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Optimization of Parameters in Macromolecular Potential Energy Functions by Conformational Space Annealing
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Prediction of Protein Structure by Template-Based Modeling Combined with the UNRES Force Field
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Chemoinformatics Methods for Studying Biomolecules
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Direct measurements, numerical predictions and simple formula estimations of welding-induced biaxial residual stresses in a full-scale steel stiffened plate structure
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Wave propagation in a sensor/actuator diffusion bond model
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Effect of Hydroxypropylation and Beta-Amylase Treatment on Complexation of Debranched Starch With Naringenin
PublicationNaringenin exhibits many health benefits but it has limited water solubility and consequently low bioavailability. The objective of this study is to investigate the effect of hydroxypropylation and enzymatic treatments on starch complexation with naringenin. Potato starch and Hylon VII are hydroxypropylated to two substitution degrees and then debranched or debranched/β‐amylase treated prior to complexing with naringenin. Both...
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Effect of Acetylation and Beta‐Amylase Treatment on Complexation of Debranched Starch with Naringenin
PublicationStarch inclusion complexation has been shown to improve solubility of water insoluble molecules. Potato starch and Hylon VII are acetylated at two levels and then debranched alone or combined with β‐amylase hydrolysis, and its complexes with naringenin are prepared in aqueous conditions and characterized in this study. Both soluble and insoluble complexes are formed with the soluble complex present in the supernatant and the insoluble...
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Adding Intelligence to Cars Using the Neural Knowledge DNA
PublicationIn this paper we propose a Neural Knowledge DNA based framework that is capable of learning from the car’s daily operation. The Neural Knowledge DNA is a novel knowledge representation and reasoning approach designed to support discovering, storing, reusing, improving, and sharing knowledge among machines and computing devices. We examine our framework for drivers' classification based on their driving behaviour. The experimental...
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An Instantaneous Engine Speed Estimation Method Using Multiple Matching Synchrosqueezing Transform
PublicationInstantaneous rotational speed measurement of the engine is crucial in routine inspection and maintenance of an automobile engine. Since the contact measurement of rotational speed is not always available, the vibration measurement has been used for noncontact rotational speed estimation methods. Unfortunately, the accuracy of the noncontact estimation methods by analyzing engine vibration frequency is not satisfactory due to the...
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Thermal analysis and experimental verification of permanent magnet synchronous motor by combining lumped-parameter thermal networks with analytical method
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ThreSpect – A Program for the Determination of the Appearance Energies of Neutral and Ionized Species
PublicationCollisions of photons and charged particles with molecules lead to their excitation, ionization, and dissociation into neutral and ionized fragments. Accurately determining thresholds of the formation of particular products plays a vital role in analyzing processes occurring during these interactions. Therefore, we present a computer program, “ThreSpect,” that allows calculating threshold energies of various species generated in...
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Wykorzystanie sztucznych sieci neuronowych do szacowania wpływu drgań na budynki jednorodzinne
PublicationW artykule przedstawiono metodę prognozowania wpływu drgań na budynki mieszkalne z wykorzystaniem sztucznych sieci neuronowych. Drgania komunikacyjne mogą doprowadzić do uszkodzenia elementów konstrukcyjnych, a nawet do awarii budynku. Najczęstszym efektem są jednak rysy, pękanie tynku i wypraw. Metody oparte na sztucznej inteligencji są przybliżone, ale stanowią wystarczająco dokładną i ekonomiczną alternatywę dla tradycyjnych...
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Urban Food Self-Production in the Perspective of Social Learning Theory: Empowering Self-Sustainability
PublicationUrban food production is becoming an increasingly significant topic in the context of climate change and food security. Conducting research on this subject is becoming an essential element of urban development, deepening knowledge regarding the benefits, challenges, and potential for the development of urban agriculture as an alternative form of food production. Responding to this need, this monograph presents the results of...
