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Structure-property relationships disclosed in the family of acridinium esters – chemiluminogenic molecules of great practical importance
PublikacjaAcridinium esters (AE), since their introduction to the analytics 30 years ago, make one of the most important groups of chemiluminogenic (CL) systems, that have been employed in medical diagnostics and environmental analysis today. So far, however, no systematic studies on the structureproperty relationships were carried out in this family of compounds. The latter features likely determine their practical utility and facilitate...
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(R,R)-1-Acetyl-1'-(2,4,6-trinitrophenyl)-2,2'-bipyrrolidine
Publikacja(R,R)-1-Acetyl-1'-(2,4,6-trinitrophenyl)-2,2'-bipyrrolidine has been synthesized and its rentgenostructure has been determined. The structure of the title molecule, C16H19N5O7, is mainly determined by the steric effect of a bulky 2,4,6-trinitrophenyl group attached to the N atom of a pyrrolidine ring. Both pyrrolidine rings adopt an envelope conformation, with one of the methylene C atoms as the flap in each case, and the N-C-C-N...
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Phylogenetic relationship and antimicrobial resistance in Escherichia coli isolated from the Reda River and the Oliwski Stream, Northern Poland = Lekooporność i przynależność filogenetyczna szczepów Escherichia Coli izolowanych z rzeki Redy i Potoku Oliwskiego
PublikacjaThe high abundance of fecal bacteria in surface water is usually related to poor agricultural practice, pollution caused by domesticated and wild animals as well as with septic tank failures. Identification of fecal contamination sources seems to be crucial in order to effectively estimate the inherent risk. In this study, the phylogenetic relationship of 30 isolates of E. coli, originated from surface water, was estimated by employing...
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DMSO hydration redefined: Unraveling the hydrophobic hydration of solutes with a mixed hydrophilic–hydrophobic characteristic
PublikacjaHydrophobic hydration of solutes with a mixed hydrophilic--hydrophobic characteristics is still poorly understood. This is because both experimental and theoretical methods find it difficult to see the ice-like water structure around the nonpolar solute groups, unlike hydrogen bonds with the hydrophilic groups. In order to unravel this problem, we have investigated DMSO hydration by means of infrared spectroscopy and theoretical...
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Adipokine and cytokine levels in non-functioning adrenal incidentalomas (NFAI)
PublikacjaDue to the fact that overweight or obesity is accompanied by hormonally active adrenal tumors: Cushing Syndrome-(CS) and Subclinical Cushing Syndrome (SCS), it is of high interest the correlation between different adipokines and cytokines secreted by adipose tissue, with metabolic disorders and hormonal activity in this group. Even in non-functioning adrenal incidentalomas (NFAI) elevated risk for cardiovascular disease and metabolic...
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Evaluation of flavour profiles in e-cigarette refill solutions using gas chromatography–tandem mass spectrometry
PublikacjaMany flavour compounds that are present in e-liquids for e-cigarettes are responsible for specific tastes and smoking sensations for users. Data concerning content and specific types of flavours is often limited and unknown to users. The aim of the research was to define and compare flavour profiles of e-liquids with the same group taste from different manufacturers. Gas chromatography coupled with tandem mass spectrometry (GC–MS/MS)...
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Soft-mode enhanced type-I superconductivity in LiPd2Ge
PublikacjaThe synthesis, crystal structure, and physical properties (magnetization, resistivity, heat capacity) in combination with theoretical calculations of the electronic structure and phonon properties are reported for intermetallic compounds LiPd2X (X = Si, Ge, and Sn). LeBail refinement of powder x-ray diffraction data confirms that all compounds belong to the Heusler family (space group Fm-3m, No. 225). The lattice parameter increases...
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Psychosocial risks associated with the profession of train driver
PublikacjaExcellent competencies as well as a good physical and mental health are required in train drivers’ profession. Despite the changes in the structure of employment the train drivers above 46 years and job tenure longer than 30 years are the largest group. The generation gap is becoming more pronounced, and its fulfilment will not be easy. It is related not only to training of new personnel but also promotion of healthy work environment...
