-contextual Assessment of Sentence Credibility
PublikacjaThis paper presents several methods of automatic context enrichment of sentences that need to be evaluated, tagged or fact-checked by human judges. We have created a corpus of medical Web articles. Sentences from this corpus have been fact-checked by medical experts in two modes: contextually (reading the entire article and evaluating sentence by sentence) and without context (evaluating sentences from all articles in random order)....
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Genetic and biochemical characterization of yeasts isolated from Antarctic soil samples
PublikacjaThe Polish Arctowski Station is situated in the maritime Antarctic on the western shore ot' Admiralty Bay and encompasses terrestrial habitats which are not perma-nently covered by ice, in contrast to morę than 90% of the island's surface area. Over the past several decades, stud-ies exploring the soils of those habitats have revealed a considerable diversity of bacteria, filamentous fungi, and, to a lesser extent, yeasts; however,...
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Modelling of in-plane wave propagation in a plate using spectral element method and Kane-Mindlin theory with application to damage detection
PublikacjaThis paper presents results of experimental and numerical analyses of in-plane waves propagatingin a 5 mm-thick steel plate in the frequency range of 120-300 kHz. For such a thickness/frequency ratio,extensional waves reveal dispersive character. To model in-plane wave propagation taking into account thethickness-stretch effect, a novel 2D spectral element, based on the Kane-Mindlin theory, was formulated. Anapplication of in-plane...
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Recognizing emotions on the basis of keystroke dynamics
PublikacjaThe article describes a research on recognizing emotional states on the basis of keystroke dynamics. An overview of various studies and applications of emotion recognition based on data coming from keyboard is presented. Then, the idea of an experiment is presented, i.e. the way of collecting and labeling training data, extracting features and finally training classifiers. Different classification approaches are proposed to be...
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Inequivalence of entanglement, steering, and Bell nonlocality for general measurements
PublikacjaEinstein-Podolsky-Rosen steering is a form of inseparability in quantum theory commonly acknowledged to be intermediate between entanglement and Bell nonlocality. However, this statement has so far only been proven for a restricted class of measurements, namely, projective measurements. Here we prove that entanglement, one-way steering, two-way steering, and nonlocality are genuinely different considering general measurements,...
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1,3-alternate calix[4]arene-bonded silica stationary phases. Effect of calixarene skeleton substituents on the retention mechanism and column selectivity
PublikacjaFour novel 1,3-alternate calix[4]arene-bonded silica gel stationary phases possessing different aromatic and aliphatic substituents at the upper rim (CalixNph, CalixBph, CalixHex and CalixDdc) were prepared and structurally characterized. The comparison and selectivity of these phases was done by using alkylbenzenes, fatty acid p-bromophenacyl esters, aromatic positional isomers and polynuclear aromatic hydrocarbons as analytes....
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The “autumn effect” in the gold market—does it contradict the Adaptive Market Hypothesis?
PublikacjaThe present study aims to verify the autumn effect in the gold market, first presented 10 years ago by Dirk Baur in the paper “The autumn effect of gold” and to investigate the calendar effects occurring for other precious metals. This empirical research is presented in a way to place the results obtained in the context of the Efficient Market Hypothesis (EMH) and the more current Adaptive Market Hypothesis (AMH). The study was...
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Methods of Incomplete and Uncertain Knowledge Acquisition in the Knowledge Processing Environemnt
PublikacjaThe authors in this paper present a concept of the environment to acquire and process knowledge about information technology. This solution is part of a project of which the objective is to build a system for the evaluation of IT tools and methodologies. Knowledge within this domain is always either uncertain or incomplete. Therefore, the authors focused on designing a dedicated algorithm for its acquisition and processing. One...
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An integrated framework for security protocol analysis
PublikacjaAssurance of security protocols needs particular attention. Flaws in a protocol can devastate security of the applications that rely on it. Analysis of the protocols is difficult and it is recommended that formal methods are employed to provide for higher levels of assurance. However, the formal methods can cover only a part of the scope of the problem. It is important that the formal models are valid representations of the protocol...
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Detection of ferromagnetic objects in local magnetic anomaly of the Baltic Sea
PublikacjaIn geological researches several kinds of methods are applied to discovering the natural resources. Planes, helicopters and UAVs (UnmAnned Vehicle) are used in researches in large areas. The gravity, electromagnetic and magnetic methods, which are used in geological researches, are presented in this paper. The special attention was paid to magnetic systems installed on mobile platforms. The magnetic field of the Earth obtained...
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Mixed conductivity in tungstenite-phosphate glasses containing alkali metal ions
PublikacjaThe conductivity of glasses in the 50WO3-(50-x)P2O5-xA2O (A = Na, K, Cs) system has been investigated as a function of composition. It is shown that in tungstenite-phosphate glasses containing different alkali metal ions the conductivity decreases with an increase in the alkali metal ion content. A decrease in conductivity is larger for heavier ions and reaches more than seven orders of magnitude in the case of glass containing...
