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Synthesis of new antrapyridazone derivatives - a novel group of anticancer agents active on a multidrugresistant(MDR) tumor cell lines
PublikacjaNovel antrapyridazone derivatives were synthesized and biologically evaluated in order tobroaden the data on structure-activity relationship of this class of cytostatics. Recent literaturedata prove that acetamides react better with aryl chlorides. A new approach based onintroduction of other amides form into aromatic ring in Ullmann was tested. This new methodcould give better yields and make purification step more convenient.
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New approach to noncausal identification of nonstationary stochastic systems subject to both smooth and abrupt parameter changes
PublikacjaIn this paper we consider the problem of finiteintervalparameter smoothing for a class of nonstationary linearstochastic systems subject to both smooth and abrupt parameterchanges. The proposed parallel estimation scheme combines theestimates yielded by several exponentially weighted basis functionalgorithms. The resulting smoother automatically adjustsits smoothing bandwidth to the type and rate of nonstationarityof the identified...
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Integrated production technology of cylindrical surfaces by turning and burnishing
PublikacjaThe method is based on a combination of previously used two separate operations namely machining and burnishing in a one complex operation implemented on a lathe.In the case of machining shafts and hydraulic cylinders of steel C45 is possible to obtain a surface roughness Ra=0,16 - 0,32 micrometers, dimensional accuracy class 7-8 according to ISO standards, and increase in the hardness of the surface up to 40%.
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Bilateral Multi-Issue Negotiation Between Active Documents and Execution Devices
PublikacjaMobile document-agents are often in conflict with execution devices when attempting to perform activities of the business process they implement, since preferences of device owners may change depending on their current location and the actual class of the device in use. The paper proposes a bilateral negotiation mechanism based on a simple bargaining game that can effectively resolve such conflicts without any third party support.
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Homoclinics for singular strong force Lagrangian systems
PublikacjaWe study the existence of homoclinic solutions for a class of generalized Lagrangian systems in the plane, with a C1-smooth potential with a single well of infinite depth at a point ξ and a unique strict global maximum 0 at the origin.Under a strong force condition around the singular point ξ, via minimization of an action integral, we will prove the existence of at least two geometrically distinct homoclinic solutions.
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UKŁADY KONSTRUKCYJNE LEKKIEJ OBUDOWY
PublikacjaW artykule przedstawiono rozwiązania konstrukcyjne przegród zewnętrznych lekkiej obudowy jednowarstwowych (nieizolowanych termicznie), wielowarstwowych (izolowanych termicznie) oraz szklano-metalowych. Omówiono procesy modyfikacji konstrukcji ścian. Podano przykładowe rozwiązania.
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Maximum temperature of 0.5-W infrared laser-Illuminated gold nanorod platforms
Dane BadawczeData concern a system consisted of two pieces of borosilicate glass surrounded by air and joined together by a transparent glue, which is to serve as a thermal transducer. On the top and bottom sides of the smaller piece, gold nanorods are dislocated. Glass is prepared here due to its high transparency, facilitating heat to be produced within the system....
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The structure of lead-borate glasses containing nanocrystallites of iron oxides
Dane BadawczeThe structure of iron-doped glasses and glass-ceramics were studied. Glass samples of composition of xFe2O3–(100 − x)(B2O3–2PbO) (2.5 b x b 37, in mol%) were prepared by the conventional melt quenching technique. The melting was conducted in alumina crucibles at the temperature of 1523 K. The melts were poured on a preheated (573 K) brass plate and...
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Nonlinear impedance as a function of A.C. voltage for glass 40Bi2VO5.5-60SrB4O7 annealed at 473 K for 3h and next fully crystallized measured with impedance spectroscopy method at high temperature region
Dane BadawczeThe nonlinear electrcial properties as a function of A.C. voltage for annealed at 473 K for 3h and next fully crystallized 40Bi2VO5.5-60SrB4O7 glass was measured by impedance spectroscopy method.
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Divide and not forget: Ensemble of selectively trained experts in Continual Learning
PublikacjaClass-incremental learning is becoming more popular as it helps models widen their applicability while not forgetting what they already know. A trend in this area is to use a mixture-of-expert technique, where different models work together to solve the task. However, the experts are usually trained all at once using whole task data, which makes them all prone to forgetting and increasing computational burden. To address this limitation,...
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COMPUTER-AIDED CONSTRUCTION AT DESIGNING REINFORCED CONCRETE COLUMNS AS PER EC
PublikacjaThe article presents the author’s computer program for designing and dimensioning columns in reinforced concrete structures taking into account phenomena affecting their behaviour and information referring to design as per EC. The computer program was developed with the use of C++ programming language. The program guides the user through particular dimensioning stages: from introducing basic data such as dimensions, concrete...