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Selection of effective cocrystals former for dissolution rate improvement of active pharmaceutical ingredients based on lipoaffinity index
PublicationNew theoretical screening procedure was proposed for appropriate selection of potential cocrystal formers possessing the ability of enhancing dissolution rates of drugs. The procedure relies on the training set comprising 102 positive and 17 negative cases of cocrystals found in the literature. Despite the fact that the only available data were of qualitative character, performed statistical analysis using binary classification...
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Distinguishing of cocrystals from simple eutectic mixtures: phenolic acids as potential pharmaceutical coformers
PublicationThe multiparameter model comprising 1D and 2D QSPR/QSAR descriptors was proposed and validated for phenolic acid binary systems. This approach is based on the optimization of regression coefficients for maximization of the percentage of true positives in the pool of systems comprising either simple binary eutectics or cocrystals. The training set consisted of 58 eutectics and 168 cocrystals. The solid dispersions collection used...
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Fertility rebound and economic growth. New evidence for 18 countries over the period 1970-2011.
PublicationLong-run impact of economic growth on fertility trends is ambiguous and sensitive for in-time variations. Noticeably, over last decades, economic growth has led in many countries to significant falls in total fertility rates. However, recently, in high-income economies a kind of ‘fertility rebound’ emerged (Goldstein, 2009; Luci and Thevenon, 2011; Day, 2012), which supports the hypothesis that reversal trends in total fertility...
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From phosphanylphosphaalkenes to coordination copper and silver polymers containing P–P bonds
PublicationThis study was focused on the activation of the C[double bond, length as m-dash]P bond via reactions of Ph2C[double bond, length as m-dash]P-PtBu2 (1) with 1,6-hexanediol and selected dithiols (1,4-butanedithiol, 1,4-benzenedithiol and 1,4-benzenedimethanethiol). These reactions proceed according to a 1,2-addition mechanism, providing new compounds with formulas {(Ph)2(H)C-P-PtBu2}{μ2-(O-(CH2)6-O)}{tBu2P-P-C(H)(Ph)2} (2), {(Ph)2(H)C-P-PtBu2}{μ2-(S-(CH2)4-S)}{tBu2P-P-C(H)(Ph)2}...
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Sonocatalytic degradation of tetracycline antibiotic using zinc oxide nanostructures loaded on nano-cellulose from waste straw as nanosonocatalyst
PublicationThe aim of the present investigation was the combination of ZnO nanostructures with nano-cellulose (NC) for the efficient degradation of tetracycline (TC) antibiotic under ultrasonic irradiation. The removal efficiency of 12.8% was obtained by the sole use of ultrasound (US), while the removal efficiency increased up to 70% by the US/ZnO treatment process. Due to the integration of ZnO nanostructures with NC, the removal efficiency...
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Telomere uncapping by common oxidative guanine lesions: Insights from atomistic models
PublicationOxidative damage to DNA is widely known to contribute to aging and disease. This relationship has been extensively studied for telomeres – structures that cap chromosome ends – due to their role in cell proliferation and senescence, and exceptional susceptibility to oxidation. Indeed, the repetitive telomeric DNA sequence contains the 5′-GGG-3′ motif that has the lowest ionization potential of all trinucleotides. Accordingly, experiments...
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Thermostability and photophysical properties of mixed-ligand carboxylate/benzimidazole Zn(II)-coordination polymers
PublicationThe reaction between Zn(NO3)2*6H2O or Zn(CH3COO)2*2H2O and isophthalic acid (1,3-H2bdc) in the presence of benzimidazole (Hbzim) in dimethylformamide (DMF)/ethanol (EtOH)/H2O solvent mixture at room temperature yielded two structurally different coordination polymers: [Zn2(1,3-bdc)2(Hbzim)2] (1) and [Zn2(1,3-bdc)(bzim)2] (2). (1) is a 2D-layered framework with a molecule of benzimidazole coordinated to the Zn center, whereas (2)...