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Measuring Pulse Rate with a Webcam
PublikacjaIn this paper a simple method of measuring the pulse rate is presented. Elaborated algorithm allows for efficient pulse rate registration directly from face images captured from a webcam. The desired signal is obtained by proper channel selection and principal component analysis. To determine the accuracy of the method an ECG signal is collected together with a video recordings. The effectiveness of the algorithm is considered...
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Testing Watermark Robustness against Application of Audio Restoration Algorithms
PublikacjaThe purpose of this study was to test to what extent watermarks embedded in distorted audio signals are immune to audio restoration algorithm performing. Several restoration routines such as noise reduction, spectrum expansion, clipping or clicks reduction were applied in the online website system. The online service was extended with some copyright protection mechanisms proposed by the authors. They contain low-level music features...
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Multiacces quantum communication and product higher rank numerical range
PublikacjaIn the present paper we initiate the study of the product higher rank numerical range. The latter, being a variant of the higher rank numerical range, is a natural tool for study- ing a construction of quantum error correction codes for multiple access channels. We review properties of this set and relate it to other numerical ranges, which were recently introduced in the literature. Further, the concept is applied to the construction...
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Heat transfer in plate heat exchanger channels: experimental validation of selected correlation equations
PublikacjaThis study is focused on experimental investigation of selected type of brazed plate heat exchanger. The Wilson approach was applied in order to estimate heat transfer coefficients for the PHEx passages. The main aim of the paper was to experimentally check ability of several correlations published in the literature to predict heat transfer coefficients by comparison experimentally obtained data with appropriate predictions. The...
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Content-Based Approach to Automatic Recommendation of Music
PublikacjaThis paper presents a content-based approach to music recommendation. For this purpose, a database which contains more than 50000 music excerpts acquired from public repositories was built. Datasets contain tracks of distinct performers within several music genres. All music pieces were converted to mp3 format and then parameterized based on MPEG-7, mel-cepstral and time-related dedicated parameters. All feature vectors are stored...
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Ion Chromatography in Environmental Analysis of Selected Organic Acids
PublikacjaLow molecular mass carboxylic acids (LCAs) occur in many environmental compartments dueto natural processes and human activity. When volatile and nonvolatile acids are to be monitored then liquidchromatography, including ion chromatography seems a method of choice. At high pH the acids are inionized form and can be separated as carboxylats by means of anion exchange chromatography. LCAs canalso be separated at low pH by ion exclusion...
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Hydro Lubricants: Water-based lubricants for hydropower applications
PublikacjaSeveral different base oil types exist in the market including mineral and synthetic oils (e.g. polyalphaolefins, ester, polyglycol, etc.) and are currently widely in use. Although synthetic oils have drawn great attention over the past few decades in terms of their tribological benefits, mineral oils are still widely used in hydropower applications due primarily to their low cost and easy miscibility with other oils. However,...
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Second-order Stark effect and polarizability of a relativistic two-dimensional hydrogenlike atom in the ground state
PublikacjaThe second-order Stark effect for a planar Dirac one-electron atom in the ground state is analyzed within the framework of the Rayleigh-Schrödinger perturbation theory, with the use of the Sturmian series expansion of the generalized Dirac-Coulomb Green's function. A closed-form analytical expression for the static dipole polarizability of that system is found. The formula involves the generalized hypergeometric function ${}_{3}F_{2}$...
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Multi-pulse VSC arrangements with coupled reactors
PublikacjaThis paper presents a novel approach to the multipulse VSC (Voltage Source Converter) arrangements based on several conventional inverter modules connected in parallel by using coupled reactors. This solution reduces the THD of the output voltage, despite the low switching frequency of transistors. The advantage of the proposed solution is also a relatively small rated power of the reactors. Proposed new arrangements for different...
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Evaluation of Path Based Methods for Conceptual Representation of the Text
PublikacjaTypical text clustering methods use the bag of words (BoW) representation to describe content of documents. However, this method is known to have several limitations. Employing Wikipedia as the lexical knowledge base has shown an improvement of the text representation for data-mining purposes. Promising extensions of that trend employ hierarchical organization of Wikipedia category system. In this paper we propose three path-based...
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Localization of impulsive disturbances in archive audio signals using predictive matched filtering
PublikacjaThe problem of elimination of impulsive disturbances from archive audio signals is considered and its new solution, called predictive matched filtering, is proposed. The new approach is based on the observation that a large percentage of noise pulses corrupting archive audio recordings have highly repetitive shapes that match several typical “patterns”, called click templates. To localize noise pulses, click templates can be correlated...
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Symmetry-Breaking Bifurcation for Free Elastic Shell of Biological Cluster, Part 2
PublikacjaWe will be concerned with a two-dimensional mathematical model for a free elastic shell of biological cluster. The cluster boundary is connected with its kernel by elastic links. The inside part is filled with compressed gas or fluid. Equilibrium forms of the shell of biological cluster may be found as solutions of a certain nonlinear functional-differential equation with several physical parameters. For each multiparameter this...
