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Search results for: 1,8-DIAZAFLUOREN-9-ONE
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Synthesis, Molecular Structure, Anticancer Activity, and QSAR Study of N-(aryl/heteroaryl)-4-(1H-pyrrol-1-yl)Benzenesulfonamide Derivatives
PublicationA series of N-(aryl/heteroaryl)-4-(1H-pyrrol-1-yl)benzenesulfonamides were synthesized from 4-amino-N-(aryl/heteroaryl)benzenesulfonamides and 2,5-dimethoxytetrahydrofuran. All the synthesized compounds were evaluated for their anticancer activity on HeLa, HCT-116, and MCF-7 human tumor cell lines. Compound 28, bearing 8-quinolinyl moiety, exhibited the most potent anticancer activity against the HCT-116, MCF-7, and HeLa cell lines,...
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Deep eutectic solvent based method for analysis of Niclosamide in pharmaceutical and wastewater samples – A green analytical chemistry approach
PublicationThe paper presents a simple, but very effective and sensitive spectrophotometric method for trace analysis of Niclosamide based on liquid–liquid microextraction using deep eutectic solvents (DESs) prior to its quantification. Here, different DES systems, such as Choline chloride (ChCl) + Urea, ChCl + Citric acid, ChCl + Ethylene glycol and ChCl + Phenol, were synthesized and evaluated at different molar ratios, selecting ChCl + Phenol...
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Stress–strain model of lower corroded steel plates of normal strength for fitness-for-purpose analyses
PublicationThis study investigates the mechanical properties of specimens made of normal strength steel subjected to lower marine immersed corrosion degradation levels (below 25 %). The specimens were corroded in laboratory conditions, and only natural factors were controlled to raise the corrosion rate (reaching the level of 1 mm/year). Three different thicknesses of plates made of normal strength of shipbuilding steel are investigated (between...
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The best porous asphalt pavement in Sweden so far
PublicationIn 2010 a double-layer porous asphalt concrete (DPAC) pavement was constructed in various versions on the E4 motorway through the Swedish city Huskvarna. As a result of a court decision the Swedish Transport Administration had to reduce noise emission by applying a low noise road surface that would reduce A-weighted noise levels by 5 dB, as an average. Earlier experience in Sweden indicated that it was possible to obtain a high...
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Optical Sensor Based Gestures Inference Using Recurrent Neural Network in Mobile Conditions
PublicationIn this paper the implementation of recurrent neural network models for hand gesture recognition on edge devices was performed. The models were trained with 27 hand gestures recorded with the use of a linear optical sensor consisting of 8 photodiodes and 4 LEDs. Different models, trained off-line, were tested in terms of different network topologies (different number of neurons and layers) and different effective sampling frequency...
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Trees as a Shading System for Streets on the East–West Axis: Computer Simulations for the Selected Geometrical Proportions of Building Developments in Humid Continental Climate
PublicationThe study is aimed at investigating the possibilities for solar protection provided to the street canyon located on the E–W axis and with the following profiles: shallow (height/width (H/W) = 0.2, 0.6, and 1) and deep (H/W = 2) by two rows of trees located at a distance of 3 m away from southern and northern façades. The research was based on numerical simulation analyses conducted in the Rhinoceros® program, with the application...
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Piotr Płotka dr hab. inż.
PeoplePiotr Płotka received the M.Sc. and D.Eng. degrees in electronic engineering from the Gdansk University of Technology, Poland, in 1976 and 1985. In 2008 he received D.Sc. (Dr.Hab.) degree, also in electronic engineering, from the Institute of Electron Technology at Warsaw, Poland. From 1977 he was with Academy of Technology and Agriculture at Bydgoszcz, Poland and from 1981 with the Gdansk University of Technology. In cooperation...
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WPŁYW TRANSFORMACJI DANYCH NA JAKOŚĆ OPRACOWANYCH METOD TOŻSAMOŚCIOWYCH W SPEKTROSKOPII BLISKIEJ PODCZERWIENI
PublicationSpektroskopia bliskiej podczerwieni (NIR) wykorzystuje absorpcję promieniowania elektromagnetycznego w zakresie 12000-4000 cm-1, (780¬-2500 nm). Absorpcja NIR pochodzi od nadtonów i drgań kombinacyjnych wiązań C-H, N-H, O-H. Widmo uzyskane techniką NIR jest unikatowym "odciskiem palca" badanej substancji gdyż zależy zarówno od właściwości fizyko-chemicznych próbki jak i od stanu fazowego oraz postaci krystalicznej jej składników.Zaletami...