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Copper(I) halide cluster-based coordination polymers modulated by chiral ditopic dithiodianthranilide ligands: synthesis, crystal structure and photoluminescence
PublicationReaction of copper(I) halides with chiral dithiodianthranilidesmdtaandbdtaafforded polymeric complexeswhere polynuclear CuX clusters were linked together by ditopic bridging ligands into 1D chains or 2D layerstructures. In the case of racemic ligands double stranded chain polymers were formed where the Cu4X4(X = I or Br) cores are connected by enantiomeric pairs of the ditopic ligands. In contrast, a homochiralmdtaligand created...
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Changes in the structure of Armenia’s labour resources between 1993 and 2020
PublicationThe article characterises the structure of Armenia’s labour resources in the period between1993 and 2020. It aims to assess the changes on the Armenian labour market by means of a deductive analysis of historical data and observation of changes in the structure of resources based on generally available macroeconomic data. The authors evaluate these processes against the background of demographic and economic changes, by presenting...
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Bitumen-Based Poroelastic Pavements: Successful Improvements and Remaining Issues
PublicationThis article presents the development process of designing and testing poroelastic pavement based on highly polymer-modified bitumen. Poroelastic wearing course was composed of mineral and rubber aggregate mixed with highly polymer-modified bitumen, in contrast to previous trials, during which polyurethane resins were mainly used as binder, which led to several serious technological problems concerning difficult production, insufficient...
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Instrumented end notched flexure - Crack propagation and process zonemonitoring Part II: Data reduction and experimental
PublicationA mode II instrumented end notched flexure three point bending (ENF) adhesion test is described. The adhesive joint consists of two aluminium alloy (AW7075-T6) plates bonded with a structural epoxy adhesive (Hysol EA 9395™). Strain gauges are attached to the outer surface (backface) of the substrates in the lengthwise direction to measure local surface strain during crack propagation. Simultaneously, load/displacement measurements...
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Evolution of Ag nanostructures created from thin films: UV–vis absorption and its theoretical predictions
PublicationAg-based plasmonic nanostructures were manufactured by thermal annealing of thin metallic films. Structure and morphology were studied using scanning electron microscopy (SEM), transmission electron microscopy (TEM), high-resolution transmission electron microscopy (HR-TEM) and X-ray photoelectron spectroscopy (XPS). SEM images show that the formation of nanostructures is influenced by the initial layer thickness as well as the...
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Perceptual and Motor Effects of Muscle Co-activation in a Force Production Task
PublicationWe tested several predictions of the theory of motor control with spatial referent coordinates related to effects of muscle coactivation on force production and perception. In particular, we predicted that subjects would produce unintentional force increase by finger flexors and be unaware of this force increase. Healthy subjects performed steady force production task in isometric conditions with visual feedback on the force level....
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Novel N-(aryl/heteroaryl)-2-chlorobenzenesulfonamide derivatives: synthesis and anticancer activity evaluation
PublicationA new series of N-(aryl/heteroaryl)-2-chlorobenzenesulfonamide derivatives 4-21 have been synthesized, and evaluated at the National Cancer Institute (USA) for their in vitro activities against a panel of 60 different human cancer cell lines. Among them, compounds 16, 20 and 21 exhibited remarkable cytotoxic activity against numerous human cancer cell lines. We found that sulfonamide derivative 21 appeared to be more selective...
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Unidirectional thyristor-based DC-DC converter for HVDC connection of offshore wind farms
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Channel Blockage and Flow Maldistribution during Unsteady Flow in a Model Microchannel Plate heat Exchanger
PublicationThis paper describes the problem of channel blockage as a result of flow maldistribution between the channels of a model mini channel plate heat exchanger consisting of one pass on each leg. Each leg of the heat exchanger contains 51 parallel and rectangular minichannels of four hydraulic diameters namely 461 μm, 571 μm, 750 μm and 823 μm. In addition, a more complex geometry has been investigated where for the sake of breaking...
