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(4-(Bis(4-Fluorophenyl)Methyl)Piperazin-1-yl)(Cyclohexyl)Methanone Hydrochloride (LDK1229): A New Cannabinoid CB1 Receptor Inverse Agonist from the Class of Benzhydryl Piperazine Analogs
PublicationSome inverse agonists of cannabinoid receptor type 1 (CB1) have been demonstrated to be anorectic antiobesity drug candidates. However, the first generation of CB1 inverse agonists, represented by rimonabant (SR141716A), otenabant, and taranabant, are centrally active, with a high level of psychiatric side effects. Hence, the discovery of CB1 inverse agonists with a chemical scaffold distinct from these holds promise for developing...
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PODEJŚCIE WARIANTOWE WE WSTĘPNYM PROJEKTOWANIU STATKÓW Variant methods approach to the preliminary ship design.
PublicationKlasyczna metoda projektowania okrętów jest metodą iteracyjną, bazującą na zgromadzonym doświadczeniu ze statków już zbu-dowanych. Natomiast w przypadku statku całkowicie nowego typu, bez „posagu wcześniejszych doświadczeń”, projektowanie polega na opracowaniu szeregu równoległych, wariantowych rozwiązań z wykorzystaniem optymalizacji. Artykuł wskazuje wybrane metody projektowe wykorzystujące optymalizacje, używane we wstępnym...
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The role and importance of WIMAX mobile system as a high-performance data transfer technology in wireless sensor networks for wide area monitoring applications
PublicationThe study discuses basic features and functional design of WiMAX Mobile system, based on the IEEE 802.16e (Release 1.5 Rev. 2.0) standard. The analysis has been made in terms of ability to use this system to transmit video stream related to monitoringof large agglomeration areas. What is more, the study includes comparison of technical parameters of WiMAX Mobile system with competitive systems such as: HSPA+ and UMTS-LTE, which...
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ANALYSIS OF THE INCREASE OF CONSTRUCTION COSTS IN URBAN REGENERATION PROJECTS
PublicationThe subject of this paper is the analysis and evaluation of the reasons for construction costs increases in urban regeneration projects. The analysis considers major refurbishments of real estates’, as well as heavy repair and modernization of the road system. For the period mentioned, the costs from works and expenditure schedules were compared with the costs of additional works, which shows the percentage cost increase in relation...
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Implementation of TVDI calculation for coastal zone
PublicationPaper will show an implementation of TVDI (Temperature-Vegetation-Dryness Index) algorithm on GPU (Graphics Processing Unit). Calculation of this index is based on LST (Land Surface Temperature) and NDVI (Normalized Difference Vegetation Index). Discussed results are based on multi-spectral imagery retrieved from AVHRR3 sensors for area of Poland, especially from region of Gdańsk coastal zone. All phases of TVDI implementation...
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The impact of environmentally friendly refrigerants on heat pump efficiency
PublicationThis paper discusses the issue of heat pump simulation. Lower operating costs can be achieved through good equipment design and appropriate operation. Detailed technical and economic analysis inform the selection of system components with the highest possible efficiency and lower energy demand. The use of systems based on environmentally friendly refrigerants can deliver long product life, which is associated with a shorter payback...
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Maritime heritage of small port towns of the Polish coast
PublicationThe article describes problems of the gradual disappearance of real maritime heritage in small Polish port cities. The maritime heritage of small port cities was shaped by coastal processes and urban historical conditions what has led to creation of specific types of landscapes. Special architectural objects of the post-port heritage of small ports of the Polish coast are hydrotechnical constructions (i.e. breakwaters, quays),...
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Impact of probability distribution on the uncertainty of resistance measurement
PublicationThe paper presents studies on the influence of probability distributions on the expanded uncertainty of the resistance measurement. Choosing the correct probability distribution is very important to estimate of measurement uncertainty. The paper presents the results of analysis of the resistance measurement uncertainty using the technical method of resistance: 100 G. The analysis of the uncertainty...
