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Optimization of Chemical Functionalities of Indole-2-carboxamides To Improve Allosteric Parameters for the Cannabinoid Receptor 1 (CB1)
Publication5-Chloro-3-ethyl-N-(4-(piperidin-1-yl)phenethyl)-1H-indole-2-carboxamide (1; ORG27569) is a prototypical allosteric modulator for the cannabinoid type 1 receptor (CB1). Here, we reveal key structural requirements of indole-2-carboxamides for allosteric modulation of CB1: a critical chain length at the C3-position, an electron withdrawing group at the C5-position, the length of the linker between the amide bond and the phenyl ring...
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Cellular Effects of Selected Unsymmetrical Bisacridines on the Multicellular Tumor Spheroids of HCT116 Colon and A549 Lung Cancer Cells in Comparison to Monolayer Cultures
PublicationMulticellular tumor spheroids are a good tool for testing new anticancer drugs, including those that may target cancer stem cells (CSCs), which are responsible for cancer progression, metastasis, and recurrence. Therefore, we applied this model in our studies of highly active antitumor unsymmetrical bisacridines (UAs). We investigated the cellular response induced by UAs in 2D and 3D cultures of HCT116 colon and A549 lung cancer...
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Reduction of steel chimney vibrations with a pendlum damper.
PublicationKarman vortices observed around chimneys may induce dangerous structural vi-brations at certain wind velocities. The aim of this paper is to analyse theeffectiveness of pendulum damper in vibration reduction of a steel chimney. A two degree-of-freedom system is used to model the behaviour of the struc-ture equipped with a damper. The results of the study show that the use of pendulum with tuned frequency leads to significant...
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Bacteriophages as potential tools for use in antimicrobial therapy and vaccine development
PublicationThe constantly growing number of people suffering from bacterial, viral, or fungal infections, parasitic diseases, and cancers prompts the search for innovative methods of disease prevention and treatment, especially based on vaccines and targeted therapy. An additional problem is the global threat to humanity resulting from the increasing resistance of bacteria to commonly used antibiotics. Conventional vaccines based on bacteria...
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A New Approach for the Mitigating of Flow Maldistribution in Parallel Microchannel Heat Sink
PublicationThe problem of flow maldistribution is very critical in microchannel heat sinks (MCHS). It induces temperature nonuniformity, which may ultimately lead to the breakdown of associated system. In the present communication, a novel approach for the mitigation of flow maldistribution problem in parallel MCHS has been proposed using variable width microchannels. Numerical simulation of copper made parallel MCHS consisting of 25 channels...
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A study about daylighting knowledge and education in Europe. Results from the first phase of the DAYKE project
PublicationThis paper presents selected results from the first stage of DAYKE (Daylight Knowledge in Europe), a 3- phase project that investigates the knowledge on daylighting in buildings among architecture students and practitioners across Europe. Subjective judgements from 561 students from 8 architecture universities in the EU, collected through two surveys in 2018. The key findings are: (i) the spatial distribution of comfort and mood...
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On the problem of optimised allocation of water quality sensors and actuators in DWDS
PublicationThe problems of water quality sensors and actuators placement in drinking water distribution systems (DWDSs) are addressed as separate, primarily. However, against the background of control systems theory, the nature of DWDSs dynamics indicates that these both problems are interdependent and impact the design of related water quality monitoring and control structures and algorithms. The research work presented in this paper is...
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Influence of Shunt Compensation with SVC Devices on Resonance Risk in Power Systems
PublicationMany analyses are required to locate a new reactive power source in a power system. The choice of a location is a very complex matter which requires various aspects to be considered. Selecting a location also entails the necessity to assess it from the point of view of the selected compensator’s structure as well as the system’s performance in various states with the new device on. The paper presents the issues of assessing compensator...