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Investigation of interaction between xanthene dye rhodamine B and metagenomic-derivated methylthioadenosine phosphorylase RSFP
PublikacjaIn the previous study we found that the expression of the metagenomic - derived methylthioadenosine phosphorylase gene (rsfp) in E. coli cells and the presence of rhodamine B in the growth medium were crucial for the pink fluorescence of one E. coli colony from Antarctic soil metagenomic library (Cieśliński et al., 2009). In this study, rsfp gene expression was induced by an arabinose promoter in an LMG194 E. coli strain and the...
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KOMPUTER W LABORATORIUM VS LABORATORIUM W KOMPUTERZE
PublikacjaAbstract. In March 2020, all of the sudden, university teachers have been made to run all the classes remotely. But, how to deal with lab classes for future engineers? Different aspects of teaching labs on Moodle, that should be taken in consideration, are not only connected with the content of the class, but also with transferring the knowledge and materials to the students in a way that would avoid distractions and help students...
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Tight bounds on the complexity of semi-equitable coloring of cubic and subcubic graphs
PublikacjaWe consider the complexity of semi-equitable k-coloring, k>3, of the vertices of a cubic or subcubic graph G. In particular, we show that, given a n-vertex subcubic graph G, it is NP-complete to obtain a semi-equitable k-coloring of G whose non-equitable color class is of size s if s>n/3, and it is polynomially solvable if s, n/3.
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Bell-Type Inequalities from the Perspective of Non-Newtonian Calculus
PublikacjaA class of quantum probabilities is reformulated in terms of non-Newtonian calculus and projective arithmetic. The model generalizes spin-1/2 singlet state probabilities discussed in Czachor (Acta Physica Polonica:139 70–83, 2021) to arbitrary spins s. For s → ∞ the formalism reduces to ordinary arithmetic and calculus. Accordingly, the limit “non-Newtonian to Newtonian” becomes analogous to the classical limit of a quantum theory
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Prediction of Processor Utilization for Real-Time Multimedia Stream Processing Tasks
PublikacjaUtilization of MPUs in a computing cluster node for multimedia stream processing is considered. Non-linear increase of processor utilization is described and a related class of algorithms for multimedia real-time processing tasks is defined. For such conditions, experiments measuring the processor utilization and output data loss were proposed and their results presented. A new formula for prediction of utilization was proposed...
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Aleksandra Parteka dr hab. inż.
OsobyAbout me: I am an associate professor and head of doctoral studies at the Faculty of Management and Economics, Gdansk University of Technology (GdanskTech, Poland). I got my MSc degree in Economics from Gdansk University of Technology (2003) and Universita’ Politecnica delle Marche (2005), as well as MA degree in Contemporary European Studies from Sussex University (2006, with distinction). I received my PhD in Economics...
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Continuation classes for a two-patch vaccination model
Dane BadawczeThis dataset contains selected results of rigorous numerical computations described in Section 5 of the paper "Rich bifurcation structure in a two-patch vaccination model" by D.H. Knipl, P. Pilarczyk, G. Röst, published in SIAM Journal on Applied Dynamical Systems (SIADS), Vol. 14, No. 2 (2015), pp. 980–1017, doi: 10.1137/140993934.
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On time-dependent nonlinear dynamic response of micro-elastic solids
PublikacjaA new approach to the mechanical response of micro-mechanic problems is presented using the modified couple stress theory. This model captured micro-turns due to micro-particles' rotations which could be essential for microstructural materials and/or at small scales. In a micro media based on the small rotations, sub-particles can also turn except the whole domain rotation. However, this framework is competent for a static medium....
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Physical and sealing properties of BaO–Al2O3–SiO2–CaO–V2O5 glasses for solid oxide fuel cell applications
PublikacjaIn this study, the properties of BaO–Al2O3–SiO2 (SAB) glasses incorporated with CaO and V2O5 as the network modifier and additive, respectively, are evaluated. The electrical resistivities of the glasses decrease upon the addition of CaO but increase upon increasing their V2O5 content because the V5+ species lower the ionic mobility of the glasses. The addition of V2O5 improves the wettability of the glasses on the Crofer 22 APU...
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Clay-filled starch films. Part I: Effect of clay kind and glycerol concentration on functional properties of composites
PublikacjaThe aim of this work was to improve the mechanical and water barrier properties of composite filmsprepared from starch and clays, plasticized with glycerol at different concentrations. The effects ofhydrophilic Closite Naþand Nanomer PGV were compared with that exerted by organicallymodifiedmorehydrophobicNanofil2 and NanoBent ZR-1. The antimicrobial activity of compositescontaining hydrophobic clays was also investigated. The hydrophilic...
