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Search results for: STATIC IN VITRO DISSOLUTION
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Fluvial ecology disasters: the impact of the Gliwice Canal on the ecological crisis in the Oder River basin, Poland (2022)
PublicationIn August 2022, the Oder River experienced an ecological disaster, resulting in the extinction of hundreds of aquatic organ- isms. Mass fsh deaths also occurred during that time in the Gliwice Canal, located in southern Poland, which connects to the upper section of the Oder River. The aim of the article was to assess the impact of the waters from the Gliwice Canal on the water quality changes in the Oder River, as expressed by...
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Classification of submandibular salivary stones based on ultrastructural studies
PublicationIntroduction: Sialolithiasis remains a clinical problem with unclear etiopathogenesis, lack of prevention methods, and only surgical treatment. Materials and methods: An ultrastructure examination of submandibular sialoliths obtained from patients with chronic sialolithiasis was conducted using a scanning electron microscope and X‐ray photoelectron spectroscopy. Results: Based on the results, we divided sialoliths into three types:...
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Experimental Study on Dynamics of Wooden House Wall Panels with Different Thermal Isolation
PublicationWood frame buildings are very popular in regions that are exposed to different dynamic excitations including earthquakes. Therefore, their seismic resistance is really important in order to prevent structural damages and human losses. The aim of the present paper is to show the results of experimental tests focused on the dynamic response of wall panels of a wooden frame building with thermal isolation made of mineral wool and...
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Correlation–polarization effects in electron/positron scattering from acetylene: A comparison of computational models
PublicationDifferent computational methods are employed to evaluate elastic (rotationally summed) integral and differential cross sections for low energy (below about 10 eV) positron scattering off gas-phase C2H2 molecules. The computations are carried out at the static and static-plus-polarization levels for describing the interaction forces and the correlation–polarization contributions are found to be an essential component for the correct...
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Generating optimal paths in dynamic environments using RiverFormation Dynamics algorithm
PublicationThe paper presents a comparison of four optimisation algorithms implemented for the purpose of finding the shortest path in static and dynamic environments with obstacles. Two classical graph algorithms –the Dijkstra complete algorithm and A* heuristic algorithm – were compared with metaheuristic River Formation Dynamics swarm algorithm and its newly introduced modified version. Moreover, another swarm algorithm has been compared...
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Dynamic model of nuclear power plant turbine
PublicationThe paper presents the dynamic multivariable model of Nuclear Power Plant steam turbine. Nature of the processes occurring in a steam turbine causes a task of modeling it very difficult, especially when this model is intended to be used for on-line optimal process control (model based) over wide range of operating conditions caused by changing power demand. Particular property of developed model is that it enables calculations...
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Curing characteristics, mechanical and thermal properties of reclaimed ground tire rubber cured with various vulcanizing systems
PublicationGround tire rubber was thermo-mechanical reclaimed at 120 °C using a co-rotating twin screw extruder. The effect of vulcanizing system type on curing characteristics, static mechanical properties (tensile strength, elongation-at-break, hardness and resilience), dynamic mechanical properties and thermal properties of reclaimed ground tire rubber was investigated. Reclaimed rubber was cured using different types of vulcanization...
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Estimation of nonstructural stiffness in instrumented steel frames
PublicationLateral stiffness of nonstructural components may significantly influence the initial stiffness of the entire structure and consequently alter its dynamic characteristics. While methods for simulating structural members are well-established, approaches for modeling nonstructural components that also participate in seismic response are notably less developed. In this paper a simplified, physically-intuitive approach for estimating...
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Interlaboratory Test to Characterize the Cyclic Behavior of Bituminous Interlayers: An Overview of Testing Equipment and Protocols
PublicationThe performance assessment of multi-layered pavements strongly depends on the mechanical behavior of the interface between bituminous layers. So far, comprehensive studies have been carried out mainly using quasi-static laboratory tests focusing on the interlayer shear strength at failure. However, it is generally recognized that cyclic shear testing will lead to the determination of parameters which are more closely linked to...