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Pavement ageing influence on tyre/road noise
PublicationRoad surface should be constructed in a way that ensures safe and comfortable traffic conditions, not only when it is newly paved but also during its entire lifetime. An important factor in the asphalt mixture design process is also the expected pavement durability and stability of pavement properties over time. In many countries, road surface starts to play a significant role in traffic noise reduction actions. Selecting a particular...
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Ultrasonic wave propagation, digital image correlation and X-ray micro-computed tomography measurements of concrete during splitting (cube #1)
Open Research DataThe DataSet contains the results of the mechanical behaviour of a concrete cube under the splitting test. The cube had dimensions 70 x 70 x 70 cm3 and was made of concrete with the following ingredients: cement type CEM I 42.5R (330 kg/m3), water (165 kg/m3), aggregate 0/2 mm (710 kg/m3), aggregate 2/8 mm (664 kg/m3), aggregate 8/16 mm (500 kg/m3),...
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The XPS spectra of AlOOH/1%Cu prepared using wet impregnation method
Open Research DataThe dataset includes XPS spectra of AlOOH/1%Cu catalyst sintered under air atmosphere. Samples were produced using aqueous soft chemistry methods and incipient wettness impregnation using nitrate solution. The XPS spectra were collected for all species.
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Analysis of the impact of socio-economic development on road safety based on the example of Baltic Sea Region countries
PublicationBaltic Sea Region (BSR) is a specific region of Europe, bringing together countries with different levels of socio-economic development. The main common point is territorial access to the Baltic Sea and the importance of maritime transport in the transportation of goods. The region consists of 9 countries, including Germany, Poland, Lithuania, Latvia, Estonia, Finland, Sweden, Denmark and Russia (more specifically, Kaliningrad...
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Video traffic data - Interchange Bielany (A4-5) - weaving, Poland
Open Research DataThe data includes video traffic data registered with 12 video cameras at weaving area (weaving section type A) of the Bielany interchange within A4 motorway in Poland (interchange of motorway A4 and nacional road 5), located in the Silesian Agglomeration.The data covers the one day: 07.06.2017 (motorway A4)
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Kazimierz Darowicki prof. dr hab. inż.
PeopleStudia wyższe ukończyłem w czerwcu 1981 roku po zdaniu egzaminu dyplomowego i obronie pracy magisterskiej. Opiekunem pracy magisterskiej był dr hab. inż. Tadeusz Szauer. W roku 1991-11-27 uzyskałem stopień naukowy broniąc pracę doktorską zatytułowaną „Symulacyjna i korelacyjna analiza widm immitancyjnych inhibitowanej reakcji elektrodowej”. Promotorem pracy był prof. dr hab. inż. Józef Kubicki (Wydział...
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Video traffic data - Interchange Sosnica (A1 - 902), Poland
Open Research DataThe data includes video traffic data registered with 8 video cameras at weaving area (weaving section type A) of the Sosnica interchange within A1 motorway in Poland (interchange of motorway A1 and regional road 902, located in the Silesian Agglomeration).The data covers the two days: 12.09.2017 (motorway A1) and 11.09.2017 (road 902).
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Szkolenie NCBiR dot. zamykania projektu
EventsNarodowe Centrum Badań i Rozwoju zaprasza do udziału w szkoleniu online pt. Zamykanie projektu – najważniejsze informacje jak przygotować wniosek końcowy. Wskazówki dla beneficjentów POWER.
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Acoustic emission signals in concrete beams under 3-point bending (plain concrete, steel fibre reinforced concrete, steel bar reinforced concrete)
Open Research DataThe DataSet contains the results of the mechanical behaviour of concrete beams with dimensions 40 x 40 x 160 cm3under the 3-point bending. Two concrete mixes, both based on the same design, were produced in the test programme. Mixture #1 was the plain concrete (PC), consisting of cement CEM I 42.5R (380 kg/m3), water (165 kg/m3), aggregate 0/2 mm (648...
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Dataset of non-isomorphic graphs of the coloring types (K3,Km;n), 2<m<7, 1<n<R(3,m)
Open Research DataFor K3 and Km graphs, a coloring type (K3,Km;n) is such an edge coloring of the full Kn graph, which does not have the K3 subgraph in the first color (representing by no edges in the graph) or the Km subgraph in the second color (representing by edges in the graph).The Ramsey number R(3,m) is the smallest natural number n such that for any edge coloring...