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A Device for Measuring Auditory Brainstem Responses to Audio
PublicationStandard ABR devices use clicks and tone bursts to assess subjects’ hearing in an objective way. A new device was developed that extends the functionality of a standard ABR audiometer by collecting and analyzing auditory brainstem responses (ABR). The developed accessory allows for the use of complex sounds (e.g., speech or music excerpts) as stimuli. Therefore, it is possible to find out how efficiently different types of sounds...
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TIRE/ROAD NOISE AND TIRE ROLLING RESISTANCE ON PROTOTYPE PERS SURFACE
PublicationPoroelastic road surfaces are characterized by low noise of tires running on them.Road pavements of this type are promising solution to problems related to traffic noise in cities and on rural roads. Some technical problems still have to be solved, in particular regarding durability and skid resistance on wet surface. Ongoing and planned works are to contribute to create a quiet, durable and safe road surface, which will become...
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Interdisciplinarity in Smart Sustainable City education: exploring educational offerings and competencies worldwide
PublicationMore and more higher education institutions are offering specialized study programs for current and future managers of Smart Sustainable Cities (SSCs). In the process, they try to reconcile the interdisciplinary nature of such studies, covering at least the technical and social aspects of SSC management, with their own traditionally discipline-based organization. However, there is little guidance on how such interdisciplinarity...
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The role of robotisation in improving bakery product quality
PublicationThe article aims to present the role of robotisation in increasing bakery product quality, as it is closely linked to machine reliability, as well as hygienic and sanitary conditions. All machines employed in the production process ought to be maintained at full production potential and reliability, which also has a fundamental influence on the final product’s quality. While participating in the 2014-2020 Smart Growth Operational...
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Analysis of the state of preservation the historic arcaded houses in Vistula Delta listed in the National Inventory of Historical Monuments
PublicationHistoric arcaded houses are part of the material heritage of the Vistula Delta. Unfortunately, their number is decreasing year by year. The article is the result of a query of available sources and field research carried out by the author in 2015-2020. The paper presents the current state of preservation the historic arcaded houses in Vistula Delta listed in the National Inventory of Historical Monuments. Criteria for the selection...
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Assessment of Wooden Beams from Historical Buildings Using Ultrasonic Transmission Tomography
PublicationThe main goal of this study was non-destructive evaluation of wooden elements using ultrasonic waves. The inspection was carried out on wooden beams from a historical object. Elastic wave signals were processed by ultrasonic transmission tomography to obtain imaging of the internal structure of tested elements without disturbing their state and integrity. The focus was on the influence of wood anisotropy on the propagation of ultrasonic...
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COMPARATIVE ANALYSIS OF TRANSPORT ORGANIZATION AND FUNCTIONING OF WATER TRAMS IN GDAŃSK, BYDGOSZCZ AND KRAKÓW
PublicationThe subject of this work is to identify and juxtapose solutions implemented in transport provided by water trams for the following cities: Gdańsk, Bydgoszcz and Kraków. As a result of the conducted analysis of transport factors, the degree of conformity of project objectives to the actual role of the water tram has been determined. It was found that the Kraków Water Tram (also known as Cracow Water Tram) is characterized by the...
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Ocena stanu technicznego konstrukcji zgarniaczy będących na wyposażeniu osadników wstępnych Grupowej Oczyszczalni Ścieków „DĘBOGÓRZE
PublicationOsadniki wstępne typu DORRA – 4 szt., o pojemności 1830 m3, wyposażone są w elementy mechaniczne do kierunkowego przemieszczania się osadu w kierunku leja centralnego. Celem pracy jest ocena stany technicznego części mechanicznej, a w szczególności: - konstrukcji zespołu zgarniania części pływających oraz osadu. - zespołu napędu i sterowania, - zespołu napędu i jazdy. Pierwsze dwa zespoły będą oceniane również z punktu widzenia...