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Crystallographic study of self-organization in the solid state including quasi-aromatic pseudo-ring stacking interactions in 1-benzoyl-3-(3,4-dimethoxyphenyl)thiourea and 1-benzoyl-3-(2-hydroxypropyl)thiourea
Publikacja1-Benzoylthioureas contain both carbonyl and thiocarbonyl functional groups and are of interest for their biological activity, metal coordination ability and involvement in hydrogen-bond formation. Two novel 1-benzoylthiourea derivatives, namely 1-benzoyl-3-(3,4-dimethoxyphenyl)thiourea, C₁₆H₁₆N₂O₃S, (I), and 1-benzoyl-3-(2-hydroxypropyl)thiourea, C₁₁H₁₄N₂O₂S, (II), have been synthesized and characterized. Compound (I) crystallizes...
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Upward convergence patterns in chosen environmental-related SDGs
PublikacjaSustainable development is a challenge facing humanity. EU countries not only strive to reach their specific objectives, but they also work collaboratively towards shared goals. There is a need to balance synergies and compromises to address these objectives effectively. When discussing countries' development and people's well-being, one often focuses on socio-economic development. However, it is crucial not to overlook the environmental...
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Measurement of temperature at sliding polymer surface by grindable thermocouples
PublikacjaThis paper is devoted to experimental study of capabilities and limitations of grindable thermocouples as applied to polymer materials sliding on metal. Chromel–alumel and chromel–copel grindable thermocouples have been developed and tested for wide ranges of contact pressure and sliding velocity. The background temperature of the sliding surface can be determined as the lower envelope of the signal from the grindable thermocouple....
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The Influence of Cooperation on the Operation of an MPC Controller Pair in a Nuclear Power Plant Turbine Generator Set
PublikacjaThe paper discusses the problem of cooperation between multiple model predictive control (MPC) systems. This approach aims at improving the control quality in electrical energy generation and forms the next step in a series of publications by the authors focusing on the optimization and control of electric power systems. Cooperation and cooperative object concepts in relation to a multi MPC system are defined and a cooperative control...
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Visual Data Encryption for Privacy Enhancement in Surveillance Systems
PublikacjaIn this paper a methodology for employing reversible visual encryption of data is proposed. The developed algorithms are focused on privacy enhancement in distributed surveillance architectures. First, motivation of the study performed and a short review of preexisting methods of privacy enhancement are presented. The algorithmic background, system architecture along with a solution for anonymization of sensitive regions of interest...
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Gaze tracking in multi-display environment
PublikacjaThis paper presents the basic ideas of eye and gaze tracking in multiple-display environment. The algorithm for display detection and identification is described as well as the rules for gaze interaction in multi display environment. The core of the method is to use special LED markers and eye and scene tracking glasses. Scene tracking camera registers markers position which is then represented as a cloud of points. Analyzing the...
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Modelling of Mechatronic Systems with Distributed Parameter Components
PublikacjaThe paper presents an uniform, port-based approach to modelling of both lumped and distributed parameter systems. Port-based model of distributed system has been defined by application of the bond graph methodology and the distributed transfer function method (DTFM). The proposed method of modelling enables to formulate input data for computer analysis by application of the DTFM. The computational package for the analysis of complex...
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Low Power Baseband Processor for M2M Reconfigurable Radio Test Platform
PublikacjaSoftware Defined Radio (SDR) is becoming more andmore frequently used technique for wireless communication. Itfacilitates as fast prototyping and is a versatile method fordeveloping new communication systems. SDR can be realizedbased on high computational capacity platform, where powerconsumption is no a primary concern like i.e. DVB or BTStransmitters. Another trend are low power systems, whereavailable power in reduced and more...
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Distributed wireless sensor for measuring humidity and temperature
PublikacjaHumidity and temperature monitoring is often required in industrial halls and laboratories and can be crucial, because many properties of electrical devices deteriorates under influence of these parameters. There are several useful commercial methods for measuring humidity and temperature, such as commercial hygrometers and humidity recorders. However, they do not allow data acquisition simultaneously from multiple sensors. This...