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Towards a classification of networks with asymmetric inputs
PublikacjaCoupled cell systems associated with a coupled cell network are determined by (smooth) vector fields that are consistent with the network structure. Here, we follow the formalisms of Stewart et al (2003 SIAM J. Appl. Dyn. Syst. 2, 609–646), Golubitsky et al (2005 SIAM J. Appl. Dyn. Syst. 4, 78–100) and Field (2004 Dyn. Syst. 19, 217–243). It is known that two non-isomorphic n-cell coupled networks can determine the same sets of...
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Bioavailability of Tannins and Other Oligomeric Polyphenols: a Still to Be Studied Phenomenon
PublikacjaPurpose of Review Polyphenols are a group of plant secondary metabolites characterized with the presence ofmultiples of phenol structural units. Tannins are plant originated phenolic substances, which play an important role in plant defense system as well as have found applications in medicine, industry, and other fields of human activity. Despite these, the mechanisms of bioavailability of these substances are poorly studied and...
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UV Light-Modulated Fluctuation-Enhanced Gas Sensing by Layers of Graphene Flakes/TiO2 Nanoparticles
PublikacjaWe present experimental results of fluctuation-enhanced gas sensing by low-cost resistive sensors made of a mixture of graphene flakes and TiO2 nanoparticles. Both components are photocatalytic and activated by UV light. Two UV LEDs of different wavelengths (362 and 394 nm) were applied to modulate the gas sensing of the layers. Resistance noise was recorded at low frequencies, between 8 Hz and 10 kHz. The sensors’ response was...
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Non-Gaussian Resistance Fluctuations in Gold-Nanoparticle-Based Gas Sensors: An Appraisal of Different Evaluation Techniques
PublikacjaVolatile organic compounds, such as formaldehyde, can be used as biomarkers in human exhaled breath in order to non-invasively detect various diseases, and the same compounds are of much interest also in the context of environmental monitoring and protection. Here, we report on a recently-developed gas sensor, based on surface-functionalized gold nanoparticles, which is able to generate voltage noise with a distinctly non-Gaussian...
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Critical Remarks on Landauer’s principle of erasure– dissipation: Including notes on Maxwell demons and Szilard engines
PublikacjaWe briefly address Landauer’s Principle and some related issues in thermal demons. We show that an error-free Turing computer works in the zero-entropy limit, which proves Landauer’s derivation incorrect. To have a physical logic gate, memory or information-engine, a few essential components necessary for the operation of these devices are often neglected, such as various aspects of control, damping and the fluctuation–dissipation...
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Resistive gas sensors – Perspectives on selectivity and sensitivity improvement
PublikacjaResistive gas sensors are very popular and relatively inexpensive; they can operate at elevated or room temperature for years on end. The main disadvantage of resistive gas sensors is their limited selectivity and sensitivity, but various methods have been applied to improve their behavior. The composition of the porous gas sensing layer, or changes in the sensor’s operating temperature, can enhance the gas detection ability. Furthermore, emerging...
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Influence of controlled crystallization and SrF2 content on the structure and properties of Eu3+ doped phosphate glasses
PublikacjaNew phosphate glasses and glass-ceramics P2O5–Bi2O3–K2O–Nb2O5-SrF2 doped with Eu were synthesized and studied in this work. The influence of the SrF2 content (0–15 mol%) and the parameters of the heat treatment on their structural and optical properties were investigated. For the above purpose, the structural characterization by FTIR spectroscopy and XRD measurements was carried out, which showed a significant effect of SrF2 on...
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Szyby zespolone w systemach fasadowych
PublikacjaW artykule przedstawiono wybrane kryteria techniczne stosowane do oceny jakościowej izolacyjnych szyb zespolonych. Bazując na własnych doświadczeniach, autor zwrócił uwagę na pojawiające się problemy w trakcie odbiorów technicznych na budowie. Przedstawiono także krótki przegląd literatury z zakresu szkła budowlanego i szyb zespolonych.
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DBpedia and YAGO as Knowledge Base for Natural Language Based Question Answering—The Evaluation
PublikacjaThe idea of automatic question answering system has a very long history. Despite constant improvement of the systems asking questions in the natural language requires very complex solutions. In this paper the DBpedia and YAGO are evaluated as a knowledge bases for simple class 1 and 2 question answering system. For this purpose a question answering system was designed and implemented. The proposed solution and the knowledge bases...