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Bilansowanie lokalne w systemie elektroenergetycznym
PublicationWprowadzenie rozliczeń rynkowych w handlu energią elektryczną wymusiło nowe podejście do krótkookresowego bilansowania energii w systemie elektroenergetycznym. Dla sprawnego funkcjonowania handlu energią, konieczne było wprowadzenie Rynku Bilansującego, łączącego realizację zadań technicznych i handlowych. Obecnie bilansowanie systemu rozwiązywane jest ogólnosystemowo. Decentralizacja procesu wytwarzania energii, rozwój niespokojnych...
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Does technology matter for economic development? Empirical evidence for Latin American Countries
PublicationThe spread of new Information and Communication Technologies (ICTs) has been recognized worldwide. ICTs are broadly perceived as tools facilitating economic growth and development, especially in backward countries. They are easy and cheap to adopt, require minimum skills for effective use, and bring opportunities for disadvantaged societies. They enable education, knowledge dissemination and sharing, and processing and storing...
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Machine Learning Techniques in Concrete Mix Design
PublicationConcrete mix design is a complex and multistage process in which we try to find the best composition of ingredients to create good performing concrete. In contemporary literature, as well as in state-of-the-art corporate practice, there are some methods of concrete mix design, from which the most popular are methods derived from The Three Equation Method. One of the most important features of concrete is compressive strength, which...
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RACIAL COMPOSITION OF COMMUNITIES AND PARTICIPATION OF ADOLESCENTS
PublicationThe investigation used the Add Health data set to examine the association between communities’ composition with respect to race and participation in extracurricular school activities in secondary education. Results of this analysis show that the composition of adolescents’ communities matters for individuals’ participation outcomes in extracurricular school activities. The results find further support in previous research connecting...
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TEORIA DECYZYJNYCH PROCESÓW SEMI-MARKOWA I JEJ ZASTOSOWANIE W PROJEKTOWANIU I EKSPLOATACJI OKRĘTOWYCH SILNIKÓW GŁÓWNYCH I INNYCH URZĄDZEŃ SIŁOWNI OKRĘTOWYCH
PublicationW referacie zaprezentowano znaczenie teorii procesów semi-Markowa w naukach technicznych, zwłaszcza w teorii niezawodności urządzeń technicznych, teorii bezpieczeństwa ich działania oraz statystycznej teorii podejmowania decyzji eksploatacyjnych. W referacie wyeksponowano także przydatność teorii procesów semi-Markowa w teorii i praktyce eksploatacji wspomnianych urządzeń technicznych na przykładzie tak istotnych urządzeń w transporcie...
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Analiza drgań przewodu jezdnego sieci trakcyjnej w aspekcie oceny jej stanu technicznego.
PublicationGórna sieć trakcyjna jest nadal najefektywniejszym sposobem zasilania kolejowych pojazdów elektrycznych. Sieć jezdna nie ma możliwości technicznych redundancji, co wymaga okresowej oceny stanu technicznego w celu zapewnienia prawidłowej współpracy z odbierakami prądu pojazdów. W artykule przedstawiono aspekty oceny stanu technicznego górnej sieci trakcyjnej na podstawie modelowania matematycznego i wybranych badań laboratoryjnych....
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WYMAGANIA STAWIANE LEKKIEJ OBUDOWIE
PublicationW artykule omówiono wymagania stawiane lekkim obudowom. Przywołano odpowiednie normy i rozporządzenia dotyczące zagadnień ogólnobudowlanych i techniczno-użytkowych.
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Razem czy osobno - zespoły a działania przedsiębiorcze
PublicationPrzedsiębiorczość rozumiana jako atrybut jednostki, charakteryzowana jest ponad 40 pojęciami. Wiadomo jest jednak, że zakres i różnorodność kompetencji pojedynczej osoby jest zazwyczaj mniejszy niż zespołu. Jednostka może posiadać wybitną wiedzę, niezwykły poziom umiejętności i ogromne doświadczenie, ale ich zakres może zostać rozszerzony o właściwie dobrane kompetencje innej jednostki. Z drugiej strony zarówno działania zespołowe...