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Badania doświadczalne segmentu walidacyjnego kompozytowej kładki pieszo-rowerowej
PublicationW artykule przedstawiono zakres badań zrealizowanych na segmencie walidacyjnym o długości ~3 m będącym wycinkiem docelowej kompozytowej, powłokowej kładki pieszo-rowerowej. Wykonane testy statyczne i dynamiczne pozwoliły na ocenę pracy konstrukcji i potwierdziły przyjęte na etapie projektowania założenia teoretyczne.
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Dynamic Content Internationalization in Web Applications
PublicationThis paper shows a concept for providing dynamic internationalization to web applications. Presented work is based on the Java Web Platform but described concepts can be successfully implemented on other platforms. It shows how textual data being part of web pages static and dynamic content can be localized dynamically during application runtime. All concepts presented were or are still being developed in an existing conference...
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Design and simulation of a new prototype of piezoelectric cantilever sensor/actuator for analysis of the soft tissues properties
PublicationThis paper is devoted to a new prototype of piezoelectric cantilever transducer dedicated for the characterization of the mechanical properties of soft tissues. General description of the actuator’s structure is presented including the basic principles of the measurement. The chosen geometry of the prototype is discussed and compared with the existing one. Constitutive equations are presented for the active and passive layer of...
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A new prototype of piezoelectric bending resonant transducer for analysis of soft tissues properties
PublicationThis paper is devoted to a new piezoelectric bending resonant transducer prototype dedicated to the characterization of the mechanical properties of soft tissue. A general description of the actuator’s structure is presented including the basic principles of the measurement. The chosen geometry of the prototype is discussed and compared with the existing version. Constitutive equations are presented for the active and passive layer...
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Efficient synthesis and antifungal investigation of nucleosides’ quaternary ammonium salt derivatives
PublicationQuaternary ammonium salts are a group of compounds with diverse biological properties, the most important of which are their antiviral, antibacterial, and antifungal activities. The quaternization reactions of 5'-O-tosyl derivatives of uridine and thymidine with triethylamine, trimethylamine, 4-(N ,N -dimethylamino)pyridine, 2-methylpyridine, and pyridine are described in this article. Two of the synthesized compounds are exceptional...
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Voriconazole and multidrug resistance in Candida albicans
PublicationPorównano aktywność grzybostatyczną in vitro worikonazolu, flukonazolu, ketokonazolu i klotrimazolu wobec opornych na flukonazol szczepów klinicznych Candida albicans oraz rekombinowanych szczepów Saccharomyces cerevisiae eksprymujących jeden z genów kodujących białka oporności wielolekowej (MDR) C. albicans: Cdr1p. Cdr2p lub CaMdr1p. Stwierdzono, że nadekspresja genów MDR czyni komórki drożdżaków mniej wrażliwymi na działanie...
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Initial Report on Numerical Modeling of Blood Flow in Myocardial Bridge Region of Coronary Artery: Concept of Model Validation
PublicationThe paper presents a numerical method of blood flow simulation within the coronary artery covered by the myocardial bridge. The myocardial bridge is a congenital coronary abnormality caused by the blood vessel location under one of the heart muscles. In this case, the blood flow within the vessel is partially disturbed which can cause several consequences. The presented numerical simulation allowed us to estimate the blood flow...
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Reduced order model of 2d system
PublicationA new method of modelling is developed for static and dynamic analysis of two-dimensional elastic bodies. In the analysis, an elastic body is divided into strips. For each one-dimensional strip the reduced modal model is build up. The modal model contains appropriate number of inputs and outputs to connect lumped interaction that occur between strips. Proposed method of modelling enables to obtain more accurate and more simple...
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Dynamic polarizability of the relativistic hydrogenlike atom: Application of the Sturmian expansion of the Dirac-Coulomb Green function
PublicationWe utilize the Sturmian expansion of the Dirac-Coulomb Green function [R. Szmytkowski, J. Phys. B 30, 825 (1997)] to obtain components of the dynamic dipole polarizability tensor of the relativistic hydrogenlike atom in the ground state. It is found that the tensor may be expressed in terms of two independent quantities: a scalar polarizability and a vector polarizability, the latter being of the relativistic origin. In the static...