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Future research directions in design of reliable communication systems
PublikacjaIn this position paper on reliable networks, we discuss new trends in the design of reliable communication systems. We focus on a wide range of research directions including protection against software failures as well as failures of communication systems equipment. In particular, we outline future research trends in software failure mitigation, reliability of wireless communications, robust optimization and network design, multilevel...
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Effect of bitumen characteristics obtained according to EN and Superpave specifications on asphalt mixture performance in low-temperature laboratory tests
PublikacjaThe paper aims to identify those characteristics of bitumen which have the greatest impact on asphalt mixture low-temperature performance. It was observed that stiffness and m-value of bitumen from BBR test were moderately related to stiffness and m-value of asphalt mixture obtained from 3 PB test. Simultaneously those rheological properties significantly impact on cryogenic stresses induced during TSRST test. The multiple regression...
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Selected studies of flow maldistribution in a minichannel plate heat exchanger
PublikacjaAnalysis of the state of-the-art in research of minichannel heat exchangers, especially on the topic of flow maldistribution in multiple channels, has been accomplished. Studies on minichannel plate heat exchanger with 51 parallel minichannels with four hydraulic diameters, i.e., 461 μm, 574 μm, 667 μm, and 750 μm have been presented. Flow at the instance of filling the microchannel with water at low flow rates has been visualized. The...
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COMPREHENSIVE MODELLING OF THE COST EFFECTIVNESS OF RAILWAY LINE ELECTRIFICATION
PublikacjaSubject of this paper is the mathematical model estimating the Economical threshold between usage of combustion engine traction and electrical traction for new and modernized railway passenger communication lines. Currently available models do not coincide with the whole complexity of the problem. The proposed model was implemented into Matlab and then validated on “Pomorska Kolej Metropolitalna” investment time-frame and its cost...
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Unraveling Energy Transfer and Fluorescence Quenching Dynamics in Biomolecular Complexes: A Comprehensive Study of Imiquimod-Rifampicin Interaction.
PublikacjaIn nature, numerous biomolecules are implicated in charge transfer (CT) and energy transfer (ET) mechanisms crucial for fundamental processes such as photosynthesis. Unveiling these mechanisms is pertinent to multiple disciplines including chemistry, engineering and biochemistry. This letter presents a study involving two molecules forming a model system with efficient ET properties. Specifically, their complex exhibits dark quenching...
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Energy efficient indoor localisation for narrowband internet of things
PublikacjaThere are an increasing number of Narrow Band IoT devices being manufactured as the technology behind them develops quickly. The high co-channel interference and signal attenuation was seen in edge Narrow Band IoT devices make it challenging to guarantee the service quality of these devices. To maximize the data rate fairness of Narrow Band IoT devices, a multi-dimensional indoor localization model is devised, consisting of...
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Design and Optimization of a Compact Super-Wideband MIMO Antenna with High Isolation and Gain for 5G Applications
PublikacjaThis paper presents a super-wideband multiple-input multiple-output (SWB MIMO) antenna with low profile, low mutual coupling, high gain and compact size for microwave and millimeter wave (mm-wave) fifth-generation (5G) applications. A single antenna is a simple elliptical-square shape with a small physical size of 20 × 20 × 0.787 mm3. The combination of both square and elliptical shapes results in an exceptionally broad impedance...
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A Planar-Structured Circularly Polarized Single-Layer MIMO Antenna for Wideband Millimetre-Wave Applications
PublikacjaIn this paper, a simple geometry, planar-structured printed multiple-input-multiple-output (MIMO) antenna utilizing dual circular polarization (CP) is presented. The proposed numerically and experimentally validated design features a fully grounded coplanar waveguide (CPW) and a systematically perturbed feedline radiator. The fringing electric (E) field along the feedline is altered by extruding periodic stubs on each side of the...