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Determination of volatile organic compounds in water samples using membrane-solid phase microextraction (M-SPME) (headspace version)
PublicationThe results of a study on the use of membrane-solid phase microextraction (M-SPME) for sampling volatile organic compounds (VOCs) from the headspace above the liquid medium are presented. The sampled VOCs were subsequently quantified by gas chromatography (GC). Two systems were compared in this study, i.e. a novel two-phase sorption system (M-SPME), and a commercial fibre. Headspace sampling using SPME was optimized with respect...
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Annual variability of heavy metal content in Svalbard reindeer faeces as a result of dietary preferences
PublicationDuring both winter and summer, Svalbard reindeer selectively feed on different types of vegetation that are not only a source of nutritional value, but also a place of heavy metal accumulation. In the present study, the content of cadmium, chromium, copper, iron, lead, nickel, manganese, and zinc in reindeer excrement was measured. The main aims were to determine the seasonal content of several heavy metals in Svalbard reindeer...
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EXPERIMENTAL ANALYSIS OF RUBBER AND STYROFOAM BUMPERS INFLUENCE ON THE COLLIDING STRUCTURES
PublicationPast and recent investigations of colliding structures under seismic excitation confirmed that pounding may have a significant influence on the structural response. Interactions between adjacent buildings may cause serious damage to the structures, leading even to its total collapse. The main reason of earthquake-induced pounding, besides insufficient distance between structures, are differences in stiffness or mass of colliding structures....
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Effect of dendrimer-based interlayers for enzyme immobilization on a model electrochemical sensing system for glutamate
PublicationIn this paper, we discuss dendrimer usage in enzyme-based electrochemical biosensors, particularly with respect to biomolecule loading on the sensing surface. A novel approach to design bioactive layers with immobilized enzymes for electrochemical biosensors using the surface plasmon resonance (SPR) method in combination with electrochemical impedance spectroscopy was presented. The gold surface was modified with linear linkers...
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Assessment of the technological reliability of a hybrid constructed wetland for wastewater treatment in a mountain eco-tourist farm in Poland
PublicationThe aim of the present study was to assess the technological reliability of a domestic hybrid wastewater treatment installation consisting of a classic three-chambered (volume 6 m3) septic tank, a vertical flow trickling bed filled with granules of a calcinated clay material (KERAMZYT), a special wetland bed constructed on a slope, and a permeable pond used as a receiver. The test treatment plant was located at a mountain eco-tourist...
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Mikrostruktura kompozytów poliuretanowo-gumowych, otrzymywanych in situ z elastomerów uretanowych i recyklatów gumowych
PublicationW pracy przedstawiono wyniki badań dotyczące mikrostruktury nowej grupy kompozytów poliuretanowo-gumowych (KPG). Materiały kompozytowe otrzymano in situ z lanych elastomerów ure-tanowych (LEU) i różnej ilości recyklatu gumowego (RG), uzyskiwanego w wyniku kriogenicznego rozdrabniania poużytkowych opon samochodowych. Mikrostrukturę przełomów KPG zbadano przy wykorzystaniu mikroskopii optycznej (OM) oraz transmisyjnej mikroskopii...
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What about the multidrug resistance in fungi? - comparison of voriconazole and ''old'' azoles.
PublicationPorównano wyniki oznaczeń aktywności przeciwgrzybowej voriconazolu- nowego leku przeciwgrzybowego z pierścieniem azolowym, z lekami poprzedniej generacji. Zaobserwowano znaczny spadek aktywności biologicznej voriconazolu (podobnie jak starszych leków, takich jak fluconazol czy ketoconazol) względem komórek wielolekoopornych, co stanowi przesłankę, że nowy lek jest substratem dla głównych pomp kształtujących zjawisko wielolekooporności...