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Structural Factors Affecting Cytotoxic Activity of (E)-1-(Benzo[d ][1,3]oxathiol-6-yl)-3-phenylprop-2-en-1-one Derivatives
PublikacjaDerivatives of (E)-1-(5-alkoxybenzo[d][1,3]oxathiol-6-yl)-3-phenylprop-2-en-1-one (1) demonstrated exceptionally high in vitro cytotoxic activity, with IC50 values of the most active derivatives in the nanomolar range. To identify structural fragments necessary for the activity, several analogs deprived of selected fragments were prepared, and their cytotoxic activity was tested. It was found that the activity depends on combined effects...
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REAL-TIME VOICE QUALITY MONITORING TOOL FOR VOIP OVER IPV6 NETWORKS
PublikacjaThe primary aim of this paper is to present a new application which is at this moment the only open source real-time VoIP quality monitoring tool that supports IPv6 networks. The application can keep VoIP system administrators provided at any time with up-to-date voice quality information. Multiple quality scores that are automatically obtained throughout each call reflect influence of variable packet losses and delays on voice...
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Analysis and Detection of Faults at Insulated Conductors of Overhead Medium Voltage Lines
PublikacjaThe paper dealt with the issue of breakdowns detection of isolated hanging wires on the medium-voltage transmission. The main aim of article is to describe the function of created breakdowns detector and evaluation its. The breakdowns detector is created based in indicators of faults such as touch between tree limbs and insulated wire, touch tree limbs with several phases or fall insulated wire on the ground. Breakdowns detector...
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A Hyperdense Semantic Domain for Discontinuous Behavior in Physical System Models
PublikacjaMultiple time models have been proposed for the formalization of hybrid dynamic system behavior. The superdense notion of time is a well-known time model for describing event-based systems where several events can occur simultaneously. Hyperreals provide a domain for defining the semantics of hybrid models that is elegantly aligned with first principles in physics. This paper discusses the value of both time models and shows how...
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Parallel computations in the volunteer based Comcute system
PublikacjaThe paper presents Comcute which is a novel multi-level implemen- tation of the volunteer based computing paradigm. Comcute was designed to let users donate the computing power of their PCs in a simplified manner, requiring only pointing their web browser at a specific web address and clicking a mouse. The server side appoints several servers to be in charge of execution of particular tasks. Thanks to that the system can survive...
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Clustering Context Items into User Trust Levels
PublikacjaAn innovative trust-based security model for Internet systems is proposed. The TCoRBAC model operates on user profiles built on the history of user with system interaction in conjunction with multi-dimensional context information. There is proposed a method of transforming the high number of possible context value variants into several user trust levels. The transformation implements Hierarchical Agglomerative Clustering strategy....
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Extra-curricular project-oriented education in optoelectronics in the Faculty of Electronics, Telecommunications and Informatics at Gdańsk University of Technology, Poland
PublikacjaProject-oriented education constitutes a key part of the curriculum in the Faculty of Electronics, Telecommunications and Informatics of Gdańsk University of Technology (Gdańsk Tech), Poland. Students on the Engineer and Master of Science level studies take part in several projects, both individually and in teams. In addition to compulsory activities, students have the opportunity to take part in the activities of student scientific...
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Heat transfer in plate heat exchanger channels: experimental validation of selected correlation equations
PublikacjaThis study is focused on experimental investigation of selected type of brazed plate heat exchanger. The Wilson approach was applied in order to estimate heat transfer coefficients for the PHEx passages. The main aim of the paper was to experimentally check ability of several correlations published in the literature to predict heat transfer coefficients by comparison experimentally obtained data with appropriate predictions. The...
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Poultry meat freshness evaluation using electronic nose technology and ultra-fast gas chromatography
PublikacjaTo ensure that chicken meat products are safe to consume, it is important to be able to reliably determine its shelf-life. To assess the applicability of ultra-fast gas chromatography and electronic nose technology in evaluation of poultry, an analysis of the headspace of ground chicken meat samples refrigerated over a period of 7 days was performed. Chemometric techniques were used to mine additional information from a multiparametric...
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DMI measurements impact on a position estimation with lack of GNSS signals during Mobile Mapping
PublikacjaNowadays, Mobile Laser Scanning is common in use in addition to geodesy measurements. The data which are provided by the system characterizes with high precision and flexibility. To precise mapping, the accuracy of the data should be maintained. In Poland, according to the minister’s dispositions, the accuracy of the data should not exceeded 10 cm. With fully operated system it is easy to uphold, but there is a situation when a...
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Arctic Freshwater Environment Altered by the Accumulation of Commonly Determined and Potentially New POPs
PublikacjaChemical composition of Arctic freshwater ecosystems depends on several factors. They include characteristics of the surrounding landscape, its lithology, geomorphology, vegetation, and hydrological features, as well as accumulation of anthropogenic pollution. In the Arctic, the problem of environmental contamination is widespread. That is why research on lakes and river catch-ments in terms of their chemical composition has enjoyed...
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Report of Eurocode 7 application for pile foundation design in Poland
PublikacjaThe EC7 rules of geotechnical design are in use in Poland for several years, even though there is no National annex. With regard to pile foundations, there are valid EC7 recommendations concerning design approaches, load partial coefficients, correlation coefficients and capacity partial coefficients. Polish designers can be quite flexible when it comes to choose a method for static, bearing capacity and settlement calculations....