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A Compact Circularly Polarized Dielectric Resonator Antenna with MIMO Characterizations for UWB Applications
PublikacjaUltra-wideband (UWB) technology is extensively used in indoor navigation, medical applications, and Internet of Things (IoT) devices due to its low power consumption and resilience against multipath fading and losses. This paper examines a multiple input multiple-output (MIMO), circularly polarized (CP) dielectric resonator antenna (DRA) for UWB systems. Compact form factor, high gain, wideband response, improved port isolation,...
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Enhanced-Performance Circularly Polarized MIMO Antenna with Polarization/Pattern Diversity
PublikacjaDesign of a compact wideband circularly polarized (CP) multiple-input multiple-output (MIMO) antenna with polarization diversity is proposed and characterized for off-body communication. The antenna is based on a simple coplanar waveguide (CPW)-fed monopole extension of the microstrip line. The orthogonal field components required by CP are induced using a simply modified right/left side ground plane. In particular, a stub extending...
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Distinct cellular uptake patterns of two anticancer unsymmetrical bisacridines and their metabolic transformation in tumor cells.
PublikacjaUnsymmetrical bisacridines (UAs) represent a novel class of anticancer agents. Their high cytotoxicity towards multiple human cancer cell lines and inhibition of human tumor xenograft growth in nude mice signal their potential for cancer treatment. Therefore, the mechanism of their strong biological activity is broadly investigated. Here, we explore the efflux and metabolism of UAs, as both strongly contribute to the development...
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Integrated membrane bioreactors modelling: A review on new comprehensive modelling framework
PublikacjaIntegrated Membrane Bioreactor (MBR) models, combination of biological and physical models, have been representing powerful tools for the accomplishment of high environmental sustainability. This paper, produced by the International Water Association (IWA) Task Group on Membrane Modelling and Control, reviews the state-of-the-art, identifying gaps for future researches, and proposes a new integrated MBR modelling framework. In...
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Pomoszcz Ministerstwa Inostrannych del Polszy Armenji, Azerbejdzżany i Gruzji = Polish Development Assistance for Armenia, Azerbaijan and Georgia
PublikacjaGeorgia has been one of the priority areas of development assistance of Polish Ministry of Foreign Affairs from 2004, because it plays a important role in Polish forsign policy in the framework of the Eastern Partnership. The largest amounts of development aid supporting the transformation were allocated for this country. Since founding the Eastern Partnership initiative in 2009 also Azerbaijan and Armenia have been included to...
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Experimental Comparison of Straight Lines and Polynomial Interpolation Modeling Methods in Ship Evolutionary Trajectory Planning Problem
PublikacjaPaper presents the application of evolutionary algorithms and polynomial interpolation in ship evolutionary trajectory planning method and its comparison to classic approach, where trajectory is modeled by straight lines. Evolutionary algorithms are group of methods that allows\ to find a collision free trajectory in real time, while polynomial interpolation allows to model smooth trajectory, which keeps continuity of velocity...
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Exploring ontological approach for user requirements elicitation in design of online virtual agents
PublikacjaEffective user requirements elicitation is a key factor for the success of software development projects. There are many qualitative and quantitative research studies that promulgate particular methods and show the application of user requirements elicitation in particular domains. However, few try to eliminate the burden of ambiguity in gathered data, naturally occurring in different groups of stakeholders. This paper deals with...
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Online stores' credibility: the moderating role of customers' gender and self-efficacy
PublikacjaThe evaluation of online stores’ credibility by customers in regard of gender and self-efficacy is presented. Two groups of attributes, usability and informational content, were characteristics of credibility. The survey involved students as representatives of the largest group of the Internet users. As shown by the results obtained, the informational content of online stores (such as recommendations) and its professionalism was...
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Auditory-visual attention stimulator
PublikacjaNew approach to lateralization irregularities formation was proposed. The emphasis is put on the relationship between visual and auditory attention stimulation. In this approach hearing is stimulated using time scale modified speech and sight is stimulated by rendering the text of the currently heard speech. Moreover, displayed text is modified using several techniques i.e. zooming, highlighting etc. In the experimental part of...