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High Resolution Sea Ice Floe Size and Shape Data from Knox Coast, East Antarctica
PublicationThis dataset contains floe size distribution data from a very high resolution (pixel size: 0.3 m) optical satellite image of sea ice, acquired on 16 Feb. 2019 off the Knox Coast (East Antarctica). The image shows relatively small ice floes produced by wave-induced breakup of landfast ice between Mill Island and Bowman Island. The ice floes are characterised by a narrow size distribution and angular, polygonal shapes, typical...
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Potential applicability of ontologies for the evaluation of information technology
PublicationIn this article we present the possibilities of using ontologies as a part of a multi-agent system (MAS) designed for the evaluation of information technologies. This is a part of a broader idea devel-oped by the team of researchers at Gdańsk University of Technology. The article deals with defining ontologies, presenting main technologies for their design and implementation and proposes, initially, domains of the ontologies' interest...
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Local atomic order in low Pt-content nanocatalysts investigated in situ by XAS
PublicationThe unique features of X-ray absorption spectroscopy allow investigations of nanosized catalysts for fuel cells under working conditions. We present the results of an experiment carried out on a low Pt content electrocatalyst supported by a mesoporous heteropolyacid salt and used at the cathode of a proton exchange membrane fuel cell (PEMFC). The analysis of the EXAFS signal at the Pt L3-edge indicates that upon operating the fuel...
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Evaluation of a sat-type fairness mechanism implemented in a dual-ring network
PublicationThe fairness problem was presented. Popular fairness concepts and measures were shown. The RPR fairness mechanism and the SAT mechanism were described. A modification of the SAT algorithm, adapted to the possibilities of Ethernet cards used for implementation of a dual-ring RPR-based network, was proposed. Performance of the proposed modification was measured. Jain's and Chen's fairness indexes were calculated. Effectiveness comparison...
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Dynamics Conscious Approach to Tribometer Design and Tribo-testing
PublicationIn the paper findings are discussed on the issue of dynamic characteristics of a tribometer as a factor influencing the result of the tribological experiment. An advanced approach to tribo-testing is attempted with integrated dynamic analysis of the tribometer and the sliding pair. The fundamental idea is explored of the tribometer being regarded as any machine in which friction is inflicted with all the resulting consequences...
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Magnetism and charge density waves in RNiC2(R=Ce,Pr,Nd)
PublicationWe have compared the magnetic, transport, galvanomagnetic, and specific-heat properties of CeNiC2, PrNiC2, and NdNiC2 to study the interplay between charge density waves (CDW) and magnetism in these compounds. The negative magnetoresistance in NdNiC2 is discussed in terms of the partial destruction of charge density waves and an irreversible phase transition stabilized by the field-induced ferromagnetic transformation is reported....
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DYNAMIC RESPONSE OF FORUM GDANSK STRUCTURE DUE TO RAIL TRAFFIC
PublicationThe paper presents the study of the impact of vibration induced by the movement of the railway rolling stock on the Forum Gdańsk structure. This object is currently under construction and is located over the railway tracks in the vicinity of the Gdańsk Główny and Gdańsk Śródmieście railway stations. The analysis covers the influence of vibrations on the structure itself and on the people within. The in situ measurements on existing...
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VUV irradiation studies of plasmid DNA in aqueous solution
PublicationInteractions of VUV light and DNA samples in aqueous solutions are reported. The damage induced by such radiation is quantified by monitoring both loss of supercoiled DNA and formation of single and double strand breaks using agarose gel electrophoresis. Irradiations were performed using synchrotron VUV photons of 130, 150, 170 and 190 nm. VUV irradiation experiments revealed enhanced damage upon irradiation with 170 nm photons...
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Retrieval with Semantic Sieve
PublicationThe article presents an algorithm we called Semantic Sieve applied for refining search results in text documents repository. The algorithm calculates socalled conceptual directions that enables interaction with the user and allows to narrow the set of results to the most relevant ones. We present the system where the algorithm has been implemented. The system also offers in the presentation layer clustering of the results into...