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New Technique of preparation of standard gas mixtures needed for validation of analytical procedures used in environmental studies
PublicationStandard gas mixtures are indispensable reference materials for ensuring the reliability of analytical work. Paper presents one novel approach in the field of production of gaseous reference materials based on the application of thermal decomposition process of proper surface compound for obtaining the desired gaseous analyte. The main fields of application of reference materials are presented. The field of application of thermal...
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Influence of span length and impulse front time on earthing measurement accuracy of power line towers
PublicationThe article discusses the issue of measuring and assessing the features of power line tower earthings using fast-changing waveform. The study analyses the effect of impulse front time and the line span length on errors made during these measurements using impulse meters. It has been found that the assessment conditions similar to the static measurement results occur for the use of 4 μs current impulses and such procedure is useful...
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Low energy elastic scattering of electrons from hexafluoropropene (C3F6)
PublicationWe present cross sections from a joint experimental and theoretical study on elastic electron scattering from hexafluoropropene (C3F6) in the gas phase. The experimental results, using low energy electron spectroscopy, were obtained at incident electron energies of 0.5, 1, 1.5, 2, 3, 4, 5, 6, 10, 12, 15 and 20 eV, for scattering angles ranging from 10°to 130°. The theoretical method used in the computation of the integral, momentum...
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Retrievable strain measuring system in screw displacement piles - readings and results interpretation problems
PublicationStatic load tests on foundation piles are generally carried out in order to determine load – displacement characteristic of the pile. For more detailed information, e.g. force distribution along the shaft, load transfer mechanism and characteristics of soil-structure interaction (unit resistance curves t-z, q-z) additional pile instrumentation is required. Most popular techniques focus on direct concrete strain measurements and...
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Atomic-Scale Finite-Element Modeling of Elastic Mechanical Anisotropy in Finite-Sized Strained Phosphorene Nanoribbons
PublicationNanoribbons are crucial nanostructures due to their superior mechanical and electrical properties. This paper is devoted to hybrid studies of the elastic mechanical anisotropy of phosphorene nanoribbons whose edges connect the terminals of devices such as bridges. Fundamental mechanical properties, including Young’s modulus, Poisson’s ratio, and density, were estimated from first-principles calculations for 1-layer, 3-layer, and...
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Impact of rotor geometry optimization on the off-design ORC turbine performance
PublicationThe paper describes the method of CFD based Nelder-Mead optimization of a 10 kW single-stage axial turbine operating in an ORC system working on R7100. The total-to-static isentropic efficiency is defined as an objective function. Multi-point linear regression is carried out to determine the significance of the objective function arguments and to pick up the set of particular variables and characteristic quantities (e.g. flow angles)...
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Chemometric methods for determination of mechanisms of action of anticancer compounds
PublicationW 1990 amerykański Narodowy Instytut Raka (NCI) wprowadził szeroki test przesiewowy in vitro mający na celu poszukiwanie nowych związków przeciwnowotworowych. Test został wdrożony po przebadaniu 171 standardowych związków przeciwnowotworowych. Przedmiotem niniejszej pracy jest próba stworzenia reguł klasyfikacji związków standardowych ze względu na ich mechanizm działania przeciwnowotworowego na podstawie wyników z testu NCI. Potwierdzono...
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Arch bridges under test loadings
PublicationThis paper illustrates experience in arch bridges test loadings of the research team of Department of Structural Mechanics and Bridge Structures from the Gdansk University of Technology. The presented calculations results constist the analysis of spatial construction schemes made using the finite elements method (FEM) and its comparison to the field studies. Arch bridges with the longest spans, visualisation of the computational...