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Synthesis of 2-amino-2,6-dideoxy-D-glucitol-6-sulfonic acid as a potential antifungal agent.
PublikacjaGlucosamine-6P (GlcN-6P) synthase catalyzes the first committed step in the biosynthetic pathway leading to the formation of UDP-GlcNAc, a sugar nucleotide precursor providing D-glucosamine for the formation of chitin and manoproteins. 2-Amino-2,6-dideoxy-D-glucitol-6-sulfonic acid is an analog of 2-amino-2-deoxy-D-glucitol 6-phosphate (GlcN-ol-6-P), a known inhibitor of GlcN-6-P synthase, in which the phosphate group of the latter...
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Synthesis and biological activity of mycophenolic acid-amino acid derivatives
PublikacjaIn search of new immunosuppressants, mycophenolic acid (MPA) was coupled with amino acid methyl esters followed by hydrolysis to analogs bearing free carboxylic groups. The obtained compunds were tested in vitro as growth inhibitors of lymphoid cell line (Jurkat) and human peripheral blood mononuclear cells (PBMC) from healthy donors. According to obtained results recovering of free carboxylic group increased their activity. Additionally,...
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High-precision bearing estimation for active sonar with cylindrical array performed by interpolated array transformation
PublikacjaThe article presents a method for improving the accuracy of bearing in multibeam sonar with a cylindrical array. The antenna’s non-linear shape and the resulting non-uniform sampling of the signal in space, mean that known methods of high-resolution spectral analysis cannot be used. In order to apply an algorithm from this group, a linear virtual antenna must be produced. The paper presents a technique of mapping a cylindrical...
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Design, synthesis, and molecular docking of new 5-HT reuptake inhibitors based on modified 1,2-dihydrocyclopenta[b] indol-3(4H)-one scaffold
PublikacjaA new group of serotonin reuptake inhibitors containing 1,2-dihydrocyclopenta[b]indol-3(4H)-one scaffoldwas synthesized, starting from indole 5-((1H-indol-3-yl)(1,3-dioxane-4,6-diones as a key intermediates. Following three transformations including intramolecular cyclization and formation of imines, a series of new ligand for human serotonin transporter was obtained. The ability of these ligands to inhibit human TS3 serotonin transporter...
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DEEP CONVOLUTIONAL NEURAL NETWORKS AS A DECISION SUPPORT TOOL IN MEDICAL PROBLEMS – MALIGNANT MELANOMA CASE STUDY
PublikacjaThe paper presents utilization of one of the latest tool from the group of Machine learning techniques, namely Deep Convolutional Neural Networks (CNN), in process of decision making in selected medical problems. After the survey of the most successful applications of CNN in solving medical problems, the paper focuses on the very difficult problem of automatic analyses of the skin lesions. The authors propose the CNN structure...
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Determinanty zakupu usług ubezpieczeniowych przez osoby powyżej 50. roku zycia
PublikacjaArtykuł dotyczy usług ubezpieczeniowych oraz determinant korzystania z tych usług przez osoby powyżej 50. roku życia. Mimo że popyt na usługi ubezpieczeniowe wśród osób w tym wieku jest mniejszy niż wśród osób młodszych, można wyodrębnić w tej grupie mniejsze grupy istotnie zróżnicowane pod względem potencjalnego popytu. W celu wyodrębnienia tych grup oraz zidentyfikowania pozostałych powodów determinantów korzystania z ubezpieczeń...
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Identyfikacja trajektorii obiektów dynamicznych w przestrzeni kartezjańskiej na podstawie informacji z wielu estymatorów stanu
PublikacjaW rozprawie przedstawiono metodologię umożliwiającą implementację rozproszonego asynchronicznego systemu wyznaczania trajektorii. System tego typu jest złożony ze zbioru tzw. węzłów (estymatorów lokalnych), które komunikują się ze sobą. Każdy węzeł wyznacza trajektorię obserwowanego obiektu/procesu na podstawie dwóch zbiorów danych. Pierwszym zbiorem są pomiary dostarczane przez skojarzone z danym...
