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Tetrahydroquinolinone derivatives exert antiproliferative effect on lung cancer cells through apoptosis induction
PublikacjaThe anticancer properties of quinolones is a topic of interest among researchers in the scientific world. Because these compounds do not cause side effects, unlike the commonly used cytostatics, they are considered a promising source of new anticancer drugs. In this work, we designed a brief synthetic pathway and obtained a series of novel 8-phenyltetrahydroquinolinone derivatives functionalized with benzyl-type moieties at position...
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A general theory for anisotropic Kirchhoff–Love shells with in-plane bending of embedded fibers
PublikacjaThis work presents a generalized Kirchhoff–Love shell theory that can explicitly capture fiber-induced anisotropy not only in stretching and out-of-plane bending, but also in in-plane bending. This setup is particularly suitable for heterogeneous and fibrous materials such as textiles, biomaterials, composites and pantographic structures. The presented theory is a direct extension of classical Kirchhoff–Love shell theory to incorporate...
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Phytoextraction and recovery of rare earth elements using willow (Salix spp.)
PublikacjaSoil and water contaminations are caused by rare earth elements (REEs) due to mining and industrial activities, that threaten the ecosystem and human health. Therefore, phytoremediation methods need to be developed to overcome this problem. To date, little research has been conducted concerning the phytoremediation potential of Salix for REEs. In this study, two Salix species (Salix myrsinifolia and Salix schwerinii) and two Salix...
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Electrochemical capacitor temperature fluctuations during charging/discharging processes
PublikacjaThepaperpresentsaproposalofusingadditionalstatisticalparameterssuchas:standarddeviation,variance, maximum and minimum increases of the observed value that were determined during measurements of temperature fields created on the surface of the tested electrochemical capacitor. The measurements were carriedoutusingthermographicmethodsinordertosupportassessmentoftheconditionofelectrochemical capacitorunderclassicdurabilitytestsbasedonmethodsofdeterminationofcapacityandequivalentseries...
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Technologia drewna , W/L, Oceanotechnika, sem.6, lato 23, (O:098640)
Kursy OnlineCelem przedmiotu jest przedstawienie wybranych zagadnień związanych z zastosowaniem i przetwarzaniem drewna do budowy jednostek pływających. W ramach przedmiotu zostaną poruszone zagadnienia materiałowe, podstawowych procesów wytwarzania, w tym metrologiczne a także wybranych problemów łączenia i konserwacji drewna. Zakres przedmiotu obejmuje: Wykład: Historia drewna...
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Nowoczesne układy przekształtników wielopoziomowych do zasilania statków z lądu
PublikacjaW artykule poruszono tematykę zasilania statków zacumowanych w porcie z lądowej sieci elektroenergetycznej poprzez wykorzystanie nowoczesnych konstrukcji przekształtników energoelektronicznych. W treści pracy zaprezentowano porównanie dwóch topologii wysokonapięciowych przekształtników wielopoziomowych. Porównano konstrukcje przekształtników z klasycznym transformatorem wielouzwojeniowym oraz z transformatorami wysokoczęstotliwościowymi.
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Modernity and postmodernity in architectural education
PublikacjaThe purpose of this article is to present a philosophical education strategy for architecture and interior architecture faculties. The approach is the result of trial and error in lectures and debates with students of philosophical courses in these fields. The presented article is not a result of empirical research, but rather a report on the problems encountered and proposals for their solution. The experience gained from conducting...
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Impacts in case of triple unilaterally constrained system
PublikacjaThe this paper focus on the behaviour of a “rigid” body biting into another “rigid” body, with some nonzero relative velocity. In the presently considered case, the introduced collision appears between a selected element of a multibody structure and its reference body being interpreted as the motionless ground. Instead of the classic case, described in a number of dissertations, where a single impacting contact is considered, three...
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Al-Kindi’s “The Real One”: Considerations of a mathematician or of a metaphysician?
PublikacjaThe aim of the article is to analyze Al-Kindi’s concept of the True (Essential) One and certain additional issues, also taking into account the influence on his position from both classical philosophy and source texts of Islam. In the opening part of the article, Al-Kindi’s innovative approach to the application of mathematics in research in other areas of knowledge is discussed. In the next part,...
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Refining of Secondary Pb with Retention of Sn Using Al and Ca Additions
PublikacjaLead grid from spent lead-acid batteries contains significant amounts of tin and antimony. In classical pyro-refining processes of lead, tin oxidizes and is transferred to dross, making its recovery problematic and expensive. This paper presents an innovative method of pyro-refining lead using metallic aluminum and calcium to purify the lead from contaminants while retaining a higher amount of tin than in the traditional process....