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Detection of defects in PMMA beam using shear waves - numerical simulation and experiment
PublicationTest doświadczalny falami sprężystymi jest częścią systemu diagnostycznego belek. Autorzy badają pole przyspieszeń wywołane przepływem fal ultradźwiękowych i jego modyfikacje wynikające z wprowadzonych uszkodzeń belki. Artykuł porównuje wyniki eksperymentalne z symulacjami numerycznymi MES. The experimental test introduced in the paper is the part of the diagnostic system utilizing the elastic waves. The authors investigate the...
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Entropy Measures in the Assessment of Heart Rate Variability in Patients with Cardiodepressive Vasovagal Syncope
PublicationSample entropy (SampEn) was reported to be useful in the assessment of the complexity of heart rate dynamics. Permutation entropy (PermEn) is a new measure based on the concept of order and was previously shown to be accurate for short, non-stationary datasets. The aim of the present study is to assess if SampEn and PermEn obtained from baseline recordings might differentiate patients with various outcomes of the head-up tilt test...
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The microbial and sensory quality of mackerel hot smoked in mild conditions
PublicationThe quality indices of Atlantic mackerel, hot smoked at core temperature not exceeding 60°C, containing 14–27 g salt and 580–670 g water per kg meat, was determined just after smoking and during storage. The aerobic plate count after smoking, chilling and packing in cardboard boxes was 0–12 cfu/25 cm2of the skin of the smoked fish and 10–240 cfu/g of flesh. It was 1.9 log cycle lower than that in the frozen raw material. At 2°C,...
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Experimental and predicted physicochemical properties of monopropanolamine-based deep eutectic solvents
PublicationIn this work, the novel deep eutectic solvents (DESs) based on 3-amino-1-propanol (AP) as hydrogen bond donor (HBD) and tetrabutylammonium bromide (TBAB) or tetrabutylammonium chloride (TBAC) or tetraethylammonium chloride (TEAC) as hydrogen bond acceptors (HBAs) were synthesized with different molar ratios of 1: 4, 1: 6 and 1: 8 salt to AP. Fourier Transform Infrared Spectroscopy measurements were performed to provide an evidence...
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Experimental and predicted physicochemical properties of monopropanolamine-based deep eutectic solvents
PublicationIn this work, the novel deep eutectic solvents (DESs) based on 3-amino-1-propanol (AP) as hydrogen bond donor (HBD) and tetrabutylammonium bromide (TBAB) or tetrabutylammonium chloride (TBAC) or tetraethylammonium chloride (TEAC) as hydrogen bond acceptors (HBAs) were synthesized with different molar ratios of 1:4, 1:6 and 1:8 salt to AP. Fourier Transform Infrared Spectroscopy measurements were performed to provide an evidence...
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Pounding Between Superstructure Segments in Multi-Supported Elevated Bridge with Three-Span Continuous Deck Under 3D Non-Uniform Earthquake Excitation
PublicationReports after severe ground motions show that the earthquake-induced structural pounding may lead to significant damage in elevated bridges. The aim of this paper is to analyse pounding between superstructure segments of a highway elevated bridge with three-span continuous deck under 3D non-uniform earthquake excitation, which is induced by spatial seismic effects related to the propagation of seismic wave. The conditional stochastic...
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Redox State Sensitive Spectroscopy of the Model Compound [(H-dcbpy)(2)Ru-II(NCS)(2)](2-) (dcbpy=2,2 '-Bipyridine-4,4 '-dicarboxylato)
PublicationThe charge transfer reaction mechanism in a ruthenium polypyridine model complex with isothiocyanato ligands, i.e., [(H-dcbpy)(2)Ru(NCS)(2)](2-) 2Bu(4)N(+) (Ru2H) (dcbpy = 2,2'-bipyridine-4,4'-dicarboxylato), has been investigated by combining UV-vis absorption, resonance Raman spectroscopy, and electrochemical methods. Understanding the photophysics of light-harvesting complexes of this class is an indispensable prerequisite to...