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Karolina Lademann mgr
PeopleCurriculum vitae
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Value of tax preferences by areas of support and types of taxes in 2013
Open Research DataThese data contain information prepared by the Ministry of Finance on the value of tax preferences by areas of support and types of taxes in 2013.
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Killing kinetics analysis of C-1311 derivative with octaarginine (Compound 1-R8) against Candida albicans
Open Research DataThe datasets contain the results of killing kinetics analysis of imidazoacridinone derivative and fluconazole against C. albicans ATCC 10231. The suspensions of Candida albicans ATCC 10231 cells (500 µL) in RPMI 1640 at cell density of 104 cells /mL were added to 500 µL of RPMI 1640 medium with various concentrations of the compounds, corresponding...
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Value of tax preferences by areas of support and types of taxes in 2014
Open Research DataThese data contain information prepared by the Ministry of Finance on the value of tax preferences by areas of support and types of taxes in 2014.
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Value of tax preferences by areas of support and types of taxes in 2011
Open Research DataThese data contain information prepared by the Ministry of Finance on the value of tax preferences by areas of support and types of taxes in 2009.
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Value of tax preferences by areas of support and types of taxes in 2009
Open Research DataThese data contain information prepared by the Ministry of Finance on the value of tax preferences by areas of support and types of taxes in 2009.
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Value of tax preferences by areas of support and types of taxes in 2010
Open Research DataThese data contain information prepared by the Ministry of Finance on the value of tax preferences by areas of support and types of taxes in 2010.
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Value of tax preferences by areas of support and types of taxes in 2012
Open Research DataThese data contain information prepared by the Ministry of Finance on the value of tax preferences by areas of support and types of taxes in 2012.
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Performance of the Direct Sequence Spread Spectrum Underwater Acoustic Communication System with Differential Detection in Strong Multipath Propagation Conditions
PublicationThe underwater acoustic communication (UAC) operating in very shallow-water should ensure reliable transmission in conditions of strong multipath propagation, significantly disturbing the received signal. One of the techniques to achieve this goal is the direct sequence spread spectrum (DSSS) technique, which consists in binary phase shift keying (BPSK) according to a pseudo-random spreading sequence. This paper describes the DSSS...
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Assestment of the anti-cancer activity of the copper complexes with imidazole and pivalato ligands
PublicationDespite the development of science and technology progress so far there have not been found effective drugs for cancer. Many coordination compounds were investigated due to their antitumor potential. The most known cis-diamminedichloroplatinum(II) is used as anti-cancer therapeutic agent. The copper complexes are the coordination compounds possessing anti-tumour properties. Their capability to kill cancer cells is mainly linked...
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SYNAT Music Genre Parameters PCA 19
Open Research DataThe dataset contains feature vector after Principal Component Analysis (PCA) performing, so there are 11 music genres and 19-element vector derived from music excerpts. Originally, a feature vector containing 173 elements was conceived in earlier research studies carried out by the team of authors [1-6]. A collection of 52532 music excerpts described...
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SYNAT_PCA_48
Open Research DataThere is a series of datasets containing feature vectors derived from music tracks. The dataset contains 51582 music tracks (22 music genres) and feature vector after Principal Component Analysis (PCA) performing, so there are 48-element vectors derived from music excerpts. Originally, a feature vector containing 173 elements was conceived in earlier...
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SYNAT_PCA_11
Open Research DataThe dataset contains 51582 music tracks (22 music genres) and feature vector after Principal Component Analysis (PCA) performing, so there are 11-element vectors derived from music excerpts. Originally, a feature vector containing 173 elements was conceived in earlier research studies carried out by the team of authors [1-6]. A collection of more than...
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Analiza porównawcza metod zwiększania nośności i sztywności stalowych, doczołowych węzłów śrubowych.
PublicationInnowacyjna, w porównaniu z dotychczas stosowanym sposobem, metoda obliczania nośności stalowych węzłów została wdrożona wraz z normami europejskimi. Pozwala ona dokładniej odwzo-rować rzeczywistą pracę poszczególnych części węzła, gdyż wynik obliczeń uzależniony jest od znacznie większej liczby zmiennych. Dzięki postępowi technologicznemu w zakresie metalurgii oraz badaniom naukowym obecnie możliwe jest wzmacnianie połączeń...