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Porous Phantoms Mimicking Tissues—Investigation of Optical Parameters Stability Over Time
PublikacjaOptical phantoms are used to validate optical measurement methods. The stability of their optical parameters over time allows them to be used and stored over long-term periods, while maintaining their optical parameters. The aim of the presented research was to investigate the stability of fabricated porous phantoms, which can be used as a lung phantom in optical system. Measurements were performed in multiple series with an interval...
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CFD analysis of fluid flow through the labyrinth seal
PublikacjaSteam and gas turbines are some of the fundamental means of power generation. The energy efficiency of the turbines, however, is not satisfactory. Ever since the start-up of the first turbine in the world, engineers have been striving for their increased efficiency. Multiple solutions to the problem of steam loss in an operating turbine are available. The use of seals is one of them. Empirical methods or numerical calculations...
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REAL-TIME VOICE QUALITY MONITORING TOOL FOR VOIP OVER IPV6 NETWORKS
PublikacjaThe primary aim of this paper is to present a new application which is at this moment the only open source real-time VoIP quality monitoring tool that supports IPv6 networks. The application can keep VoIP system administrators provided at any time with up-to-date voice quality information. Multiple quality scores that are automatically obtained throughout each call reflect influence of variable packet losses and delays on voice...
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A Hyperdense Semantic Domain for Discontinuous Behavior in Physical System Models
PublikacjaMultiple time models have been proposed for the formalization of hybrid dynamic system behavior. The superdense notion of time is a well-known time model for describing event-based systems where several events can occur simultaneously. Hyperreals provide a domain for defining the semantics of hybrid models that is elegantly aligned with first principles in physics. This paper discusses the value of both time models and shows how...
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Multiacces quantum communication and product higher rank numerical range
PublikacjaIn the present paper we initiate the study of the product higher rank numerical range. The latter, being a variant of the higher rank numerical range, is a natural tool for study- ing a construction of quantum error correction codes for multiple access channels. We review properties of this set and relate it to other numerical ranges, which were recently introduced in the literature. Further, the concept is applied to the construction...
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Fast implementation of FDTD-compatible green's function on multicore processor
PublikacjaIn this letter, numerically efficient implementation of the finite-difference time domain (FDTD)-compatible Green's function on a multicore processor is presented. Recently, closed-form expression of this discrete Green's function (DGF) was derived, which simplifies its application in the FDTD simulations of radiation and scattering problems. Unfortunately, the new DGF expression involves binomial coefficients, whose computations...
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Resonance Frequency Calculation of a Multilayer and Multipatch Spherical Microstrip Structure Using a Hybrid Technique
PublikacjaThis communication offers a rigorous analysis of the resonance frequency problem of a spherical microstrip structure mounted on a multilayer, dielectric-coated metallic sphere, with an electrically small radius. The structure consists of single or multiple metallic patches with arbitrary shapes. A full-wave analysis is employed with the use of proposed hybrid approach, combining the finite-difference technique with a spectral domain...
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Parameters optimization in medicine supporting image recognition algorithms
PublikacjaIn this paper, a procedure of automatic set up of image recognition algorithms' parameters is proposed, for the purpose of reducing the time needed for algorithms' development. The procedure is presented on two medicine supporting algorithms, performing bleeding detection in endoscopic images. Since the algorithms contain multiple parameters which must be specified, empirical testing is usually required to optimise the algorithm's...
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On the impact of Big Data and Cloud Computing on a scalable multimedia archiving system
PublikacjaMultimedia Archiver (MA) is a system build upon the promise and fascination of the possibilities emerging from cloud computing and big data. We aim to present and describe how the Multimedia Archiving system works for us to record, put in context and allow a swift access to large amounts of data. We introduce the architecture, identified goals and needs taken into account while designing a system processing data with Big Data...