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Formaldehyde detection with chemical gas sensors based on WO3 nanowires decorated with metal nanoparticles under dark conditions and UV light irradiation
PublicationWe report results of formaldehyde gas (CH2O) detection under dark conditions and UV light irradiation with pristine tungsten trioxide nanowires (WO3 NWs) and metal nanoparticles decorated WO3 NWs gas sensing layers. The resistive layers were deposited by one step aerosol assisted chemical vapor deposition (AACVD) on commercial alumina substrates with 10-pair interdigitated platinum electrodes. The elaborated gas sensors, based...
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CYP3A4-dependent cellular response does not relate to CYP3A4-catalysed metabolites of C-1748 and C-1305 acridine antitumor agents in HepG2 cells
PublicationHigh CYP3A4 expression sensitizes tumor cells to certain antitumor agents while for others it can lower their therapeutic ef fi cacy. We have elucidated the in fl uence of CYP3A4 overexpression on the cellular response induced by antitumor acridine derivatives, C-1305 and C-1748, in two hepatocellular carcinoma (HepG2) cell lines, Hep3A4 stably transfected with CYP3A4 isoenzyme, and HepC34 expressing empty vector. The compounds...
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Ruch wirowy wywoływany przez ultradźwięk w płynach z relaksacją
PublicationRozprawa doktorska poświęcona jest badaniu ruchu wirowego wywoływanego przez ultradźwięk w różnych modelach płynów z relaksacją. Ma ona charakter teoretyczny, jednak wykorzystanie uzyskanych dzięki niej wyników może przynieść lepsze zrozumienie ruchu wirowego wywoływanego przez siłę akustyczną. W I rozdziale rozprawy przedstawione zostały ogólne rozważania dotyczące akustyki nieliniowej. Rozdział II dotyczy ruchu wirowego wywoływanego...
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Nadmiarowe zgony podczas pandemii COVID-19 w Polsce i ocena skuteczności szczepień
PublicationZ powodu pandemii COVID-19 zmarły miliony ludzi na całym świecie. Jak wynika z wielu badań, szczepienia przeciw chorobie wywołanej wirusem SARS-CoV-2 okazały się środ-kiem ograniczającym skalę zachorowań i liczbę zgonów. Celem badania omawianego w artyku-le jest pomiar skali pandemii w Polsce za pomocą liczby nadmiarowych zgonów w podregio-nach według klasyfikacji NUTS 3 i w grupach wieku, a następnie określenie zależności pomiędzy...
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Consideration of the safety of bungee jumping in relation to mechanical properties of the instalation based on a jump accident in Gdynia
PublicationThis paper considers a bungee jumping accident that took place in July 2019 in Gdynia, Poland. The authors conducted an investigation to determine the cause of the bungee rope failure. It was based on mechanical tests concerning the strength of the rope as well as the calculation of the force induced in the rope during the jump. Based on the theoretical and experimental results, the rope safety factor was estimated. It appeared...
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The Relationship between Gene Activity and Nitrous Oxide Production during Nitrification in Activated Sludge Systems
PublicationNitrite is an important factor which inhibits the first stage of the nitrification, the effect is stronger with the decrease of the DO concentrations. NO2- presence at concentration above 15 mg N – NO2 in the aeration tanks stimulates N2O production regardless of the DO concentration. The significant nirS gene induction, observed especially during the experiments with the nitrite addition indicates that N2O production is basically...
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Resonance problems in UHV transmission lines
PublicationThe paper presents resonance phenomena observed in 400 kV transmission lines in the Polish power system. Two events are analysed, when shunt reactors used for reactive power compensation, caused overvoltages and overcurrent protection tripping as a result of resonance. An oscillographic fault recordings from protection devices are compared to time domain simulation results. The obtained simulation results match fault recordings,...
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Effects of Xanthan Gum Biopolymer on the Permeability, Odometer, Unconfined Compressive and Triaxial Shear Behavior of a Sand
PublicationBiopolymers, which are microbially induced polymers, can be used as an alternative material to improve engineering performance of soils. In this paper, a laboratory study of 0.075-1.0 mm size sand and biopolymer (i.e., xanthan gum) mixtures with various mix ratios (0%, 0.5%, 1.0%, and 1.5%) was performed. The materials, specimen preparation, and test methods are described, as are the results of a suite of permeability, odometer, unconfined...