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Generating optimal paths in dynamic environments using RiverFormation Dynamics algorithm
PublikacjaThe paper presents a comparison of four optimisation algorithms implemented for the purpose of finding the shortest path in static and dynamic environments with obstacles. Two classical graph algorithms –the Dijkstra complete algorithm and A* heuristic algorithm – were compared with metaheuristic River Formation Dynamics swarm algorithm and its newly introduced modified version. Moreover, another swarm algorithm has been compared...
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Thermodynamic Cycle Concepts for High-Efficiency Power Plants. Part B: Prosumer and Distributed Power Industry
PublikacjaAn analysis was carried out for different thermodynamic cycles of power plants with air turbines. A new modification of a gas turbine cycle with the combustion chamber at the turbine outlet has been described in the paper. A special air by-pass system of the combustor was applied, and in this way, the efficiency of the turbine cycle was increased by a few points. The proposed cycle equipped with an effective heat exchanger could...
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Flexomagneticity in buckled shear deformable hard-magnetic soft structures
PublikacjaThis research work performs the first time exploring and addressing the flexomagnetic property in a shear deformable piezomagnetic structure. The strain gradient reveals flexomagneticity in a magnetization phenomenon of structures regardless of their atomic lattice is symmetrical or asymmetrical. It is assumed that a synchronous converse magnetization couples both piezomagnetic and flexomagnetic features into the material structure....
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How high-tech solutions support the fight against IUU and ghost fishing: a review of innovative approaches, methods, and trends
PublikacjaIllegal, Unreported, and Unregulated fishing is a major threat to human food supply and marine ecosystem health. Not only is it a cause of significant economic loss but also its effects have serious long-term environmental implications, such as overfishing and ocean pollution. The beginning of the fight against this problem dates since the early 2000s. From that time, a number of approaches and methods have been developed and reported....
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Hyperbolic heat conduction at a microscopic sliding contact with account of adhesion-deformational heat generation and wear
PublikacjaDifferent non-Fourier models were proposed to simulate temperatures in materials subjected to extremely fast thermal disturbances, when the speed of heat propagation should be concerned. The present study investigated temperature and heat balance at a microscopic sliding contact during a single frictional interaction based on the Cattaneo-Vernotte hyperbolic heat conduction equation. Two fundamental features of friction, namely,...
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Power System Dynamics. Stability and Control. 3rd edition
PublikacjaComprehensive, state-of-the-art review of information on the electric power system dynamics and stability. It places the emphasis first on understanding the underlying physical principles before proceeding to more complex models and algorithms. The book explores the influence of classical sources of energy, wind farms and virtual power plants, power plants inertia and control strategy on power system stability. The book cover...
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Pressure effects on the electronic structure and superconductivity of (TaNb)0.67(HfZrTi)0.33 high entropy alloy
PublikacjaEffects of pressure on the electronic structure, electron-phonon interaction, and superconductivity of the high entropy alloy ( TaNb ) 0.67 ( HfZrTi ) 0.33 are studied in the pressure range 0–100 GPa. The electronic structure is calculated using the Korringa-Kohn-Rostoker method with the coherent potential approximation. Effects of pressure on the lattice dynamics are simulated using the Debye-Grüneisen model and the Grüneisen...
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An Innovative Approach to the Forecasting of Energetic Effects While Wood Sawing
PublikacjaIn the classical approach, energetic effects (cutting forces and cutting power) of wood sawing process are generally calculated on the basis of the specifi c cutting resistance, which is in the case of wood cutting the function of more or less important factors. On the other hand, the cutting forces (power) problem may be tackled with an innovative, up-to-date fundamental analysis of the mechanics of sawing based on modern fracture mechanics....
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The Use of Wavelet Analysis to Denoising of Electrocardiography Signal
PublikacjaThe electrocardiography examination, due to its accessibility and simplicity, has an important role in diagnostics of the heart ailments. It enables quick detection of various heart defects, undetectable by other kinds of diagnostic tools, so it is very popular. Nevertheless, the measured signal is exposed to a different disturbances. Among them, the electromagnetic interferences, drift of reference electrode and high frequency...
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An innovative approach to the forecasting of energetic effects while wood sawing
PublikacjaIn the classical approach, energetic effects (cutting forces and cutting power) of wood sawing process are generally calculated on the basis of the specific cutting resistance, which is in the case of wood cutting the function of more or less important factors. On the other hand, the cutting forces (power) problem may be tackled with an innovative, up-to-date fundamental analysis of the mechanics of sawing based on modern fracture...