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Students from the Russian Federation at Polish Universities
PublicationSince the dissolution of the USSR, students from the Russian Federation have been able to study at Polish universities on the basis of bilateral agreements between the Polish and Russian governments. The purpose of this article is to analyse the legal basis enabling Russian citizens to obtain education in Poland, analyse the numbers of such students and the principles and procedure they followed to begin studies at Polish universities...
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FTIR, Raman spectroscopy and HT-XRD in compatibility study between naproxen and excipients
PublicationDetection of incompatibility between an active pharmaceutical ingredient (API) and excipients, including the selection of the most biopharmaceutical advantageous excipients is extremely important in the pre-formulation process of developing a solid dosage form technology. Therefore, having fast and reliable methods for identifying incompatibility is fundamental in pharmaceutical technology. For this purpose, combined Fourier transform...
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Evolution of the nanostructure of Pt and Pt–Co polymer electrolyte membrane fuel cell electrocatalysts at successive degradation stages probed by X-ray photoemission
PublicationWe present a set of XPS (X-ray photoemission spectroscopy) measurements and detailed data-analysis of electrodes for polymer electrolyte membrane fuel cell (PEMFC) based on carbon supported catalysts (Pt and Pt–Co) subjected to a step-like potential cycling (accelerated degradation test). The results of the measurements complete and corroborate parallel TEM (transmission electron microscopy), XRD (X-ray diffraction) and XAS (X-ray...
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Electrochemical simulation of metabolism for antitumor-active imidazoacridinone C-1311 and in silico prediction of drug metabolic reactions
PublicationThe metabolism of antitumor-active 5-diethylaminoethylamino-8-hydroxyimidazoacridinone (C-1311) has been investigated widely over the last decade but some aspects of molecular mechanisms of its metabolic transformation are still not explained. In the current work, we have reported a direct and rapid analytical tool for better prediction of C-1311 metabolism which is based on electrochemistry (EC) coupled on-line with electrospray...
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Anticancer Properties of Amino Acid and Peptide Derivatives of Mycophenolic Acid
PublicationBackground: Although Mycophenolic Acid (MPA) is applied as prodrugs in clinic as an immunosuppressant, it also possesses anticancer activity. MPA acts as Inosine-5’-Monophosphate Dehydrogenase (IMPDH) inhibitor, where the carboxylic group at the end of the side chain interacts with Ser 276 of the enzyme via hydrogen bonds. Therefore, MPA derivatives with other polar groups indicated high inhibition too. On the other hand, potent...
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Mission impossible for cellular internalization: When porphyrin alliance with UiO-66-NH2 MOF gives the cell lines a ride
PublicationIs it possible to accelerate cell internalization by hybridization of nanomaterials? Herein we support the realization of using metal-organic frameworks (MOFs) with the assistance of rigid porphyrin structure (H2TMP) aimed at drug loading, drug release, relative cell viability, and targeted in vitro drug delivery. There are several MOFs, i.e., UiO-66-NH2 (125 ± 12.5 nm), UiO-66-NH2 @H2TMP (160 ± 14 nm), UiO-66-NH2 @H2TMP@DOX, and...
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OPTICAL STRAIN MEASUREMENT OF CONCRETE VERSUS MANUAL EXTENSOMETER MEASUREMENT BASED ON THE TEST RC DEEP BEAM IN A COMPLEX STATE OF STRESS
PublicationThe purpose of this study is to compare the strain measurement techniques of concrete in R-C element subjected to the monotonic load up to the failure. In the analysis manual extensometer methods of measurements and the optical system ARAMIS for non-contact three-dimensional measurements of deformation was used. The test sample was a cantilever deep beam loaded throughout the depth which was a part of the reinforced concrete deep...
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Establishing Relationships between Parameters of the controlled Compaction Soil by Using Various In-Situ Tests
PublicationThe aim of research was evaluating reliable correlations between chosen soil parameters describing state of surface layers of soil. The paper presents site comparative tests based on the light falling weight deflectometer (LFWD), the static plate load tester (VSS), the dynamic probing light tester (DPL) and the bearing ratio tester (CBR in-situ) with relationships between soil state parameters. All featured in-situ...