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Quality Evaluation of Speech Transmission via Two-way BPL-PLC Voice Communication System in an Underground Mine
PublicationIn order to design a stable and reliable voice communication system, it is essential to know how many resources are necessary for conveying quality content. These parameters may include objective quality of service (QoS) metrics, such as: available bandwidth, bit error rate (BER), delay, latency as well as subjective quality of experience (QoE) related to user expectations. QoE is expressed as clarity of speech and the ability...
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Subjective Quality Evaluation of Underground BPL-PLC Voice Communication System
PublicationDesigning a reliable voice transmission system is not a trivial task. Wired media, thanks to their resistance to mechanical damage, seem an ideal solution. The BPL-PLC (Broadband over Power Line – Power Line Communication) cable is resilient to electricity stoppage and partial damage of phase conductors. It maintains continuity of transmission in case of an emergency situation, including paramedic rescue operations. These features...
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Synthesis of highly crystalline photocatalysts based on TiO2 and ZnO for the degradation of organic impurities under visible-light irradiation
PublicationA TiO2–ZnO binary oxide system (with molar ratio TiO2:ZnO = 8:2) was synthesized by a hydrothermal method, assisted by calcination at temperatures of 500, 600 and 700 °C, using zinc citrate as the precursor of ZnO. The morphology (SEM, TEM), crystalline structure (XRD, Raman spectroscopy), diffuse reflectance spectra (DRS), chemical surface composition (EDXRF), porous structure parameters (low-temperature N2 sorption) and characteristic...
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Rysunek Techniczny i Planistyczny
e-Learning CoursesKurs jest przeznaczony dla studentów 1 semestru kierunku GOSPODARKA PRZESTRZENNA, studia inżynierskie I stopnia. Celem zajęć jest przekazanie wiedzy i wykształcenie praktycznych umiejętności przydatnych przy sporządzaniu rysunków technicznych i planistycznych w zawodzie architekta urbanisty i zawodach pokrewnych związanych z gospodarką przestrzenną. Zajęcia odbywają się w formie ćwiczeń - 7 spotkań (rysunek odręczny) oraz w laboratorium...
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Miscanthus × giganteus root anatomical traits measurements
Open Research DataThis data set presents the optical microscope measurements/ images of Miscanthus × giganteus (M×g) roots. The experiment was performed under work package 1: "Properties characterisation of two types of biochar", task D_RT: Phyto-analyses (stress response of plants on biochar amendments) in cooperation with Aarhus University. A short term pot experiment...
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Ferromagnetic nanoparticles imaging by means of Magnetic Force Microscopy
Open Research DataFerromagnetic nanoparticles can be used as building blocks for advanced thin film magnets, and can also be used in data storage and biomedical technologies. Nano-crystalline ferrites with the chemical formula NixZn (1 - x) Fe2O4, where x = 0, 0.2, 0.4, 0.6, 0.8, 1.0 show anti-corrosion properties and suppress electromagnetic interference, in the case...
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Effects of liquid phase modification on the values of surface tension of trickling liquid
Open Research DataDataset presents the values of surface tension of trickling liquid sampled from three running biotrickling filters.
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Impact of laser beam welding on mechanical behaviour of 2.25Cr–1Mo (P22) steel
PublicationThe use of welding processes in the manufacturing and repair of structures intended for the energy industry plays a key role in the guarantee of a continuous supply of fossil fuels, which is the basic condition for ensuring energy security. A square butt joint of 10 mm thick plate of 2.25Cr–1Mo (P22) steel was fabricated by autogenous laser beam welding process and then post-weld heat treatment (PWHT) for two sets of process parameters...
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Dataset of non-isomorphic graphs of the coloring types (K3,Km-e;n), 2<m<7, 1<n<R(K3,Km-e).
Open Research DataFor K3 and Km-e graphs, a coloring type (K3,Km-e;n) is such an edge coloring of the full Kn graph, which does not have the K3 subgraph in the first color (representing by no edges in the graph) or the Km-e subgraph in the second color (representing by edges in the graph). Km-e means the full Km graph with one edge removed.The Ramsey number R(K3,Km-e)...