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The complexity of zero-visibility cops and robber
PublikacjaWe consider the zero-visibility cops & robber game restricted to trees. We produce a characterisation of trees of copnumber k and We consider the computational complexity of the zero-visibility Cops and Robber game. We present a heavily modified version of an already-existing algorithm that computes the zero-visibility copnumber of a tree in linear time and we show that the corresponding decision problem is NP-complete on a nontrivial...
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Some Progress on Total Bondage in Graphs
PublikacjaThe total bondage number b_t(G) of a graph G with no isolated vertex is the cardinality of a smallest set of edges E'⊆E(G) for which (1) G−E' has no isolated vertex, and (2) γ_t(G−E')>γ_t(G). We improve some results on the total bondage number of a graph and give a constructive characterization of a certain class of trees achieving the upper bound on the total bondage number.
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History of World Architecture I 2021/22
Kursy OnlineThe course History of World Architecture (HWA I) is obligatory on the first semester of study at the Faculty of Architecture at Gdańsk University ofTechnology. It lasts 15 weeks, finishes with the exam, and consists of 15 two-hour lectures and 15 two-hour exercises. The merit of the course includes Western World architecture, beginning from Prehistory and Antiquity (Sumer, Egypt, Greece, Rome), up to the end of the Middle Ages....
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The generalization by simplification operator with Sester’s method of objects representing groups of buildings in Gdańsk district - scale 1:10000. Data from OSM
Dane BadawczeThe process of automatic generalization is one of the elements of spatial data preparation for the purpose of creating digital cartographic studies. The presented data include a part of the process of generalization of building groups obtained from the Open Street Map databases (OSM) [1].
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Effect of composition on the thermal properties and structure of M-Al-Si-O-N glasses, M = Na, Mg, Ca
PublikacjaThe primary objective of this study is to explore the relationship between the composition, structure, and thermal characteristics of M-Al-Si-O-N glasses, with M representing sodium (Na), magnesium (Mg), or calcium (Ca). The glasses were prepared by melting in a quartz crucible at 1650 °C and AlN precursor (powder) was utilized as a nitrogen source. The measured thermal properties studied were glass transition temperature (Tg),...
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General paradigm for distilling classical key from quantum states
PublikacjaIn this paper, we develop a formalism for distilling aclassical key from a quantum state in a systematic way, expandingon our previous work on a secure key from bound entanglement(Horodecki et al., 2005). More detailed proofs, discussion, andexamples are provided of the main results. Namely, we demonstratethat all quantum cryptographic protocols can be recast in away which looks like entanglement theory, with the only changebeing...
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eGlasses e-Glass - Interaktywne okulary dla potrzeb mobilnego przetwarzania informacji o postrzeganym otoczeniu
ProjektyProjekt realizowany w Katedra Inżynierii Biomedycznej zgodnie z porozumieniem ERA-NET-CHIST-ERA-II /01/ 2013 z dnia 2013-12-31
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A graphical approach to yield and boundary surfaces of selected hypoplastic constitutive equations
PublikacjaThe article describes how to identify the boundary and yield surface for hypoplastic constitutive equations proposed by Wu, Gudehus and Bauer. It is shown how to identify and plot the surfaces for any equation in this class. Calculation errors are analyzed characteristic for appleid set of numerical formulas. In the paper there are computer links to the source code prepared in the MATLAB system, based on istructions in the article....
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Generalized Gradient Equivariant Multivalued Maps, Approximation and Degree
PublikacjaConsider the Euclidean space Rn with the orthogonal action of a compact Lie group G. We prove that a locally Lipschitz G-invariant mapping f from Rn to R can be uniformly approximated by G-invariant smooth mappings g in such a way that the gradient of g is a graph approximation of Clarke’s generalized gradient of f . This result enables a proper development of equivariant gradient degree theory for a class of set-valued gradient...
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The database of indices computed from RR-intervals of length 512 of 41 patients at rest hospitalized due to the episode of acute ischemic stroke
Dane BadawczeThis dataset contains the data that was a basis for the results discussed in the paper “Persistent homology as a new method of the assessment of heart rate variability” by Grzegorz Graff, Beata Graff, Paweł Pilarczyk, Grzegorz Jabłoński, Dariusz Gąsecki, Krzysztof Narkiewicz, Plos One (2021), DOI: 10.1371/journal.pone.0253851.
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The database of interpolated RR-intervals of original length 512 of 41 patients at rest hospitalized due to the episode of acute ischemic stroke
Dane BadawczeThis dataset contains the data that was a basis for the results discussed in the paper “Persistent homology as a new method of the assessment of heart rate variability” by Grzegorz Graff, Beata Graff, Paweł Pilarczyk, Grzegorz Jabłoński, Dariusz Gąsecki, Krzysztof Narkiewicz, Plos One (2021), DOI: 10.1371/journal.pone.0253851.