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Selected problems of sensitivity and reliability of a jack-up platform
PublicationThe paper deals with sensitivity and reliability applications to numerical studies of an off-shore platform model. Structural parameters and sea conditions are referred to the Baltic jack-up drilling platform. The study aims at the influence of particular basic variables on static and dynamic response as well as the probability of failure due to water waves and wind loads. The paper presents the sensitivity approach to a generalized...
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EXPERIMENTS AND SIMULATIONS FOR LAPAROSCOPICVENTRAL HERNIA REPAIR IMPROVEMENT
PublicationThe authors conducted a wide experimental and numerical study in order to determine effective approaches in the laparoscopic VH repair. At first the study covered identification of mechanical properties of the abdominal fascia, implants, tacks and transabdominalsutures. Basis on these data, the one and two-dimensional mathematical models were formulated and a number of numerical static and dynamic analyses were carried out. Then...
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EXPERIMENTAL ANALYSIS OF CONNECTION BETWEEN OBJECT-ORIENTED METRICS AND SOFTWARE CHANGEABILITY
PublicationFor the purpose of video surveillance software quality assessment in this work the ISO/IEC-9126 norm was used with a particular focus on maintainability of the software system. The paper presents a study on the connection between software metrics derived from the static analysis of the source code and changeability of the video surveillance software system. It is shown that meeting requirements of software quality metrics may result...
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Control of a vapour microturbine set in cogeneration applications
PublicationSystems with microturbines are implemented for local generation of heat and electricity. This paper presents the analysis of control concepts for a vapour microturbine set with a generator with permanent magnets, intended to work in small heat and power plants. Control system variants differed by the selection of controlled signals and set parameters. Possible ways of control were discussed and compared with experimentally determined...
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Load test of new European record holder in span length among extradosed type bridges
PublicationThe article presents acceptance load tests of a newly built extradosed MS-3 bridge located along the national road DK-16 near Ostróda (Poland). The structure features significant dimension in European reference scale. It is a new record holder in span length regarding this distinct bridge category. Its length ranges 206 m. Static and dynamic load tests were performed here. The program was extended by entire structural laser scanning...
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Innovative Cold-formed GEB Section under Bending
PublicationThis paper is concerned with the numerical bending capacity study of the innovative cold-formed GEB sections. Both linear buckling analysis and non-linear static analysis incorporating geometric and material nonlinearity were carried out employing a shell structural model. The magnitudes of buckling load and limit load with respect to GEB section depth and thickness were obtained. The opened cold-formed section was tested assuming...
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Analiza statyczna i wytrzymałościowa konstrukcji wiszącej zadaszenia Stadionu Śląskiego
PublicationW artykule scharakteryzowano konstrukcję nośną zadaszenia Stadionu Śląskiego w Chorzowie, system statyczny i przyjęte rozwiązania konstrukcyjne. Przedstawiono poziom wytężenia kluczowych elementów oraz wytyczne dotyczące wzmocnienia. Analizy przeprowadzono w ramach audytu dokumentacji projektowej wykonanego na zlecenie inwestora.
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Nonlinear free and forced vibrations of a dielectric elastomer-based microcantilever for atomic force microscopy
PublicationThe majority of atomic force microcode (AFM) probes work based on piezoelectric actuation. However, some undesirable phenomena such as creep and hysteresis may appear in the piezoelectric actuators that limit their applications. This paper proposes a novel AFM probe based on dielectric elastomer actuators (DEAs). The DE is modeled via the use of a hyperelastic Cosserat model. Size effects and geometric nonlinearity are included...
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Optoelectronic investigation of nanodiamond interactions with human blood
PublicationWe present optoelectronic investigation of in vitro interactions of whole human blood with different nanodiamond biomarkers. Plasmo-chemical modifications of detonation nanodiamond particles gives the possibility for controlling their surface for biological applications. Optical investigations reveal the biological activity of nanodiamonds in blood dependent on its surface termination. We compare different types of nanodiamonds:...