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Investigation of RTS Noise in Reverse Polarized Silicon Carbide Schottky Diodes
PublicationOne of the method of electronic device quality and reliability evaluation is observation of its inherent noise. The RTS phenomena usually indicates the presence of large defects in the structure of the material of the device, therefore it can be treated as an indicator of technology quality. In the paper authors present results of RTS investigations in reverse polarized Silicon Carbide Schottky diodes. Devices being studied are...
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A Study in Experimental Methods of Human-Computer Communication for Patients After Severe Brain Injuries
PublicationExperimental research in the domain of multimedia technology applied to medical practice is discussed, employing a prototype of integrated multimodal system to assist diagnosis and polysensory stimulation of patients after severe brain injury. The system being developed includes among others: eye gaze tracker, and EEG monitoring of non-communicating patients after severe brain injuries. The proposed solutions are used for collecting...
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An Approach to Mean Path Loss Model Estimation for Off-Body Channels
PublicationThis paper presents an approach to estimation of the mean path loss model parameters in off-body Body Area Networks channels. In this approach, the path loss exponent is constrained to a value obtained for the line-of-sight (LoS) propagation in the co-polarised channel, considering a generalised static scenario. The comparison of the goodness of fit between the proposed approach and other approaches, for a set of measurements obtained...
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Issues of Measuring the Course of Batch Production Processes
PublicationIn order to meet demands induced by development of manufacturing processes and production systems, new criteria and indicators that would allow a multiple aspect and realistic rating of batch production process courses are necessary. The objective of this paper is to present the correlation between production processes measurement, its rating and production control, basing on case study analysis from production enterprise. A new...
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Literature review of user needs, toward user requirements
PublicationThis report has been developed in the frame of the IEA SHC Task 61 Subtask A “User requirements”. The main objective was to rethink and reformulate user requirements to lighting (daylighting and electric lighting) in public buildings on the basis of a thorough literature study. The work is a joint effort of a number of scientists and represents collective knowledge in this topic. The concept of Lighting quality is the one, among...
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Banking concentration in the Baltic and Western Balkan states — selected issues
PublicationResearch background: In a rapidly changing economic environment companies deepen their cooperation, which entails in all sectors of the economy. The progressive increase in market concentration, especially in the banking sector, is caused by various reasons. Purpose of the article: The purpose of this article is to compare the tendencies within market structures in few countries which origin from similar political systems and...
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Some variants of perfect graphs related to the matching number, the vertex cover and the weakly connected domination number
PublicationGiven two types of graph theoretical parameters ρ and σ, we say that a graph G is (σ, ρ)- perfect if σ(H) = ρ(H) for every non-trivial connected induced subgraph H of G. In this work we characterize (γw, τ )-perfect graphs, (γw, α′)-perfect graphs, and (α′, τ )-perfect graphs, where γw(G), τ (G) and α′(G) denote the weakly connected domination number, the vertex cover number and the matching number of G, respectively. Moreover,...
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How Do Ionic Liquids Affect the Surface Structure of Titania Photocatalyst? An Electron-Trap Distribution-Analysis Study
PublicationTitanium(IV) oxide, titania, photocatalyst particles were prepared from titanium alkoxide in the presence of several kinds of ionic liquids, and it was clarified that a group of samples exhibited photocatalytic activity for phenol degradation under the irradiation of light of wavelength >400 nm higher than those of the other group of samples. Although the conventional structural analytical results could not be related to the activity,...
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Generalised heart rate statistics reveal neurally mediated homeostasis transients
PublicationDistributions of accelerations and decelerations, obtained from increments of heart rate recorded during a head-up tilt table (HUTT) test provide short-term characterization of the complex cardiovascular response to a rapid controlled dysregulation of homeostasis. A generalised statistic is proposed for evaluating the neural reflexes responsible for restoring the homeostatic dynamics. An evaluation of the effects on heart rate...