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Grade of service determination methodology in IP networks with SIP protocol
PublicationAlthough Grade of Service is very important in VoIP providers evaluation, We wasn't able to find any paper regarding the topic of measuring GoS variables for IP networks utilizing SIP, which are defined like for PSTN/ISDN/GSM networks (post-selection delay, answering delay, release delay, or probability of end-to-end blocking). Due to the lack of research in this field, it was necessary to start from defining measures and cover...
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Modern approaches to file system integrity checking
PublicationOne of the means to detect intruder's activity is totrace all unauthorized changes in a file system.Programs which fulfill this functionality are called fileintegrity checkers. This paper concerns modernapproach to file system integrity checking. It reviewsarchitecture of popular systems that are widely used inproduction environment as well as scientific projects,which not only detect intruders but also take actions tostop their...
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Finite Element Method Applied in Electromagnetic NDTE: - A Review
PublicationThe paper contains an original comprehensive review of finite element analysis (FEA) applied by researchers to calibrate and improve existing and developing electromagnetic non-destructive testing and evaluation techniques, including but not limited to magnetic flux leakage (MFL), eddy current testing, electromagnetic-acoustic transducers (EMATs). Premium is put on the detection and modelling of magnetic field, as the vast majority...
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New oryginal generic technologies: A Polish R&D strategic implementation programme
PublicationPolands's pharmaceutical industry is of great significance to the whole economy. According to Forbs (2 October 2012), the cost of launching a new drug varies from USD 1 to 11 bilion. There is little Chance of a Polish pharmaceutical company developing an original drug due to financial reason.Many research teams in Poland take up research projects aimed at new biologically active compounds. But such an objective has no broader perspective,...
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Extraction of information from born-digital PDF documents for reproducible research
PublicationBorn-digital PDF electronic documents might reasonably be expected to preserve useful data units of their source originals that suffice to produce executable papers for reproducible research. Unfortunately, developers of authoring tools may adopt arbitrary PDF generation strategies, producing a plethora of internal data representations. Such common information units as text paragraphs, tables, function graphs and flow diagrams,...
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Ergonomics in Polish outpatient clinics
PublicationOutpatient clinics are structures In which ergonomics play a key role. This fact is associated with an often occurring risk of developing hospital-acquired infection. The risk increases with mistakes made in wrong planning the functional and spatial lay-out is subordinated to high utilitarian requirements, including hygienic and sanitary, and technological requirements. A properly planned structure allows to reduce dangers more...
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Inseparability criteria based on matrices of moments
PublicationInseparability criteria for continuous and discrete bipartite quantum states based on moments of annihilationand creation operators are studied by developing the idea of Shchukin-Vogel criterion Phys. Rev. Lett. 95,230502 2005. If a state is separable, then the corresponding matrix of moments is separable too. Thus, wederive generalized criteria based on the separability properties of the matrix of moments. In particular, acriterion...
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The study of Arduino Uno feasibility for DAQ purposes
PublicationUsing microcontroller systems becomes a routine in various measurement and control tasks. Their wide availability together with a huge potential of extending their functionality by additional modules allows developing advanced measuring and monitoring systems by non-specialists. However, using popular example codes often leads the user to pass over or not to be aware of the limitations of the system and drawing too far-reaching...
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Sewage sludge pretreatment by low thermal disintegration for better efficacy of sludge digestion process
PublicationThe wastewater water treatment plant (WWTP) sector and it is developing technologies strive to be implement circular economy. The methane production from the sludge digestion process constitute promising source of the renewable energy for WWTP and approaching circular economy assumptions. For this reason, the objective of the study was to examine the modification of sludge characteristics due to the low temperature pretreatment....