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A Convenient Way to Methylated 2-Imidazolines. Syntheses of Fluorene and Triazine Cyclic Diamidines
PublicationOne N-methyl- and 4-substituted 2-imidazolines are described. Fluorene bisimidazolines were obtained in good yield (64-92%), starting from 2,7-dicyanofluorene and ammonium sulfide. In a two-step procedure the crude bisthioamide was reacted with excess diaminoalkane-ethanol (1:1 mixt.) in an oil bath. This new procedure is superior over std. methods. For the sake of comparison, a new triazine bisimidazoline (I) was prepd. by...
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Computational studies of friction forces for hard tissue cultivation in bioreactor.
PublicationPonieważ wymiana naturalego stawu na endoprotezę może być dokonywana 2-3 razy w życiu, problem leczenia przez transplantację tkanek chrzęstnych nabiera dużego znaczenia. Przeszczepów tkanki można dokonywać z sukcesem wiele razy. W bioreaktorach, środowisko hydrodynamiczne kształtuje hodowlę tkanek in vitro w obecności sił tarcia, poprzez bezpośrednie działanie na morfologię komórek a także poprzez pośrednie działanie na tkankę...
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The activity of latent benzoperimidine esters to inhibit P-glycoprotein and multidrug resistance-associated protein 1 dependent efflux of pirarubicin from several lines of multidrug resistant tumor cells.
PublicationZaprezentowano wyniki badań biologicznych przeprowadzonych dla nowej grupy związków: estrów benzoperymidyny z zastosowaniem wybranych linii komórek nowotworowych: wrażliwych i opornych o oporności P-gp-zależnej, MRP1-zależnej i o oporności związanej z nadekspresją białek MRP1/LRP. Metodą spektrofluorymetryczną zbadano zdolność estrów benzoperymidyny do hamowania eksportu aktywnego pirarubicyny z komórek opornych. Estry benzoperymidyny...
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Structural Factors Affecting Cytotoxic Activity of (E)-1-(Benzo[d ][1,3]oxathiol-6-yl)-3-phenylprop-2-en-1-one Derivatives
PublicationDerivatives of (E)-1-(5-alkoxybenzo[d][1,3]oxathiol-6-yl)-3-phenylprop-2-en-1-one (1) demonstrated exceptionally high in vitro cytotoxic activity, with IC50 values of the most active derivatives in the nanomolar range. To identify structural fragments necessary for the activity, several analogs deprived of selected fragments were prepared, and their cytotoxic activity was tested. It was found that the activity depends on combined effects...
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Numerical analysis of pile installation effects in cohesive soils
PublicationIn this thesis the empirical equation for radial effective stress calculation after displacement pile installation and following consolidation phase has been proposed. The equation is based on the numerical studies performed with Updated Lagrangian, Arbitrary Lagrangian-Eulerian and Coupled Eulerian-Lagrangian formulations as well as the calibration procedure with database containing world-wide 30 pile static loading tests in cohesive...
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Wykorzystanie metody Neldera-Meada do identyfikacji wartości parametrów niequasi-statycznego modelu małosygnałowego tranzystora MOS
PublicationW artykule zaprezentowano wyniki zastosowania metody sympleksu Neldera-Meada do ekstrakcji wartości parametrów niequasi-stycznego modelu małosygnałowego tranzystora MOS. Przedstawiono równoważny elektryczny schemat zastępczy i model matematyczny nowego modelu małosygnałowego MOSFETa dla częstotliwości mikrofalowych. Opisano zaimplementowany algorytm i otrzymane rezultaty badań.
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Chemical denudation and the role of sulfide oxidation at Werenskioldbreen, Svalbard
PublicationThis study aims to determine the rate of chemical denudation and the relationships between dominant geochemical reactions operating in the proglacial and subglacial environments of the polythermal glacier Werenskioldbreen (SW Svalbard) during an entire ablation season. Water sampling for major ion chemistry was performed at a proglacial hydrometric station and from subglacial outflows from May to September 2011. These data were...