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Możliwości wykorzystania protokołów typu LLDP do określania położenia urządzenia VOIP
PublicationW pracy scharakteryzowano protokoły typu LLDP. Oceniono możliwość wykorzystania rozwiązań proponowanych w standardzie ANSI/TIA-1057 do umiejscawiania urządzeń VoIP w rozbudowanej sieci komputerowej. Opisano korzyści stwarzane przez implementacje protokołów LLDP dla służb ratowniczych przy identyfikacji urządzenia VoIP użytkownika wzywającego pomocy. Wskazano na niebezpieczeństwa związane z implementacją protokołu LLDP-MED.
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Velocity Field Characteristics at the Inlet to a Pipe Culvert
PublicationA poorly designed culvert inlet structure causes scouring, which can lead to the collapse of the culvert and significant damage to the neighboring land. A set of laboratory tests was evaluated to examine velocity distribution at the culvert inlet. A three-dimensional acoustic Doppler velocimeterwas used to measure instantaneous flowvelocity upstream of the culvert. The analysis of mean velocities, turbulence strength, and Reynolds...
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Neufunde von fossilen Harzen aus dem Mitteldeutschen Braunkohlenrevier
PublicationEs werden einige Neufunde von fossilen Harzen aus ded tertiaren Braunkohlenvorkommen Mitteldeutschlands aus Sachsen-Anhalt vorgestellt. Die Fundstucke wurden mit dem Vergleichsmaterial der Harzammulung des Geiseltalmuseums in Halle/Saale und den privaten Harzsammlungen von G. Krumbiegiel und R. Wimmer makropetrographisch verglichen. Sie werden erstmalig beschrieben und die Ergebnisse der Infrarotabsorptions-Spektroskopie prasentiert.
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Music Recommendation System
PublicationThe paper focuses on optimization vector content feature for the music recommendation system. For the purpose of experiments a database is created consisting of excerpts of music les. They are assigned to 22 classes corresponding to dierent music genres. Various feature vectors based on low-level signal descriptors are tested and then optimized using correlation analysis and Principal Component Analysis (PCA). Results of the experiments...
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Environmental impact of construction. Methods of conscious shaping architecture in terms of ecological solutions
PublicationShaping an ecologically conscious society is a process that also affects architecture. Currently, designers are eagerly looking for solutions that are beneficial in terms of carbon footprint. For the proper multi-criteria assessment and selection of adequate solutions, it is necessary to use appropriate tools such as, for example, the Life Cycle Assessment (LCA) method or the rules of ecological certification (BREEAM and LEED)....
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Badania nad wykorzystaniem fotokatalizatorów WO3/TiO2 do degradacji wybranych zanieczyszczeń organicznych
PublicationW dysertacji skupiono się na: preparatyce fotokatalizatorów WO3/TiO2, weryfikacji efektywności działania kompozytów w kierunku fotokatalitycznego usuwania zanieczyszczeń oraz analizie wyników pod kątem zaprojektowania i skonstruowania fotoreaktora wyposażonego w sterowane źródło światła LED do fotokatalitycznej degradacji zanieczyszczeń. Fotokatalizatory otrzymano łącząc dwie metody preparatyki – zol-żel i hydrotermalną. Otrzymano...
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Opinions and view of entrepreneurs regerding the single european Market-Analytical Model. W: Entrepreneurship and small business development in the21st century. Przedsiębiorczość i rozwój małych i średnich przedsiebiorstww XI wieku. Ed. B. Piasecki. Łódź: Uniw. Łódź**2002 s. 109-117.**2002 s. 109 - 117 Opinie i poglądy przedsiębiorców na temat Jednolitego Rynku Europejskiego - model analityczny.
PublicationArtykuł zawiera propozycje modelu czynników kształtujących świadomość pol-skich przedsiębiorców odnośnie szans i zagrożeń w związku z otwarciem gospodarki Polski na Jednolitu Rynek Europejski. Model ten musi być wykorzystany przy projektowaniu badań opinii i poglądów przedsiębiorców.