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Structural Reliability Assessment Of Corroded Tanker Ship Based On Experimentally Estimated Ultimate Strength
PublicationThis work deals with the reliability assessment of a tanker ship hull structure subjected to a vertical bending moment and corrosion degradation. The progressive collapse and ultimate load carrying capacity are estimated based on experimentally tested scaled box-shaped-specimens. The translation of the strength estimate of the scaled specimen to the real tanker ship hull structure is performed based on the dimensional theory developing...
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OPTIMALIZATION OF SORBENT FEEDING IN THE DRY METHOD OF FLUE GAS DESULFURIZATION
PublicationThe swiftly developing sea transport contributes to a considerable increase of fuel usage in the international shipping, which results in the escalation of toxic compounds emitted into the atmosphere. It is followed by the constantly heightened requirements limiting those emissions. In the case of sulfur oxide emission, inside of SECA (Sulfur Emission Control Area), the maximum content of sulfur in the shipping fuels used on the...
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Development of tools for road infrastructure safety management for the provinces (voivodeships) in Poland
PublicationThe development of modern tools for road infrastructure safety management will help to reduce the number of fatalities and serious injuries as one of the main objectives adopted in 2013 in the National Road Safety Programme 2014-2020 and the new Road Safety Programme 2011-2020 in the EU. Risk Management in Highway Engineering can be applied in developing tools essential in the process of safety management. Risk Management in Highway...
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From Linear Classifier to Convolutional Neural Network for Hand Pose Recognition
PublicationRecently gathered image datasets and the new capabilities of high-performance computing systems have allowed developing new artificial neural network models and training algorithms. Using the new machine learning models, computer vision tasks can be accomplished based on the raw values of image pixels instead of specific features. The principle of operation of deep neural networks resembles more and more what we believe to be happening...
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Design of control algorithms for mobile robots in an environment with static and dynamic obstacles
PublicationThis article proposes the construction of autonomous mobile robots and designing of obstacle avoidance algorithms for them. Nowadays, mobile robots are gaining more and more popularity on the customer as well as industrial market, for example as automatic vacuum cleaners or lawnmowers. Obstacle avoidance algorithms play an important role in performance of this types of robots. The proposed algorithms were designed for builds with...
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Parametric method applicable in assessing breakout force and time for lifting slender bodies from seabed
PublicationThe article presents a parametric method applicable in assessing the suction force of a slender body to the seabed, and prognosing the body extrication time. Along with the body weight in water, the information on the suction force is essential for assessing the force needed to lift the object from the seabed. Based on the Foda theory and the resulting integral equation, which relates the maximum suction force with basic parameters...
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Evolutionary Sets of Safe Ship Trajectories: improving the method by adjusting evolutionary techniques and parameters
PublicationThe paper presents some of the evolutionary techniques used by the evolutionary sets of safe ship trajectories method. In general, this method utilizes a customized evolutionary algorithm to solve a constrained optimization problem. This problem is defined as finding a set of cooperating trajectories (here the set is an evolutionary individual) of all the ships involved in the encounter situation. The resulting trajectories are...
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WHAT DRIVES CROSS-COUNTRY DIFFERENCES IN EXPORT VARIETY? A BILATERAL PANEL APPROACH
PublicationA worldwide event like the 2020 Coronavirus outbreak can only reinforce the interest in modelling trade diversification as a key factor in countries’ vulnerability to external shocks. This paper adopts a detailed relative framework to study the determinants of product-level export variety in a large bilateral panel of developing and developed economies (16,770 country pairs in the period 1988–2014). We find that country pairs characterized...
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Preeclampsia Risk Prediction Using Machine Learning Methods Trained on Synthetic Data
PublicationThis paper describes a research study that investigates the use of machine learning algorithms on synthetic data to classify the risk of developing preeclampsia by pregnant women. Synthetic datasets were generated based on parameter distributions from three real patient studies. Four models were compared: XGBoost, Support Vector Machine (SVM), Random Forest, and Explainable Boosting Machines (EBM). The study found that the XGBoost...