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Feasibility of combined diesel engine - steam turbine in power station operating in the maritime
PublikacjaCompression-ignition engines used in ship technology as main propulsion engines are large units reaching even to 50-60 MW. Currently, the efficiency of such engines amounts to 45-50%. With such a large power unit, exhaust gases leaving the engine contain very large quantities of heat available for further treatment. Exhaust gases from the piston engine contain about 25% of the heat supplied to the engine in the fuel. Using the...
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Risk factor assessment in agricultural supply chain by fuzzy logic
PublikacjaSignificant uncertainty characterizes the harvest period. This aspect is due to various risks impacting agrifood supply chains. The occurrence of risks is due to hazards: technological failures, technical breakdowns, or adverse weather conditions. Hence, the operational time of the agricultural supply chain during the harvest period increases due to such risk factors. In essence, some hazards are fuzzy, and the nature of most threats...
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NUMERICAL MODEL OF PLASTIC DESTRUCTION OF THICK STEEL STRUCTURAL ELEMENTS
PublikacjaIn the shipbuilding industry, the risk of brittle fracture of the structure is limited by using certified materials with specified impact strength, determined by the Charpy method (for a given design temperature) and by supervising the welding processes (technology qualification, production supervision, non-destructive testing). For off-shore constructions, classical shipbuilding requirements may not be sufficient. Therefore, the...
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Comparison of noise reduction methods in radiometric correlation measurements of two-phase liquid-gas flows
PublikacjaTwo-phase liquid-gas flows occur frequently in the mining, energy, chemical, and petrochemical industries. One of non-contact methods used to analyse these flows is the gamma ray absorption method. However, the signals received from radiation detectors contain a significant stochastic noise, which makes them difficult to analyse. The article describes four methods of noise reduction in cross-correlation measurements of water-air...
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A methodology for ultimate strength assessment of ship hull girder accounting for enhanced corrosion degradation modelling
PublikacjaThe presented work shows a methodology for the ultimate strength assessment of a ship hull, considering enhanced corrosion modelling. The approach is based on the classical Smith method. However, the recent findings regarding the impact of corrosion degradation on ultimate strength are incorporated. To this end, the stress–strain relationships for particular elements composing ship hull cross-section are modified using a specially...
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Solid and liquid fractionation of sugarcane and Agave bagasse during ozonolysis and enzymatic hydrolysis: Impact on biohydrogen and biogas production
PublikacjaSustainable and cost-efficient lignocellulosic biomass-to-energy bioprocesses require assessing the main components released during biomass fractionation. This study assessed the mesophilic biochemical potential of biohydrogen (BHP) and methane production (BMP) from sugarcane bagasse (SCB) and cooked (CAB) and uncooked (UAB) Agave bagasse. A systematic comparative analysis was performed for the liquid and solid fractions derived...
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A new anisotropic bending model for nonlinear shells: Comparison with existing models and isogeometric finite element implementation
PublikacjaA new nonlinear hyperelastic bending model for shells formulated directly in surface form is presented, and compared to four existing prominent bending models. Through an essential set of elementary nonlinear bending test cases, the membrane and bending stresses of each model are examined analytically. Only the proposed bending model passes all the test cases, while the other bending models either fail or only pass the test cases for...
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Selecting the optimum location for logistics facilities using Solver
PublikacjaSiting logistics facilities strategically in the most costeffective geographic location is one of the key decisions a contemporary company will make. The aim of the paper is to present a solution to this problem using the Solver add-on. In the case study discussed in the paper, the company’s central warehouse location was selected based on the classic location theory, which addresses the need to minimize the cost of transport....
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Investigation of the Aerodynamics of an Innovative Vertical-Axis Wind Turbine
PublikacjaThe paper presents the results of an experimental investigation and a three dimensional numerical analysis of the transient aerodynamic phenomena occurring in the innovative modification of classic Savonius wind turbine. An attempt to explain the increased efficiency of the innovative design a comparison with the traditional solution is undertaken. A vorticity measure based on the integral of the velocity gradient tensor second...
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Infinite chromatic games
PublikacjaIn the paper we introduce a new variant of the graph coloring game and a new graph parameter being the result of the new game. We study their properties and get some lower and upper bounds, exact values for complete multipartite graphs and optimal, often polynomial-time strategies for both players provided that the game is played on a graph with an odd number of vertices. At the end we show that both games, the new and the classic...