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Production activity control in a flexible machining cell considering part measuring condition. W: Computer integrated manufacturing. Advanced design and management. Ed.: B. Skołud, D. Krenczyk. Warszawa: Wydaw. Nauk.-Tech. **2003 s. 494-501, 6 rys. 1 tabl. bibliogr. 9 poz. Sterowanie procesu produkcyjnego w elastycznym gnieździe obróbkowym z uwzg- lędnieniem funkcji kontroli wytwarzanych przedmiotów.
PublicationPrzedstawiono modele struktur organizacyjnych przebiegu procesu organizacyj-nego w rzeczywistym zrobotyzowanym elastycznym gnieździe obróbki (EGO) z udziałem współrzędnościowej maszyny pomiarowej CNC. Badano eksperymentalnie występujące współzależności pomiędzy analizowanymi planami kontroli przed-miotów wytwarzanych i strategiami szeregowania operacji procesu technologi-cznego obróbki, z wykorzystaniem zintegrowanych modeli...
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Capacitively coupled ECG measurements - a CMRR circuit improvement
PublicationA typical galvanic-connected electrocardiogram (ECG) measurement system utilizes two signal’s electrodes and a third one in driven-right-leg (DRL) circuit for improving a common-mode rejection ratio(CMRR) of the acquisition system. In capacitive-coupled ECG similar techniques are used, however it is expected, that the utilized DRL subsystem is formed using a capacitive coupling approach, too. An improvement of the acquisition system...
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Konstrukcje morskich farm wiatrowych – wyzywanie dla projektantów
PublicationPozyskanie energii wiatru jest jednym z najbardziej obiecujących źródeł energii odnawialnej. W artykule przestawiono zagadnienia związane z rozwojem energetyki wiatrowej, w tym budową morskich farm wiatrowych. W szczególności zaś zaprezentowano podstawy energetyki wiatrowej, stan aktualny i perspektywy rozwoju morskich farm wiatrowych, elementy konstrukcyjne morskich turbin wiatrowych oraz infrastrukturę przesyłania energii na...
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NOBLE METAL MODIFIED TiO2 FOR PHOTOCATALYTIC AIR PURIFICATION
PublicationTiO2 was surface modified with silver, gold, palladium and platinum ion clusters to improve its photocatalytic activity. The effect of metal content, the kind of dopant used during preparation procedure on the photoactivity were investigated. in toluene removal which was used as a model volatile organic compound. Toluene, at the concentration of about 100 ppm, was irradiated over noble metal modified TiO2 using light-emitting diodes...
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Design of Inner Gate for CRIST Shipyard Dry Dock
PublicationThe paper deals with a removable steel inner gate which was designed to separate two parts of a dry dock of about 70 m in width and 380 m in length. The gate allows for independent assembly of ship structures in two separated parts of the dock. The fore part of the dock can be flooded while the after part is dry. Tthe gate was designed by IDEK Company Ltd in 2011 and it was soon constructed and used by CRIST Shipyard in Gdynia.
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S&YP + Mentors + Peace + Love = Science and Growing
PublicationIn this extraordinarily difficult time, we understand better that only peace, love, and cooperation are the keys to growing in technology for humanity. Let us learn from our mentors how they grow from their hard work and international cooperation. Thanks to Prof. Giuseppe Buja and Prof. Zbigniew Krzemiński, we have unique schools of adjustable speed drives that are helping people convert electrical to mechanical power and vice...
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Co-gasification of waste biomass-low grade coal mix using downdraft gasifier coupled with dual-fuel engine system: Multi-objective optimization with hybrid approach using RSM and Grey Wolf Optimizer
PublicationThe looming global crisis over increasing greenhouse gases and rapid depletion of fossil fuels are the motivation factors for researchers to search for alternative fuels. There is a need for more sustainable and less polluting fuels for internal combustion engines. Biomass offers significant potential as a feed material for gasification to produce gaseous fuel. It is carbon neutral, versatile, and abundant on earth. The present...