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The database of indices computed from RR-intervals of length 512 of 46 healthy subjects at rest
Dane BadawczeThis dataset contains the data that was a basis for the results discussed in the paper “Persistent homology as a new method of the assessment of heart rate variability” by Grzegorz Graff, Beata Graff, Paweł Pilarczyk, Grzegorz Jabłoński, Dariusz Gąsecki, Krzysztof Narkiewicz, Plos One (2021), DOI: 10.1371/journal.pone.0253851.
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The database of interpolated RR-intervals of length 512 of 46 healthy subjects at rest
Dane BadawczeThis dataset contains the data that was a basis for the results discussed in the paper “Persistent homology as a new method of the assessment of heart rate variability” by Grzegorz Graff, Beata Graff, Paweł Pilarczyk, Grzegorz Jabłoński, Dariusz Gąsecki, Krzysztof Narkiewicz, Plos One (2021), DOI: 10.1371/journal.pone.0253851.
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PROJEKT ZESPOŁOWY [DK][2023/24]
Kursy OnlineCCCLECTURE and Classes: Power supply systems for industrial facilities. Devices and main circuits of MV power stations. Short-circuit calculation. Power protection automation. Security classification according to American ANSI standards used in the EU. Microprocessor protection relays. Drive systems for medium power and medium voltage pumps. Roving inverters. PROJECT: Design of a MV switching station for a medium-power pumping...
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PROJEKT ZESPOŁOWY [ET][DK][2024/25]
Kursy OnlineCCCLECTURE and Classes: Power supply systems for industrial facilities. Devices and main circuits of MV power stations. Short-circuit calculation. Power protection automation. Security classification according to American ANSI standards used in the EU. Microprocessor protection relays. Drive systems for medium power and medium voltage pumps. Roving inverters. PROJECT: Design of a MV switching station for a medium-power pumping...
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Wiktor Sieklicki dr inż.
OsobyTytuł magistra oraz inżyniera uzyskał w specjalności Automatyka i Robotyka w Katedrze Mechaniki i Wytrzymałości Materiałów Wydziału Mechanicznego Politechniki Gdańskiej (2006). Tytuł doktora nauk technicznych w dyscyplinie Budowa Maszyn uzyskał w 2010 roku na Wydziale Mechanicznym PG (2010). Od 2010 roku zatrudniony na stanowisku Adiunkta w Katedrze Mechaniki i Mechatroniki Wydziału Mechanicznego PG. W latach 2011-2013 zatrudniony...
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On the origin of surface imposed anisotropic growth of salicylic and acetylsalicylic acids crystals during droplet evaporation
PublikacjaIn this paper droplet evaporative crystallization of salicylic acid (SA) and acetylsalicylic acid (ASA) crystals on different surfaces, such as glass, polyvinyl alcohol (PVA), and paraffin was studied. The obtained crystals were analyzed using powder X-ray diffraction (PXRD) technique. In order to better understand the effect of the surface on evaporative crystallization, crystals deposited on glass were scraped off. Moreover,...
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DC and AC Conductivity, Biosolubility and Thermal Properties of Mg-Doped Na2O–CaO–P2O5 Glasses
PublikacjaBioactive glasses have recently been extensively used to replace, regenerate, and repair hard tissues in the human body because of their ability to bond with living tissue. In this work, the effects of replacing Na2O with MgO on the electrical, biosolubility, and thermal properties of the target glass 10Na2O–60P2O5–30CaO (in mol%) were investigated. The electrical properties of the glasses were studied with the impedance spectroscopy...
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New Approach to Noncasual Identification of Nonstationary Stochastic FIR Systems Subject to Both Smooth and Abrupt Parameter Changes
PublikacjaIn this technical note, we consider the problem of finite-interval parameter smoothing for a class of nonstationary linear stochastic systems subject to both smooth and abrupt parameter changes. The proposed parallel estimation scheme combines the estimates yielded by several exponentially weighted basis function algorithms. The resulting smoother automatically adjusts its smoothing bandwidth to the type and rate of nonstationarity...
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Quantum corrections to quasi-periodic solution of Sine-Gordon model and periodic solution of phi^4 model
PublikacjaAnalytical form of quantum corrections to quasi-periodic solution of Sine-Gordon model and periodic solution of phi^4 model is obtained through zeta function regularisation with account of all rest variables of a d-dimensional theory. Qualitative dependence of quantum corrections on parameters of the classical systems is also evaluated for a much broader class of potentials u(x) = b^2 f(bx) + C with b and C as arbitrary real constants