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XPS data of deuterium and hydrogen grown boron-doped diamond
Open Research DataThe high-resolution C1s X-ray absorption spectra of BDD@H and BDD@D samples were measured using the facilities of the HE-SGM beamline (HE-SGM) at the BESSY II synchrotron radiation source of Helmholtz–Zentrum Berlin (HZB).[90] The measurements were carried out under ultra-high vacuum conditions: P ≈ 2×10−9 Torr at T = 300 K. The NEXAFS spectra were...
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PCR Melting Profile method for genotyping analysis of vancomycin-resistant Enterococcus faecium isolates from Hematological Unit patients
PublicationW ostatnich latach znacząco wzrasta liczba szczepów Enterococcus opornych na wankomycynę. Stwarzają one problemy medyczne u pacjentów skolonizowanych czy zainfekowanych tymi drobnoustrojami. W przedstawionych badaniach, określiliśmy genetyczne podobieństwo pomiędzy izolatami E. faecium VRE, pozyskiwanymi w okresie od kwietnia 2003 do kwietnia 2005 od pojedynczych pacjentów oddziału Hematologicznego Specjalistycznego Publicznego...
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Silicon’s Influence on Polyphenol and Flavonoid Profiles in Pea (Pisum sativum L.) under Cadmium Exposure in Hydroponics: A Study of Metabolomics, Extraction Efficacy, and Antimicrobial Properties of Extracts
PublicationThe current study aimed to investigate the impact of silicon (Si) supplementation in the form of Na2SiO3 on the metabolome of peas under normal conditions and following exposure to cadmium (Cd) stress. Si is known for its ability to enhance stress tolerance in various plant species, including the mitigation of heavy metal toxicity. Cd, a significant contaminant, poses risks to...
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Bee Pollen and Bee Bread as a Source of Bacteria Producing Antimicrobials
PublicationThe principal objective of the study was the isolation and identification of bacteria that are present in mature bee bread (BB) and dried (ready for selling and consumption) bee pollen (BP). Obtained isolates were screened for their potential to inhibit select human pathogenic bacteria and their ability to produce enzymes of particular industrial importance. Four and five samples of BP and BB, respectively, were used for the study....
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Orbital blowout trauma occurring at the workplace – clinical, biomechanical and legal aspects
PublicationIntroduction and objective: Craniofacial injury at the workplace may lead to orbital blowout fractures. The aim of the study is the development of own numerical model of the eye orbit, assessment of the damage zones, and comparing them with clinical examinations. In addition, the current legal status of patients after injuries is presented Material and methods: In laboratory tests performed on bones collected from the upper and...
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Badania eksperymentalne intensyfikacji wymiany ciepła wymiennika U-rurowego z wykorzystaniem turbulizatora helikoidalnego
PublicationW niniejszej pracy zostały zaprezentowane możliwości intensyfikacji wymiany ciepła po stronie płaszcza wymiennika U-rurowego. Badania eksperymentalne zostały przeprowadzone zarówno dla wymienników referencyjnych tj. prosty – rura w rurze, U-rurowy bez turbulizacji jak i wymiennika z turbulizatorem helikoidalnym. Dla konstrukcji rura w rurze w celu uzyskania wartości referencyjnych przeprowadzono pomiary w układzie woda-woda oraz...
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Detection of the Incoming Sound Direction Employing MEMS Microphones and the DSP
PublicationA 3D acoustic vector sensor based on MEMS microphones and its application to road traffic monitoring is presented in the paper. The sensor is constructed from three pairs of digital MEMS microphones, mounted on the orthogonal axes. Signals obtained from the microphones are used to compute sound intensity vectors in each direction. With this data, it is possible to compute the horizontal and vertical angle of an incoming sound....
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Properties and applications of thermostable proteases sourced from Deinococcus geothermalis.
PublicationThe growing interest of extremophiles results from the fact that their enzymes arestable and active under harsh environment conditions. These type of biocatalysts are attractivedue to the fact that can be used in industrial processes that were previously regarded asincompatible with biological materials. Among extremozymes the largest group constitutethermozymes. Currently it is estimated that approximately 40% of enzymes used...
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FURTHER REMARKS ON THE NEO-CLASSICAL NAVIER-STOKES EQUATIONS
PublicationThe seminal Navier-Stokes equations have been stated yet before creation of principles of thermodynamics and the first and second laws. In the literature there is the common opinion that the Navier-Stokes equations cannot be taken as a thermodynamically correct model of “working fluid” which is able to describe transformation of “ heat” into “work” and vice versa. Therefore, in the paper, a new exposition of thermodynamically...