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Method of sacrificial anode transistor-driving in cathodic protection system
PublikacjaA magnesium anode driving system has been proposed. A PNP driving transistor has been used. Electrochemical testing in 3%NaCl, results and comparison of the driving system and classic direct anode to cathode connection are presented. The driving system reduced the protection current and stabilized the working conditions of the anode. Higher anode efficiency was achieved. Overprotection and hydrogen embrittlement threats were prevented...
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Distributed Evolutionary Algorithm for Path Planning in Navigation Situation
PublikacjaThis article presents the use of a multi-population distributed evolutionary algorithm for path planning in navigation situation. The algorithm used is with partially exchanged population and migration between independently evolving populations. In this paper a comparison between a multi-population and a classic single-population algorithm takes place. The impact on the ultimate solution has been researched. It was shown that using...
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Analysis of distance measurement errors in CW FM sonar with MLS code modulation
PublikacjaAlthough used in the classic silent sonar, the CW FM sounding signal has a major flaw which is its inaccuracy in determining the distance to a target. The authors of the article have developed a concept of silent sonar using frequency modulation signals switched by pseudorandom codes, already discussed in their previous work. This article presents a detailed analysis of errors in CW FM sonar with pseudo-random sequence code modulation...
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Spectroscopic studies on physicochemical properties of selected unsymmetrical bisacridine derivatives and NMR analysis of their interactions with the model sequence Pu22 aided by molecular dynamics
PublikacjaIn recent years, new promising acridine derivatives have appeared, belonging to the unsymmetrical bisacridines (UAs) family with high anticancer activity. Both their physicochemical properties and their mechanism of action at the molecular level have not been thoroughly analyzed so far. Four derivatives were selected for the study, termed as: C-2028, C-2041, C-2045 and C-2053. The first aim of this work was to determine the protonation...
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Non-Adaptive Speed and Position Observer of Doubly-Fed Induction Generator
PublikacjaThe non-adaptive speed and position estimation of a doubly-fed induction generator (DFIG) is presented in this paper. The speed observer is based on the mathematical model of DFIG and to stabilize the structure the Lyapunov method is used. The classic stator field-oriented control to active and reactive power control is used in the sensorless control system. The performance of the proposed algorithm of a speed observer is validated...
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Space-mapping-based design flow of miniaturized broadband matching transformer with perforated metallization
PublikacjaA fast design procedure of unconventional passive components has been presented and experimentally validated on the basis of a wideband microstrip four-section matching transformer (50:6 OHm). A classic impedance matching circuit has been miniaturized by means of compact microstrip resonant cells (CMRCs) leading to a considerable length reduction (34%) together with minor degradation in its performance. The spacemapping-based design...
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Evaluation of Readiness of IT Organizations to Agile Transformation Based on Case-Based Reasoning
PublikacjaNowadays many of IT organization decides to change the way of delivering from classic, waterfall approach to agile. This transition is called “agile transformation” (AT). The problem of this process is that part of companies started AT without any analysis. This causes that many of transitions fails and organizations must return to old methods of delivering. Cost of return is significant and number of projects with violated project...
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Tyre dynamic radius determination
PublikacjaW artykule opisano stanowisko wykorzystywane do badania oporu toczenia opon samochodowych znajdujące się w Katedrze Konstrukcji Maszyn i Pojazdów Wydziału Mechanicznego Politechniki Gdańskiej. Przedstawiono wyniki badań promienia dynamicznego opony Michelin 165/80R13 83T z bieżnikiem CLASSIC przeprowadzone z wykorzystaniem tego stanowiska na nawierzchni Safety Walk 80. Badania przeprowadzono zmieniając: prędkość jazdy, obciążenie...
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Application of artificial intelligence into/for control of flexible manufacturing cell
PublikacjaThe application of artificial intelligence in technological processes control is usually limited. One problem is how to respond to changes in the environment of manufacturing system. A way to overcome the above shortcoming is to use fuzzy logic for representation of the inexact information. In this paper fundamentals of artificial intelligence and fuzzy logic are introduced from a theoretical point of view. Still more the fuzzy...
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An energetic analysis of a gas turbine with regenerative heating using turbine extraction at intermediate pressure - Brayton cycle advanced according to Szewalski's idea
PublikacjaIn this paper, a modification of a simple gas turbine into the Brayton cycle with regenerative heating, using turbine extraction at intermediate pressure, is presented. The main concept of the retrofitting is based on the transfer of heat from the turbine exhaust gases to the air entering the combustion chamber. The extracted gas transfers heat to air via the divided regenerative heat exchanger and after that is compressed and...