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Ultrasonic diagnostics of concrete T-beams used in bridge structures
PublicationThis paper describes a method of ultrasonic diagnostics used for prefabricated concrete elements. The studies are focused on the applicability of nondestructive techniques based on impulse and wave packet induced elastic waves for the condition assessment of T-shaped bridge beams. Experimental tests were performed for the prestressed beam used for the superstructure of the viaduct on A1 highway near Toruń. In addition numerical...
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Detection of damages in a rivetted plate
PublicationThe paper presents the results of damage detection in a riveted aluminium plate. The detection method has been based on Lamb wave propagation. The plate has been analysed numerically and experimentally. Numerical calculations have been carried out by the use of the time-domain spectral finite element method, while for the experimental analysis laser scanning Doppler vibrometry (LSDV) has been utilised. The panel has been excited...
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Localization and identyfication of ferromagnetic objects
PublicationA compact ferromagnetic object placed in the earthly magnetic field causes disturbance of this field. This disturbance is associated with magnetization of the object. Ferromagnetic objects have induced and can also have permanent magnetization. In methods of locating and identifying ferromagnetic objects usually is using the model of the dipol moment. Determination of the position and values of the extremes of the magnetic field...
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A new methodological approach to the noise threat evaluation based on the selected physiological properties of the human hearing system
PublicationA new way of assessment of noise-induced harmful effects on human hearing system is presented in the paper. The method takes into consideration properties of the selected physiological human hearing system. On the basis of the hearing examinations and noise measurements results and psychoacoustical noise dosimeter performance the new indicators of the noise harmfulness were proposed. The evaluation of the proposed indicators were...
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Regional observatory as a part of road safety information system
PublicationEU experience clearly indicates that it is necessary to inform and motivate the public on road unsafety to undertake specific preventive efforts, as well as making road users feel responsible for the state of road safety and seek to improve this state gradually to protect their health and life. The implementation of the Warmia-Mazury Road Safety Observatory project will not only be an excellent addition to the activities carried...
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The influence of rubber recyclate morphology on the properties of rubber-asphalt composite
PublicationIn the paper wastes, mostly in the form of used tires, were analyzed. One of the methods of waste tires application use them as a modifier of asphalt. However, the properties of rubber-asphalt composites depend on the morphology of waste tiregranulate and kind of tire recycled (car/truck). In this chapter, the influence of grinding methods of waste tire on the prop¬erties of rubber-asphalt composites were studied. SEM analysis...
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Dynamics analysis of footbridge mode shapes the s8 expressway on the basis of the results of in situ tests
PublicationNon-destructive diagnostics for structure may use dynamic measurements realized during vibrations of a facility induced by dynamic environmental impact, enforced by the use of inductors or impulse impact. Dynamic tests and the analysis were undertaken for a footbridge situated over the expressway S8. The studies in situ allowed for dynamic characteristics to be determined: frequency, shape modes and damping for respective frequency...
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Numerical simulation of the influence of the selected factors on the performance of a concrete road barrier H2/W5/B
PublicationThis paper discuss the influence of selected factors on the performance of a concrete road barrier H2/W5/B. Modelling techniques of a concrete road safety system were briefly discussed. Comparison to the full scale crash test results has been shown. The concrete road safety barrier has been investigated for evaluation of the overall damage after collision under various initial conditions. The failure assessment criterion has been...
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High-temperature kinetics study of 430L steel powder oxidized in air at 600–850 °C
PublicationThe 430L stainless steel powder with a mean particle size of 95 μm was studied to determine its high-temperature oxidation properties. Continuous thermogravimetric measurements were carried out for 100 h in air at temperatures in the range of 600–850 °C. Even though a considerable amount of Cr (up to ˜5 wt.% Cr) inside the grains was depleted – especially inside small grains – no breakaway oxidation was observed. This indicates...