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Trends in the new generation of green solvents in extraction processes
PublicationAnalytical chemistry, like other scientific fields, has undergone a number of changes to make it more consistent with the concept of sustainable development. Among the various steps of chemical analysis, without a doubt, sample preparation is the bottleneck in regard to following a green protocol, especially in terms of solvent consumption. Therefore, many attempts have been made to improve the environmental friendliness of this...
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Diiodo-BODIPY Sensitizing of the [Mo3S13]2– Cluster for Noble-Metal-Free Visible-Light-Driven Hydrogen Evolution within a Polyampholytic Matrix
PublicationWe report on a photocatalytic setup that utilizes the organic photosensitizer (PS) diiodo-BODIPY and the non-precious-metal-based hydrogen evolution reaction (HER) catalyst (NH4)2[Mo3S13] together with a polyampholytic unimolecular matrix poly(dehydroalanine)-graft-poly(ethyleneglycol) (PDha-g-PEG) in aqueous media. The system shows exceptionally high performance with turnover numbers (TON > 7300) and turnover frequencies (TOF...
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The Lost Kinetic Architecture and How to Reintroduce it in the Landscape – The Case Study of the Drainage Windmills in the Vistula Delta
PublicationRecreating the lost kinetic landscape of the Vistula Delta is a considerable challenge. The study aims to propose a method for reproducing windmills and their effect on the landscape. The paper suggests a method based on the transposition of the forms of movement from windmills historically present in the region to modern forms. The method is based on a series of analyses starting with the study of the region and its history followed...
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Towards Cancer Patients Classification Using Liquid Biopsy
PublicationLiquid biopsy is a useful, minimally invasive diagnostic and monitoring tool for cancer disease. Yet, developing accurate methods, given the potentially large number of input features, and usually small datasets size remains very challenging. Recently, a novel feature parameterization based on the RNA-sequenced platelet data which uses the biological knowledge from the Kyoto Encyclopedia of Genes and Genomes, combined with a classifier...
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A numerical and experimental analysis of multi-hole orifice in turbulent flow
PublicationIn this research study, the comprehensive metrological analysis is investigated for a 4-hole orifice with module m = 0.25 installed in the pipeline with an internal diameter of 50 mm. A detailed numerical simulation was performed for the turbulence models: k-ε-realizable and k-ω-BSL. The novelties of the research include model validation by comparing the results of numerical studies with the experiment conducted in the area of...
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Selected biotrends in development of epoxy resins and their composites
PublicationEpoxy resins and their fibre or particulate composites are widely used in various industries, including building, naval, aircraft, automotive and aerospace. Modern polymer science and technology focus on the development of green polymers and composites. There are two major areas of interest in the case of epoxy resins: the development of bio-based resins and the production of composites with natural fibers. One of the most interesting...
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Numerical Model of the Aortic Valve Implanted Within Real Human Aorta
PublicationCardiovascular system diseases are the main cause of deaths in developed and developing countries. The main reasons are myocardial infarction, heart failure, stroke and valvular diseases. These are caused mainly by arteriosclerosis. The valvular diseases involve a significant burden for the health care system and their frequency is rising with the patient age. This work describes the tools and numerical models appropriate for modeling...
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Miniaturized Solid Phase Extraction techniques for different kind of pollutants analysis: State of the art and future perspectives – PART 1
PublicationSolid Phase Extraction (SPE) has been practiced in a modern form for more than half a century. It was constantly developing, driven by the analysts needs. These needs are coming from the importance to select an appropriate analytical method, which should have satisfactory accuracy, precision and sensitivity. In the case of sorbent-based microextraction techniques, the choice of miniaturized variants that meet these requirements...