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Application of GC-MS/MS technique for the determination of benzodiazepines in blood samples
PublikacjaAbstract Benzodiazepines (BZD) are widely used as pharmaceuticals in medicine. However, due to psychostimulatory effect of BZD, in the last decade, they are more and more often used as drugs of abuse. These compounds produce similar effects to classical illicit drugs and are sold as “legal” alternatives to them as new psychoactive substances (NPS). Currently new BZD, named designer benzodiazepines (DBZD), are synthesized each year...
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GreedyMAX-type Algorithms for the Maximum Independent Set Problem
PublikacjaA maximum independent set problem for a simple graph G = (V,E) is to find the largest subset of pairwise nonadjacent vertices. The problem is known to be NP-hard and it is also hard to approximate. Within this article we introduce a non-negative integer valued functionp defined on the vertex set V(G) and called a potential function of agraph G, while P(G) = max{vinV(G)| p(v)} is called a potential of G. For any graph P(G) <= D(G),...
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On the deformation and frequency analyses of SARS-CoV-2 at nanoscale
PublikacjaThe SARS-CoV-2 virus, which has emerged as a Covid-19 pandemic, has had the most significant impact on people's health, economy, and lifestyle around the world today. In the present study, the SARS-CoV-2 virus is mechanically simulated to obtain its deformation and natural frequencies. The virus under analysis is modeled on a viscoelastic spherical structure. The theory of shell structures in mechanics is used to derive the governing...
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Active Control of Highly Autocorrelated Machinery Noise in Multivariate Nonminimum Phase Systems
PublikacjaIn this paper, a novel multivariate active noise control scheme, designed to attenuate disturbances with high autocorrelation characteristics and preserve background signals, is proposed. The algorithm belongs to the class of feedback controllers and, unlike the popular feedforward FX-LMS approach, does not require availability of a reference signal. The proposed approach draws its inspiration from the iterative learning control...
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Lagrangian model of an isolated dc-dc converter with a 3-phase medium frequency transformer accounting magnetic cross saturation
PublikacjaThis article presents a nonlinear equivalent circuit model of an isolated dc-dc converter with a 3-phase medium frequency transformer. The model takes into account the magnetic cross saturation of the 3-phase core-type magnetic circuit. The model is suitable in detailed electromagnetic transient simulations of power systems involving isolated dc-dc converters. The model is developed using the Lagrange energy method. It involves...
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Arithmetic Loophole in Bell's Theorem: Overlooked Threat to Entangled-State Quantum Cryptography
PublikacjaBell’s theorem is supposed to exclude all local hidden-variable models of quantum correlations. However,an explicit counterexample shows that a new class of local realistic models, based on generalized arith-metic and calculus, can exactly reconstruct rotationally symmetric quantum probabilities typical oftwo-electron singlet states. Observable probabilities are consistent with the usual arithmetic employedby macroscopic observers...
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Market Structure and Market Power in Selected Sectors of The Polish Economy Based on COICOP Classification
PublikacjaThis paper present new and simple measures of market structure and market power. Based on the classical models of market structures, where a given structure is determined by the number of enterprises, indexes of degree of monopoly have been estimated, representing an average number of entities per branch. Additionally, market power indexes have been determined as an average revenue per an enterprise in a given branch. This approach...
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Bridging challenges of clinical decision support systems with a semantic approach. A case study on breast cancer
PublikacjaThe integration of Clinical Decision Support Systems (CDSS) in nowadays clinical environments has not been fully achieved yet. Although numerous approaches and technologies have been proposed since 1960, there are still open gaps that need to be bridged. In this work we present advances from the established state of the art, overcoming some of the most notorious reported difficulties in: (i) automating CDSS, (ii) clinical workflow...
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Dynamic mass measurement in checkweighers using a discrete time-variant low-pass filter
PublikacjaConveyor belt type checkweighers are complex mechanical systems consisting of a weighing sensor (strain gauge load cell, electrodynamically compensated load cell), packages (of different shapes, made of different materials) and a transport system (motors, gears, rollers). Disturbances generated by the vibrating parts of such a system are reflected in the signal power spectra in a form of strong spectral peaks, located usually in...
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Numerical analysis of elastic wave propagation in unbounded structures
PublikacjaThe main objective of this paper is to show the effectiveness and usefulness of the concept of an absorbing layer with increasing damping (ALID) in numerical investigations of elastic wave propagation in unbounded engineering structures. This has been achieved by the authors by a careful investigation of three different types of structures characterised by gradually increasing geometrical and mathematical description complexities....